References analysis of the Wikipedia article "Adenosine A2A receptor" in the English version

doi.org

Libert F, Parmentier M, Lefort A, Dinsart C, Van Sande J, Maenhaut C, et al. (May 1989). "Selective amplification and cloning of four new members of the G protein-coupled receptor family". Science. 244 (4904): 569–72. Bibcode:1989Sci...244..569L. doi:10.1126/science.2541503. PMID 2541503.

Libert F, Passage E, Parmentier M, Simons MJ, Vassart G, Mattei MG (September 1991). "Chromosomal mapping of A1 and A2 adenosine receptors, VIP receptor, and a new subtype of serotonin receptor". Genomics. 11 (1): 225–7. doi:10.1016/0888-7543(91)90125-X. PMID 1662665.

PDB: 3EML; Jaakola VP, Griffith MT, Hanson MA, Cherezov V, Chien EY, Lane JR, et al. (November 2008). "The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist". Science. 322 (5905): 1211–7. Bibcode:2008Sci...322.1211J. doi:10.1126/science.1164772. PMC 2586971. PMID 18832607.

Liu W, Chun E, Thompson AA, Chubukov P, Xu F, Katritch V, et al. (July 2012). "Structural basis for allosteric regulation of GPCRs by sodium ions". Science. 337 (6091): 232–6. Bibcode:2012Sci...337..232L. doi:10.1126/science.1219218. PMC 3399762. PMID 22798613.

Ciruela F, Casadó V, Rodrigues RJ, Luján R, Burgueño J, Canals M, et al. (February 2006). "Presynaptic control of striatal glutamatergic neurotransmission by adenosine A1-A2A receptor heteromers". The Journal of Neuroscience. 26 (7): 2080–7. doi:10.1523/JNEUROSCI.3574-05.2006. PMC 6674939. PMID 16481441.

Ferre S, Ciruela F, Borycz J, Solinas M, Quarta D, Antoniou K, et al. (January 2008). "Adenosine A1-A2A receptor heteromers: new targets for caffeine in the brain". Frontiers in Bioscience. 13 (13): 2391–9. doi:10.2741/2852. PMID 17981720. Archived from the original on 2023-03-06. Retrieved 2009-04-20.

Fuxe K, Ferré S, Canals M, Torvinen M, Terasmaa A, Marcellino D, et al. (2005). "Adenosine A2A and dopamine D2 heteromeric receptor complexes and their function". Journal of Molecular Neuroscience. 26 (2–3): 209–20. doi:10.1385/JMN:26:2-3:209. PMID 16012194. S2CID 427930.

Torvinen M, Marcellino D, Canals M, Agnati LF, Lluis C, Franco R, Fuxe K (February 2005). "Adenosine A2A receptor and dopamine D3 receptor interactions: evidence of functional A2A/D3 heteromeric complexes". Molecular Pharmacology. 67 (2): 400–7. doi:10.1124/mol.104.003376. PMID 15539641. S2CID 24475855.

Zezula J, Freissmuth M (March 2008). "The A(2A)-adenosine receptor: a GPCR with unique features?". British Journal of Pharmacology. 153 Suppl 1 (S1): S184-90. doi:10.1038/sj.bjp.0707674. PMC 2268059. PMID 18246094.

Ferré S, Goldberg SR, Lluis C, Franco R (2009). "Looking for the role of cannabinoid receptor heteromers in striatal function". Neuropharmacology. 56 (Suppl 1): 226–34. doi:10.1016/j.neuropharm.2008.06.076. PMC 2635338. PMID 18691604.

Marcellino D, Carriba P, Filip M, Borgkvist A, Frankowska M, Bellido I, et al. (April 2008). "Antagonistic cannabinoid CB1/dopamine D2 receptor interactions in striatal CB1/D2 heteromers. A combined neurochemical and behavioral analysis". Neuropharmacology. 54 (5): 815–23. doi:10.1016/j.neuropharm.2007.12.011. PMID 18262573. S2CID 195685369.

