Tatsumi M, Groshan K, Blakely RD, Richelson E (December 1997). "Pharmacological profile of antidepressants and related compounds at human monoamine transporters". European Journal of Pharmacology. 340 (2–3): 249–258. doi:10.1016/s0014-2999(97)01393-9. PMID9537821.
Hoffman BJ, Scheffel U, Lever JR, Karpa MD, Hartig PR (January 1987). "N1-methyl-2-125I-lysergic acid diethylamide, a preferred ligand for in vitro and in vivo characterization of serotonin receptors". Journal of Neurochemistry. 48 (1): 115–124. doi:10.1111/j.1471-4159.1987.tb13135.x. PMID3794694. S2CID23311638.
Arias-Montaño JA, Young JM (May 1993). "Characteristics of histamine H1 receptors on HeLa cells". European Journal of Pharmacology. 245 (3): 291–295. doi:10.1016/0922-4106(93)90110-u. PMID8335064.
West RE, Zweig A, Granzow RT, Siegel MI, Egan RW (November 1990). "Biexponential kinetics of (R)-alpha-[3H]methylhistamine binding to the rat brain H3 histamine receptor". Journal of Neurochemistry. 55 (5): 1612–1616. doi:10.1111/j.1471-4159.1990.tb04946.x. PMID2213013. S2CID83953993.
Yasuda SU, Yasuda RP (April 1999). "Affinities of brompheniramine, chlorpheniramine, and terfenadine at the five human muscarinic cholinergic receptor subtypes". Pharmacotherapy. 19 (4): 447–451. doi:10.1592/phco.19.6.447.31041. PMID10212017. S2CID39502992.
Simons FE (November 2004). "Advances in H1-antihistamines". The New England Journal of Medicine. 351 (21): 2203–2217. doi:10.1056/NEJMra033121. PMID15548781.
Leurs R, Church MK, Taglialatela M (April 2002). "H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects". Clinical and Experimental Allergy. 32 (4): 489–498. doi:10.1046/j.0954-7894.2002.01314.x. PMID11972592. S2CID11849647.
Cusack B, Nelson A, Richelson E (May 1994). "Binding of antidepressants to human brain receptors: focus on newer generation compounds". Psychopharmacology. 114 (4): 559–565. doi:10.1007/bf02244985. PMID7855217. S2CID21236268.
Carlsson A, Lindqvist M (July 1969). "Central and peripheral monoaminergic membrane-pump blockade by some addictive analgesics and antihistamines". The Journal of Pharmacy and Pharmacology. 21 (7): 460–464. doi:10.1111/j.2042-7158.1969.tb08287.x. PMID4390069. S2CID39627573.
Booth RG, Moniri NH, Bakker RA, Choksi NY, Nix WB, Timmerman H, Leurs R (July 2002). "A novel phenylaminotetralin radioligand reveals a subpopulation of histamine H(1) receptors". The Journal of Pharmacology and Experimental Therapeutics. 302 (1): 328–336. doi:10.1124/jpet.302.1.328. PMID12065734. S2CID2600032.
Djerassi C, Scholz CR (January 1948). "Brominations with pyridine hydrobromide perbromide". Journal of the American Chemical Society. 70 (1): 417–418. doi:10.1021/ja01181a508. PMID18918843.
drugs.com
"Chlorpheniramine". Drugs.com. American Society of Health-System Pharmacists. 26 July 2023. Archived from the original on 20 August 2023. Retrieved 20 August 2023.
Tatsumi M, Groshan K, Blakely RD, Richelson E (December 1997). "Pharmacological profile of antidepressants and related compounds at human monoamine transporters". European Journal of Pharmacology. 340 (2–3): 249–258. doi:10.1016/s0014-2999(97)01393-9. PMID9537821.
Hoffman BJ, Scheffel U, Lever JR, Karpa MD, Hartig PR (January 1987). "N1-methyl-2-125I-lysergic acid diethylamide, a preferred ligand for in vitro and in vivo characterization of serotonin receptors". Journal of Neurochemistry. 48 (1): 115–124. doi:10.1111/j.1471-4159.1987.tb13135.x. PMID3794694. S2CID23311638.
Sanders-Bush E, Breeding M (October 1988). "Putative selective 5-HT-2 antagonists block serotonin 5-HT-1c receptors in the choroid plexus". The Journal of Pharmacology and Experimental Therapeutics. 247 (1): 169–173. PMID3139864.
Arias-Montaño JA, Young JM (May 1993). "Characteristics of histamine H1 receptors on HeLa cells". European Journal of Pharmacology. 245 (3): 291–295. doi:10.1016/0922-4106(93)90110-u. PMID8335064.
West RE, Zweig A, Granzow RT, Siegel MI, Egan RW (November 1990). "Biexponential kinetics of (R)-alpha-[3H]methylhistamine binding to the rat brain H3 histamine receptor". Journal of Neurochemistry. 55 (5): 1612–1616. doi:10.1111/j.1471-4159.1990.tb04946.x. PMID2213013. S2CID83953993.
Yasuda SU, Yasuda RP (April 1999). "Affinities of brompheniramine, chlorpheniramine, and terfenadine at the five human muscarinic cholinergic receptor subtypes". Pharmacotherapy. 19 (4): 447–451. doi:10.1592/phco.19.6.447.31041. PMID10212017. S2CID39502992.
