Green, Brian; Flatt, Peter; Bailey, Clifford (December 2006), "Dipeptidyl peptidase IV (DPP IV) inhibitors: a newly emerging drug class for the treatment of type 2 diabetes", Diabetes and Vascular Disease Research, 3 (3): 159–165, doi:10.3132/dvdr.2006.024, PMID17160910
Sebokova, Elena; Christ, Andreas; Boehringer, Markus; Mizrahi, Jacques (May 2006), "Dipeptidyl peptidase IV inhibitors: The next generation of new promising therapies for the management of type 2 diabetes", Current Topics in Medicinal Chemistry, 7 (6): 547–555, doi:10.2174/156802607780091019, PMID17352676
Ahn, Jin Hee; Shin, Mi Sik; June, Mi Ae; Jung, Sun Ho; Kang, Seung Kyu; Kim, Kwang Rok; Rhee, Sang Dal; Kang, Nam Sook; Kim, Seung Kyu (February 2007), "Synthesis, biological evaluation and structural determination of β-aminoacyl-containing cyclic hydrazine derivatives as dipeptidyl peptidase IV (DPP-IV) inhibitors", Bioorganic & Medicinal Chemistry Letters, 17 (9): 2622–2628, doi:10.1016/j.bmcl.2007.01.111, PMID17331715
Lu, I-Lin; Tsai, Keng-Chang; Chiang, Yi-Kun; Jiaang, Weir-Torn; Wu, Ssu-Hui; Mahindroo, Neeraj; Chien, Chia-Hui; Lee, Shiow-Ju; Chen, Xin; Wu, Su-Ying (January 2008), "A three-dimensional pharmacophore model for dipeptidyl peptidase IV inhibitors", European Journal of Medicinal Chemistry, 43 (8): 1603–1611, doi:10.1016/j.ejmech.2007.11.014, PMID18207285
Peters, Jens-Uwe (March 2007), "11 years of Cyanopyrrolidines as DPP-IV Inhibitors", Current Topics in Medicinal Chemistry, 7 (6): 579–595, doi:10.2174/156802607780091000, PMID17352679
Cox, Jason; Harper, Bart; Mastracchio, Anthony; Leiting, Barbara; Roy, Ranabir; Reshma, Patel; Wu, Joseph; Lyons, Kathryn; He, Huaibing; Edmondson, Scott (June 2007), "Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors", Bioorganic & Medicinal Chemistry, 17 (16): 4579–4583, doi:10.1016/j.bmcl.2007.05.087, PMID17562364
Idris, Iskandar; Donnely, Richard (January 2007), "Dipeptidyl peptidase-IV inhibitors: a major new class of oral antidiabetic drug", Diabetes, Obesity and Metabolism, 9 (2): 153–165, doi:10.1111/j.1463-1326.2007.00705.x, PMID17300591, S2CID3102605
Kuhn, Bernd; Hennig, Michael; Mattei, Patrizio (March 2007), "Molecular Recognition of Ligands in Dipeptidyl Peptidase IV", Current Topics in Medicinal Chemistry, 7 (6): 609–619, doi:10.2174/156802607780091064, PMID17352681
Veken, Pieter Van der; Haemers, Achiel; Augustyns, Koen (May 2007), "Prolyl peptidase related to dipeptidyl peptidase IV: Potential of specific inhibitors in drug discovery", Current Topics in Medicinal Chemistry, 7 (6): 621–635, doi:10.2174/156802607780091046, PMID17352682
Deng, Guanghui; Ye, Deju; Li, Yuanyuan; He, Lingyan; Zhou, Yu; Wang, Jiang; Li, Jia; Jiang, Hualiang; Liu, Hong (September 2008), "Synthesis of (S)-, (R)-, and (rac)-2-amino-3,3-bis(4-fluorophenyl)propanoic acids and an evaluation of the DPP-IV inhibitory activity of Denagliptin diastereomers", Tetrahedron, 64 (46): 10512–10516, doi:10.1016/j.tet.2008.08.097
