References analysis of the Wikipedia article "Discovery and development of antiandrogens" in the English version

doi.org

Denmeade SR, Isaacs JT (May 2002). "A history of prostate cancer treatment". Nature Reviews. Cancer. 2 (5): 389–96. doi:10.1038/nrc801. PMC 4124639. PMID 12044015.

Gao W (October 2010). "Androgen receptor as a therapeutic target". Advanced Drug Delivery Reviews. 62 (13): 1277–84. doi:10.1016/j.addr.2010.08.002. PMID 20708648.

Singh SM, Gauthier S, Labrie F (February 2000). "Androgen receptor antagonists (antiandrogens): structure-activity relationships". Current Medicinal Chemistry. 7 (2): 211–47. doi:10.2174/0929867003375371. PMID 10637363.

Williams L, Thompson LD, Seethala RR, Weinreb I, Assaad AM, Tuluc M, et al. (May 2015). "Salivary duct carcinoma: the predominance of apocrine morphology, prevalence of histologic variants, and androgen receptor expression". The American Journal of Surgical Pathology. 39 (5): 705–13. doi:10.1097/pas.0000000000000413. PMID 25871467. S2CID 24737257.

Gucalp A, Traina TA (Jan–Feb 2010). "Triple-negative breast cancer: role of the androgen receptor". Cancer Journal. 16 (1): 62–5. doi:10.1097/PPO.0b013e3181ce4ae1. PMID 20164692. S2CID 6922842.

Urban D, Rischin D, Angel C, D'Costa I, Solomon B (March 2015). "Abiraterone in metastatic salivary duct carcinoma". Journal of the National Comprehensive Cancer Network. 13 (3): 288–90. doi:10.6004/jnccn.2015.0040. PMID 25736005.

Haendler B, Cleve A (April 2012). "Recent developments in antiandrogens and selective androgen receptor modulators". Molecular and Cellular Endocrinology. 352 (1–2): 79–91. doi:10.1016/j.mce.2011.06.002. PMID 21704118. S2CID 36184991.

Gao W (2010). "Peptide antagonist of the androgen receptor". Current Pharmaceutical Design. 16 (9): 1106–13. doi:10.2174/138161210790963850. PMID 20030610.

Gao W, Kim J, Dalton JT (August 2006). "Pharmacokinetics and pharmacodynamics of nonsteroidal androgen receptor ligands". Pharmaceutical Research. 23 (8): 1641–58. doi:10.1007/s11095-006-9024-3. PMC 2072875. PMID 16841196.

Narayanan R, Mohler ML, Bohl CE, Miller DD, Dalton JT (2008). "Selective androgen receptor modulators in preclinical and clinical development". Nuclear Receptor Signaling. 6: e010. doi:10.1621/nrs.06010. PMC 2602589. PMID 19079612.

Gelmann EP (July 2002). "Molecular biology of the androgen receptor". Journal of Clinical Oncology. 20 (13): 3001–15. doi:10.1200/jco.2002.10.018. PMID 12089231.

Poyet P, Labrie F (October 1985). "Comparison of the antiandrogenic/androgenic activities of flutamide, cyproterone acetate and megestrol acetate". Molecular and Cellular Endocrinology. 42 (3): 283–8. doi:10.1016/0303-7207(85)90059-0. PMID 3930312. S2CID 24746807.

Yin D, He Y, Perera MA, Hong SS, Marhefka C, Stourman N, et al. (January 2003). "Key structural features of nonsteroidal ligands for binding and activation of the androgen receptor". Molecular Pharmacology. 63 (1): 211–23. doi:10.1124/mol.63.1.211. PMC 2040236. PMID 12488554.

Miyamoto H, Rahman MM, Chang C (January 2004). "Molecular basis for the antiandrogen withdrawal syndrome". Journal of Cellular Biochemistry. 91 (1): 3–12. doi:10.1002/jcb.10757. PMID 14689576. S2CID 5773128.

Jiang Y, Palma JF, Agus DB, Wang Y, Gross ME (September 2010). "Detection of androgen receptor mutations in circulating tumor cells in castration-resistant prostate cancer" (PDF). Clinical Chemistry. 56 (9): 1492–5. doi:10.1373/clinchem.2010.143297. PMID 20581083. Archived (PDF) from the original on 2017-08-17. Retrieved 2019-09-02.

Suzuki H, Akakura K, Komiya A, Aida S, Akimoto S, Shimazaki J (September 1996). "Codon 877 mutation in the androgen receptor gene in advanced prostate cancer: relation to antiandrogen withdrawal syndrome". The Prostate. 29 (3): 153–8. doi:10.1002/1097-0045(199609)29:3<153::aid-pros2990290303>3.0.co;2-5. PMID 8827083. S2CID 22806905.

Bohl CE, Gao W, Miller DD, Bell CE, Dalton JT (April 2005). "Structural basis for antagonism and resistance of bicalutamide in prostate cancer". Proceedings of the National Academy of Sciences of the United States of America. 102 (17): 6201–6. Bibcode:2005PNAS..102.6201B. doi:10.1073/pnas.0500381102. PMC 1087923. PMID 15833816.

Sadar MD, Williams DE, Mawji NR, Patrick BO, Wikanta T, Chasanah E, et al. (November 2008). "Sintokamides A to E, chlorinated peptides from the sponge Dysidea sp. that inhibit transactivation of the N-terminus of the androgen receptor in prostate cancer cells". Organic Letters. 10 (21): 4947–50. doi:10.1021/ol802021w. PMID 18834139.

Gao W, Dalton JT (March 2007). "Expanding the therapeutic use of androgens via selective androgen receptor modulators (SARMs)". Drug Discovery Today. 12 (5–6): 241–8. doi:10.1016/j.drudis.2007.01.003. PMC 2072879. PMID 17331889.

