Libert F, Parmentier M, Lefort A, Dinsart C, Van Sande J, Maenhaut C, Simons MJ, Dumont JE, Vassart G (May 1989). „Selective amplification and cloning of four new members of the G protein-coupled receptor family”. Science244 (4904): 569–72. DOI:10.1126/science.2541503. PMID2541503.
Libert F, Passage E, Parmentier M, Simons MJ, Vassart G, Mattei MG (September 1991). „Chromosomal mapping of A1 and A2 adenosine receptors, VIP receptor, and a new subtype of serotonin receptor”. Genomics11 (1): 225–7. DOI:10.1016/0888-7543(91)90125-X. PMID1662665.
Ciruela F, Casadó V, Rodrigues RJ, Luján R, Burgueño J, Canals M, Borycz J, Rebola N, Goldberg SR, Mallol J, Cortés A, Canela EI, López-Giménez JF, Milligan G, Lluis C, Cunha RA, Ferré S, Franco R (February 2006). „Presynaptic control of striatal glutamatergic neurotransmission by adenosine A1-A2A receptor heteromers”. The Journal of Neuroscience : the Official Journal of the Society for Neuroscience26 (7): 2080–7. DOI:10.1523/JNEUROSCI.3574-05.2006. PMID16481441.
Simola N, Morelli M, Pinna A (2008). „Adenosine A2A receptor antagonists and Parkinson's disease: state of the art and future directions”. Current Pharmaceutical Design14 (15): 1475–89. DOI:10.2174/138161208784480072. PMID18537671.
Morelli M, Di Paolo T, Wardas J, Calon F, Xiao D, Schwarzschild MA (December 2007). „Role of adenosine A2A receptors in parkinsonian motor impairment and l-DOPA-induced motor complications”. Progress in Neurobiology83 (5): 293–309. DOI:10.1016/j.pneurobio.2007.07.001. PMID17826884.
Brown RM, Short JL (November 2008). „Adenosine A(2A) receptors and their role in drug addiction”. The Journal of Pharmacy and Pharmacology60 (11): 1409–30. DOI:10.1211/jpp/60.11.0001. PMID18957161.
Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Monopoli A, Ongini E, Varani K, Borea PA (January 2002). „7-Substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: a study on the importance of modifications at the side chain on the activity and solubility”. Journal of Medicinal Chemistry45 (1): 115–26. DOI:10.1021/jm010924c. PMID11754583.
Baraldi PG, Fruttarolo F, Tabrizi MA, Preti D, Romagnoli R, El-Kashef H, Moorman A, Varani K, Gessi S, Merighi S, Borea PA (March 2003). „Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists”. Journal of Medicinal Chemistry46 (7): 1229–41. DOI:10.1021/jm021023m. PMID12646033.
Cristalli G, Cacciari B, Dal Ben D, Lambertucci C, Moro S, Spalluto G, Volpini R (March 2007). „Highlights on the development of A(2A) adenosine receptor agonists and antagonists”. ChemMedChem2 (3): 260–81. DOI:10.1002/cmdc.200600193. PMID17177231.
Cristalli G, Lambertucci C, Marucci G, Volpini R, Dal Ben D (2008). „A2A adenosine receptor and its modulators: overview on a druggable GPCR and on structure-activity relationship analysis and binding requirements of agonists and antagonists”. Current Pharmaceutical Design14 (15): 1525–52. DOI:10.2174/138161208784480081. PMID18537675.
Gillespie RJ, Adams DR, Bebbington D, Benwell K, Cliffe IA, Dawson CE, Dourish CT, Fletcher A, Gaur S, Giles PR, Jordan AM, Knight AR, Knutsen LJ, Lawrence A, Lerpiniere J, Misra A, Porter RH, Pratt RM, Shepherd R, Upton R, Ward SE, Weiss SM, Williamson DS (May 2008). „Antagonists of the human adenosine A2A receptor. Part 1: Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives”. Bioorganic & Medicinal Chemistry Letters18 (9): 2916–9. DOI:10.1016/j.bmcl.2008.03.075. PMID18406614.
Gillespie RJ, Cliffe IA, Dawson CE, Dourish CT, Gaur S, Giles PR, Jordan AM, Knight AR, Lawrence A, Lerpiniere J, Misra A, Pratt RM, Todd RS, Upton R, Weiss SM, Williamson DS (May 2008). „Antagonists of the human adenosine A2A receptor. Part 2: Design and synthesis of 4-arylthieno[3,2-d]pyrimidine derivatives”. Bioorganic & Medicinal Chemistry Letters18 (9): 2920–3. DOI:10.1016/j.bmcl.2008.03.076. PMID18407496.
