References analysis of the Wikipedia article "Antalarmin" in the English version

doi.org

Zoumakis E, Rice KC, Gold PW, Chrousos GP (November 2006). "Potential uses of corticotropin-releasing hormone antagonists". Annals of the New York Academy of Sciences. 1083 (1): 239–51. Bibcode:2006NYASA1083..239Z. doi:10.1196/annals.1367.021. PMID 17148743. S2CID 7731338.

Webster EL, Lewis DB, Torpy DJ, Zachman EK, Rice KC, Chrousos GP (December 1996). "In vivo and in vitro characterization of antalarmin, a nonpeptide corticotropin-releasing hormone (CRH) receptor antagonist: suppression of pituitary ACTH release and peripheral inflammation". Endocrinology. 137 (12): 5747–50. doi:10.1210/endo.137.12.8940412. PMID 8940412.

Deak T, Nguyen KT, Ehrlich AL, Watkins LR, Spencer RL, Maier SF, et al. (January 1999). "The impact of the nonpeptide corticotropin-releasing hormone antagonist antalarmin on behavioral and endocrine responses to stress". Endocrinology. 140 (1): 79–86. doi:10.1210/endo.140.1.6415. PMID 9886810.

Nielsen DM, Carey GJ, Gold LH (September 2004). "Antidepressant-like activity of corticotropin-releasing factor type-1 receptor antagonists in mice". European Journal of Pharmacology. 499 (1–2): 135–46. doi:10.1016/j.ejphar.2004.07.091. PMID 15363960.

McCarthy JR, Heinrichs SC, Grigoriadis DE (May 1999). "Recent advances with the CRF1 receptor: design of small molecule inhibitors, receptor subtypes and clinical indications". Current Pharmaceutical Design. 5 (5): 289–315. doi:10.2174/138161280505230110095255. PMID 10213797.

Chen YL, Mansbach RS, Winter SM, Brooks E, Collins J, Corman ML, et al. (May 1997). "Synthesis and oral efficacy of a 4-(butylethylamino)pyrrolo[2,3-d]pyrimidine: a centrally active corticotropin-releasing factor1 receptor antagonist". Journal of Medicinal Chemistry. 40 (11): 1749–54. doi:10.1021/jm960861b. PMID 9171885.

Schoeffter P, Feuerbach D, Bobirnac I, Gazi L, Longato R (1999). "Functional, endogenously expressed corticotropin-releasing factor receptor type 1 (CRF1) and CRF1 receptor mRNA expression in human neuroblastoma SH-SY5Y cells". Fundamental & Clinical Pharmacology. 13 (4): 484–9. doi:10.1111/j.1472-8206.1999.tb00007.x. PMID 10456290. S2CID 31280442.

Gully D, Geslin M, Serva L, Fontaine E, Roger P, Lair C, et al. (April 2002). "4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1,3-thiazol-2-amine hydrochloride (SSR125543A): a potent and selective corticotrophin-releasing factor(1) receptor antagonist. I. Biochemical and pharmacological characterization". The Journal of Pharmacology and Experimental Therapeutics. 301 (1): 322–32. doi:10.1124/jpet.301.1.322. PMID 11907190.

Schulz DW, Mansbach RS, Sprouse J, Braselton JP, Collins J, Corman M, et al. (September 1996). "CP-154,526: a potent and selective nonpeptide antagonist of corticotropin releasing factor receptors". Proceedings of the National Academy of Sciences of the United States of America. 93 (19): 10477–82. Bibcode:1996PNAS...9310477S. doi:10.1073/pnas.93.19.10477. PMC 38410. PMID 8816826.

Lundkvist J, Chai Z, Teheranian R, Hasanvan H, Bartfai T, Jenck F, et al. (August 1996). "A non peptidic corticotropin releasing factor receptor antagonist attenuates fever and exhibits anxiolytic-like activity". European Journal of Pharmacology. 309 (2): 195–200. doi:10.1016/0014-2999(96)00337-8. PMID 8874139.

Gottowik J, Goetschy V, Henriot S, Kitas E, Fluhman B, Clerc RG, et al. (October 1997). "Labelling of CRF1 and CRF2 receptors using the novel radioligand, [3H]-urocortin". Neuropharmacology. 36 (10): 1439–46. doi:10.1016/S0028-3908(97)00098-1. PMID 9423932. S2CID 6235036.

Keller C, Bruelisauer A, Lemaire M, Enz A (February 2002). "Brain pharmacokinetics of a nonpeptidic corticotropin-releasing factor receptor antagonist". Drug Metabolism and Disposition. 30 (2): 173–6. doi:10.1124/dmd.30.2.173. PMID 11792687. S2CID 26144504.