Ferré S, Ciruela F, Quiroz C, Luján R, Popoli P, Cunha RA, et al. (November 2007). "Adenosine receptor heteromers and their integrative role in striatal function". TheScientificWorldJournal. 7: 74–85. doi:10.1100/tsw.2007.211. PMC 5901194. PMID 17982579.

Wardas J (May 2008). "Potential role of adenosine A2A receptors in the treatment of schizophrenia". Frontiers in Bioscience. 13 (13): 4071–96. doi:10.2741/2995. PMID 18508501.

Simola N, Morelli M, Pinna A (2008). "Adenosine A2A receptor antagonists and Parkinson's disease: state of the art and future directions". Current Pharmaceutical Design. 14 (15): 1475–89. doi:10.2174/138161208784480072. PMID 18537671.

Cekic C, Linden J (December 2014). "Adenosine A2A receptors intrinsically regulate CD8+ T cells in the tumor microenvironment". Cancer Research. 74 (24): 7239–49. doi:10.1158/0008-5472.CAN-13-3581. PMC 4459794. PMID 25341542.

Carpenter B, Nehmé R, Warne T, Leslie AG, Tate CG (August 2016). "Structure of the adenosine A(2A) receptor bound to an engineered G protein". Nature. 536 (7614): 104–7. Bibcode:2016Natur.536..104C. doi:10.1038/nature18966. PMC 4979997. PMID 27462812.

Ohta A, Sitkovsky M (2001). "Role of G-protein-coupled adenosine receptors in downregulation of inflammation and protection from tissue damage". Nature. 414 (6866): 916–20. Bibcode:2001Natur.414..916O. doi:10.1038/414916a. PMID 11780065. S2CID 4386419. Archived from the original on 2020-09-16. Retrieved 2019-07-05.

Hack SP, Christie MJ (2003). "Adaptations in adenosine signaling in drug dependence: therapeutic implications". Critical Reviews in Neurobiology. 15 (3–4): 235–74. doi:10.1615/CritRevNeurobiol.v15.i34.30. PMID 15248812.

Morelli M, Di Paolo T, Wardas J, Calon F, Xiao D, Schwarzschild MA (December 2007). "Role of adenosine A2A receptors in parkinsonian motor impairment and l-DOPA-induced motor complications". Progress in Neurobiology. 83 (5): 293–309. doi:10.1016/j.pneurobio.2007.07.001. PMID 17826884. S2CID 27478825.

Schiffmann SN, Fisone G, Moresco R, Cunha RA, Ferré S (December 2007). "Adenosine A2A receptors and basal ganglia physiology". Progress in Neurobiology. 83 (5): 277–92. doi:10.1016/j.pneurobio.2007.05.001. PMC 2148496. PMID 17646043.

Ferré S, Diamond I, Goldberg SR, Yao L, Hourani SM, Huang ZL, et al. (December 2007). "Adenosine A2A receptors in ventral striatum, hypothalamus and nociceptive circuitry implications for drug addiction, sleep and pain". Progress in Neurobiology. 83 (5): 332–47. doi:10.1016/j.pneurobio.2007.04.002. PMC 2141681. PMID 17532111.

Brown RM, Short JL (November 2008). "Adenosine A(2A) receptors and their role in drug addiction". The Journal of Pharmacy and Pharmacology. 60 (11): 1409–30. doi:10.1211/jpp/60.11.0001 (inactive 3 December 2024). PMID 18957161.{{cite journal}}: CS1 maint: DOI inactive as of December 2024 (link)

Cunha RA, Ferré S, Vaugeois JM, Chen JF (2008). "Potential therapeutic interest of adenosine A2A receptors in psychiatric disorders". Current Pharmaceutical Design. 14 (15): 1512–24. doi:10.2174/138161208784480090. PMC 2423946. PMID 18537674.

Mingote S, Font L, Farrar AM, Vontell R, Worden LT, Stopper CM, et al. (September 2008). "Nucleus accumbens adenosine A2A receptors regulate exertion of effort by acting on the ventral striatopallidal pathway". The Journal of Neuroscience. 28 (36): 9037–46. doi:10.1523/JNEUROSCI.1525-08.2008. PMC 2806668. PMID 18768698.

