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Relugolix (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "Relugolix" in English language version.

refsWebsite
Global rank English rank
15nih.gov
4th place
4th place
10doi.org
2nd place
2nd place
4semanticscholar.org
11th place
8th place
3europa.eu
68th place
117th place
2web.archive.org
1st place
1st place
2springer.com
274th place
309th place
1legislation.gov.au
6,658th place
4,027th place
1canada.ca
1,712th place
1,063rd place
1hpfb-dgpsa.ca
low place
low place
1aska-pharma.co.jp
low place
low place
1prnewswire.com
406th place
258th place
1patents.google.com
1,182nd place
725th place
1fda.gov
447th place
338th place
1kegg.jp
low place
low place
1mhra.gov.uk
low place
low place
1nice.org.uk
3,258th place
2,666th place
1worldcat.org
5th place
5th place

aska-pharma.co.jp

canada.ca

doi.org

  • Barra F, Seca M, Della Corte L, Giampaolino P, Ferrero S (August 2019). "Relugolix for the treatment of uterine fibroids". Drugs of Today. 55 (8): 503–512. doi:10.1358/dot.2019.55.8.3020179. PMID 31461087. S2CID 201654739.
  • Miwa K, Hitaka T, Imada T, Sasaki S, Yoshimatsu M, Kusaka M, et al. (July 2011). "Discovery of 1-{4-[1-(2,6-difluorobenzyl)-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl]phenyl}-3-methoxyurea (TAK-385) as a potent, orally active, non-peptide antagonist of the human gonadotropin-releasing hormone receptor". Journal of Medicinal Chemistry. 54 (14): 4998–5012. doi:10.1021/jm200216q. PMID 21657270.
  • Nakata D, Masaki T, Tanaka A, Yoshimatsu M, Akinaga Y, Asada M, et al. (January 2014). "Suppression of the hypothalamic-pituitary-gonadal axis by TAK-385 (relugolix), a novel, investigational, orally active, small molecule gonadotropin-releasing hormone (GnRH) antagonist: studies in human GnRH receptor knock-in mice". European Journal of Pharmacology. 723: 167–174. doi:10.1016/j.ejphar.2013.12.001. PMID 24333551.
  • Tukun FL, Olberg DE, Riss PJ, Haraldsen I, Kaass A, Klaveness J (December 2017). "Recent Development of Non-Peptide GnRH Antagonists". Molecules. 22 (12): 2188. doi:10.3390/molecules22122188. PMC 6149776. PMID 29232843.
  • MacLean DB, Shi H, Faessel HM, Saad F (December 2015). "Medical Castration Using the Investigational Oral GnRH Antagonist TAK-385 (Relugolix): Phase 1 Study in Healthy Males". The Journal of Clinical Endocrinology and Metabolism. 100 (12): 4579–4587. doi:10.1210/jc.2015-2770. PMC 4667159. PMID 26502357.
  • Streuli I, de Ziegler D, Borghese B, Santulli P, Batteux F, Chapron C (March 2012). "New treatment strategies and emerging drugs in endometriosis". Expert Opinion on Emerging Drugs. 17: 83–104. doi:10.1517/14728214.2012.668885. PMID 22439891. S2CID 27472695.
  • Struthers RS, Nicholls AJ, Grundy J, Chen T, Jimenez R, Yen SS, Bozigian HP (February 2009). "Suppression of gonadotropins and estradiol in premenopausal women by oral administration of the nonpeptide gonadotropin-releasing hormone antagonist elagolix". The Journal of Clinical Endocrinology and Metabolism. 94 (2): 545–551. doi:10.1210/jc.2008-1695. PMC 2646513. PMID 19033369.
  • Goenka L, George M, Sen M (June 2017). "A peek into the drug development scenario of endometriosis - A systematic review". Biomedicine & Pharmacotherapy. 90: 575–585. doi:10.1016/j.biopha.2017.03.092. PMID 28407578.
  • Dellis A, Papatsoris A (October 2017). "Therapeutic outcomes of the LHRH antagonists". Expert Review of Pharmacoeconomics & Outcomes Research. 17 (5): 481–488. doi:10.1080/14737167.2017.1375855. PMID 28870102. S2CID 38014222.
  • Elancheran R, Maruthanila VL, Ramanathan M, Kabilan S, Devi R, Kunnumakara A, Kotoky J (2015). "Recent discoveries and developments of androgen receptor based therapy for prostate cancer". Med. Chem. Commun. 6 (5): 746–768. doi:10.1039/C4MD00416G. ISSN 2040-2503. S2CID 72654573.

europa.eu

ema.europa.eu

  • "Orgovyx EPAR". European Medicines Agency. 22 February 2022. Retrieved 3 March 2023. Text was copied from this source which is copyright European Medicines Agency. Reproduction is authorized provided the source is acknowledged.
  • "Orgovyx: Pending EC decision". European Medicines Agency. 24 February 2022. Archived from the original on 27 February 2022. Retrieved 27 February 2022. Text was copied from this source which is copyright European Medicines Agency. Reproduction is authorized provided the source is acknowledged.

ec.europa.eu

fda.gov

hpfb-dgpsa.ca

dhpp.hpfb-dgpsa.ca

kegg.jp

  • "Relugolix". KEGG DRUG Database. Kyoto Encyclopedia of Genes and Genomes.

