Disappearing polymorphs (English Wikipedia)

Rubin-Preminger JM, Bernstein J (2005-07-01). "3-Aminobenzenesulfonic Acid: A Disappearing Polymorph". Crystal Growth & Design. 5 (4): 1343–1349. doi:10.1021/cg049680y. ISSN 1528-7483.
Bučar DK, Lancaster RW, Bernstein J (June 2015). "Disappearing polymorphs revisited". Angewandte Chemie. 54 (24): 6972–6993. doi:10.1002/anie.201410356. PMC 4479028. PMID 26031248.
Dunitz JD, Bernstein J (1995-04-01). "Disappearing Polymorphs". Accounts of Chemical Research. 28 (4): 193–200. doi:10.1021/ar00052a005. ISSN 0001-4842.
Surov AO, Vasilev NA, Churakov AV, Stroh J, Emmerling F, Perlovich GL (2019). "Solid Forms of Ciprofloxacin Salicylate: Polymorphism, Formation Pathways and Thermodynamic Stability". Crystal Growth & Design. 19 (5): 2979–2990. doi:10.1021/acs.cgd.9b00185. S2CID 132854494.
Ward MD (February 2017). "Perils of Polymorphism: Size Matters". Israel Journal of Chemistry. 57 (1–2): 82–92. doi:10.1002/ijch.201600071. ISSN 0021-2148.
Threlfall T (2000-09-01). "Crystallisation of Polymorphs: Thermodynamic Insight into the Role of Solvent". Organic Process Research & Development. 4 (5): 384–390. doi:10.1021/op000058y. ISSN 1083-6160.
Vure P (2011). "Polymorph patents; how strong they are really?". International Journal of Intellectual Property Management. 4 (4): 297. doi:10.1504/IJIPM.2011.043875. ISSN 1478-9647.
Rakoczy WA, Mazzochi DM (January 2006). "The Case of the Disappearing Polymorph: 'Inherent Anticipation' and the Impact of SmithKline Beecham Corp. v Apotex Corp. (Paxil®) on Patent Validity and Infringement by Inevitable Conversion". Journal of Generic Medicines: The Business Journal for the Generic Medicines Sector. 3 (2): 131–139. doi:10.1057/palgrave.jgm.4940110. ISSN 1741-1343.
Pina MF, Pinto JF, Sousa JJ, Fábián L, Zhao M, Craig DQ (December 2012). "Identification and characterization of stoichiometric and nonstoichiometric hydrate forms of paroxetine HCl: reversible changes in crystal dimensions as a function of water absorption". Molecular Pharmaceutics. 9 (12): 3515–3525. doi:10.1021/mp3003573. PMID 23051151.
Morissette SL, Soukasene S, Levinson D, Cima MJ, Almarsson O (March 2003). "Elucidation of crystal form diversity of the HIV protease inhibitor ritonavir by high-throughput crystallization". Proceedings of the National Academy of Sciences of the United States of America. 100 (5): 2180–2184. doi:10.1073/pnas.0437744100. PMC 151315. PMID 12604798.
Chen JJ, Swope DM, Dashtipour K, Lyons KE (December 2009). "Transdermal rotigotine: a clinically innovative dopamine-receptor agonist for the management of Parkinson's disease". Pharmacotherapy. 29 (12): 1452–1467. doi:10.1592/phco.29.12.1452. PMID 19947805. S2CID 40466260.
Davies S (September 2009). "Rotigotine for restless legs syndrome". Drugs of Today. 45 (9): 663–668. doi:10.1358/dot.2009.45.9.1399952. PMID 19956807.
Lancaster RW, Karamertzanis PG, Hulme AT, Tocher DA, Lewis TC, Price SL (December 2007). "The polymorphism of progesterone: stabilization of a 'disappearing' polymorph by co-crystallization". Journal of Pharmaceutical Sciences. 96 (12): 3419–3431. doi:10.1002/jps.20983. PMID 17621678.
Kim HS, Jeffrey GA (1969-12-15). "The crystal structure of xylitol". Acta Crystallographica Section B: Structural Crystallography and Crystal Chemistry. 25 (12): 2607–2613. doi:10.1107/S0567740869006133. ISSN 0567-7408.
Trask AV (2007). "An overview of pharmaceutical cocrystals as intellectual property". Molecular Pharmaceutics. 4 (3): 301–9. doi:10.1021/mp070001z. PMID 17477544.
"{BLR 2023} Azeotroping Process – CAFC – Glaxo – Novopharm – Ranitidine". Biotechnology Law Report. 14 (3): 423–504. May 1995. doi:10.1089/blr.1995.14.423. ISSN 0730-031X.
Hicks AJ (2020-05-18). "Cat's Cradle". Posthumanism in the Novels of Kurt Vonnegut. Routledge. pp. 25–51. doi:10.4324/9780367521646-3. ISBN 9780367521646.