Battmann T, Branche C, Bouchoux F, Cerede E, Philibert D, Goubet F, et al. (January 1998). "Pharmacological profile of RU 58642, a potent systemic antiandrogen for the treatment of androgen-dependent disorders". The Journal of Steroid Biochemistry and Molecular Biology. 64 (1–2): 103–11. doi:10.1016/S0960-0760(97)00151-9. PMID 9569015. S2CID 290926.

Hamann LG, Higuchi RI, Zhi L, Edwards JP, Wang XN, Marschke KB, et al. (February 1998). "Synthesis and biological activity of a novel series of nonsteroidal, peripherally selective androgen receptor antagonists derived from 1,2-dihydropyridono[5,6-g]quinolines". Journal of Medicinal Chemistry. 41 (4): 623–39. doi:10.1021/jm970699s. PMID 9484511.

Tran C, Ouk S, Clegg NJ, Chen Y, Watson PA, Arora V, et al. (May 2009). "Development of a second-generation antiandrogen for treatment of advanced prostate cancer". Science. 324 (5928): 787–90. Bibcode:2009Sci...324..787T. doi:10.1126/science.1168175. PMC 2981508. PMID 19359544.

Scher HI, Beer TM, Higano CS, Anand A, Taplin ME, Efstathiou E, et al. (April 2010). "Antitumour activity of MDV3100 in castration-resistant prostate cancer: a phase 1-2 study". Lancet. 375 (9724): 1437–46. doi:10.1016/S0140-6736(10)60172-9. PMC 2948179. PMID 20398925.

Rathkopf D, Liu G, Carducci MA, Eisenberger MA, Anand A, Morris MJ, et al. (February 2011). "Phase I dose-escalation study of the novel antiandrogen BMS-641988 in patients with castration-resistant prostate cancer". Clinical Cancer Research. 17 (4): 880–7. doi:10.1158/1078-0432.CCR-10-2955. PMC 3070382. PMID 21131556.

Foster WR, Car BD, Shi H, Levesque PC, Obermeier MT, Gan J, et al. (April 2011). "Drug safety is a barrier to the discovery and development of new androgen receptor antagonists". The Prostate. 71 (5): 480–8. doi:10.1002/pros.21263. PMID 20878947. S2CID 24620044.

Kawata H, Arai S, Nakagawa T, Ishikura N, Nishimoto A, Yoshino H, et al. (September 2011). "Biological properties of androgen receptor pure antagonist for treatment of castration-resistant prostate cancer: optimization from lead compound to CH5137291". The Prostate. 71 (12): 1344–56. doi:10.1002/pros.21351. PMID 21308717. S2CID 42009977.

Yoshino H, Sato H, Shiraishi T, Tachibana K, Emura T, Honma A, et al. (December 2010). "Design and synthesis of an androgen receptor pure antagonist (CH5137291) for the treatment of castration-resistant prostate cancer". Bioorganic & Medicinal Chemistry. 18 (23): 8150–7. doi:10.1016/j.bmc.2010.10.023. PMID 21050768.

Schleich S, Papaioannou M, Baniahmad A, Matusch R (July 2006). "Extracts from Pygeum africanum and other ethnobotanical species with antiandrogenic activity". Planta Medica. 72 (9): 807–13. doi:10.1055/s-2006-946638. PMID 16783690. S2CID 260278595.

Roell D, Baniahmad A (January 2011). "The natural compounds atraric acid and N-butylbenzene-sulfonamide as antagonists of the human androgen receptor and inhibitors of prostate cancer cell growth" (PDF). Molecular and Cellular Endocrinology. 332 (1–2): 1–8. doi:10.1016/j.mce.2010.09.013. PMID 20965230. S2CID 26865620. Archived (PDF) from the original on 2019-10-01. Retrieved 2019-10-01.

nih.gov

pubmed.ncbi.nlm.nih.gov

Denmeade SR, Isaacs JT (May 2002). "A history of prostate cancer treatment". Nature Reviews. Cancer. 2 (5): 389–96. doi:10.1038/nrc801. PMC 4124639. PMID 12044015.

Gao W (October 2010). "Androgen receptor as a therapeutic target". Advanced Drug Delivery Reviews. 62 (13): 1277–84. doi:10.1016/j.addr.2010.08.002. PMID 20708648.

Gucalp A, Traina TA (Jan–Feb 2010). "Triple-negative breast cancer: role of the androgen receptor". Cancer Journal. 16 (1): 62–5. doi:10.1097/PPO.0b013e3181ce4ae1. PMID 20164692. S2CID 6922842.

Gao W (2010). "Peptide antagonist of the androgen receptor". Current Pharmaceutical Design. 16 (9): 1106–13. doi:10.2174/138161210790963850. PMID 20030610.

Gelmann EP (July 2002). "Molecular biology of the androgen receptor". Journal of Clinical Oncology. 20 (13): 3001–15. doi:10.1200/jco.2002.10.018. PMID 12089231.

Hara T, Miyazaki J, Araki H, Yamaoka M, Kanzaki N, Kusaka M, et al. (January 2003). "Novel mutations of androgen receptor: a possible mechanism of bicalutamide withdrawal syndrome". Cancer Research. 63 (1): 149–53. PMID 12517791.

ncbi.nlm.nih.gov

semanticscholar.org

api.semanticscholar.org

Gucalp A, Traina TA (Jan–Feb 2010). "Triple-negative breast cancer: role of the androgen receptor". Cancer Journal. 16 (1): 62–5. doi:10.1097/PPO.0b013e3181ce4ae1. PMID 20164692. S2CID 6922842.

Discovery and development of antiandrogens (English Wikipedia)

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