Biginelli reaction (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "Biginelli reaction" in English language version.

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20doi.org

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6nih.gov

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2zenodo.org

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2worldcat.org

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1semanticscholar.org

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doi.org

Biginelli, P. (1891). "Ueber Aldehyduramide des Acetessigäthers". Chemische Berichte. 24: 1317–1319. doi:10.1002/cber.189102401228.
Biginelli, P. (1891). "Ueber Aldehyduramide des Acetessigäthers. II". Chemische Berichte. 24 (2): 2962–2967. doi:10.1002/cber.189102402126.
Zaugg, H. E.; Martin, W. B. (1965). "Α-Amidoalkylations at Carbon". Org. React. 14: 88. doi:10.1002/0471264180.or014.02. ISBN 0471264180.
Kappe, C. O. (1993). "100 years of the biginelli dihydropyrimidine synthesis". Tetrahedron. 49 (32): 6937–6963. doi:10.1016/S0040-4020(01)87971-0.
Kappe, C. O.; Stadler, A. (2004). "The Biginelli Dihydropyrimidine Synthesis". Organic Reactions. 63: 1–116. doi:10.1002/0471264180.or063.01. ISBN 0471264180.
Song, Dailei; Wang, Runxia; Chen, Yongli; Zhang, Shaohua; Liu, Chunsheng; Luo, Genxiang (2008). "Copper(II) trifluoroacetate catalyzed synthesis of 3,4- dihydropyrimidin-2(1H)-ones under solvent-free conditions". Reaction Kinetics and Catalysis Letters. 95 (2): 385. doi:10.1007/s11144-008-5379-2. S2CID 93287161.
Hu, E. H.; Sidler, D. R.; Dolling, U.-H. (1998). "Unprecedented Catalytic Three Component One-Pot Condensation Reaction: An Efficient Synthesis of 5-Alkoxycarbonyl- 4-aryl-3,4-dihydropyrimidin-2(1H)-ones". J. Org. Chem. 63 (10): 3454. doi:10.1021/jo970846u.
Wipf, P.; Cunningham, A. (1995). "A solid phase protocol of the biginelli dihydropyrimidine synthesis suitable for combinatorial chemistry". Tetrahedron Lett. 36 (43): 7819–7822. doi:10.1016/0040-4039(95)01660-A.
Kappe, C. O. (2000). "Highly versatile solid phase synthesis of biofunctional 4-aryl-3,4-dihydropyrimidines using resin-bound isothiourea building blocks and multidirectional resin cleavage". Bioorg. Med. Chem. Lett. 10 (1): 49–51. doi:10.1016/S0960-894X(99)00572-7. PMID 10636241.
Rovnyak, G. C.; Atwal, K. S.; Hedberg, A.; Kimball, S. D.; Moreland, S.; Gougoutas, J. Z.; O'Reilly, B. C.; Schwartz, J.; Malley, M. F. (1992). "Dihydropyrimidine calcium channel blockers. 4. Basic 3-substituted-4-aryl-1,4-dihydropyrimidine-5-carboxylic acid esters. Potent antihypertensive agents". J. Med. Chem. 35 (17): 3254–3263. doi:10.1021/jm00095a023. PMID 1387168.
Crespo, Abel; El Maatougui, Abdelaziz; Biagini, Pierfrancesco; Azuaje, Jhonny; Coelho, Alberto; Brea, José; Loza, María Isabel; Cadavid, María Isabel; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2013-10-03). "Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists". ACS Medicinal Chemistry Letters. 4 (11): 1031–1036. doi:10.1021/ml400185v. ISSN 1948-5875. PMC 4027370. PMID 24900602.
El Maatougui, Abdelaziz; Azuaje, Jhonny; González-Gómez, Manuel; Miguez, Gabriel; Crespo, Abel; Carbajales, Carlos; Escalante, Luz; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2016-03-10). "Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes". Journal of Medicinal Chemistry. 59 (5): 1967–1983. doi:10.1021/acs.jmedchem.5b01586. ISSN 0022-2623. PMID 26824742.
Folkers, K.; Johnson, T. B. (1933). "Researches on Pyrimidines. CXXXVI. The Mechanism of Formation of Tetrahydropyrimidines by the Biginelli Reaction1". J. Am. Chem. Soc. 55 (9): 3784–3791. doi:10.1021/ja01336a054.
Sweet, F.; Fissekis, J. D. (1973). "Synthesis of 3,4-dihydro-2(1H)-pyrimidinones and the mechanism of the Biginelli reaction". J. Am. Chem. Soc. 95 (26): 8741–8749. doi:10.1021/ja00807a040.
Folkers, K.; Harwood, H. J.; Johnson, T. B. (1932). "Researches on Pyrimidines. Cxxx. Synthesis of 2-Keto-1,2,3,4-Tetrahydropyrimidines". J. Am. Chem. Soc. 54 (9): 3751–3758. doi:10.1021/ja01348a040.
Kappe, C.O. (1997). "A Reexamination of the Mechanism of the Biginelli Dihydropyrimidine Synthesis. Support for anN-Acyliminium Ion Intermediate1". J. Org. Chem. 62 (21): 7201–7204. doi:10.1021/jo971010u. PMID 11671828.
O'Reilly, B. C.; Atwal, K. S. (1987). "Synthesis of Substituted 1,2,3,4-Tetrahydro-6-methyl-2-oxo-5-pyrimidinecarboxylic Acid Esters: The Biginelli Condensation Revisited". Heterocycles. 26 (5): 1185–1188. doi:10.3987/R-1987-05-1185.
O'Reilly, B. C.; Atwal, K. S. (1987). "Synthesis of Substituted 1,2,3,4-Tetrahydro-6-methyl-2-thioxo-5-pyrimidinecarboxylic Acid Esters". Heterocycles. 26 (5): 1189–1192. doi:10.3987/R-1987-05-1189.
Kumar, Atul; Maurya, Ram Awatar (2007). "An efficient bakers' yeast catalyzed synthesis of 3,4-dihydropyrimidin-2-(1H)-ones". Tetrahedron Letters. 48 (26): 4569. doi:10.1016/j.tetlet.2007.04.130.
Panda, S.S.; Khanna, P.; Khanna, L. (2012). "Biginelli Reaction: A Green Perspective". Curr. Org. Chem. 16 (4): 507–520. doi:10.2174/138527212799499859.

