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Befiradol (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "Befiradol" in English language version.

refsWebsite
Global rank English rank
18nih.gov
4th place
4th place
15doi.org
2nd place
2nd place
8semanticscholar.org
11th place
8th place
1psu.edu
207th place
136th place
1neurolixis.com
low place
low place
1michaeljfox.org
low place
low place
1parkinsons.org.uk
low place
low place
1prlog.org
9,932nd place
6,569th place
1thetimes.com
low place
low place
1prnewswire.com
406th place
258th place
1clinicaltrials.gov
5,225th place
4,062nd place
1einnews.com
low place
low place
1independent.co.uk
36th place
33rd place

clinicaltrials.gov (Global: 5,225th place; English: 4,062nd place)

  • Clinical trial number NCT05148884 for "Study to Assess the Safety, Tolerability and Preliminary Efficacy of NLX-112 Versus Placebo in L-dopa-induced Dyskinesia" at ClinicalTrials.gov

doi.org (Global: 2nd place; English: 2nd place)

  • Newman-Tancredi A, Martel JC, Cosi C, Heusler P, Lestienne F, Varney MA, et al. (September 2017). "Distinctive in vitro signal transduction profile of NLX-112, a potent and efficacious serotonin 5-HT1A receptor agonist". The Journal of Pharmacy and Pharmacology. 69 (9): 1178–1190. doi:10.1111/jphp.12762. PMID 28612503. S2CID 13676820.
  • Lladó-Pelfort L, Assié MB, Newman-Tancredi A, Artigas F, Celada P (May 2012). "In vivo electrophysiological and neurochemical effects of the selective 5-HT1A receptor agonist, F13640, at pre- and postsynaptic 5-HT1A receptors in the rat". Psychopharmacology. 221 (2): 261–272. doi:10.1007/s00213-011-2569-9. PMID 22147258. S2CID 18779324.
  • Bardin L, Tarayre JP, Malfetes N, Koek W, Colpaert FC (April 2003). "Profound, non-opioid analgesia produced by the high-efficacy 5-HT(1A) agonist F 13640 in the formalin model of tonic nociceptive pain". Pharmacology. 67 (4): 182–194. doi:10.1159/000068404. PMID 12595749. S2CID 25882138.
  • Bruins Slot LA, Koek W, Tarayre JP, Colpaert FC (April 2003). "Tolerance and inverse tolerance to the hyperalgesic and analgesic actions, respectively, of the novel analgesic, F 13640". European Journal of Pharmacology. 466 (3): 271–279. doi:10.1016/S0014-2999(03)01566-8. PMID 12694810.
  • Bardin L, Assié MB, Pélissou M, Royer-Urios I, Newman-Tancredi A, Ribet JP, et al. (March 2005). "Dual, hyperalgesic, and analgesic effects of the high-efficacy 5-hydroxytryptamine 1A (5-HT1A) agonist F 13640 [(3-chloro-4-fluoro-phenyl)-[4-fluoro-4-{[(5-methyl-pyridin-2-ylmethyl)-amino]-methyl}piperidin-1-yl]methanone, fumaric acid salt]: relationship with 5-HT1A receptor occupancy and kinetic parameters". The Journal of Pharmacology and Experimental Therapeutics. 312 (3): 1034–1042. doi:10.1124/jpet.104.077669. PMID 15528450. S2CID 42446435.
