References analysis of the Wikipedia article "Receptor antagonist" in the English version

books.google.com

eds, David E. Golan, ed.-in-chief; Armen H. Tashjian Jr., deputy ed.; Ehrin J. Armstrong, April W. Armstrong, associate (2008). Principles of pharmacology: the pathophysiologic basis of drug therapy (2nd ed.). Philadelphia, Pa., [etc.]: Lippincott Williams & Wilkins. p. 25. ISBN 978-0-7817-8355-2. Retrieved 2012-02-05.{{cite book}}: CS1 maint: multiple names: authors list (link)

doi.org

Hopkins AL, Groom CR (September 2002). "The druggable genome". Nature Reviews. Drug Discovery. 1 (9): 727–30. doi:10.1038/nrd892. PMID 12209152. S2CID 13166282.

May LT, Avlani VA, Sexton PM, Christopoulos A (2004). "Allosteric modulation of G protein-coupled receptors". Current Pharmaceutical Design. 10 (17): 2003–13. doi:10.2174/1381612043384303. PMID 15279541. S2CID 36602982.

Christopoulos A (March 2002). "Allosteric binding sites on cell-surface receptors: novel targets for drug discovery". Nature Reviews. Drug Discovery. 1 (3): 198–210. doi:10.1038/nrd746. PMID 12120504. S2CID 13230838.

Bleicher KH, Green LG, Martin RE, Rogers-Evans M (June 2004). "Ligand identification for G-protein-coupled receptors: a lead generation perspective". Current Opinion in Chemical Biology. 8 (3): 287–96. doi:10.1016/j.cbpa.2004.04.008. PMID 15183327.

Rees S, Morrow D, Kenakin T (2002). "GPCR drug discovery through the exploitation of allosteric drug binding sites". Receptors & Channels. 8 (5–6): 261–8. doi:10.1080/10606820214640. PMID 12690954.

Negus SS (June 2006). "Some implications of receptor theory for in vivo assessment of agonists, antagonists and inverse agonists". Biochemical Pharmacology. 71 (12): 1663–70. doi:10.1016/j.bcp.2005.12.038. PMC 1866283. PMID 16460689.

Stephenson RP (February 1997). "A modification of receptor theory. 1956". British Journal of Pharmacology. 120 (4 Suppl): 106–20, discussion 103–5. doi:10.1111/j.1476-5381.1997.tb06784.x. PMC 3224279. PMID 9142399. of the original article.

Vauquelin G, Van Liefde I (February 2005). "G protein-coupled receptors: a count of 1001 conformations". Fundamental & Clinical Pharmacology. 19 (1): 45–56. doi:10.1111/j.1472-8206.2005.00319.x. PMID 15660959. S2CID 609867.

Urban JD, Clarke WP, von Zastrow M, Nichols DE, Kobilka B, Weinstein H, Javitch JA, Roth BL, Christopoulos A, Sexton PM, Miller KJ, Spedding M, Mailman RB (January 2007). "Functional selectivity and classical concepts of quantitative pharmacology". The Journal of Pharmacology and Experimental Therapeutics. 320 (1): 1–13. doi:10.1124/jpet.106.104463. PMID 16803859. S2CID 447937.

Lees P, Cunningham FM, Elliott J (December 2004). "Principles of pharmacodynamics and their applications in veterinary pharmacology". Journal of Veterinary Pharmacology and Therapeutics. 27 (6): 397–414. doi:10.1111/j.1365-2885.2004.00620.x. PMID 15601436.

Swinney DC (September 2004). "Biochemical mechanisms of drug action: what does it take for success?". Nature Reviews. Drug Discovery. 3 (9): 801–8. doi:10.1038/nrd1500. PMID 15340390. S2CID 28668800.

Wyllie DJ, Chen PE (March 2007). "Taking the time to study competitive antagonism". British Journal of Pharmacology. 150 (5): 541–51. doi:10.1038/sj.bjp.0706997. PMC 2189774. PMID 17245371.

Colquhoun D (December 2007). "Why the Schild method is better than Schild realised". Trends in Pharmacological Sciences. 28 (12): 608–14. doi:10.1016/j.tips.2007.09.011. PMID 18023486.

Schild HO (February 1975). "An ambiguity in receptor theory". British Journal of Pharmacology. 53 (2): 311. doi:10.1111/j.1476-5381.1975.tb07365.x. PMC 1666289. PMID 1148491.

Cheng Y, Prusoff WH (December 1973). "Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction". Biochemical Pharmacology. 22 (23): 3099–108. doi:10.1016/0006-2952(73)90196-2. PMID 4202581.

Neubig RR, Spedding M, Kenakin T, Christopoulos A (December 2003). "International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on terms and symbols in quantitative pharmacology" (PDF). Pharmacological Reviews. 55 (4): 597–606. doi:10.1124/pr.55.4.4. PMID 14657418. S2CID 1729572.

Vauquelin G, Van Liefde I, Birzbier BB, Vanderheyden PM (August 2002). "New insights in insurmountable antagonism". Fundamental & Clinical Pharmacology. 16 (4): 263–72. doi:10.1046/j.1472-8206.2002.00095.x. PMID 12570014. S2CID 6145796.

Surin A, Pshenichkin S, Grajkowska E, Surina E, Wroblewski JT (March 2007). "Cyclothiazide selectively inhibits mGluR1 receptors interacting with a common allosteric site for non-competitive antagonists". Neuropharmacology. 52 (3): 744–54. doi:10.1016/j.neuropharm.2006.09.018. PMC 1876747. PMID 17095021.

