Lipinski's rule of five (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "Lipinski's rule of five" in English language version.

refsWebsite

Global rank English rank

14nih.gov

4^th place

12doi.org

2^nd place

1semanticscholar.org

11^th place

8^th place

1harvard.edu

18^th place

17^th place

1psu.edu

207^th place

136^th place

doi.org

Lipinski CA, Lombardo F, Dominy BW, Feeney PJ (January 1997). "Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings". Advanced Drug Delivery Reviews. 46 (1–3): 3–26. doi:10.1016/S0169-409X(00)00129-0. PMID 11259830.
Lipinski CA (December 2004). "Lead- and drug-like compounds: the rule-of-five revolution". Drug Discovery Today: Technologies. 1 (4): 337–341. doi:10.1016/j.ddtec.2004.11.007. PMID 24981612.
Oprea TI, Davis AM, Teague SJ, Leeson PD (2001). "Is there a difference between leads and drugs? A historical perspective". Journal of Chemical Information and Computer Sciences. 41 (5): 1308–1315. doi:10.1021/ci010366a. PMID 11604031.
Leeson PD, Springthorpe B (November 2007). "The influence of drug-like concepts on decision-making in medicinal chemistry". Nature Reviews. Drug Discovery. 6 (11): 881–890. doi:10.1038/nrd2445. PMID 17971784. S2CID 205476574.
O Hagan S, Swainston N, Handl J, Kell DB (2015). "A 'rule of 0.5' for the metabolite-likeness of approved pharmaceutical drugs". Metabolomics. 11 (2): 323–339. doi:10.1007/s11306-014-0733-z. PMC 4342520. PMID 25750602.
Doak BC, Over B, Giordanetto F, Kihlberg J (September 2014). "Oral druggable space beyond the rule of 5: insights from drugs and clinical candidates". Chemistry & Biology. 21 (9): 1115–1142. doi:10.1016/j.chembiol.2014.08.013. PMID 25237858.
de Oliveira EC, Santana K, Josino L, Lima E, Lima AH, de Souza de Sales Júnior C (April 2021). "Predicting cell-penetrating peptides using machine learning algorithms and navigating in their chemical space". Scientific Reports. 11 (1): 7628. Bibcode:2021NatSR..11.7628D. doi:10.1038/s41598-021-87134-w. PMC 8027643. PMID 33828175.
Doak BC, Kihlberg J (February 2017). "Drug discovery beyond the rule of 5 - Opportunities and challenges". Expert Opinion on Drug Discovery. 12 (2): 115–119. doi:10.1080/17460441.2017.1264385. PMID 27883294.
Lipinski CA, Lombardo F, Dominy BW, Feeney PJ (March 2001). "Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings". Advanced Drug Delivery Reviews. 46 (1–3): 3–26. doi:10.1016/S0169-409X(00)00129-0. PMID 11259830.
Ghose AK, Viswanadhan VN, Wendoloski JJ (January 1999). "A knowledge-based approach in designing combinatorial or medicinal chemistry libraries for drug discovery. 1. A qualitative and quantitative characterization of known drug databases". Journal of Combinatorial Chemistry. 1 (1): 55–68. doi:10.1021/cc9800071. PMID 10746014.
Veber DF, Johnson SR, Cheng HY, Smith BR, Ward KW, Kopple KD (June 2002). "Molecular properties that influence the oral bioavailability of drug candidates". Journal of Medicinal Chemistry. 45 (12): 2615–2623. CiteSeerX 10.1.1.606.5270. doi:10.1021/jm020017n. PMID 12036371.
Congreve M, Carr R, Murray C, Jhoti H (October 2003). "A 'rule of three' for fragment-based lead discovery?". Drug Discovery Today. 8 (19): 876–877. doi:10.1016/S1359-6446(03)02831-9. PMID 14554012.

harvard.edu

ui.adsabs.harvard.edu

de Oliveira EC, Santana K, Josino L, Lima E, Lima AH, de Souza de Sales Júnior C (April 2021). "Predicting cell-penetrating peptides using machine learning algorithms and navigating in their chemical space". Scientific Reports. 11 (1): 7628. Bibcode:2021NatSR..11.7628D. doi:10.1038/s41598-021-87134-w. PMC 8027643. PMID 33828175.