Ongini E, Monopoli A, Cacciari B, Baraldi PG (2001). "Selective adenosine A2A receptor antagonists". Farmaco. 56 (1–2): 87–90. doi:10.1016/S0014-827X(01)01024-2. PMID 11347973.
Burton JH, Mass M, Menegazzi JJ, Yealy DM (August 1997). "Aminophylline as an adjunct to standard advanced cardiac life support in prolonged cardiac arrest". Annals of Emergency Medicine. 30 (2): 154–8. doi:10.1016/S0196-0644(97)70134-3. PMID 9250637.
Khoury MY, Moukarbel GV, Obeid MY, Alam SE (May 2001). "Effect of aminophylline on complete atrioventricular block with ventricular asystole following blunt chest trauma". Injury. 32 (4): 335–8. doi:10.1016/S0020-1383(00)00222-9. PMID 11325371.
Mader TJ, Bertolet B, Ornato JP, Gutterman JM (October 2000). "Aminophylline in the treatment of atropine-resistant bradyasystole". Resuscitation. 47 (2): 105–12. doi:10.1016/S0300-9572(00)00234-3. PMID 11008148.
Mader TJ, Smithline HA, Durkin L, Scriver G (March 2003). "A randomized controlled trial of intravenous aminophylline for atropine-resistant out-of-hospital asystolic cardiac arrest". Academic Emergency Medicine. 10 (3): 192–7. doi:10.1197/aemj.10.3.192. PMID 12615581.
Mader TJ, Gibson P (August 1997). "Adenosine receptor antagonism in refractory asystolic cardiac arrest: results of a human pilot study". Resuscitation. 35 (1): 3–7. doi:10.1016/S0300-9572(97)01097-6. PMID 9259053.
Perouansky M, Shamir M, Hershkowitz E, Donchin Y (July 1998). "Successful resuscitation using aminophylline in refractory cardiac arrest with asystole". Resuscitation. 38 (1): 39–41. doi:10.1016/S0300-9572(98)00079-3. PMID 9783508.
Viskin S, Belhassen B, Roth A, Reicher M, Averbuch M, Sheps D, et al. (February 1993). "Aminophylline for bradyasystolic cardiac arrest refractory to atropine and epinephrine". Annals of Internal Medicine. 118 (4): 279–81. doi:10.7326/0003-4819-118-4-199302150-00006. PMID 8420445. S2CID 44883687.
Jenner P (December 2003). "A2A antagonists as novel non-dopaminergic therapy for motor dysfunction in PD". Neurology. 61 (11 Suppl 6): S32-8. doi:10.1212/01.WNL.0000095209.59347.79. PMID 14663007. S2CID 28897242.
Mori A, Shindou T (December 2003). "Modulation of GABAergic transmission in the striatopallidal system by adenosine A2A receptors: a potential mechanism for the antiparkinsonian effects of A2A antagonists". Neurology. 61 (11 Suppl 6): S44-8. doi:10.1212/01.WNL.0000095211.71092.A0. PMID 14663009. S2CID 26827799.
Pinna A, Wardas J, Simola N, Morelli M (November 2005). "New therapies for the treatment of Parkinson's disease: adenosine A2A receptor antagonists". Life Sciences. 77 (26): 3259–67. doi:10.1016/j.lfs.2005.04.029. PMID 15979104.
Kelsey JE, Langelier NA, Oriel BS, Reedy C (January 2009). "The effects of systemic, intrastriatal, and intrapallidal injections of caffeine and systemic injections of A2A and A1 antagonists on forepaw stepping in the unilateral 6-OHDA-lesioned rat". Psychopharmacology. 201 (4): 529–39. doi:10.1007/s00213-008-1319-0. PMID 18791705. S2CID 24159282.
Jacobson KA, Gao ZG (March 2006). "Adenosine receptors as therapeutic targets". Nature Reviews. Drug Discovery. 5 (3): 247–64. doi:10.1038/nrd1983. PMC 3463109. PMID 16518376. table 1 lists affinities
Burstein S (7 February 2015). "Cannabidiol (CBD) and its analogs: a review of their effects on inflammation". Bioorganic & Medicinal Chemistry. 23 (7): 1377–1385. doi:10.1016/j.bmc.2015.01.059. PMID 25703248.
Amelia T, Van Veldhoven JP, Falsini M, Liu R, Heitman LH, Van Westen GJ, Segala E, Verdon G, Cheng RK, Cooke RM, Van Der Es D, Ijzerman AP (2021). "Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A_2A Receptor". Journal of Medicinal Chemistry. 64 (7): 3827–3842. doi:10.1021/acs.jmedchem.0c01856. PMC 8154574. PMID 33764785.
Bolcato G, Pavan M, Bassani D, Sturlese M, Moro S (2022). "Ribose and Non-Ribose A2A Adenosine Receptor Agonists: Do They Share the Same Receptor Recognition Mechanism?". Biomedicines. 10 (2): 515. doi:10.3390/biomedicines10020515. PMC 8962312. PMID 35203724.