  • Colpaert FC, Deseure K, Stinus L, Adriaensen H (February 2006). "High-efficacy 5-hydroxytryptamine 1A receptor activation counteracts opioid hyperallodynia and affective conditioning". The Journal of Pharmacology and Experimental Therapeutics. 316 (2): 892–899. doi:10.1124/jpet.105.095109. PMID 16254131. S2CID 8820667.
  • Deseure K, Bréand S, Colpaert FC (July 2007). "Curative-like analgesia in a neuropathic pain model: parametric analysis of the dose and the duration of treatment with a high-efficacy 5-HT(1A) receptor agonist". European Journal of Pharmacology. 568 (1–3): 134–141. doi:10.1016/j.ejphar.2007.04.022. PMID 17512927.
  • Bollinger S, Hübner H, Heinemann FW, Meyer K, Gmeiner P (October 2010). "Novel pyridylmethylamines as highly selective 5-HT(1A) superagonists". Journal of Medicinal Chemistry. 53 (19): 7167–7179. doi:10.1021/jm100835q. PMID 20860381.
  • Vacher B, Bonnaud B, Funes P, Jubault N, Koek W, Assié MB, et al. (May 1999). "Novel derivatives of 2-pyridinemethylamine as selective, potent, and orally active agonists at 5-HT1A receptors". Journal of Medicinal Chemistry. 42 (9): 1648–1660. CiteSeerX 10.1.1.325.8872. doi:10.1021/jm9806906. PMID 10229633.
  • Iderberg H, McCreary AC, Varney MA, Kleven MS, Koek W, Bardin L, et al. (September 2015). "NLX-112, a novel 5-HT1A receptor agonist for the treatment of L-DOPA-induced dyskinesia: Behavioral and neurochemical profile in rat". Experimental Neurology. 271: 335–350. doi:10.1016/j.expneurol.2015.05.021. PMID 26037043. S2CID 35525495.
  • McCreary AC, Varney MA, Newman-Tancredi A (June 2016). "The novel 5-HT1A receptor agonist, NLX-112 reduces l-DOPA-induced abnormal involuntary movements in rat: A chronic administration study with microdialysis measurements". Neuropharmacology. 105: 651–660. doi:10.1016/j.neuropharm.2016.01.013. PMID 26777281. S2CID 1979117.
  • Depoortere R, Johnston TH, Fox SH, Brotchie JM, Newman-Tancredi A (September 2020). "The selective 5-HT1A receptor agonist, NLX-112, exerts anti-dyskinetic effects in MPTP-treated macaques". Parkinsonism & Related Disorders. 78: 151–157. doi:10.1016/j.parkreldis.2020.08.009. PMID 32846366. S2CID 221343904.
  • Fisher R, Hikima A, Morris R, Jackson MJ, Rose S, Varney MA, et al. (May 2020). "The selective 5-HT1A receptor agonist, NLX-112, exerts anti-dyskinetic and anti-parkinsonian-like effects in MPTP-treated marmosets". Neuropharmacology. 167 107997. doi:10.1016/j.neuropharm.2020.107997. PMC 7103782. PMID 32057799.
  • Colom M, Vidal B, Fieux S, Redoute J, Costes N, Lavenne F, et al. (2021). "[18F]F13640, a 5-HT1A Receptor Radiopharmaceutical Sensitive to Brain Serotonin Fluctuations". Frontiers in Neuroscience. 15 622423. doi:10.3389/fnins.2021.622423. PMC 7982540. PMID 33762906.
  • Courault P, Lancelot S, Costes N, Colom M, Le Bars D, Redoute J, et al. (May 2023). "[18F]F13640: a selective agonist PET radiopharmaceutical for imaging functional 5-HT1A receptors in humans". European Journal of Nuclear Medicine and Molecular Imaging. 50 (6): 1651–1664. doi:10.1007/s00259-022-06103-1. PMC 10119077. PMID 36656363.

