Becker KL (2001). "Endometriosis". Principles and Practice of Endocrinology and Metabolism. Lippincott Williams & Wilkins. pp. 975–. ISBN978-0-7817-1750-2. Archived from the original on 2022-06-10. Retrieved 2018-07-26.
Lemke TL, Williams DA (24 January 2012). "Womens Health". Foye's Principles of Medicinal Chemistry. Lippincott Williams & Wilkins. pp. 1411–. ISBN978-1-60913-345-0. Archived from the original on 21 December 2016. Retrieved 24 October 2016.
Matsumoto AM, Bremmer WJ (1 January 2016). "Testicular Disorders". In Melmed S (ed.). Williams Textbook of Endocrinology. Elsevier Health Sciences. pp. 752–. ISBN978-0-323-29738-7. Archived from the original on 27 July 2020. Retrieved 26 July 2018.
McCartney CR, Marshall JC (13 September 2013). "Endocrinology of Reproduction". In Strauss III JF, Barbieri RL (eds.). Yen and Jaffe's Reproductive Endocrinology. Elsevier Health Sciences. pp. 19–. ISBN978-1-4557-2758-2. Archived from the original on 10 June 2022. Retrieved 26 July 2018.
Clemenza S, Sorbi F, Noci I, Capezzuoli T, Turrini I, Carriero C, Buffi N, Fambrini M, Petraglia F (February 2018). "From pathogenesis to clinical practice: Emerging medical treatments for endometriosis". Best Pract Res Clin Obstet Gynaecol. 51: 92–101. doi:10.1016/j.bpobgyn.2018.01.021. PMID29559388. S2CID3952054.
Chen C, Wu D, Guo Z, Xie Q, Reinhart GJ, Madan A, Wen J, Chen T, Huang CQ, Chen M, Chen Y, Tucci FC, Rowbottom M, Pontillo J, Zhu YF, Wade W, Saunders J, Bozigian H, Struthers RS (December 2008). "Discovery of sodium R-(+)-4-{2-[5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-[trifluoromethyl]benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2H-pyrimidin-1-yl]-1-phenylethylamino}}butyrate (elagolix), a potent and orally available nonpeptide antagonist of the human gonadotropin-releasing hormone receptor". J. Med. Chem. 51 (23): 7478–85. doi:10.1021/jm8006454. PMID19006286.
Tan O, Carr BR, Beshay VE, Bukulmez O (January 2013). "The extrapituitary effects of GnRH antagonists and their potential clinical implications: a narrated review". Reprod Sci. 20 (1): 16–25. doi:10.1177/1933719112459244. PMID23012318. S2CID21376889.
Tucci FC, Zhu YF, Struthers RS, Guo Z, Gross TD, Rowbottom MW, Acevedo O, Gao Y, Saunders J, Xie Q, Reinhart GJ, Liu XJ, Ling N, Bonneville AK, Chen T, Bozigian H, Chen C (February 2005). "3-[(2R)-Amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)- 6-methylpyrimidin-2,4-dione (NBI 42902) as a potent and orally active antagonist of the human gonadotropin-releasing hormone receptor. Design, synthesis, and in vitro and in vivo characterization". J. Med. Chem. 48 (4): 1169–78. doi:10.1021/jm049218c. PMID15715483.
Clemenza S, Sorbi F, Noci I, Capezzuoli T, Turrini I, Carriero C, Buffi N, Fambrini M, Petraglia F (February 2018). "From pathogenesis to clinical practice: Emerging medical treatments for endometriosis". Best Pract Res Clin Obstet Gynaecol. 51: 92–101. doi:10.1016/j.bpobgyn.2018.01.021. PMID29559388. S2CID3952054.
Chen C, Wu D, Guo Z, Xie Q, Reinhart GJ, Madan A, Wen J, Chen T, Huang CQ, Chen M, Chen Y, Tucci FC, Rowbottom M, Pontillo J, Zhu YF, Wade W, Saunders J, Bozigian H, Struthers RS (December 2008). "Discovery of sodium R-(+)-4-{2-[5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-[trifluoromethyl]benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2H-pyrimidin-1-yl]-1-phenylethylamino}}butyrate (elagolix), a potent and orally available nonpeptide antagonist of the human gonadotropin-releasing hormone receptor". J. Med. Chem. 51 (23): 7478–85. doi:10.1021/jm8006454. PMID19006286.
