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Metribolone (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "Metribolone" in English language version.

refsWebsite
Global rank English rank
9doi.org
2nd place
2nd place
8nih.gov
4th place
4th place
4books.google.com
3rd place
3rd place
1semanticscholar.org
11th place
8th place
1psu.edu
207th place
136th place
1usatoday.com
41st place
34th place

books.google.com

  • Elks J (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. pp. 654–. ISBN 978-1-4757-2085-3.
  • William Llewellyn's Anabolics. Molecular Nutrition LLC. 2011. pp. 546–. ISBN 978-0-9828280-1-4.
  • Phillipps GH (22 October 2013). "Structure-Activity Relationships in Steroid Anaesthetics". In James VJ, Pasqualini JR (eds.). Proceedings of the Fourth International Congress on Hormonal Steroids: Mexico City, September 1974. Elsevier Science. p. 618. ISBN 978-1-4831-4566-2. R-2956 [41-43], a dimethyl derivative of an extremely potent androgen, R 1881 [44], is a powerful testosterone antagonist with very low androgenic activity.
  • Harms AF (1 January 1986). Innovative Approaches in Drug Research: Proceedings of the Third Noordwijkerhout Symposium on Medicinal Chemistry, Held in the Netherlands, September 3-6, 1985. Elsevier. ISBN 978-0-444-42606-2. At this stage, RU 2956 exerts a competitive effect about 4 times less marked than metribolone may be because the steric hindrance of the dimethyl group in position C-2 interferes with H-bond formation between the C-3 oxygen and the receptor protein, i.e., with the recognition step, and consequently, with the association rate.

doi.org

  • Brinkmann AO, Kuiper GG, de Boer W, Mulder E, Bolt J, van Steenbrugge GJ, van der Molen HJ (January 1986). "Characterization of androgen receptors after photoaffinity labelling with [3H]methyltrienolone (R1881)". Journal of Steroid Biochemistry. 24 (1): 245–249. doi:10.1016/0022-4731(86)90058-0. PMID 2422446.
  • Brueggemeier RW (2006). "Sex Hormones (Male): Analogs and Antagonists". In Meyers RA (ed.). Encyclopedia of Molecular Cell Biology and Molecular Medicine. Vol. 13 (2nd ed.). doi:10.1002/3527600906.mcb.200500066. ISBN 3527600906.
  • Singh SM, Gauthier S, Labrie F (February 2000). "Androgen receptor antagonists (antiandrogens): structure-activity relationships". Current Medicinal Chemistry. 7 (2): 211–247. doi:10.2174/0929867003375371. PMID 10637363.
  • Ho-Kim MA, Tremblay RR, Dubé JY (November 1981). "Binding of methyltrienolone to glucocorticoid receptors in rat muscle cytosol". Endocrinology. 109 (5): 1418–1423. doi:10.1210/endo-109-5-1418. PMID 6975208.
  • Takeda AN, Pinon GM, Bens M, Fagart J, Rafestin-Oblin ME, Vandewalle A (February 2007). "The synthetic androgen methyltrienolone (r1881) acts as a potent antagonist of the mineralocorticoid receptor". Molecular Pharmacology. 71 (2): 473–482. doi:10.1124/mol.106.031112. PMID 17105867. S2CID 28647372.
  • Krüskemper HL, Noell G (July 1966). "Liver toxicity of a new anabolic agent: methyltrienolone (17-alpha-methyl-4,9,11-estratriene-17 beta-ol-3-one)". Steroids. 8 (1): 13–24. doi:10.1016/0039-128x(66)90114-0. PMID 5955468.
  • Delettré J, Mornon JP, Lepicard G, Ojasoo T, Raynaud JP (January 1980). "Steroid flexibility and receptor specificity". Journal of Steroid Biochemistry. 13 (1): 45–59. doi:10.1016/0022-4731(80)90112-0. PMID 7382482.
  • Ojasoo T, Delettré J, Mornon JP, Turpin-VanDycke C, Raynaud JP (1987). "Towards the mapping of the progesterone and androgen receptors". Journal of Steroid Biochemistry. 27 (1–3): 255–269. doi:10.1016/0022-4731(87)90317-7. PMID 3695484.
  • Saartok T, Dahlberg E, Gustafsson JA (June 1984). "Relative binding affinity of anabolic-androgenic steroids: comparison of the binding to the androgen receptors in skeletal muscle and in prostate, as well as to sex hormone-binding globulin". Endocrinology. 114 (6): 2100–2106. doi:10.1210/endo-114-6-2100. PMID 6539197.