Gillespie RJ, Cliffe IA, Dawson CE, Dourish CT, Gaur S, Jordan AM, Knight AR, Lerpiniere J, Misra A, Pratt RM, Roffey J, Stratton GC, Upton R, Weiss SM, Williamson DS (May 2008). „Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines”. Bioorganic & Medicinal Chemistry Letters18 (9): 2924–9. DOI:10.1016/j.bmcl.2008.03.072. PMID18411049.
Lappas CM, Sullivan GW, Linden J (July 2005). „Adenosine A2A agonists in development for the treatment of inflammation”. Expert Opinion on Investigational Drugs14 (7): 797–806. DOI:10.1517/13543784.14.7.797. PMID16022569.
Lobato KR, Binfaré RW, Budni J, Rosa AO, Santos AR, Rodrigues AL (May 2008). „Involvement of the adenosine A1 and A2A receptors in the antidepressant-like effect of zinc in the forced swimming test”. Progress in Neuro-psychopharmacology & Biological Psychiatry32 (4): 994–9. DOI:10.1016/j.pnpbp.2008.01.012. PMID18289757.
Mader TJ, Bertolet B, Ornato JP, Gutterman JM (2000). „Aminophylline in the treatment of atropine-resistant bradyasystole”. Resuscitation47 (2): 105–12. DOI:10.1016/S0300-9572(00)00234-3. PMID11008148.
Mader TJ, Smithline HA, Durkin L, Scriver G (2003). „A randomized controlled trial of intravenous aminophylline for atropine-resistant out-of-hospital asystolic cardiac arrest”. Academic emergency medicine : official journal of the Society for Academic Emergency Medicine10 (3): 192–7. DOI:10.1197/aemj.10.3.192. PMID12615581.
Pinna A, Wardas J, Simola N, Morelli M (November 2005). „New therapies for the treatment of Parkinson's disease: adenosine A2A receptor antagonists”. Life Sciences77 (26): 3259–67. DOI:10.1016/j.lfs.2005.04.029. PMID15979104.
Hodgson RA, Bertorelli R, Varty GB, Lachowicz JE, Forlani A, Fredduzzi S, Cohen-Williams ME, Higgins GA, Impagnatiello F, Nicolussi E, Parra LE, Foster C, Zhai Y, Neustadt BR, Stamford AW, Parker EM, Reggiani A, Hunter JC (March 2009). „Characterization of the Potent and Highly Selective A2A Receptor Antagonists Preladenant and SCH 412348 in Rodent Models of Movement Disorders and Depression”. The Journal of Pharmacology and Experimental Therapeutics330 (1): 294–303. DOI:10.1124/jpet.108.149617. PMID19332567.
Pinna A, Fenu S, Morelli M (March 2001). „Motor stimulant effects of the adenosine A2A receptor antagonist SCH 58261 do not develop tolerance after repeated treatments in 6-hydroxydopamine-lesioned rats”. Synapse39 (3): 233–8. DOI:10.1002/1098-2396(20010301)39:3<233::AID-SYN1004>3.0.CO;2-K. PMID11284438.
Rose S, Jackson MJ, Smith LA, Stockwell K, Johnson L, Carminati P, Jenner P (September 2006). „The novel adenosine A2a receptor antagonist ST1535 potentiates the effects of a threshold dose of L-DOPA in MPTP treated common marmosets”. European Journal of Pharmacology546 (1-3): 82–7. DOI:10.1016/j.ejphar.2006.07.017. PMID16925991.
Kamiya, Toshio; Saitoh Osamu, Yoshioka Kazuaki, Nakata Hiroyasu (June 2003). „Oligomerization of adenosine A2A and dopamine D2 receptors in living cells”. Biochem. Biophys. Res. Commun. (United States) 306 (2): 544–9. DOI:10.1016/S0006-291X(03)00991-4. ISSN0006-291X. PMID12804599.
Libert F, Parmentier M, Lefort A, Dinsart C, Van Sande J, Maenhaut C, Simons MJ, Dumont JE, Vassart G (May 1989). „Selective amplification and cloning of four new members of the G protein-coupled receptor family”. Science244 (4904): 569–72. DOI:10.1126/science.2541503. PMID2541503.