einnews.com (Global: low place; English: low place)

independent.co.uk (Global: 36th place; English: 33rd place)

michaeljfox.org (Global: low place; English: low place)

neurolixis.com (Global: low place; English: low place)

nih.gov (Global: 4th place; English: 4th place)

pubmed.ncbi.nlm.nih.gov

  • Newman-Tancredi A, Martel JC, Cosi C, Heusler P, Lestienne F, Varney MA, et al. (September 2017). "Distinctive in vitro signal transduction profile of NLX-112, a potent and efficacious serotonin 5-HT1A receptor agonist". The Journal of Pharmacy and Pharmacology. 69 (9): 1178–1190. doi:10.1111/jphp.12762. PMID 28612503. S2CID 13676820.
  • Lladó-Pelfort L, Assié MB, Newman-Tancredi A, Artigas F, Celada P (May 2012). "In vivo electrophysiological and neurochemical effects of the selective 5-HT1A receptor agonist, F13640, at pre- and postsynaptic 5-HT1A receptors in the rat". Psychopharmacology. 221 (2): 261–272. doi:10.1007/s00213-011-2569-9. PMID 22147258. S2CID 18779324.
  • Bardin L, Tarayre JP, Malfetes N, Koek W, Colpaert FC (April 2003). "Profound, non-opioid analgesia produced by the high-efficacy 5-HT(1A) agonist F 13640 in the formalin model of tonic nociceptive pain". Pharmacology. 67 (4): 182–194. doi:10.1159/000068404. PMID 12595749. S2CID 25882138.
  • Bruins Slot LA, Koek W, Tarayre JP, Colpaert FC (April 2003). "Tolerance and inverse tolerance to the hyperalgesic and analgesic actions, respectively, of the novel analgesic, F 13640". European Journal of Pharmacology. 466 (3): 271–279. doi:10.1016/S0014-2999(03)01566-8. PMID 12694810.
  • Bardin L, Assié MB, Pélissou M, Royer-Urios I, Newman-Tancredi A, Ribet JP, et al. (March 2005). "Dual, hyperalgesic, and analgesic effects of the high-efficacy 5-hydroxytryptamine 1A (5-HT1A) agonist F 13640 [(3-chloro-4-fluoro-phenyl)-[4-fluoro-4-{[(5-methyl-pyridin-2-ylmethyl)-amino]-methyl}piperidin-1-yl]methanone, fumaric acid salt]: relationship with 5-HT1A receptor occupancy and kinetic parameters". The Journal of Pharmacology and Experimental Therapeutics. 312 (3): 1034–1042. doi:10.1124/jpet.104.077669. PMID 15528450. S2CID 42446435.
  • Colpaert FC, Deseure K, Stinus L, Adriaensen H (February 2006). "High-efficacy 5-hydroxytryptamine 1A receptor activation counteracts opioid hyperallodynia and affective conditioning". The Journal of Pharmacology and Experimental Therapeutics. 316 (2): 892–899. doi:10.1124/jpet.105.095109. PMID 16254131. S2CID 8820667.
  • Deseure K, Bréand S, Colpaert FC (July 2007). "Curative-like analgesia in a neuropathic pain model: parametric analysis of the dose and the duration of treatment with a high-efficacy 5-HT(1A) receptor agonist". European Journal of Pharmacology. 568 (1–3): 134–141. doi:10.1016/j.ejphar.2007.04.022. PMID 17512927.
  • Bollinger S, Hübner H, Heinemann FW, Meyer K, Gmeiner P (October 2010). "Novel pyridylmethylamines as highly selective 5-HT(1A) superagonists". Journal of Medicinal Chemistry. 53 (19): 7167–7179. doi:10.1021/jm100835q. PMID 20860381.
  • Vacher B, Bonnaud B, Funes P, Jubault N, Koek W, Assié MB, et al. (May 1999). "Novel derivatives of 2-pyridinemethylamine as selective, potent, and orally active agonists at 5-HT1A receptors". Journal of Medicinal Chemistry. 42 (9): 1648–1660. CiteSeerX 10.1.1.325.8872. doi:10.1021/jm9806906. PMID 10229633.
  • Iderberg H, McCreary AC, Varney MA, Kleven MS, Koek W, Bardin L, et al. (September 2015). "NLX-112, a novel 5-HT1A receptor agonist for the treatment of L-DOPA-induced dyskinesia: Behavioral and neurochemical profile in rat". Experimental Neurology. 271: 335–350. doi:10.1016/j.expneurol.2015.05.021. PMID 26037043. S2CID 35525495.
  • McCreary AC, Varney MA, Newman-Tancredi A (June 2016). "The novel 5-HT1A receptor agonist, NLX-112 reduces l-DOPA-induced abnormal involuntary movements in rat: A chronic administration study with microdialysis measurements". Neuropharmacology. 105: 651–660. doi:10.1016/j.neuropharm.2016.01.013. PMID 26777281. S2CID 1979117.
  • Depoortere R, Johnston TH, Fox SH, Brotchie JM, Newman-Tancredi A (September 2020). "The selective 5-HT1A receptor agonist, NLX-112, exerts anti-dyskinetic effects in MPTP-treated macaques". Parkinsonism & Related Disorders. 78: 151–157. doi:10.1016/j.parkreldis.2020.08.009. PMID 32846366. S2CID 221343904.
  • Fisher R, Hikima A, Morris R, Jackson MJ, Rose S, Varney MA, et al. (May 2020). "The selective 5-HT1A receptor agonist, NLX-112, exerts anti-dyskinetic and anti-parkinsonian-like effects in MPTP-treated marmosets". Neuropharmacology. 167 107997. doi:10.1016/j.neuropharm.2020.107997. PMC 7103782. PMID 32057799.
  • Colom M, Vidal B, Fieux S, Redoute J, Costes N, Lavenne F, et al. (2021). "[18F]F13640, a 5-HT1A Receptor Radiopharmaceutical Sensitive to Brain Serotonin Fluctuations". Frontiers in Neuroscience. 15 622423. doi:10.3389/fnins.2021.622423. PMC 7982540. PMID 33762906.
  • Courault P, Lancelot S, Costes N, Colom M, Le Bars D, Redoute J, et al. (May 2023). "[18F]F13640: a selective agonist PET radiopharmaceutical for imaging functional 5-HT1A receptors in humans". European Journal of Nuclear Medicine and Molecular Imaging. 50 (6): 1651–1664. doi:10.1007/s00259-022-06103-1. PMC 10119077. PMID 36656363.