Lipton SA (January 2004). "Failures and successes of NMDA receptor antagonists: molecular basis for the use of open-channel blockers like memantine in the treatment of acute and chronic neurologic insults". NeuroRx. 1 (1): 101–10. doi:10.1602/neurorx.1.1.101. PMC 534915. PMID 15717010.

Parsons CG, Stöffler A, Danysz W (November 2007). "Memantine: a NMDA receptor antagonist that improves memory by restoration of homeostasis in the glutamatergic system—too little activation is bad, too much is even worse". Neuropharmacology. 53 (6): 699–723. doi:10.1016/j.neuropharm.2007.07.013. PMID 17904591. S2CID 6599658.

Fletcher A, Cliffe IA, Dourish CT (December 1993). "Silent 5-HT1A receptor antagonists: utility as research tools and therapeutic agents". Trends in Pharmacological Sciences. 14 (12): 41–48. doi:10.1016/0165-6147(93)90185-m. PMID 8122313. S2CID 4274320.

Patil PN (2002). "Everhardus J. Ariëns (1918–2002): a tribute". Trends in Pharmacological Sciences. 23 (7): 344–5. doi:10.1016/S0165-6147(02)02068-0.

Bosier B, Hermans E (August 2007). "Versatility of GPCR recognition by drugs: from biological implications to therapeutic relevance". Trends in Pharmacological Sciences. 28 (8): 438–46. doi:10.1016/j.tips.2007.06.001. PMID 17629964.

Pulvirenti L, Koob GF (April 2002). "Being partial to psychostimulant addiction therapy". Trends in Pharmacological Sciences. 23 (4): 151–3. doi:10.1016/S0165-6147(00)01991-X. PMID 11931978.

Vadivelu N, Hines RL (2007). "Buprenorphine: a unique opioid with broad clinical applications". Journal of Opioid Management. 3 (1): 49–58. doi:10.5055/jom.2007.0038. PMID 17367094.

Greasley PJ, Clapham JC (December 2006). "Inverse agonism or neutral antagonism at G-protein coupled receptors: a medicinal chemistry challenge worth pursuing?". European Journal of Pharmacology. 553 (1–3): 1–9. doi:10.1016/j.ejphar.2006.09.032. PMID 17081515.

Kenakin T (January 2004). "Efficacy as a vector: the relative prevalence and paucity of inverse agonism". Molecular Pharmacology. 65 (1): 2–11. doi:10.1124/mol.65.1.2. PMID 14722230. S2CID 115140.

Leurs R, Church MK, Taglialatela M (April 2002). "H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects". Clinical and Experimental Allergy. 32 (4): 489–98. doi:10.1046/j.0954-7894.2002.01314.x. PMID 11972592. S2CID 11849647.

Frang H, Cockcroft V, Karskela T, Scheinin M, Marjamäki A (August 2001). "Phenoxybenzamine binding reveals the helical orientation of the third transmembrane domain of adrenergic receptors". The Journal of Biological Chemistry. 276 (33): 31279–84. doi:10.1074/jbc.M104167200. PMID 11395517.

nih.gov

pubmed.ncbi.nlm.nih.gov

Hopkins AL, Groom CR (September 2002). "The druggable genome". Nature Reviews. Drug Discovery. 1 (9): 727–30. doi:10.1038/nrd892. PMID 12209152. S2CID 13166282.

Ariens EJ (September 1954). "Affinity and intrinsic activity in the theory of competitive inhibition. I. Problems and theory". Archives Internationales de Pharmacodynamie et de Thérapie. 99 (1): 32–49. PMID 13229418.

Wyllie DJ, Chen PE (March 2007). "Taking the time to study competitive antagonism". British Journal of Pharmacology. 150 (5): 541–51. doi:10.1038/sj.bjp.0706997. PMC 2189774. PMID 17245371.

Colquhoun D (December 2007). "Why the Schild method is better than Schild realised". Trends in Pharmacological Sciences. 28 (12): 608–14. doi:10.1016/j.tips.2007.09.011. PMID 18023486.

Schild HO (February 1975). "An ambiguity in receptor theory". British Journal of Pharmacology. 53 (2): 311. doi:10.1111/j.1476-5381.1975.tb07365.x. PMC 1666289. PMID 1148491.

Pulvirenti L, Koob GF (April 2002). "Being partial to psychostimulant addiction therapy". Trends in Pharmacological Sciences. 23 (4): 151–3. doi:10.1016/S0165-6147(00)01991-X. PMID 11931978.

Vadivelu N, Hines RL (2007). "Buprenorphine: a unique opioid with broad clinical applications". Journal of Opioid Management. 3 (1): 49–58. doi:10.5055/jom.2007.0038. PMID 17367094.

ncbi.nlm.nih.gov

semanticscholar.org

api.semanticscholar.org

Hopkins AL, Groom CR (September 2002). "The druggable genome". Nature Reviews. Drug Discovery. 1 (9): 727–30. doi:10.1038/nrd892. PMID 12209152. S2CID 13166282.

unc.edu

cdr.lib.unc.edu

Receptor antagonist (English Wikipedia)

books.google.com

doi.org

etymonline.com

guidetopharmacology.org

nih.gov

pubmed.ncbi.nlm.nih.gov

ncbi.nlm.nih.gov

oed.com

semanticscholar.org

api.semanticscholar.org

tulane.edu

tmedweb.tulane.edu

uam.es

pdg.cnb.uam.es

unc.edu

cdr.lib.unc.edu

web.archive.org

worldcat.org

search.worldcat.org