legislation.gov.au

mhra.gov.uk

products.mhra.gov.uk

nice.org.uk

nih.gov

pubmed.ncbi.nlm.nih.gov

  • Barra F, Seca M, Della Corte L, Giampaolino P, Ferrero S (August 2019). "Relugolix for the treatment of uterine fibroids". Drugs of Today. 55 (8): 503–512. doi:10.1358/dot.2019.55.8.3020179. PMID 31461087. S2CID 201654739.
  • Miwa K, Hitaka T, Imada T, Sasaki S, Yoshimatsu M, Kusaka M, et al. (July 2011). "Discovery of 1-{4-[1-(2,6-difluorobenzyl)-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl]phenyl}-3-methoxyurea (TAK-385) as a potent, orally active, non-peptide antagonist of the human gonadotropin-releasing hormone receptor". Journal of Medicinal Chemistry. 54 (14): 4998–5012. doi:10.1021/jm200216q. PMID 21657270.
  • Nakata D, Masaki T, Tanaka A, Yoshimatsu M, Akinaga Y, Asada M, et al. (January 2014). "Suppression of the hypothalamic-pituitary-gonadal axis by TAK-385 (relugolix), a novel, investigational, orally active, small molecule gonadotropin-releasing hormone (GnRH) antagonist: studies in human GnRH receptor knock-in mice". European Journal of Pharmacology. 723: 167–174. doi:10.1016/j.ejphar.2013.12.001. PMID 24333551.
  • Tukun FL, Olberg DE, Riss PJ, Haraldsen I, Kaass A, Klaveness J (December 2017). "Recent Development of Non-Peptide GnRH Antagonists". Molecules. 22 (12): 2188. doi:10.3390/molecules22122188. PMC 6149776. PMID 29232843.
  • MacLean DB, Shi H, Faessel HM, Saad F (December 2015). "Medical Castration Using the Investigational Oral GnRH Antagonist TAK-385 (Relugolix): Phase 1 Study in Healthy Males". The Journal of Clinical Endocrinology and Metabolism. 100 (12): 4579–4587. doi:10.1210/jc.2015-2770. PMC 4667159. PMID 26502357.
  • Streuli I, de Ziegler D, Borghese B, Santulli P, Batteux F, Chapron C (March 2012). "New treatment strategies and emerging drugs in endometriosis". Expert Opinion on Emerging Drugs. 17: 83–104. doi:10.1517/14728214.2012.668885. PMID 22439891. S2CID 27472695.
  • Struthers RS, Nicholls AJ, Grundy J, Chen T, Jimenez R, Yen SS, Bozigian HP (February 2009). "Suppression of gonadotropins and estradiol in premenopausal women by oral administration of the nonpeptide gonadotropin-releasing hormone antagonist elagolix". The Journal of Clinical Endocrinology and Metabolism. 94 (2): 545–551. doi:10.1210/jc.2008-1695. PMC 2646513. PMID 19033369.
  • Goenka L, George M, Sen M (June 2017). "A peek into the drug development scenario of endometriosis - A systematic review". Biomedicine & Pharmacotherapy. 90: 575–585. doi:10.1016/j.biopha.2017.03.092. PMID 28407578.
  • Dellis A, Papatsoris A (October 2017). "Therapeutic outcomes of the LHRH antagonists". Expert Review of Pharmacoeconomics & Outcomes Research. 17 (5): 481–488. doi:10.1080/14737167.2017.1375855. PMID 28870102. S2CID 38014222.

ncbi.nlm.nih.gov

dailymed.nlm.nih.gov

chem.nlm.nih.gov

  • "Relugolix". ChemIDplus. U.S. National Library of Medicine.

patents.google.com

  • US 7300935, Cho N, Imada T, Hitaka T, Miwa K, Kusaka M, Suzuki N, "Thienopyrimidine compounds and use thereof", issued 27 November 2007, assigned to Takeda Pharmaceutical Co Ltd. 

prnewswire.com

semanticscholar.org

api.semanticscholar.org

  • Barra F, Seca M, Della Corte L, Giampaolino P, Ferrero S (August 2019). "Relugolix for the treatment of uterine fibroids". Drugs of Today. 55 (8): 503–512. doi:10.1358/dot.2019.55.8.3020179. PMID 31461087. S2CID 201654739.
  • Streuli I, de Ziegler D, Borghese B, Santulli P, Batteux F, Chapron C (March 2012). "New treatment strategies and emerging drugs in endometriosis". Expert Opinion on Emerging Drugs. 17: 83–104. doi:10.1517/14728214.2012.668885. PMID 22439891. S2CID 27472695.
  • Dellis A, Papatsoris A (October 2017). "Therapeutic outcomes of the LHRH antagonists". Expert Review of Pharmacoeconomics & Outcomes Research. 17 (5): 481–488. doi:10.1080/14737167.2017.1375855. PMID 28870102. S2CID 38014222.
  • Elancheran R, Maruthanila VL, Ramanathan M, Kabilan S, Devi R, Kunnumakara A, Kotoky J (2015). "Recent discoveries and developments of androgen receptor based therapy for prostate cancer". Med. Chem. Commun. 6 (5): 746–768. doi:10.1039/C4MD00416G. ISSN 2040-2503. S2CID 72654573.

springer.com

adisinsight.springer.com

web.archive.org

  • "Relumina (relugolix) Information" (PDF). ASKA Pharmaceutical (in Japanese). January 2019. Archived from the original (PDF) on 16 February 2019. Retrieved 16 February 2019.
  • "Orgovyx: Pending EC decision". European Medicines Agency. 24 February 2022. Archived from the original on 27 February 2022. Retrieved 27 February 2022. Text was copied from this source which is copyright European Medicines Agency. Reproduction is authorized provided the source is acknowledged.

worldcat.org

search.worldcat.org

  • Elancheran R, Maruthanila VL, Ramanathan M, Kabilan S, Devi R, Kunnumakara A, Kotoky J (2015). "Recent discoveries and developments of androgen receptor based therapy for prostate cancer". Med. Chem. Commun. 6 (5): 746–768. doi:10.1039/C4MD00416G. ISSN 2040-2503. S2CID 72654573.