ncbi.nlm.nih.gov

parkinsons.org.uk (Global: low place; English: low place)

prlog.org (Global: 9,932nd place; English: 6,569th place)

prnewswire.com (Global: 406th place; English: 258th place)

psu.edu (Global: 207th place; English: 136th place)

citeseerx.ist.psu.edu

  • Vacher B, Bonnaud B, Funes P, Jubault N, Koek W, Assié MB, et al. (May 1999). "Novel derivatives of 2-pyridinemethylamine as selective, potent, and orally active agonists at 5-HT1A receptors". Journal of Medicinal Chemistry. 42 (9): 1648–1660. CiteSeerX 10.1.1.325.8872. doi:10.1021/jm9806906. PMID 10229633.

semanticscholar.org (Global: 11th place; English: 8th place)

api.semanticscholar.org

  • Newman-Tancredi A, Martel JC, Cosi C, Heusler P, Lestienne F, Varney MA, et al. (September 2017). "Distinctive in vitro signal transduction profile of NLX-112, a potent and efficacious serotonin 5-HT1A receptor agonist". The Journal of Pharmacy and Pharmacology. 69 (9): 1178–1190. doi:10.1111/jphp.12762. PMID 28612503. S2CID 13676820.
  • Lladó-Pelfort L, Assié MB, Newman-Tancredi A, Artigas F, Celada P (May 2012). "In vivo electrophysiological and neurochemical effects of the selective 5-HT1A receptor agonist, F13640, at pre- and postsynaptic 5-HT1A receptors in the rat". Psychopharmacology. 221 (2): 261–272. doi:10.1007/s00213-011-2569-9. PMID 22147258. S2CID 18779324.
  • Bardin L, Tarayre JP, Malfetes N, Koek W, Colpaert FC (April 2003). "Profound, non-opioid analgesia produced by the high-efficacy 5-HT(1A) agonist F 13640 in the formalin model of tonic nociceptive pain". Pharmacology. 67 (4): 182–194. doi:10.1159/000068404. PMID 12595749. S2CID 25882138.
  • Bardin L, Assié MB, Pélissou M, Royer-Urios I, Newman-Tancredi A, Ribet JP, et al. (March 2005). "Dual, hyperalgesic, and analgesic effects of the high-efficacy 5-hydroxytryptamine 1A (5-HT1A) agonist F 13640 [(3-chloro-4-fluoro-phenyl)-[4-fluoro-4-{[(5-methyl-pyridin-2-ylmethyl)-amino]-methyl}piperidin-1-yl]methanone, fumaric acid salt]: relationship with 5-HT1A receptor occupancy and kinetic parameters". The Journal of Pharmacology and Experimental Therapeutics. 312 (3): 1034–1042. doi:10.1124/jpet.104.077669. PMID 15528450. S2CID 42446435.
  • Colpaert FC, Deseure K, Stinus L, Adriaensen H (February 2006). "High-efficacy 5-hydroxytryptamine 1A receptor activation counteracts opioid hyperallodynia and affective conditioning". The Journal of Pharmacology and Experimental Therapeutics. 316 (2): 892–899. doi:10.1124/jpet.105.095109. PMID 16254131. S2CID 8820667.
  • Iderberg H, McCreary AC, Varney MA, Kleven MS, Koek W, Bardin L, et al. (September 2015). "NLX-112, a novel 5-HT1A receptor agonist for the treatment of L-DOPA-induced dyskinesia: Behavioral and neurochemical profile in rat". Experimental Neurology. 271: 335–350. doi:10.1016/j.expneurol.2015.05.021. PMID 26037043. S2CID 35525495.
  • McCreary AC, Varney MA, Newman-Tancredi A (June 2016). "The novel 5-HT1A receptor agonist, NLX-112 reduces l-DOPA-induced abnormal involuntary movements in rat: A chronic administration study with microdialysis measurements". Neuropharmacology. 105: 651–660. doi:10.1016/j.neuropharm.2016.01.013. PMID 26777281. S2CID 1979117.
  • Depoortere R, Johnston TH, Fox SH, Brotchie JM, Newman-Tancredi A (September 2020). "The selective 5-HT1A receptor agonist, NLX-112, exerts anti-dyskinetic effects in MPTP-treated macaques". Parkinsonism & Related Disorders. 78: 151–157. doi:10.1016/j.parkreldis.2020.08.009. PMID 32846366. S2CID 221343904.

thetimes.com (Global: low place; English: low place)