Larock, R. C.; Yum, E. K. (1991). "Synthesis of indoles via palladium-catalyzed heteroannulation of internal alkynes". Journal of the American Chemical Society. 113 (17): 6689. doi:10.1021/ja00017a059.
Larock, R. C.; Yum, E. K.; Refvik, M. D. (1998). "Synthesis of 2,3-Disubstituted Indoles via Palladium-Catalyzed Annulation of Internal Alkynes". The Journal of Organic Chemistry. 63 (22): 7652. doi:10.1021/jo9803277.
Monguchi, Y.; Mori, S.; Aoyagi, S.; Tsutsui, A.; Maegawa, T.; Sajiki, H. (2010). "Palladium on carbon-catalyzed synthesis of 2- and 2,3-substituted indoles under heterogeneous conditions". Organic & Biomolecular Chemistry. 8 (14): 3338–42. doi:10.1039/c004939e. PMID20526486.
Nishikawa, T.; Wada, K.; Isobe, M. (2002). "Synthesis of Novel .ALPHA.-C-Glycosylamino Acids and Reverse Regioselectivity in Larock's Heteroannulation for the Synthesis of the Indole Nucleus". Bioscience, Biotechnology, and Biochemistry. 66 (10): 2273–8. doi:10.1271/bbb.66.2273. PMID12450149.
Ma, C.; Liu, X.; Yu, S.; Zhao, S.; Cook, J. M. (1999). "Concise synthesis of optically active ring-A substituted tryptophans". Tetrahedron Letters. 40 (4): 657. doi:10.1016/S0040-4039(98)02497-6.
Chen, C.-Y, Lieberman, D.R., Larsen, R.D., Reamer, R.A., Verhoeven, T.R., Reider, P.J., Cottrell, I.F., Houghton, P.G. (1994). "Synthesis of the 5-HT1D agonist MK-0462 via a Pd-catalyzed coupling reaction". Tetrahedron Lett.35: 6981–6984. doi:10.1016/0040-4039(94)88204-5.{{cite journal}}: CS1 maint: multiple names: authors list (link)
nih.gov
pubmed.ncbi.nlm.nih.gov
Monguchi, Y.; Mori, S.; Aoyagi, S.; Tsutsui, A.; Maegawa, T.; Sajiki, H. (2010). "Palladium on carbon-catalyzed synthesis of 2- and 2,3-substituted indoles under heterogeneous conditions". Organic & Biomolecular Chemistry. 8 (14): 3338–42. doi:10.1039/c004939e. PMID20526486.
Nishikawa, T.; Wada, K.; Isobe, M. (2002). "Synthesis of Novel .ALPHA.-C-Glycosylamino Acids and Reverse Regioselectivity in Larock's Heteroannulation for the Synthesis of the Indole Nucleus". Bioscience, Biotechnology, and Biochemistry. 66 (10): 2273–8. doi:10.1271/bbb.66.2273. PMID12450149.
patents.google.com
Li, G., Liu, J., Lu, B., Roschangar, F., Senanayake, C.H., Shen, M. (2005) "By reacting with substituted acetylenes in the presence of a phosphine ligand and a base (K2CO3); used to make drugs" U.S. patent 20,050,209,465