H3 receptor antagonist (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "H3 receptor antagonist" in English language version.

refsWebsite

Global rank English rank

19nih.gov

4^th place

15doi.org

2^nd place

5worldcat.org

5^th place

4semanticscholar.org

11^th place

8^th place

2web.archive.org

1^st place

1aspetjournals.org

6,663^rd place

5,792^nd place

1europa.eu

68^th place

117^th place

aspetjournals.org

jpet.aspetjournals.org

Ligneau X, Lin J, Vanni-Mercier G, Jouvet M, Muir JL, Ganellin CR, Stark H, Elz S, Schunack W, Schwartz J (November 1998). "Neurochemical and behavioral effects of ciproxifan, a potent histamine H₃-receptor antagonist". The Journal of Pharmacology and Experimental Therapeutics. 287 (2): 658–66. PMID 9808693. Archived from the original on 2020-05-02. Retrieved 2013-12-18.

doi.org

Yoneyama H, Shimoda A, Araki L, et al. (March 2008). "Efficient approaches to S-alkyl-N-alkylisothioureas: syntheses of histamine H3 antagonist clobenpropit and its analogues". The Journal of Organic Chemistry. 73 (6): 2096–104. doi:10.1021/jo702181x. PMID 18278935.
Fox GB, Esbenshade TA, Pan JB, Radek RJ, Krueger KM, Yao BB, Browman KE, Buckley MJ, Ballard ME, Komater VA, Miner H, Zhang M, Faghih R, Rueter LE, Bitner RS, Drescher KU, Wetter J, Marsh K, Lemaire M, Porsolt RD, Bennani YL, Sullivan JP, Cowart MD, Decker MW, Hancock AA (April 2005). "Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H₃ receptor antagonist". Journal of Pharmacology and Experimental Therapeutics. 313 (1): 176–90. doi:10.1124/jpet.104.078402. ISSN 1521-0103. PMID 15608077. S2CID 15430117.
Esbenshade TA, Fox GB, Krueger KM, Baranowski JL, Miller TR, Kang CH, Denny LI, Witte DG, Yao BB, Pan JB, Faghih R, Bennani YL, Williams M, Hancock AA (1 September 2004). "Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist". Biochemical Pharmacology. 68 (5): 933–45. doi:10.1016/j.bcp.2004.05.048. PMID 15294456.
Ligneau X, Perrin D, Landais L, Camelin JC, Calmels TP, Berrebi-Bertrand I, Lecomte JM, Parmentier R, Anaclet C, Lin JS, Bertaina-Anglade V, la Rochelle CD, d'Aniello F, Rouleau A, Gbahou F, Arrang JM, Ganellin CR, Stark H, Schunack W, Schwartz JC (January 2007). "BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology". Journal of Pharmacology and Experimental Therapeutics. 320 (1): 365–75. doi:10.1124/jpet.106.111039. PMID 17005916. S2CID 7489564.
Schwartz, Jean-Charles (2011-06-01). "The histamine H3 receptor: from discovery to clinical trials with pitolisant". British Journal of Pharmacology. 163 (4): 713–721. doi:10.1111/j.1476-5381.2011.01286.x. ISSN 1476-5381. PMC 3111674. PMID 21615387.
Sadek, Bassem; Saad, Ali; Sadeq, Adel; Jalal, Fakhreya; Stark, Holger (2016). "Histamine H3 receptor as a potential target for cognitive symptoms in neuropsychiatric diseases". Behavioural Brain Research. 312: 415–430. doi:10.1016/j.bbr.2016.06.051. PMID 27363923. S2CID 40024812.