Tan O, Carr BR, Beshay VE, Bukulmez O (January 2013). "The extrapituitary effects of GnRH antagonists and their potential clinical implications: a narrated review". Reprod Sci. 20 (1): 16–25. doi:10.1177/1933719112459244. PMID23012318. S2CID21376889.
Tucci FC, Zhu YF, Struthers RS, Guo Z, Gross TD, Rowbottom MW, Acevedo O, Gao Y, Saunders J, Xie Q, Reinhart GJ, Liu XJ, Ling N, Bonneville AK, Chen T, Bozigian H, Chen C (February 2005). "3-[(2R)-Amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)- 6-methylpyrimidin-2,4-dione (NBI 42902) as a potent and orally active antagonist of the human gonadotropin-releasing hormone receptor. Design, synthesis, and in vitro and in vivo characterization". J. Med. Chem. 48 (4): 1169–78. doi:10.1021/jm049218c. PMID15715483.
US patent 7056927, Zhiqiang Guo, Yongsheng Chen, Dongpei Wu, Chen Chen, Warren Wade, Wesley J. Dwight, Charles Q. Huang, Fabio C. Tucci, "Gonadotropin-releasing hormone receptor antagonists and methods relating thereto", published 2006-06-06Archived 2020-11-27 at the Wayback Machine
Clemenza S, Sorbi F, Noci I, Capezzuoli T, Turrini I, Carriero C, Buffi N, Fambrini M, Petraglia F (February 2018). "From pathogenesis to clinical practice: Emerging medical treatments for endometriosis". Best Pract Res Clin Obstet Gynaecol. 51: 92–101. doi:10.1016/j.bpobgyn.2018.01.021. PMID29559388. S2CID3952054.
Tan O, Carr BR, Beshay VE, Bukulmez O (January 2013). "The extrapituitary effects of GnRH antagonists and their potential clinical implications: a narrated review". Reprod Sci. 20 (1): 16–25. doi:10.1177/1933719112459244. PMID23012318. S2CID21376889.
Diamond MP, Carr B, Dmowski WP, Koltun W, O'Brien C, Jiang P, Burke J, Jimenez R, Garner E, Chwalisz K (2014). "Elagolix treatment for endometriosis-associated pain: results from a phase 2, randomized, double-blind, placebo-controlled study". Reprod Sci. 21 (3): 363–71. doi:10.1177/1933719113497292. PMID23885105. S2CID9607500.
Becker KL (2001). "Endometriosis". Principles and Practice of Endocrinology and Metabolism. Lippincott Williams & Wilkins. pp. 975–. ISBN978-0-7817-1750-2. Archived from the original on 2022-06-10. Retrieved 2018-07-26.
Lemke TL, Williams DA (24 January 2012). "Womens Health". Foye's Principles of Medicinal Chemistry. Lippincott Williams & Wilkins. pp. 1411–. ISBN978-1-60913-345-0. Archived from the original on 21 December 2016. Retrieved 24 October 2016.
Matsumoto AM, Bremmer WJ (1 January 2016). "Testicular Disorders". In Melmed S (ed.). Williams Textbook of Endocrinology. Elsevier Health Sciences. pp. 752–. ISBN978-0-323-29738-7. Archived from the original on 27 July 2020. Retrieved 26 July 2018.
McCartney CR, Marshall JC (13 September 2013). "Endocrinology of Reproduction". In Strauss III JF, Barbieri RL (eds.). Yen and Jaffe's Reproductive Endocrinology. Elsevier Health Sciences. pp. 19–. ISBN978-1-4557-2758-2. Archived from the original on 10 June 2022. Retrieved 26 July 2018.
US patent 7056927, Zhiqiang Guo, Yongsheng Chen, Dongpei Wu, Chen Chen, Warren Wade, Wesley J. Dwight, Charles Q. Huang, Fabio C. Tucci, "Gonadotropin-releasing hormone receptor antagonists and methods relating thereto", published 2006-06-06Archived 2020-11-27 at the Wayback Machine