handle.net

hdl.handle.net

World Health Organization (2019). World Health Organization model list of essential medicines: 21st list 2019. Geneva: World Health Organization. hdl:10665/325771. WHO/MVP/EMP/IAU/2019.06. License: CC BY-NC-SA 3.0 IGO.

inderscience.com

Vure P (2011). "Polymorph patents; how strong they are really?". International Journal of Intellectual Property Management. 4 (4): 297. doi:10.1504/IJIPM.2011.043875. ISSN 1478-9647.

iucr.org

scripts.iucr.org

Kim HS, Jeffrey GA (1969-12-15). "The crystal structure of xylitol". Acta Crystallographica Section B: Structural Crystallography and Crystal Chemistry. 25 (12): 2607–2613. doi:10.1107/S0567740869006133. ISSN 0567-7408.

liebertpub.com

"{BLR 2023} Azeotroping Process – CAFC – Glaxo – Novopharm – Ranitidine". Biotechnology Law Report. 14 (3): 423–504. May 1995. doi:10.1089/blr.1995.14.423. ISSN 0730-031X.

nih.gov

pubmed.ncbi.nlm.nih.gov

Bučar DK, Lancaster RW, Bernstein J (June 2015). "Disappearing polymorphs revisited". Angewandte Chemie. 54 (24): 6972–6993. doi:10.1002/anie.201410356. PMC 4479028. PMID 26031248.
Pina MF, Pinto JF, Sousa JJ, Fábián L, Zhao M, Craig DQ (December 2012). "Identification and characterization of stoichiometric and nonstoichiometric hydrate forms of paroxetine HCl: reversible changes in crystal dimensions as a function of water absorption". Molecular Pharmaceutics. 9 (12): 3515–3525. doi:10.1021/mp3003573. PMID 23051151.
Morissette SL, Soukasene S, Levinson D, Cima MJ, Almarsson O (March 2003). "Elucidation of crystal form diversity of the HIV protease inhibitor ritonavir by high-throughput crystallization". Proceedings of the National Academy of Sciences of the United States of America. 100 (5): 2180–2184. doi:10.1073/pnas.0437744100. PMC 151315. PMID 12604798.
Chen JJ, Swope DM, Dashtipour K, Lyons KE (December 2009). "Transdermal rotigotine: a clinically innovative dopamine-receptor agonist for the management of Parkinson's disease". Pharmacotherapy. 29 (12): 1452–1467. doi:10.1592/phco.29.12.1452. PMID 19947805. S2CID 40466260.
Davies S (September 2009). "Rotigotine for restless legs syndrome". Drugs of Today. 45 (9): 663–668. doi:10.1358/dot.2009.45.9.1399952. PMID 19956807.
Lancaster RW, Karamertzanis PG, Hulme AT, Tocher DA, Lewis TC, Price SL (December 2007). "The polymorphism of progesterone: stabilization of a 'disappearing' polymorph by co-crystallization". Journal of Pharmaceutical Sciences. 96 (12): 3419–3431. doi:10.1002/jps.20983. PMID 17621678.
Trask AV (2007). "An overview of pharmaceutical cocrystals as intellectual property". Molecular Pharmaceutics. 4 (3): 301–9. doi:10.1021/mp070001z. PMID 17477544.

ncbi.nlm.nih.gov

Bučar DK, Lancaster RW, Bernstein J (June 2015). "Disappearing polymorphs revisited". Angewandte Chemie. 54 (24): 6972–6993. doi:10.1002/anie.201410356. PMC 4479028. PMID 26031248.
Morissette SL, Soukasene S, Levinson D, Cima MJ, Almarsson O (March 2003). "Elucidation of crystal form diversity of the HIV protease inhibitor ritonavir by high-throughput crystallization". Proceedings of the National Academy of Sciences of the United States of America. 100 (5): 2180–2184. doi:10.1073/pnas.0437744100. PMC 151315. PMID 12604798.

openjurist.org

110 F. 3d 1562 – Glaxo Inc v. Novopharm Ltd. No. 96-1466. United States Court of Appeals, Federal Circuit. April 4, 1997.