Ferraris, Dana; Belyakov, Sergei; Li, Weixing; Oliver, Eddie; Ko, Yao-Sen; Calvin, David; Lautar, Susan; Thomas, Bert; Rojas, Camilo (March 2007), "Azetidine-Based Inhibitors of Dipeptidyl Peptidase IV (DPP IV)", Current Topics in Medicinal Chemistry, 7 (6): 597–608, doi:10.2174/156802607780090993, PMID17352680
Thornberry, Nancy A.; Weber, Ann E. (March 2007), "Discovery of JANUVIA (Sitagliptin), a Selective Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type2 Diabetes", Current Topics in Medicinal Chemistry, 7 (6): 557–568, doi:10.2174/156802607780091028, PMID17352677
Wright, Stephen; Ammirati, Mark; Andrews, Kim; Brodeur, Anne; Danley, Dennis; Doran, Shawn; Lillquist, Jay; Liu, Shenping; McClure, Lester; Cox, Eric (August 2007), "(3R,4S)-4-(2,4,5-Trifluorophenyl)-pyrrolidin-3-ylamine inhibitors of dipeptidyl peptidase IV: Synthesis, in vitro, in vivo, and X-ray crystallographic characterization", Bioorganic & Medicinal Chemistry Letters, 17 (20): 5638–5642, doi:10.1016/j.bmcl.2007.07.081, PMID17822893
Hulin, Bernard; Cabral, Shawn; Lopaze, Michael; VanVolkenburg, Maria; Andrews, Kim; Parker, Janice (August 2005), "New fluorinated pyrrolidine and azetidine amides as dipeptidyl peptidase IV inhibitors", Bioorganic & Medicinal Chemistry Letters, 15 (21): 4770–4773, doi:10.1016/j.bmcl.2005.07.026, PMID16115768
Szczepankiewicz, Bruce G.; Kurukulasuriya, Ravi (March 2007), "Aromatic Heterocycle-Based DPP-IV Inhibitors: Xanthines and Related Structural Types", Current Topics in Medicinal Chemistry, 7 (6): 569–578, doi:10.2174/156802607780091073, PMID17352678
Green, Brian; Flatt, Peter; Bailey, Clifford (December 2006), "Dipeptidyl peptidase IV (DPP IV) inhibitors: a newly emerging drug class for the treatment of type 2 diabetes", Diabetes and Vascular Disease Research, 3 (3): 159–165, doi:10.3132/dvdr.2006.024, PMID17160910
Sebokova, Elena; Christ, Andreas; Boehringer, Markus; Mizrahi, Jacques (May 2006), "Dipeptidyl peptidase IV inhibitors: The next generation of new promising therapies for the management of type 2 diabetes", Current Topics in Medicinal Chemistry, 7 (6): 547–555, doi:10.2174/156802607780091019, PMID17352676
Ahn, Jin Hee; Shin, Mi Sik; June, Mi Ae; Jung, Sun Ho; Kang, Seung Kyu; Kim, Kwang Rok; Rhee, Sang Dal; Kang, Nam Sook; Kim, Seung Kyu (February 2007), "Synthesis, biological evaluation and structural determination of β-aminoacyl-containing cyclic hydrazine derivatives as dipeptidyl peptidase IV (DPP-IV) inhibitors", Bioorganic & Medicinal Chemistry Letters, 17 (9): 2622–2628, doi:10.1016/j.bmcl.2007.01.111, PMID17331715
Lu, I-Lin; Tsai, Keng-Chang; Chiang, Yi-Kun; Jiaang, Weir-Torn; Wu, Ssu-Hui; Mahindroo, Neeraj; Chien, Chia-Hui; Lee, Shiow-Ju; Chen, Xin; Wu, Su-Ying (January 2008), "A three-dimensional pharmacophore model for dipeptidyl peptidase IV inhibitors", European Journal of Medicinal Chemistry, 43 (8): 1603–1611, doi:10.1016/j.ejmech.2007.11.014, PMID18207285