Yoneyama F, Yamada H, Satoh K, Taira N (March 1992). "Vasodepressor mechanisms of 2-(1-octynyl)-adenosine (YT-146), a selective adenosine A2 receptor agonist, involve the opening of glibenclamide-sensitive K+ channels". European Journal of Pharmacology. 213 (2): 199–204. doi:10.1016/0014-2999(92)90682-T. PMID 1521559.
Doyle SE, Breslin FJ, Rieger JM, Beauglehole A, Lynch WJ (August 2012). "Time and sex-dependent effects of an adenosine A2A/A1 receptor antagonist on motivation to self-administer cocaine in rats". Pharmacology, Biochemistry, and Behavior. 102 (2): 257–63. doi:10.1016/j.pbb.2012.05.001. PMC 3383440. PMID 22579716.
Kase H, Aoyama S, Ichimura M, Ikeda K, Ishii A, Kanda T, et al. (December 2003). "Progress in pursuit of therapeutic A2A antagonists: the adenosine A2A receptor selective antagonist KW6002: research and development toward a novel nondopaminergic therapy for Parkinson's disease". Neurology. 61 (11 Suppl 6): S97-100. doi:10.1212/01.WNL.0000095219.22086.31. PMID 14663020. S2CID 72084113.
Mott AM, Nunes EJ, Collins LE, Port RG, Sink KS, Hockemeyer J, et al. (May 2009). "The adenosine A2A antagonist MSX-3 reverses the effects of the dopamine antagonist haloperidol on effort-related decision making in a T-maze cost/benefit procedure". Psychopharmacology. 204 (1): 103–12. doi:10.1007/s00213-008-1441-z. PMC 2875244. PMID 19132351.
Hodgson RA, Bertorelli R, Varty GB, Lachowicz JE, Forlani A, Fredduzzi S, et al. (July 2009). "Characterization of the potent and highly selective A2A receptor antagonists preladenant and SCH 412348 [7-[2-[4-2,4-difluorophenyl]-1-piperazinyl]ethyl]-2-(2-furanyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine] in rodent models of movement disorders and depression". The Journal of Pharmacology and Experimental Therapeutics. 330 (1): 294–303. doi:10.1124/jpet.108.149617. PMID 19332567. S2CID 22033475.
Pinna A, Fenu S, Morelli M (March 2001). "Motor stimulant effects of the adenosine A2A receptor antagonist SCH 58261 do not develop tolerance after repeated treatments in 6-hydroxydopamine-lesioned rats". Synapse. 39 (3): 233–8. doi:10.1002/1098-2396(20010301)39:3<233::AID-SYN1004>3.0.CO;2-K. PMID 11284438. S2CID 23370571.
Rose S, Jackson MJ, Smith LA, Stockwell K, Johnson L, Carminati P, Jenner P (September 2006). "The novel adenosine A2a receptor antagonist ST1535 potentiates the effects of a threshold dose of L-DOPA in MPTP treated common marmosets". European Journal of Pharmacology. 546 (1–3): 82–7. doi:10.1016/j.ejphar.2006.07.017. PMID 16925991.
Kamiya T, Saitoh O, Yoshioka K, Nakata H (June 2003). "Oligomerization of adenosine A2A and dopamine D2 receptors in living cells". Biochemical and Biophysical Research Communications. 306 (2): 544–9. doi:10.1016/S0006-291X(03)00991-4. PMID 12804599.
Sitkovsky MV, Kjaergaard J, Lukashev D, Ohta A (October 2008). "Hypoxia-adenosinergic immunosuppression: tumor protection by T regulatory cells and cancerous tissue hypoxia". Clinical Cancer Research. 14 (19): 5947–52. doi:10.1158/1078-0432.CCR-08-0229. PMID 18829471.
Leone RD, Lo YC, Powell JD (April 2015). "A2aR antagonists: Next generation checkpoint blockade for cancer immunotherapy". Computational and Structural Biotechnology Journal. 13: 265–72. doi:10.1016/j.csbj.2015.03.008. PMC 4415113. PMID 25941561.
Pardoll DM (March 2012). "The blockade of immune checkpoints in cancer immunotherapy". Nature Reviews. Cancer. 12 (4): 252–64. doi:10.1038/nrc3239. PMC 4856023. PMID 22437870.
Willingham SB (October 2018). "A2AR Antagonism with CPI-444 Induces Antitumor Responses and Augments Efficacy to Anti-PD-(L)1 and Anti-CTLA-4 in Preclinical Models". Cancer Immunol Res. 6 (10): 1136–1149. doi:10.1158/2326-6066.CIR-18-0056. PMID 30131376.
Beavis PA, Henderson MA, Giuffrida L, Mills JK, Sek K, Cross RS, et al. (March 2017). "Targeting the adenosine 2A receptor enhances chimeric antigen receptor T cell efficacy". The Journal of Clinical Investigation. 127 (3): 929–941. doi:10.1172/JCI89455. PMC 5330718. PMID 28165340.