nih.gov

pubmed.ncbi.nlm.nih.gov

Kappe, C. O. (2000). "Highly versatile solid phase synthesis of biofunctional 4-aryl-3,4-dihydropyrimidines using resin-bound isothiourea building blocks and multidirectional resin cleavage". Bioorg. Med. Chem. Lett. 10 (1): 49–51. doi:10.1016/S0960-894X(99)00572-7. PMID 10636241.
Rovnyak, G. C.; Atwal, K. S.; Hedberg, A.; Kimball, S. D.; Moreland, S.; Gougoutas, J. Z.; O'Reilly, B. C.; Schwartz, J.; Malley, M. F. (1992). "Dihydropyrimidine calcium channel blockers. 4. Basic 3-substituted-4-aryl-1,4-dihydropyrimidine-5-carboxylic acid esters. Potent antihypertensive agents". J. Med. Chem. 35 (17): 3254–3263. doi:10.1021/jm00095a023. PMID 1387168.
Crespo, Abel; El Maatougui, Abdelaziz; Biagini, Pierfrancesco; Azuaje, Jhonny; Coelho, Alberto; Brea, José; Loza, María Isabel; Cadavid, María Isabel; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2013-10-03). "Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists". ACS Medicinal Chemistry Letters. 4 (11): 1031–1036. doi:10.1021/ml400185v. ISSN 1948-5875. PMC 4027370. PMID 24900602.
El Maatougui, Abdelaziz; Azuaje, Jhonny; González-Gómez, Manuel; Miguez, Gabriel; Crespo, Abel; Carbajales, Carlos; Escalante, Luz; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2016-03-10). "Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes". Journal of Medicinal Chemistry. 59 (5): 1967–1983. doi:10.1021/acs.jmedchem.5b01586. ISSN 0022-2623. PMID 26824742.
Kappe, C.O. (1997). "A Reexamination of the Mechanism of the Biginelli Dihydropyrimidine Synthesis. Support for anN-Acyliminium Ion Intermediate1". J. Org. Chem. 62 (21): 7201–7204. doi:10.1021/jo971010u. PMID 11671828.

ncbi.nlm.nih.gov

Crespo, Abel; El Maatougui, Abdelaziz; Biagini, Pierfrancesco; Azuaje, Jhonny; Coelho, Alberto; Brea, José; Loza, María Isabel; Cadavid, María Isabel; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2013-10-03). "Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists". ACS Medicinal Chemistry Letters. 4 (11): 1031–1036. doi:10.1021/ml400185v. ISSN 1948-5875. PMC 4027370. PMID 24900602.

researchgate.net

Panda, S.S.; Khanna, P.; Khanna, L. (2012). "Biginelli Reaction: A Green Perspective". Curr. Org. Chem. 16 (4): 507–520. doi:10.2174/138527212799499859.

semanticscholar.org

api.semanticscholar.org

Song, Dailei; Wang, Runxia; Chen, Yongli; Zhang, Shaohua; Liu, Chunsheng; Luo, Genxiang (2008). "Copper(II) trifluoroacetate catalyzed synthesis of 3,4- dihydropyrimidin-2(1H)-ones under solvent-free conditions". Reaction Kinetics and Catalysis Letters. 95 (2): 385. doi:10.1007/s11144-008-5379-2. S2CID 93287161.

worldcat.org

search.worldcat.org

Crespo, Abel; El Maatougui, Abdelaziz; Biagini, Pierfrancesco; Azuaje, Jhonny; Coelho, Alberto; Brea, José; Loza, María Isabel; Cadavid, María Isabel; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2013-10-03). "Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists". ACS Medicinal Chemistry Letters. 4 (11): 1031–1036. doi:10.1021/ml400185v. ISSN 1948-5875. PMC 4027370. PMID 24900602.
El Maatougui, Abdelaziz; Azuaje, Jhonny; González-Gómez, Manuel; Miguez, Gabriel; Crespo, Abel; Carbajales, Carlos; Escalante, Luz; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy (2016-03-10). "Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes". Journal of Medicinal Chemistry. 59 (5): 1967–1983. doi:10.1021/acs.jmedchem.5b01586. ISSN 0022-2623. PMID 26824742.

zenodo.org

Biginelli, P. (1891). "Ueber Aldehyduramide des Acetessigäthers". Chemische Berichte. 24: 1317–1319. doi:10.1002/cber.189102401228.
Biginelli, P. (1891). "Ueber Aldehyduramide des Acetessigäthers. II". Chemische Berichte. 24 (2): 2962–2967. doi:10.1002/cber.189102402126.