patents.google.com

US4007196A, Christensen, Jorgen Anders & Squires, Richard Felt, "4-Phenylpiperidine compounds", issued 1977-02-08
US4504657A, Bouzard, Daniel; Weber, Abraham & Stemer, Jacques, "Cephadroxil monohydrate", issued 1985-03-12
US3781282A, Garbrecht, W., "Cephalosporin process and product", issued 1973-12-25
US4128658A, Price, Barry J.; Clitherow, John W. & Bradshaw, John, "Aminoalkyl furan derivatives", issued 1978-12-05
US4521431A, Crookes, Derek L., "Aminoalkyl furan derivative", issued 1985-06-04
US4672133A, Crookes, Derek L., "Process for forming Form 2 ranitidine hydrochloride", issued 1987-06-09

pdf.org

"Neupro Patch Re-launches in the US". Archived from the original on 2016-03-23. Retrieved 2022-07-08.

science.org

Lowe D. "Down At the Crystal Surface". In the Pipeline. American Association for the Advancement of Science. Retrieved 2022-07-08.

semanticscholar.org

api.semanticscholar.org

Surov AO, Vasilev NA, Churakov AV, Stroh J, Emmerling F, Perlovich GL (2019). "Solid Forms of Ciprofloxacin Salicylate: Polymorphism, Formation Pathways and Thermodynamic Stability". Crystal Growth & Design. 19 (5): 2979–2990. doi:10.1021/acs.cgd.9b00185. S2CID 132854494.
Chen JJ, Swope DM, Dashtipour K, Lyons KE (December 2009). "Transdermal rotigotine: a clinically innovative dopamine-receptor agonist for the management of Parkinson's disease". Pharmacotherapy. 29 (12): 1452–1467. doi:10.1592/phco.29.12.1452. PMID 19947805. S2CID 40466260.

supercheats.com

"Game Script". Super Cheats.

web.archive.org

Lowe D (November 26, 2019). "Perverse Polymorphism". In the Pipeline. American Association for the Advancement of Science. Archived from the original on July 5, 2022. Retrieved 2022-07-04.{{cite web}}: CS1 maint: bot: original URL status unknown (link)
"Neupro Patch Re-launches in the US". Archived from the original on 2016-03-23. Retrieved 2022-07-08.

worldcat.org

search.worldcat.org

Rubin-Preminger JM, Bernstein J (2005-07-01). "3-Aminobenzenesulfonic Acid: A Disappearing Polymorph". Crystal Growth & Design. 5 (4): 1343–1349. doi:10.1021/cg049680y. ISSN 1528-7483.
Dunitz JD, Bernstein J (1995-04-01). "Disappearing Polymorphs". Accounts of Chemical Research. 28 (4): 193–200. doi:10.1021/ar00052a005. ISSN 0001-4842.
Ward MD (February 2017). "Perils of Polymorphism: Size Matters". Israel Journal of Chemistry. 57 (1–2): 82–92. doi:10.1002/ijch.201600071. ISSN 0021-2148.
Threlfall T (2000-09-01). "Crystallisation of Polymorphs: Thermodynamic Insight into the Role of Solvent". Organic Process Research & Development. 4 (5): 384–390. doi:10.1021/op000058y. ISSN 1083-6160.
Vure P (2011). "Polymorph patents; how strong they are really?". International Journal of Intellectual Property Management. 4 (4): 297. doi:10.1504/IJIPM.2011.043875. ISSN 1478-9647.
Rakoczy WA, Mazzochi DM (January 2006). "The Case of the Disappearing Polymorph: 'Inherent Anticipation' and the Impact of SmithKline Beecham Corp. v Apotex Corp. (Paxil®) on Patent Validity and Infringement by Inevitable Conversion". Journal of Generic Medicines: The Business Journal for the Generic Medicines Sector. 3 (2): 131–139. doi:10.1057/palgrave.jgm.4940110. ISSN 1741-1343.
Kim HS, Jeffrey GA (1969-12-15). "The crystal structure of xylitol". Acta Crystallographica Section B: Structural Crystallography and Crystal Chemistry. 25 (12): 2607–2613. doi:10.1107/S0567740869006133. ISSN 0567-7408.
"{BLR 2023} Azeotroping Process – CAFC – Glaxo – Novopharm – Ranitidine". Biotechnology Law Report. 14 (3): 423–504. May 1995. doi:10.1089/blr.1995.14.423. ISSN 0730-031X.