nih.gov

pubmed.ncbi.nlm.nih.gov

Wardas J (May 2008). "Potential role of adenosine A2A receptors in the treatment of schizophrenia". Frontiers in Bioscience. 13 (13): 4071–96. doi:10.2741/2995. PMID 18508501.

Ongini E, Monopoli A, Cacciari B, Baraldi PG (2001). "Selective adenosine A2A receptor antagonists". Farmaco. 56 (1–2): 87–90. doi:10.1016/S0014-827X(01)01024-2. PMID 11347973.
- Sullivan GW (November 2003). "Adenosine A2A receptor agonists as anti-inflammatory agents". Current Opinion in Investigational Drugs. 4 (11): 1313–9. PMID 14758770.
- Burton JH, Mass M, Menegazzi JJ, Yealy DM (August 1997). "Aminophylline as an adjunct to standard advanced cardiac life support in prolonged cardiac arrest". Annals of Emergency Medicine. 30 (2): 154–8. doi:10.1016/S0196-0644(97)70134-3. PMID 9250637.
- Khoury MY, Moukarbel GV, Obeid MY, Alam SE (May 2001). "Effect of aminophylline on complete atrioventricular block with ventricular asystole following blunt chest trauma". Injury. 32 (4): 335–8. doi:10.1016/S0020-1383(00)00222-9. PMID 11325371.
- Mader TJ, Bertolet B, Ornato JP, Gutterman JM (October 2000). "Aminophylline in the treatment of atropine-resistant bradyasystole". Resuscitation. 47 (2): 105–12. doi:10.1016/S0300-9572(00)00234-3. PMID 11008148.
- Mader TJ, Smithline HA, Durkin L, Scriver G (March 2003). "A randomized controlled trial of intravenous aminophylline for atropine-resistant out-of-hospital asystolic cardiac arrest". Academic Emergency Medicine. 10 (3): 192–7. doi:10.1197/aemj.10.3.192. PMID 12615581.
- Mader TJ, Gibson P (August 1997). "Adenosine receptor antagonism in refractory asystolic cardiac arrest: results of a human pilot study". Resuscitation. 35 (1): 3–7. doi:10.1016/S0300-9572(97)01097-6. PMID 9259053.
- Perouansky M, Shamir M, Hershkowitz E, Donchin Y (July 1998). "Successful resuscitation using aminophylline in refractory cardiac arrest with asystole". Resuscitation. 38 (1): 39–41. doi:10.1016/S0300-9572(98)00079-3. PMID 9783508.
- Viskin S, Belhassen B, Roth A, Reicher M, Averbuch M, Sheps D, et al. (February 1993). "Aminophylline for bradyasystolic cardiac arrest refractory to atropine and epinephrine". Annals of Internal Medicine. 118 (4): 279–81. doi:10.7326/0003-4819-118-4-199302150-00006. PMID 8420445. S2CID 44883687.
- Jenner P (December 2003). "A2A antagonists as novel non-dopaminergic therapy for motor dysfunction in PD". Neurology. 61 (11 Suppl 6): S32-8. doi:10.1212/01.WNL.0000095209.59347.79. PMID 14663007. S2CID 28897242.
- Mori A, Shindou T (December 2003). "Modulation of GABAergic transmission in the striatopallidal system by adenosine A2A receptors: a potential mechanism for the antiparkinsonian effects of A2A antagonists". Neurology. 61 (11 Suppl 6): S44-8. doi:10.1212/01.WNL.0000095211.71092.A0. PMID 14663009. S2CID 26827799.