Simons FE (November 2004). "Advances in H1-antihistamines". The New England Journal of Medicine. 351 (21): 2203–2217. doi:10.1056/NEJMra033121. PMID15548781.
Leurs R, Church MK, Taglialatela M (April 2002). "H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects". Clinical and Experimental Allergy. 32 (4): 489–498. doi:10.1046/j.0954-7894.2002.01314.x. PMID11972592. S2CID11849647.
Richelson E, Nelson A (July 1984). "Antagonism by antidepressants of neurotransmitter receptors of normal human brain in vitro". The Journal of Pharmacology and Experimental Therapeutics. 230 (1): 94–102. PMID6086881.
Cusack B, Nelson A, Richelson E (May 1994). "Binding of antidepressants to human brain receptors: focus on newer generation compounds". Psychopharmacology. 114 (4): 559–565. doi:10.1007/bf02244985. PMID7855217. S2CID21236268.
Carlsson A, Lindqvist M (July 1969). "Central and peripheral monoaminergic membrane-pump blockade by some addictive analgesics and antihistamines". The Journal of Pharmacy and Pharmacology. 21 (7): 460–464. doi:10.1111/j.2042-7158.1969.tb08287.x. PMID4390069. S2CID39627573.
Booth RG, Moniri NH, Bakker RA, Choksi NY, Nix WB, Timmerman H, Leurs R (July 2002). "A novel phenylaminotetralin radioligand reveals a subpopulation of histamine H(1) receptors". The Journal of Pharmacology and Experimental Therapeutics. 302 (1): 328–336. doi:10.1124/jpet.302.1.328. PMID12065734. S2CID2600032.
Djerassi C, Scholz CR (January 1948). "Brominations with pyridine hydrobromide perbromide". Journal of the American Chemical Society. 70 (1): 417–418. doi:10.1021/ja01181a508. PMID18918843.
Yasuda SU, Wellstein A, Likhari P, Barbey JT, Woosley RL (August 1995). "Chlorpheniramine plasma concentration and histamine H1-receptor occupancy". Clinical Pharmacology and Therapeutics. 58 (2): 210–220. doi:10.1016/0009-9236(95)90199-X. PMID7648771. S2CID35759573.
Hoffman BJ, Scheffel U, Lever JR, Karpa MD, Hartig PR (January 1987). "N1-methyl-2-125I-lysergic acid diethylamide, a preferred ligand for in vitro and in vivo characterization of serotonin receptors". Journal of Neurochemistry. 48 (1): 115–124. doi:10.1111/j.1471-4159.1987.tb13135.x. PMID3794694. S2CID23311638.
West RE, Zweig A, Granzow RT, Siegel MI, Egan RW (November 1990). "Biexponential kinetics of (R)-alpha-[3H]methylhistamine binding to the rat brain H3 histamine receptor". Journal of Neurochemistry. 55 (5): 1612–1616. doi:10.1111/j.1471-4159.1990.tb04946.x. PMID2213013. S2CID83953993.
Yasuda SU, Yasuda RP (April 1999). "Affinities of brompheniramine, chlorpheniramine, and terfenadine at the five human muscarinic cholinergic receptor subtypes". Pharmacotherapy. 19 (4): 447–451. doi:10.1592/phco.19.6.447.31041. PMID10212017. S2CID39502992.
Leurs R, Church MK, Taglialatela M (April 2002). "H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects". Clinical and Experimental Allergy. 32 (4): 489–498. doi:10.1046/j.0954-7894.2002.01314.x. PMID11972592. S2CID11849647.
Cusack B, Nelson A, Richelson E (May 1994). "Binding of antidepressants to human brain receptors: focus on newer generation compounds". Psychopharmacology. 114 (4): 559–565. doi:10.1007/bf02244985. PMID7855217. S2CID21236268.
Carlsson A, Lindqvist M (July 1969). "Central and peripheral monoaminergic membrane-pump blockade by some addictive analgesics and antihistamines". The Journal of Pharmacy and Pharmacology. 21 (7): 460–464. doi:10.1111/j.2042-7158.1969.tb08287.x. PMID4390069. S2CID39627573.
Booth RG, Moniri NH, Bakker RA, Choksi NY, Nix WB, Timmerman H, Leurs R (July 2002). "A novel phenylaminotetralin radioligand reveals a subpopulation of histamine H(1) receptors". The Journal of Pharmacology and Experimental Therapeutics. 302 (1): 328–336. doi:10.1124/jpet.302.1.328. PMID12065734. S2CID2600032.
unc.edu
kidbdev.med.unc.edu
Roth BL, Driscol J. "PDSP Ki Database". Psychoactive Drug Screening Program (PDSP). University of North Carolina at Chapel Hill and the United States National Institute of Mental Health. Archived from the original on 2 October 2020. Retrieved 14 August 2017.
"Chlorpheniramine". Drugs.com. American Society of Health-System Pharmacists. 26 July 2023. Archived from the original on 20 August 2023. Retrieved 20 August 2023.
"Cêgripe". Cegripe.pt. Archived from the original on 25 June 2022. Retrieved 10 June 2022.
Roth BL, Driscol J. "PDSP Ki Database". Psychoactive Drug Screening Program (PDSP). University of North Carolina at Chapel Hill and the United States National Institute of Mental Health. Archived from the original on 2 October 2020. Retrieved 14 August 2017.