Jagabandhu Das, Ping Chen, Derek Norris, Ramesh Padmanabha, James Lin, Robert V. Moquin, Zhongqi Shen, Lynda S. Cook, Arthur M. Doweyko, Sidney Pitt, Suhong Pang, Ding Ren Shen, Qiong Fang, Henry F. de Fex, Kim W. McIntyre, David J. Shuster, Kathleen M. Gillooly, Kamelia Behnia, Gary L. Schieven, John Wityak, Joel C. Barrish: 2-Aminothiazole as a Novel Kinase Inhibitor Template. Structure-Activity Relationship Studies toward the Discovery of N-(2-Chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl}amino)-1,3-thiazole-5-carboxamide (Dasatinib, BMS-354825) as a Potent pan-Src Kinase Inhibitor. In: Journal of Medicinal Chemistry, 49, 2006, S. 6819–6832, PMID 17154512, doi:10.1021/jm060727j.
Jagabandhu Das, Ping Chen, Derek Norris, Ramesh Padmanabha, James Lin, Robert V. Moquin, Zhongqi Shen, Lynda S. Cook, Arthur M. Doweyko, Sidney Pitt, Suhong Pang, Ding Ren Shen, Qiong Fang, Henry F. de Fex, Kim W. McIntyre, David J. Shuster, Kathleen M. Gillooly, Kamelia Behnia, Gary L. Schieven, John Wityak, Joel C. Barrish: 2-Aminothiazole as a Novel Kinase Inhibitor Template. Structure-Activity Relationship Studies toward the Discovery of N-(2-Chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl}amino)-1,3-thiazole-5-carboxamide (Dasatinib, BMS-354825) as a Potent pan-Src Kinase Inhibitor. In: Journal of Medicinal Chemistry, 49, 2006, S. 6819–6832, PMID 17154512, doi:10.1021/jm060727j.