- Pinna A, Wardas J, Simola N, Morelli M (November 2005). "New therapies for the treatment of Parkinson's disease: adenosine A2A receptor antagonists". Life Sciences. 77 (26): 3259–67. doi:10.1016/j.lfs.2005.04.029. PMID 15979104.
- Kelsey JE, Langelier NA, Oriel BS, Reedy C (January 2009). "The effects of systemic, intrastriatal, and intrapallidal injections of caffeine and systemic injections of A2A and A1 antagonists on forepaw stepping in the unilateral 6-OHDA-lesioned rat". Psychopharmacology. 201 (4): 529–39. doi:10.1007/s00213-008-1319-0. PMID 18791705. S2CID 24159282.
- Jacobson KA, Gao ZG (March 2006). "Adenosine receptors as therapeutic targets". Nature Reviews. Drug Discovery. 5 (3): 247–64. doi:10.1038/nrd1983. PMC 3463109. PMID 16518376. table 1 lists affinities
- Burstein S (7 February 2015). "Cannabidiol (CBD) and its analogs: a review of their effects on inflammation". Bioorganic & Medicinal Chemistry. 23 (7): 1377–1385. doi:10.1016/j.bmc.2015.01.059. PMID 25703248.
- Amelia T, Van Veldhoven JP, Falsini M, Liu R, Heitman LH, Van Westen GJ, Segala E, Verdon G, Cheng RK, Cooke RM, Van Der Es D, Ijzerman AP (2021). "Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A_2A Receptor". Journal of Medicinal Chemistry. 64 (7): 3827–3842. doi:10.1021/acs.jmedchem.0c01856. PMC 8154574. PMID 33764785.
- Bolcato G, Pavan M, Bassani D, Sturlese M, Moro S (2022). "Ribose and Non-Ribose A2A Adenosine Receptor Agonists: Do They Share the Same Receptor Recognition Mechanism?". Biomedicines. 10 (2): 515. doi:10.3390/biomedicines10020515. PMC 8962312. PMID 35203724.
- Yoneyama F, Yamada H, Satoh K, Taira N (March 1992). "Vasodepressor mechanisms of 2-(1-octynyl)-adenosine (YT-146), a selective adenosine A2 receptor agonist, involve the opening of glibenclamide-sensitive K+ channels". European Journal of Pharmacology. 213 (2): 199–204. doi:10.1016/0014-2999(92)90682-T. PMID 1521559.
- Doyle SE, Breslin FJ, Rieger JM, Beauglehole A, Lynch WJ (August 2012). "Time and sex-dependent effects of an adenosine A2A/A1 receptor antagonist on motivation to self-administer cocaine in rats". Pharmacology, Biochemistry, and Behavior. 102 (2): 257–63. doi:10.1016/j.pbb.2012.05.001. PMC 3383440. PMID 22579716.
- Kase H, Aoyama S, Ichimura M, Ikeda K, Ishii A, Kanda T, et al. (December 2003). "Progress in pursuit of therapeutic A2A antagonists: the adenosine A2A receptor selective antagonist KW6002: research and development toward a novel nondopaminergic therapy for Parkinson's disease". Neurology. 61 (11 Suppl 6): S97-100. doi:10.1212/01.WNL.0000095219.22086.31. PMID 14663020. S2CID 72084113.
- Mott AM, Nunes EJ, Collins LE, Port RG, Sink KS, Hockemeyer J, et al. (May 2009). "The adenosine A2A antagonist MSX-3 reverses the effects of the dopamine antagonist haloperidol on effort-related decision making in a T-maze cost/benefit procedure". Psychopharmacology. 204 (1): 103–12. doi:10.1007/s00213-008-1441-z. PMC 2875244. PMID 19132351.