Habib KE, Weld KP, Rice KC, Pushkas J, Champoux M, Listwak S, et al. (May 2000). "Oral administration of a corticotropin-releasing hormone receptor antagonist significantly attenuates behavioral, neuroendocrine, and autonomic responses to stress in primates". Proceedings of the National Academy of Sciences of the United States of America. 97 (11): 6079–84. Bibcode:2000PNAS...97.6079H. doi:10.1073/pnas.97.11.6079. PMC 18561. PMID 10823952.

Jutkiewicz EM, Wood SK, Houshyar H, Hsin LW, Rice KC, Woods JH (July 2005). "The effects of CRF antagonists, antalarmin, CP154,526, LWH234, and R121919, in the forced swim test and on swim-induced increases in adrenocorticotropin in rats". Psychopharmacology. 180 (2): 215–23. doi:10.1007/s00213-005-2164-z. PMC 1315297. PMID 15696320.

Ducottet C, Griebel G, Belzung C (June 2003). "Effects of the selective nonpeptide corticotropin-releasing factor receptor 1 antagonist antalarmin in the chronic mild stress model of depression in mice". Progress in Neuro-Psychopharmacology & Biological Psychiatry. 27 (4): 625–31. doi:10.1016/S0278-5846(03)00051-4. PMID 12787849. S2CID 32290500.

Zorrilla EP, Valdez GR, Nozulak J, Koob GF, Markou A (October 2002). "Effects of antalarmin, a CRF type 1 receptor antagonist, on anxiety-like behavior and motor activation in the rat". Brain Research. 952 (2): 188–99. doi:10.1016/S0006-8993(02)03189-X. PMID 12376179. S2CID 6797766.

Briscoe RJ, Cabrera CL, Baird TJ, Rice KC, Woods JH (October 2000). "Antalarmin blockade of corticotropin releasing hormone-induced hypertension in rats". Brain Research. 881 (2): 204–7. doi:10.1016/S0006-8993(00)02742-6. PMID 11036160. S2CID 12152273.

Seymour PA, Schmidt AW, Schulz DW (2003). "The pharmacology of CP-154,526, a non-peptide antagonist of the CRH1 receptor: a review". CNS Drug Reviews. 9 (1): 57–96. doi:10.1111/j.1527-3458.2003.tb00244.x. PMC 6741649. PMID 12595912.

Willenberg HS, Bornstein SR, Hiroi N, Päth G, Goretzki PE, Scherbaum WA, Chrousos GP (March 2000). "Effects of a novel corticotropin-releasing-hormone receptor type I antagonist on human adrenal function". Molecular Psychiatry. 5 (2): 137–41. doi:10.1038/sj.mp.4000720. PMID 10822340.

Wong ML, Webster EL, Spokes H, Phu P, Ehrhart-Bornstein M, Bornstein S, et al. (1999). "Chronic administration of the non-peptide CRH type 1 receptor antagonist antalarmin does not blunt hypothalamic-pituitary-adrenal axis responses to acute immobilization stress". Life Sciences. 65 (4): PL53-8. doi:10.1016/s0024-3205(99)00268-4. PMID 10421433.

Griebel G, Simiand J, Steinberg R, Jung M, Gully D, Roger P, et al. (April 2002). "4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1, 3-thiazol-2-amine hydrochloride (SSR125543A), a potent and selective corticotrophin-releasing factor(1) receptor antagonist. II. Characterization in rodent models of stress-related disorders". The Journal of Pharmacology and Experimental Therapeutics. 301 (1): 333–45. doi:10.1124/jpet.301.1.333. PMID 11907191. S2CID 24106723.

Kirby LG, Rice KC, Valentino RJ (February 2000). "Effects of corticotropin-releasing factor on neuronal activity in the serotonergic dorsal raphe nucleus". Neuropsychopharmacology. 22 (2): 148–62. doi:10.1016/S0893-133X(99)00093-7. PMID 10649828.

Griebel G (April 1999). "Is there a future for neuropeptide receptor ligands in the treatment of anxiety disorders?". Pharmacology & Therapeutics. 82 (1): 1–61. doi:10.1016/S0163-7258(98)00041-2. PMID 10341356.

Britton KT, Lee G, Vale W, Rivier J, Koob GF (March 1986). "Corticotropin releasing factor (CRF) receptor antagonist blocks activating and 'anxiogenic' actions of CRF in the rat". Brain Research. 369 (1–2): 303–6. doi:10.1016/0006-8993(86)90539-1. PMID 3008937. S2CID 6290497.