nih.gov

pubmed.ncbi.nlm.nih.gov

Lipinski CA, Lombardo F, Dominy BW, Feeney PJ (January 1997). "Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings". Advanced Drug Delivery Reviews. 46 (1–3): 3–26. doi:10.1016/S0169-409X(00)00129-0. PMID 11259830.
Lipinski CA (December 2004). "Lead- and drug-like compounds: the rule-of-five revolution". Drug Discovery Today: Technologies. 1 (4): 337–341. doi:10.1016/j.ddtec.2004.11.007. PMID 24981612.
Oprea TI, Davis AM, Teague SJ, Leeson PD (2001). "Is there a difference between leads and drugs? A historical perspective". Journal of Chemical Information and Computer Sciences. 41 (5): 1308–1315. doi:10.1021/ci010366a. PMID 11604031.
Leeson PD, Springthorpe B (November 2007). "The influence of drug-like concepts on decision-making in medicinal chemistry". Nature Reviews. Drug Discovery. 6 (11): 881–890. doi:10.1038/nrd2445. PMID 17971784. S2CID 205476574.
O Hagan S, Swainston N, Handl J, Kell DB (2015). "A 'rule of 0.5' for the metabolite-likeness of approved pharmaceutical drugs". Metabolomics. 11 (2): 323–339. doi:10.1007/s11306-014-0733-z. PMC 4342520. PMID 25750602.
Doak BC, Over B, Giordanetto F, Kihlberg J (September 2014). "Oral druggable space beyond the rule of 5: insights from drugs and clinical candidates". Chemistry & Biology. 21 (9): 1115–1142. doi:10.1016/j.chembiol.2014.08.013. PMID 25237858.
de Oliveira EC, Santana K, Josino L, Lima E, Lima AH, de Souza de Sales Júnior C (April 2021). "Predicting cell-penetrating peptides using machine learning algorithms and navigating in their chemical space". Scientific Reports. 11 (1): 7628. Bibcode:2021NatSR..11.7628D. doi:10.1038/s41598-021-87134-w. PMC 8027643. PMID 33828175.
Doak BC, Kihlberg J (February 2017). "Drug discovery beyond the rule of 5 - Opportunities and challenges". Expert Opinion on Drug Discovery. 12 (2): 115–119. doi:10.1080/17460441.2017.1264385. PMID 27883294.
Lipinski CA, Lombardo F, Dominy BW, Feeney PJ (March 2001). "Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings". Advanced Drug Delivery Reviews. 46 (1–3): 3–26. doi:10.1016/S0169-409X(00)00129-0. PMID 11259830.
Ghose AK, Viswanadhan VN, Wendoloski JJ (January 1999). "A knowledge-based approach in designing combinatorial or medicinal chemistry libraries for drug discovery. 1. A qualitative and quantitative characterization of known drug databases". Journal of Combinatorial Chemistry. 1 (1): 55–68. doi:10.1021/cc9800071. PMID 10746014.
Veber DF, Johnson SR, Cheng HY, Smith BR, Ward KW, Kopple KD (June 2002). "Molecular properties that influence the oral bioavailability of drug candidates". Journal of Medicinal Chemistry. 45 (12): 2615–2623. CiteSeerX 10.1.1.606.5270. doi:10.1021/jm020017n. PMID 12036371.
Congreve M, Carr R, Murray C, Jhoti H (October 2003). "A 'rule of three' for fragment-based lead discovery?". Drug Discovery Today. 8 (19): 876–877. doi:10.1016/S1359-6446(03)02831-9. PMID 14554012.

ncbi.nlm.nih.gov

O Hagan S, Swainston N, Handl J, Kell DB (2015). "A 'rule of 0.5' for the metabolite-likeness of approved pharmaceutical drugs". Metabolomics. 11 (2): 323–339. doi:10.1007/s11306-014-0733-z. PMC 4342520. PMID 25750602.
de Oliveira EC, Santana K, Josino L, Lima E, Lima AH, de Souza de Sales Júnior C (April 2021). "Predicting cell-penetrating peptides using machine learning algorithms and navigating in their chemical space". Scientific Reports. 11 (1): 7628. Bibcode:2021NatSR..11.7628D. doi:10.1038/s41598-021-87134-w. PMC 8027643. PMID 33828175.

psu.edu

citeseerx.ist.psu.edu

Veber DF, Johnson SR, Cheng HY, Smith BR, Ward KW, Kopple KD (June 2002). "Molecular properties that influence the oral bioavailability of drug candidates". Journal of Medicinal Chemistry. 45 (12): 2615–2623. CiteSeerX 10.1.1.606.5270. doi:10.1021/jm020017n. PMID 12036371.

semanticscholar.org

api.semanticscholar.org

Leeson PD, Springthorpe B (November 2007). "The influence of drug-like concepts on decision-making in medicinal chemistry". Nature Reviews. Drug Discovery. 6 (11): 881–890. doi:10.1038/nrd2445. PMID 17971784. S2CID 205476574.