Berlin, Michael; Boyce, Christopher W.; de Lera Ruiz, Manuel (2011-01-13). "Histamine H3 Receptor as a Drug Discovery Target". Journal of Medicinal Chemistry. 54 (1): 26–53. doi:10.1021/jm100064d. ISSN 0022-2623. PMID 21062081.
Wijtmans, Maikel; Leurs, Rob; Esch, Iwan de (2007-07-01). "Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas". Expert Opinion on Investigational Drugs. 16 (7): 967–985. doi:10.1517/13543784.16.7.967. ISSN 1354-3784. PMID 17594183. S2CID 21914430.
Celanire, Sylvain; Wijtmans, Maikel; Talaga, Patrice; Leurs, Rob; Esch, Iwan J.P. de (2005). "Keynote review: Histamine H3 receptor antagonists reach out for the clinic". Drug Discovery Today. 10 (23–24): 1613–1627. doi:10.1016/s1359-6446(05)03625-1. PMID 16376822.
Gemkow, Mark J.; Davenport, Adam J.; Harich, Silke; Ellenbroek, Bart A.; Cesura, Andrea; Hallett, David (2009). "The histamine H3 receptor as a therapeutic drug target for CNS disorders". Drug Discovery Today. 14 (9–10): 509–515. doi:10.1016/j.drudis.2009.02.011. PMID 19429511.
Ledneczki, Istvan; Tapolcsányi, Pál; Gábor, Eszter; Éles, János; Greiner, István; Schmidt, Éva; Némethy, Zsolt; Kedves, Rita Soukupné; Balázs, Ottilia (2017). "Discovery of novel steroidal histamine H 3 receptor antagonists/inverse agonists". Bioorganic & Medicinal Chemistry Letters. 27 (19): 4525–4530. doi:10.1016/j.bmcl.2017.08.060. PMID 28888822.
Masini, D.; Lopes-Aguiar, C.; Bonito-Oliva, A.; Papadia, D.; Andersson, R.; Fisahn, A.; Fisone, G. (2017-04-11). "The histamine H3 receptor antagonist thioperamide rescues circadian rhythm and memory function in experimental parkinsonism". Translational Psychiatry. 7 (4): e1088. doi:10.1038/tp.2017.58. PMC 5416699. PMID 28398338.
Kollb-Sielecka, Marta; Demolis, Pierre; Emmerich, Joseph; Markey, Greg; Salmonson, Tomas; Haas, Manuel (2017). "The European Medicines Agency review of pitolisant for treatment of narcolepsy: summary of the scientific assessment by the Committee for Medicinal Products for Human Use". Sleep Medicine. 33: 125–129. doi:10.1016/j.sleep.2017.01.002. PMID 28449891.
Vohora, Divya; Bhowmik, Malay (2012). "Histamine H3 receptor antagonists/inverse agonists on cognitive and motor processes: relevance to Alzheimer's disease, ADHD, schizophrenia, and drug abuse". Frontiers in Systems Neuroscience. 6: 72. doi:10.3389/fnsys.2012.00072. ISSN 1662-5137. PMC 3478588. PMID 23109919.
Scammell, Thomas E. (2015-12-30). "Narcolepsy". New England Journal of Medicine. 373 (27): 2654–2662. doi:10.1056/nejmra1500587. PMID 26716917.

europa.eu

ema.europa.eu

"European Medicines Agency - Find medicine - Wakix". www.ema.europa.eu. Archived from the original on 2017-09-27. Retrieved 2017-09-27.