Libert F, Passage E, Parmentier M, Simons MJ, Vassart G, Mattei MG (September 1991). „Chromosomal mapping of A1 and A2 adenosine receptors, VIP receptor, and a new subtype of serotonin receptor”. Genomics11 (1): 225–7. DOI:10.1016/0888-7543(91)90125-X. PMID1662665.
Ciruela F, Casadó V, Rodrigues RJ, Luján R, Burgueño J, Canals M, Borycz J, Rebola N, Goldberg SR, Mallol J, Cortés A, Canela EI, López-Giménez JF, Milligan G, Lluis C, Cunha RA, Ferré S, Franco R (February 2006). „Presynaptic control of striatal glutamatergic neurotransmission by adenosine A1-A2A receptor heteromers”. The Journal of Neuroscience : the Official Journal of the Society for Neuroscience26 (7): 2080–7. DOI:10.1523/JNEUROSCI.3574-05.2006. PMID16481441.
Simola N, Morelli M, Pinna A (2008). „Adenosine A2A receptor antagonists and Parkinson's disease: state of the art and future directions”. Current Pharmaceutical Design14 (15): 1475–89. DOI:10.2174/138161208784480072. PMID18537671.
Morelli M, Di Paolo T, Wardas J, Calon F, Xiao D, Schwarzschild MA (December 2007). „Role of adenosine A2A receptors in parkinsonian motor impairment and l-DOPA-induced motor complications”. Progress in Neurobiology83 (5): 293–309. DOI:10.1016/j.pneurobio.2007.07.001. PMID17826884.
Brown RM, Short JL (November 2008). „Adenosine A(2A) receptors and their role in drug addiction”. The Journal of Pharmacy and Pharmacology60 (11): 1409–30. DOI:10.1211/jpp/60.11.0001. PMID18957161.
Ongini E, Monopoli A, Cacciari B, Baraldi PG (2001). „Selective adenosine A2A receptor antagonists”. Farmaco (Società Chimica Italiana : 1989)56 (1-2): 87–90. PMID11347973.
Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Monopoli A, Ongini E, Varani K, Borea PA (January 2002). „7-Substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: a study on the importance of modifications at the side chain on the activity and solubility”. Journal of Medicinal Chemistry45 (1): 115–26. DOI:10.1021/jm010924c. PMID11754583.
Baraldi PG, Fruttarolo F, Tabrizi MA, Preti D, Romagnoli R, El-Kashef H, Moorman A, Varani K, Gessi S, Merighi S, Borea PA (March 2003). „Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists”. Journal of Medicinal Chemistry46 (7): 1229–41. DOI:10.1021/jm021023m. PMID12646033.
Cristalli G, Cacciari B, Dal Ben D, Lambertucci C, Moro S, Spalluto G, Volpini R (March 2007). „Highlights on the development of A(2A) adenosine receptor agonists and antagonists”. ChemMedChem2 (3): 260–81. DOI:10.1002/cmdc.200600193. PMID17177231.
Cristalli G, Lambertucci C, Marucci G, Volpini R, Dal Ben D (2008). „A2A adenosine receptor and its modulators: overview on a druggable GPCR and on structure-activity relationship analysis and binding requirements of agonists and antagonists”. Current Pharmaceutical Design14 (15): 1525–52. DOI:10.2174/138161208784480081. PMID18537675.
Gillespie RJ, Adams DR, Bebbington D, Benwell K, Cliffe IA, Dawson CE, Dourish CT, Fletcher A, Gaur S, Giles PR, Jordan AM, Knight AR, Knutsen LJ, Lawrence A, Lerpiniere J, Misra A, Porter RH, Pratt RM, Shepherd R, Upton R, Ward SE, Weiss SM, Williamson DS (May 2008). „Antagonists of the human adenosine A2A receptor. Part 1: Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives”. Bioorganic & Medicinal Chemistry Letters18 (9): 2916–9. DOI:10.1016/j.bmcl.2008.03.075. PMID18406614.
Gillespie RJ, Cliffe IA, Dawson CE, Dourish CT, Gaur S, Giles PR, Jordan AM, Knight AR, Lawrence A, Lerpiniere J, Misra A, Pratt RM, Todd RS, Upton R, Weiss SM, Williamson DS (May 2008). „Antagonists of the human adenosine A2A receptor. Part 2: Design and synthesis of 4-arylthieno[3,2-d]pyrimidine derivatives”. Bioorganic & Medicinal Chemistry Letters18 (9): 2920–3. DOI:10.1016/j.bmcl.2008.03.076. PMID18407496.
