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Faucher, A-M.; Bailey, M. D.; Beaulieu, P. L.; Brochu, C.; Duceppe, J-S.; Ferland, J-M.; Ghiro, E.; Gorys, V.; Halmos, T.; Kawai, S. H.; Poirier, M.; Simoneau, B.; Tsantrizos, Y. S.; Llinas-Brunet, M. (2004). "Synthesis of BILN 2061, an HCV NS3 protease inhibitor with proven antiviral effect in humans". Org. Lett. 6 (17): 2901–2904. doi:10.1021/ol0489907. PMID15330643.
Yee, N. K.; Farina, V.; Houpis, I. N.; Haddad, N.; Frutos, R. P.; Gallou, F.; Wang, X-J.; Wei, X.; Simpson, R. D.; Feng, X.; Fuchs, V.; Xu, Y.; Tan, J.; Zhang, L.; Xu, J.; Smith-Keenan, L. L.; Vitous, J.; Ridges, M. D.; Spinelli, E. M.; Johnson, M. (2006). "Efficient large-scale synthesis of BILN 2061, a potent HCV protease inhibitor, by a convergent approach based on ring-closing metathesis". J. Org. Chem. 71 (19): 7133–7145. doi:10.1021/jo060285j. PMID16958506.
Zeng, X.; Wei, X.; Farina, V.; Napolitano, E.; Xu, Y.; Zhang, L.; Haddad, N.; Yee, N. K.; Grinberg, N.; Shen, S.; Senanayake, C. H. (2006). "Epimerization reaction of a substituted vinylcyclopropane catalyzed by ruthenium carbenes: mechanistic analysis". J. Org. Chem. 71 (23): 8864–8875. doi:10.1021/jo061587o. PMID17081017.
Wei, X.; Shu, C.; Haddad, N.; Zeng, X.; Patel, N. D.; Tan, Z.; Liu, J.; Lee, H.; Shen, S.; Campbell, S.; Varsolona, R. J.; Busacca, C. A.; Hossain, A.; Yee, N. K.; Senanayake, C. H. (2013). "A highly convergent and efficient synthesis of a macrocyclic hepatitis C virus protease inhibitor BI 201302". Org. Lett. 15 (5): 1016–1019. doi:10.1021/ol303498m. PMID23406520.
Desai, A. A. (2011). "Sitagliptin manufacture: a compelling tale of green chemistry, process intensification, and industrial asymmetric catalysis". Angew. Chem. Int. Ed. 50 (9): 1974–1976. doi:10.1002/anie.201007051. PMID21284073.