nih.gov

pubmed.ncbi.nlm.nih.gov

Yoneyama H, Shimoda A, Araki L, et al. (March 2008). "Efficient approaches to S-alkyl-N-alkylisothioureas: syntheses of histamine H3 antagonist clobenpropit and its analogues". The Journal of Organic Chemistry. 73 (6): 2096–104. doi:10.1021/jo702181x. PMID 18278935.
Fox GB, Esbenshade TA, Pan JB, Radek RJ, Krueger KM, Yao BB, Browman KE, Buckley MJ, Ballard ME, Komater VA, Miner H, Zhang M, Faghih R, Rueter LE, Bitner RS, Drescher KU, Wetter J, Marsh K, Lemaire M, Porsolt RD, Bennani YL, Sullivan JP, Cowart MD, Decker MW, Hancock AA (April 2005). "Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H₃ receptor antagonist". Journal of Pharmacology and Experimental Therapeutics. 313 (1): 176–90. doi:10.1124/jpet.104.078402. ISSN 1521-0103. PMID 15608077. S2CID 15430117.
Ligneau X, Lin J, Vanni-Mercier G, Jouvet M, Muir JL, Ganellin CR, Stark H, Elz S, Schunack W, Schwartz J (November 1998). "Neurochemical and behavioral effects of ciproxifan, a potent histamine H₃-receptor antagonist". The Journal of Pharmacology and Experimental Therapeutics. 287 (2): 658–66. PMID 9808693. Archived from the original on 2020-05-02. Retrieved 2013-12-18.
Esbenshade TA, Fox GB, Krueger KM, Baranowski JL, Miller TR, Kang CH, Denny LI, Witte DG, Yao BB, Pan JB, Faghih R, Bennani YL, Williams M, Hancock AA (1 September 2004). "Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist". Biochemical Pharmacology. 68 (5): 933–45. doi:10.1016/j.bcp.2004.05.048. PMID 15294456.
Ligneau X, Perrin D, Landais L, Camelin JC, Calmels TP, Berrebi-Bertrand I, Lecomte JM, Parmentier R, Anaclet C, Lin JS, Bertaina-Anglade V, la Rochelle CD, d'Aniello F, Rouleau A, Gbahou F, Arrang JM, Ganellin CR, Stark H, Schunack W, Schwartz JC (January 2007). "BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology". Journal of Pharmacology and Experimental Therapeutics. 320 (1): 365–75. doi:10.1124/jpet.106.111039. PMID 17005916. S2CID 7489564.
Schwartz, Jean-Charles (2011-06-01). "The histamine H3 receptor: from discovery to clinical trials with pitolisant". British Journal of Pharmacology. 163 (4): 713–721. doi:10.1111/j.1476-5381.2011.01286.x. ISSN 1476-5381. PMC 3111674. PMID 21615387.
Sadek, Bassem; Saad, Ali; Sadeq, Adel; Jalal, Fakhreya; Stark, Holger (2016). "Histamine H3 receptor as a potential target for cognitive symptoms in neuropsychiatric diseases". Behavioural Brain Research. 312: 415–430. doi:10.1016/j.bbr.2016.06.051. PMID 27363923. S2CID 40024812.