Gillespie RJ, Cliffe IA, Dawson CE, Dourish CT, Gaur S, Jordan AM, Knight AR, Lerpiniere J, Misra A, Pratt RM, Roffey J, Stratton GC, Upton R, Weiss SM, Williamson DS (May 2008). „Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines”. Bioorganic & Medicinal Chemistry Letters18 (9): 2924–9. DOI:10.1016/j.bmcl.2008.03.072. PMID18411049.
Sullivan GW (November 2003). „Adenosine A2A receptor agonists as anti-inflammatory agents”. Current Opinion in Investigational Drugs (London, England : 2000)4 (11): 1313–9. PMID14758770.
Lappas CM, Sullivan GW, Linden J (July 2005). „Adenosine A2A agonists in development for the treatment of inflammation”. Expert Opinion on Investigational Drugs14 (7): 797–806. DOI:10.1517/13543784.14.7.797. PMID16022569.
Lobato KR, Binfaré RW, Budni J, Rosa AO, Santos AR, Rodrigues AL (May 2008). „Involvement of the adenosine A1 and A2A receptors in the antidepressant-like effect of zinc in the forced swimming test”. Progress in Neuro-psychopharmacology & Biological Psychiatry32 (4): 994–9. DOI:10.1016/j.pnpbp.2008.01.012. PMID18289757.
Mader TJ, Bertolet B, Ornato JP, Gutterman JM (2000). „Aminophylline in the treatment of atropine-resistant bradyasystole”. Resuscitation47 (2): 105–12. DOI:10.1016/S0300-9572(00)00234-3. PMID11008148.
Mader TJ, Smithline HA, Durkin L, Scriver G (2003). „A randomized controlled trial of intravenous aminophylline for atropine-resistant out-of-hospital asystolic cardiac arrest”. Academic emergency medicine : official journal of the Society for Academic Emergency Medicine10 (3): 192–7. DOI:10.1197/aemj.10.3.192. PMID12615581.
Pinna A, Wardas J, Simola N, Morelli M (November 2005). „New therapies for the treatment of Parkinson's disease: adenosine A2A receptor antagonists”. Life Sciences77 (26): 3259–67. DOI:10.1016/j.lfs.2005.04.029. PMID15979104.
Hodgson RA, Bertorelli R, Varty GB, Lachowicz JE, Forlani A, Fredduzzi S, Cohen-Williams ME, Higgins GA, Impagnatiello F, Nicolussi E, Parra LE, Foster C, Zhai Y, Neustadt BR, Stamford AW, Parker EM, Reggiani A, Hunter JC (March 2009). „Characterization of the Potent and Highly Selective A2A Receptor Antagonists Preladenant and SCH 412348 in Rodent Models of Movement Disorders and Depression”. The Journal of Pharmacology and Experimental Therapeutics330 (1): 294–303. DOI:10.1124/jpet.108.149617. PMID19332567.
Pinna A, Fenu S, Morelli M (March 2001). „Motor stimulant effects of the adenosine A2A receptor antagonist SCH 58261 do not develop tolerance after repeated treatments in 6-hydroxydopamine-lesioned rats”. Synapse39 (3): 233–8. DOI:10.1002/1098-2396(20010301)39:3<233::AID-SYN1004>3.0.CO;2-K. PMID11284438.
Rose S, Jackson MJ, Smith LA, Stockwell K, Johnson L, Carminati P, Jenner P (September 2006). „The novel adenosine A2a receptor antagonist ST1535 potentiates the effects of a threshold dose of L-DOPA in MPTP treated common marmosets”. European Journal of Pharmacology546 (1-3): 82–7. DOI:10.1016/j.ejphar.2006.07.017. PMID16925991.
Kamiya, Toshio; Saitoh Osamu, Yoshioka Kazuaki, Nakata Hiroyasu (June 2003). „Oligomerization of adenosine A2A and dopamine D2 receptors in living cells”. Biochem. Biophys. Res. Commun. (United States) 306 (2): 544–9. DOI:10.1016/S0006-291X(03)00991-4. ISSN0006-291X. PMID12804599.