- Hodgson RA, Bertorelli R, Varty GB, Lachowicz JE, Forlani A, Fredduzzi S, et al. (July 2009). "Characterization of the potent and highly selective A2A receptor antagonists preladenant and SCH 412348 [7-[2-[4-2,4-difluorophenyl]-1-piperazinyl]ethyl]-2-(2-furanyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine] in rodent models of movement disorders and depression". The Journal of Pharmacology and Experimental Therapeutics. 330 (1): 294–303. doi:10.1124/jpet.108.149617. PMID 19332567. S2CID 22033475.
- Pinna A, Fenu S, Morelli M (March 2001). "Motor stimulant effects of the adenosine A2A receptor antagonist SCH 58261 do not develop tolerance after repeated treatments in 6-hydroxydopamine-lesioned rats". Synapse. 39 (3): 233–8. doi:10.1002/1098-2396(20010301)39:3<233::AID-SYN1004>3.0.CO;2-K. PMID 11284438. S2CID 23370571.
- Rose S, Jackson MJ, Smith LA, Stockwell K, Johnson L, Carminati P, Jenner P (September 2006). "The novel adenosine A2a receptor antagonist ST1535 potentiates the effects of a threshold dose of L-DOPA in MPTP treated common marmosets". European Journal of Pharmacology. 546 (1–3): 82–7. doi:10.1016/j.ejphar.2006.07.017. PMID 16925991.
- Kamiya T, Saitoh O, Yoshioka K, Nakata H (June 2003). "Oligomerization of adenosine A2A and dopamine D2 receptors in living cells". Biochemical and Biophysical Research Communications. 306 (2): 544–9. doi:10.1016/S0006-291X(03)00991-4. PMID 12804599.
- Sitkovsky MV, Kjaergaard J, Lukashev D, Ohta A (October 2008). "Hypoxia-adenosinergic immunosuppression: tumor protection by T regulatory cells and cancerous tissue hypoxia". Clinical Cancer Research. 14 (19): 5947–52. doi:10.1158/1078-0432.CCR-08-0229. PMID 18829471.
- Leone RD, Lo YC, Powell JD (April 2015). "A2aR antagonists: Next generation checkpoint blockade for cancer immunotherapy". Computational and Structural Biotechnology Journal. 13: 265–72. doi:10.1016/j.csbj.2015.03.008. PMC 4415113. PMID 25941561.
- Pardoll DM (March 2012). "The blockade of immune checkpoints in cancer immunotherapy". Nature Reviews. Cancer. 12 (4): 252–64. doi:10.1038/nrc3239. PMC 4856023. PMID 22437870.
- Willingham SB (October 2018). "A2AR Antagonism with CPI-444 Induces Antitumor Responses and Augments Efficacy to Anti-PD-(L)1 and Anti-CTLA-4 in Preclinical Models". Cancer Immunol Res. 6 (10): 1136–1149. doi:10.1158/2326-6066.CIR-18-0056. PMID 30131376.
- Beavis PA, Henderson MA, Giuffrida L, Mills JK, Sek K, Cross RS, et al. (March 2017). "Targeting the adenosine 2A receptor enhances chimeric antigen receptor T cell efficacy". The Journal of Clinical Investigation. 127 (3): 929–941. doi:10.1172/JCI89455. PMC 5330718. PMID 28165340.
ncbi.nlm.nih.gov
- "Human PubMed Reference:". National Center for Biotechnology Information, U.S. National Library of Medicine.
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Adenosine A2A receptor (English Wikipedia)

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