Berlin, Michael; Boyce, Christopher W.; de Lera Ruiz, Manuel (2011-01-13). "Histamine H3 Receptor as a Drug Discovery Target". Journal of Medicinal Chemistry. 54 (1): 26–53. doi:10.1021/jm100064d. ISSN 0022-2623. PMID 21062081.
Wijtmans, Maikel; Leurs, Rob; Esch, Iwan de (2007-07-01). "Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas". Expert Opinion on Investigational Drugs. 16 (7): 967–985. doi:10.1517/13543784.16.7.967. ISSN 1354-3784. PMID 17594183. S2CID 21914430.
Celanire, Sylvain; Wijtmans, Maikel; Talaga, Patrice; Leurs, Rob; Esch, Iwan J.P. de (2005). "Keynote review: Histamine H3 receptor antagonists reach out for the clinic". Drug Discovery Today. 10 (23–24): 1613–1627. doi:10.1016/s1359-6446(05)03625-1. PMID 16376822.
Gemkow, Mark J.; Davenport, Adam J.; Harich, Silke; Ellenbroek, Bart A.; Cesura, Andrea; Hallett, David (2009). "The histamine H3 receptor as a therapeutic drug target for CNS disorders". Drug Discovery Today. 14 (9–10): 509–515. doi:10.1016/j.drudis.2009.02.011. PMID 19429511.
Ledneczki, Istvan; Tapolcsányi, Pál; Gábor, Eszter; Éles, János; Greiner, István; Schmidt, Éva; Némethy, Zsolt; Kedves, Rita Soukupné; Balázs, Ottilia (2017). "Discovery of novel steroidal histamine H 3 receptor antagonists/inverse agonists". Bioorganic & Medicinal Chemistry Letters. 27 (19): 4525–4530. doi:10.1016/j.bmcl.2017.08.060. PMID 28888822.
Masini, D.; Lopes-Aguiar, C.; Bonito-Oliva, A.; Papadia, D.; Andersson, R.; Fisahn, A.; Fisone, G. (2017-04-11). "The histamine H3 receptor antagonist thioperamide rescues circadian rhythm and memory function in experimental parkinsonism". Translational Psychiatry. 7 (4): e1088. doi:10.1038/tp.2017.58. PMC 5416699. PMID 28398338.
Kollb-Sielecka, Marta; Demolis, Pierre; Emmerich, Joseph; Markey, Greg; Salmonson, Tomas; Haas, Manuel (2017). "The European Medicines Agency review of pitolisant for treatment of narcolepsy: summary of the scientific assessment by the Committee for Medicinal Products for Human Use". Sleep Medicine. 33: 125–129. doi:10.1016/j.sleep.2017.01.002. PMID 28449891.
Vohora, Divya; Bhowmik, Malay (2012). "Histamine H3 receptor antagonists/inverse agonists on cognitive and motor processes: relevance to Alzheimer's disease, ADHD, schizophrenia, and drug abuse". Frontiers in Systems Neuroscience. 6: 72. doi:10.3389/fnsys.2012.00072. ISSN 1662-5137. PMC 3478588. PMID 23109919.
Scammell, Thomas E. (2015-12-30). "Narcolepsy". New England Journal of Medicine. 373 (27): 2654–2662. doi:10.1056/nejmra1500587. PMID 26716917.