Peters, Jens-Uwe (March 2007), "11 years of Cyanopyrrolidines as DPP-IV Inhibitors", Current Topics in Medicinal Chemistry, 7 (6): 579–595, doi:10.2174/156802607780091000, PMID17352679
Cox, Jason; Harper, Bart; Mastracchio, Anthony; Leiting, Barbara; Roy, Ranabir; Reshma, Patel; Wu, Joseph; Lyons, Kathryn; He, Huaibing; Edmondson, Scott (June 2007), "Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors", Bioorganic & Medicinal Chemistry, 17 (16): 4579–4583, doi:10.1016/j.bmcl.2007.05.087, PMID17562364
Idris, Iskandar; Donnely, Richard (January 2007), "Dipeptidyl peptidase-IV inhibitors: a major new class of oral antidiabetic drug", Diabetes, Obesity and Metabolism, 9 (2): 153–165, doi:10.1111/j.1463-1326.2007.00705.x, PMID17300591, S2CID3102605
Kuhn, Bernd; Hennig, Michael; Mattei, Patrizio (March 2007), "Molecular Recognition of Ligands in Dipeptidyl Peptidase IV", Current Topics in Medicinal Chemistry, 7 (6): 609–619, doi:10.2174/156802607780091064, PMID17352681
Veken, Pieter Van der; Haemers, Achiel; Augustyns, Koen (May 2007), "Prolyl peptidase related to dipeptidyl peptidase IV: Potential of specific inhibitors in drug discovery", Current Topics in Medicinal Chemistry, 7 (6): 621–635, doi:10.2174/156802607780091046, PMID17352682
Ferraris, Dana; Belyakov, Sergei; Li, Weixing; Oliver, Eddie; Ko, Yao-Sen; Calvin, David; Lautar, Susan; Thomas, Bert; Rojas, Camilo (March 2007), "Azetidine-Based Inhibitors of Dipeptidyl Peptidase IV (DPP IV)", Current Topics in Medicinal Chemistry, 7 (6): 597–608, doi:10.2174/156802607780090993, PMID17352680
Thornberry, Nancy A.; Weber, Ann E. (March 2007), "Discovery of JANUVIA (Sitagliptin), a Selective Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type2 Diabetes", Current Topics in Medicinal Chemistry, 7 (6): 557–568, doi:10.2174/156802607780091028, PMID17352677
Wright, Stephen; Ammirati, Mark; Andrews, Kim; Brodeur, Anne; Danley, Dennis; Doran, Shawn; Lillquist, Jay; Liu, Shenping; McClure, Lester; Cox, Eric (August 2007), "(3R,4S)-4-(2,4,5-Trifluorophenyl)-pyrrolidin-3-ylamine inhibitors of dipeptidyl peptidase IV: Synthesis, in vitro, in vivo, and X-ray crystallographic characterization", Bioorganic & Medicinal Chemistry Letters, 17 (20): 5638–5642, doi:10.1016/j.bmcl.2007.07.081, PMID17822893
Hulin, Bernard; Cabral, Shawn; Lopaze, Michael; VanVolkenburg, Maria; Andrews, Kim; Parker, Janice (August 2005), "New fluorinated pyrrolidine and azetidine amides as dipeptidyl peptidase IV inhibitors", Bioorganic & Medicinal Chemistry Letters, 15 (21): 4770–4773, doi:10.1016/j.bmcl.2005.07.026, PMID16115768
Szczepankiewicz, Bruce G.; Kurukulasuriya, Ravi (March 2007), "Aromatic Heterocycle-Based DPP-IV Inhibitors: Xanthines and Related Structural Types", Current Topics in Medicinal Chemistry, 7 (6): 569–578, doi:10.2174/156802607780091073, PMID17352678
Idris, Iskandar; Donnely, Richard (January 2007), "Dipeptidyl peptidase-IV inhibitors: a major new class of oral antidiabetic drug", Diabetes, Obesity and Metabolism, 9 (2): 153–165, doi:10.1111/j.1463-1326.2007.00705.x, PMID17300591, S2CID3102605