Dermitzaki E, Tsatsanis C, Gravanis A, Margioris AN (April 2002). "Corticotropin-releasing hormone induces Fas ligand production and apoptosis in PC12 cells via activation of p38 mitogen-activated protein kinase". The Journal of Biological Chemistry. 277 (14): 12280–7. doi:10.1074/jbc.M111236200. PMID 11790788.

Theoharides TC, Singh LK, Boucher W, Pang X, Letourneau R, Webster E, Chrousos G (January 1998). "Corticotropin-releasing hormone induces skin mast cell degranulation and increased vascular permeability, a possible explanation for its proinflammatory effects". Endocrinology. 139 (1): 403–13. doi:10.1210/endo.139.1.5660. PMID 9421440.

Gabry KE, Chrousos GP, Rice KC, Mostafa RM, Sternberg E, Negrao AB, et al. (2002). "Marked suppression of gastric ulcerogenesis and intestinal responses to stress by a novel class of drugs". Molecular Psychiatry. 7 (5): 474–83, 433. doi:10.1038/sj.mp.4001031. PMID 12082565.

Greenwood-Van Meerveld B, Johnson AC, Cochrane S, Schulkin J, Myers DA (June 2005). "Corticotropin-releasing factor 1 receptor-mediated mechanisms inhibit colonic hypersensitivity in rats". Neurogastroenterology and Motility. 17 (3): 415–22. doi:10.1111/j.1365-2982.2005.00648.x. PMID 15916629. S2CID 25379651.

Martinez V, Taché Y (2006). "CRF1 receptors as a therapeutic target for irritable bowel syndrome". Current Pharmaceutical Design. 12 (31): 4071–88. doi:10.2174/138161206778743637. PMID 17100612.

Mello NK, Negus SS, Rice KC, Mendelson JH (December 2006). "Effects of the CRF1 antagonist antalarmin on cocaine self-administration and discrimination in rhesus monkeys". Pharmacology, Biochemistry, and Behavior. 85 (4): 744–51. doi:10.1016/j.pbb.2006.11.008. PMID 17182090. S2CID 8186943.

Specio SE, Wee S, O'Dell LE, Boutrel B, Zorrilla EP, Koob GF (February 2008). "CRF(1) receptor antagonists attenuate escalated cocaine self-administration in rats". Psychopharmacology. 196 (3): 473–82. doi:10.1007/s00213-007-0983-9. PMC 2769571. PMID 17965976.

Stinus L, Cador M, Zorrilla EP, Koob GF (January 2005). "Buprenorphine and a CRF1 antagonist block the acquisition of opiate withdrawal-induced conditioned place aversion in rats". Neuropsychopharmacology. 30 (1): 90–8. doi:10.1038/sj.npp.1300487. PMID 15138444.

Funk CK, Zorrilla EP, Lee MJ, Rice KC, Koob GF (January 2007). "Corticotropin-releasing factor 1 antagonists selectively reduce ethanol self-administration in ethanol-dependent rats". Biological Psychiatry. 61 (1): 78–86. doi:10.1016/j.biopsych.2006.03.063. PMC 2741496. PMID 16876134.

Chu K, Koob GF, Cole M, Zorrilla EP, Roberts AJ (April 2007). "Dependence-induced increases in ethanol self-administration in mice are blocked by the CRF1 receptor antagonist antalarmin and by CRF1 receptor knockout". Pharmacology, Biochemistry, and Behavior. 86 (4): 813–21. doi:10.1016/j.pbb.2007.03.009. PMC 2170886. PMID 17482248.

Marinelli PW, Funk D, Juzytsch W, Harding S, Rice KC, Shaham Y, Lê AD (December 2007). "The CRF1 receptor antagonist antalarmin attenuates yohimbine-induced increases in operant alcohol self-administration and reinstatement of alcohol seeking in rats". Psychopharmacology. 195 (3): 345–55. doi:10.1007/s00213-007-0905-x. PMID 17705061. S2CID 25629995.

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Porsolt RD, Bertin A, Jalfre M (October 1977). "Behavioral despair in mice: a primary screening test for antidepressants". Archives Internationales de Pharmacodynamie et de Therapie. 229 (2): 327–36. PMID 596982.

Webster EL, Barrientos RM, Contoreggi C, Isaac MG, Ligier S, Gabry KE, et al. (June 2002). "Corticotropin releasing hormone (CRH) antagonist attenuates adjuvant induced arthritis: role of CRH in peripheral inflammation". The Journal of Rheumatology. 29 (6): 1252–61. PMID 12064844.

Martinez V, Taché Y (2006). "CRF1 receptors as a therapeutic target for irritable bowel syndrome". Current Pharmaceutical Design. 12 (31): 4071–88. doi:10.2174/138161206778743637. PMID 17100612.

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Antalarmin (English Wikipedia)