ncbi.nlm.nih.gov

Schwartz, Jean-Charles (2011-06-01). "The histamine H3 receptor: from discovery to clinical trials with pitolisant". British Journal of Pharmacology. 163 (4): 713–721. doi:10.1111/j.1476-5381.2011.01286.x. ISSN 1476-5381. PMC 3111674. PMID 21615387.
Masini, D.; Lopes-Aguiar, C.; Bonito-Oliva, A.; Papadia, D.; Andersson, R.; Fisahn, A.; Fisone, G. (2017-04-11). "The histamine H3 receptor antagonist thioperamide rescues circadian rhythm and memory function in experimental parkinsonism". Translational Psychiatry. 7 (4): e1088. doi:10.1038/tp.2017.58. PMC 5416699. PMID 28398338.
Vohora, Divya; Bhowmik, Malay (2012). "Histamine H3 receptor antagonists/inverse agonists on cognitive and motor processes: relevance to Alzheimer's disease, ADHD, schizophrenia, and drug abuse". Frontiers in Systems Neuroscience. 6: 72. doi:10.3389/fnsys.2012.00072. ISSN 1662-5137. PMC 3478588. PMID 23109919.

semanticscholar.org

api.semanticscholar.org

Fox GB, Esbenshade TA, Pan JB, Radek RJ, Krueger KM, Yao BB, Browman KE, Buckley MJ, Ballard ME, Komater VA, Miner H, Zhang M, Faghih R, Rueter LE, Bitner RS, Drescher KU, Wetter J, Marsh K, Lemaire M, Porsolt RD, Bennani YL, Sullivan JP, Cowart MD, Decker MW, Hancock AA (April 2005). "Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H₃ receptor antagonist". Journal of Pharmacology and Experimental Therapeutics. 313 (1): 176–90. doi:10.1124/jpet.104.078402. ISSN 1521-0103. PMID 15608077. S2CID 15430117.
Ligneau X, Perrin D, Landais L, Camelin JC, Calmels TP, Berrebi-Bertrand I, Lecomte JM, Parmentier R, Anaclet C, Lin JS, Bertaina-Anglade V, la Rochelle CD, d'Aniello F, Rouleau A, Gbahou F, Arrang JM, Ganellin CR, Stark H, Schunack W, Schwartz JC (January 2007). "BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology". Journal of Pharmacology and Experimental Therapeutics. 320 (1): 365–75. doi:10.1124/jpet.106.111039. PMID 17005916. S2CID 7489564.
Sadek, Bassem; Saad, Ali; Sadeq, Adel; Jalal, Fakhreya; Stark, Holger (2016). "Histamine H3 receptor as a potential target for cognitive symptoms in neuropsychiatric diseases". Behavioural Brain Research. 312: 415–430. doi:10.1016/j.bbr.2016.06.051. PMID 27363923. S2CID 40024812.
Wijtmans, Maikel; Leurs, Rob; Esch, Iwan de (2007-07-01). "Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas". Expert Opinion on Investigational Drugs. 16 (7): 967–985. doi:10.1517/13543784.16.7.967. ISSN 1354-3784. PMID 17594183. S2CID 21914430.

web.archive.org

Ligneau X, Lin J, Vanni-Mercier G, Jouvet M, Muir JL, Ganellin CR, Stark H, Elz S, Schunack W, Schwartz J (November 1998). "Neurochemical and behavioral effects of ciproxifan, a potent histamine H₃-receptor antagonist". The Journal of Pharmacology and Experimental Therapeutics. 287 (2): 658–66. PMID 9808693. Archived from the original on 2020-05-02. Retrieved 2013-12-18.
"European Medicines Agency - Find medicine - Wakix". www.ema.europa.eu. Archived from the original on 2017-09-27. Retrieved 2017-09-27.

worldcat.org

search.worldcat.org

Fox GB, Esbenshade TA, Pan JB, Radek RJ, Krueger KM, Yao BB, Browman KE, Buckley MJ, Ballard ME, Komater VA, Miner H, Zhang M, Faghih R, Rueter LE, Bitner RS, Drescher KU, Wetter J, Marsh K, Lemaire M, Porsolt RD, Bennani YL, Sullivan JP, Cowart MD, Decker MW, Hancock AA (April 2005). "Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H₃ receptor antagonist". Journal of Pharmacology and Experimental Therapeutics. 313 (1): 176–90. doi:10.1124/jpet.104.078402. ISSN 1521-0103. PMID 15608077. S2CID 15430117.
Schwartz, Jean-Charles (2011-06-01). "The histamine H3 receptor: from discovery to clinical trials with pitolisant". British Journal of Pharmacology. 163 (4): 713–721. doi:10.1111/j.1476-5381.2011.01286.x. ISSN 1476-5381. PMC 3111674. PMID 21615387.
Berlin, Michael; Boyce, Christopher W.; de Lera Ruiz, Manuel (2011-01-13). "Histamine H3 Receptor as a Drug Discovery Target". Journal of Medicinal Chemistry. 54 (1): 26–53. doi:10.1021/jm100064d. ISSN 0022-2623. PMID 21062081.
Wijtmans, Maikel; Leurs, Rob; Esch, Iwan de (2007-07-01). "Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas". Expert Opinion on Investigational Drugs. 16 (7): 967–985. doi:10.1517/13543784.16.7.967. ISSN 1354-3784. PMID 17594183. S2CID 21914430.
Vohora, Divya; Bhowmik, Malay (2012). "Histamine H3 receptor antagonists/inverse agonists on cognitive and motor processes: relevance to Alzheimer's disease, ADHD, schizophrenia, and drug abuse". Frontiers in Systems Neuroscience. 6: 72. doi:10.3389/fnsys.2012.00072. ISSN 1662-5137. PMC 3478588. PMID 23109919.