nih.gov

pubmed.ncbi.nlm.nih.gov

  • Brinkmann AO, Kuiper GG, de Boer W, Mulder E, Bolt J, van Steenbrugge GJ, van der Molen HJ (January 1986). "Characterization of androgen receptors after photoaffinity labelling with [3H]methyltrienolone (R1881)". Journal of Steroid Biochemistry. 24 (1): 245–249. doi:10.1016/0022-4731(86)90058-0. PMID 2422446.
  • Singh SM, Gauthier S, Labrie F (February 2000). "Androgen receptor antagonists (antiandrogens): structure-activity relationships". Current Medicinal Chemistry. 7 (2): 211–247. doi:10.2174/0929867003375371. PMID 10637363.
  • Ho-Kim MA, Tremblay RR, Dubé JY (November 1981). "Binding of methyltrienolone to glucocorticoid receptors in rat muscle cytosol". Endocrinology. 109 (5): 1418–1423. doi:10.1210/endo-109-5-1418. PMID 6975208.
  • Takeda AN, Pinon GM, Bens M, Fagart J, Rafestin-Oblin ME, Vandewalle A (February 2007). "The synthetic androgen methyltrienolone (r1881) acts as a potent antagonist of the mineralocorticoid receptor". Molecular Pharmacology. 71 (2): 473–482. doi:10.1124/mol.106.031112. PMID 17105867. S2CID 28647372.
  • Krüskemper HL, Noell G (July 1966). "Liver toxicity of a new anabolic agent: methyltrienolone (17-alpha-methyl-4,9,11-estratriene-17 beta-ol-3-one)". Steroids. 8 (1): 13–24. doi:10.1016/0039-128x(66)90114-0. PMID 5955468.
  • Delettré J, Mornon JP, Lepicard G, Ojasoo T, Raynaud JP (January 1980). "Steroid flexibility and receptor specificity". Journal of Steroid Biochemistry. 13 (1): 45–59. doi:10.1016/0022-4731(80)90112-0. PMID 7382482.
  • Ojasoo T, Delettré J, Mornon JP, Turpin-VanDycke C, Raynaud JP (1987). "Towards the mapping of the progesterone and androgen receptors". Journal of Steroid Biochemistry. 27 (1–3): 255–269. doi:10.1016/0022-4731(87)90317-7. PMID 3695484.
  • Saartok T, Dahlberg E, Gustafsson JA (June 1984). "Relative binding affinity of anabolic-androgenic steroids: comparison of the binding to the androgen receptors in skeletal muscle and in prostate, as well as to sex hormone-binding globulin". Endocrinology. 114 (6): 2100–2106. doi:10.1210/endo-114-6-2100. PMID 6539197.

psu.edu

citeseerx.ist.psu.edu

  • Zheng F (2010). "Methyltrienolone (R1881) is a Potent Inhibitor of 3B-Hydroxysteroid Dehydrogenase (3B-HSD) Activity". Characterization of Enzymes Involved in the Metabolism of Dihydrotestosterone, the Most Potent Natural Androgen (thesis). pp. 91–103. CiteSeerX 10.1.1.428.3729.

semanticscholar.org

api.semanticscholar.org

  • Takeda AN, Pinon GM, Bens M, Fagart J, Rafestin-Oblin ME, Vandewalle A (February 2007). "The synthetic androgen methyltrienolone (r1881) acts as a potent antagonist of the mineralocorticoid receptor". Molecular Pharmacology. 71 (2): 473–482. doi:10.1124/mol.106.031112. PMID 17105867. S2CID 28647372.

usatoday.com