Archer DF (August 2020). "Ospemifene: less venous thrombosis than other selective estrogen receptor modulators in postmenopausal women with vulvo vaginal atrophy". Menopause. 27 (8): 846–847. doi:10.1097/GME.0000000000001600. PMID32576803. S2CID220045301.
Riggs BL, Hartmann LC (Feb 2003). "Selective estrogen-receptor modulators -- mechanisms of action and application to clinical practice". The New England Journal of Medicine. 348 (7): 618–29. doi:10.1056/NEJMra022219. PMID12584371.
Pickar JH, Komm BS (Sep 2015). "Selective estrogen receptor modulators and the combination therapy conjugated estrogens/bazedoxifene: A review of effects on the breast". Post Reproductive Health. 21 (3): 112–21. doi:10.1177/2053369115599090. PMID26289836. S2CID206825977.
Kremoser C, Albers M, Burris TP, Deuschle U, Koegl M (Oct 2007). "Panning for SNuRMs: using cofactor profiling for the rational discovery of selective nuclear receptor modulators". Drug Discovery Today. 12 (19–20): 860–9. doi:10.1016/j.drudis.2007.07.025. PMID17933688.
Rosano C, Stec-Martyna E, Lappano R, Maggiolini M (2011). "Structure-based approach for the discovery of novel selective estrogen receptor modulators". Current Medicinal Chemistry. 18 (8): 1188–94. doi:10.2174/092986711795029645. PMID21291367.
Xu X, Yang W, Li Y, Wang Y (Jan 2010). "Discovery of estrogen receptor modulators: a review of virtual screening and SAR efforts". Expert Opinion on Drug Discovery. 5 (1): 21–31. doi:10.1517/17460440903490395. PMID22823969. S2CID207492889.
Brzozowski AM, Pike AC, Dauter Z, Hubbard RE, Bonn T, Engström O, Öhman L, Greene GL, Gustafsson JÅ, Carlquist M (1997). "Molecular basis of agonism and antagonism in the oestrogen receptor". Nature. 389 (6652): 753–8. Bibcode:1997Natur.389..753B. doi:10.1038/39645. PMID9338790. S2CID4430999.
Musa MA, Khan MO, Cooperwood JS (2007). "Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs)". Current Medicinal Chemistry. 14 (11): 1249–61. doi:10.2174/092986707780598023. PMID17504144.
Lewis JS, Jordan VC (Dec 2005). "Selective estrogen receptor modulators (SERMs): mechanisms of anticarcinogenesis and drug resistance". Mutation Research. 591 (1–2): 247–63. doi:10.1016/j.mrfmmm.2005.02.028. PMID16083919.
Fang H, Tong W, Shi LM, Blair R, Perkins R, Branham W, Hass BS, Xie Q, Dial SL, Moland CL, Sheehan DM (Mar 2001). "Structure-activity relationships for a large diverse set of natural, synthetic, and environmental estrogens". Chemical Research in Toxicology. 14 (3): 280–94. CiteSeerX10.1.1.460.20. doi:10.1021/tx000208y. PMID11258977.
Clark JH, Markaverich BM (1981). "The agonistic-antagonistic properties of clomiphene: a review". Pharmacology & Therapeutics. 15 (3): 467–519. doi:10.1016/0163-7258(81)90055-3. PMID7048350.
Singh MN, Stringfellow HF, Paraskevaidis E, Martin-Hirsch PL, Martin FL (Apr 2007). "Tamoxifen: important considerations of a multi-functional compound with organ-specific properties". Cancer Treatment Reviews. 33 (2): 91–100. doi:10.1016/j.ctrv.2006.09.008. PMID17178195.]
de Médina P, Favre G, Poirot M (Nov 2004). "Multiple targeting by the antitumor drug tamoxifen: a structure-activity study". Current Medicinal Chemistry. Anti-Cancer Agents. 4 (6): 491–508. doi:10.2174/1568011043352696. PMID15579015.
Gauthier S, Mailhot J, Labrie F (May 1996). "New Highly Stereoselective Synthesis of (Z)-4-Hydroxytamoxifen and (Z)-4-Hydroxytoremifene via McMurry Reaction". The Journal of Organic Chemistry. 61 (11): 3890–3893. doi:10.1021/jo952279l. PMID11667248.
Jordan VC (Mar 2003). "Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents". Journal of Medicinal Chemistry. 46 (7): 1081–111. doi:10.1021/jm020450x. PMID12646017.
Kung AW, Chu EY, Xu L (Jun 2009). "Bazedoxifene: a new selective estrogen receptor modulator for the treatment of postmenopausal osteoporosis". Expert Opinion on Pharmacotherapy. 10 (8): 1377–85. doi:10.1517/14656560902980228. PMID19445558. S2CID20781017.
Gennari L, Merlotti D, Valleggi F, Nuti R (Jun 2009). "Ospemifene use in postmenopausal women". Expert Opinion on Investigational Drugs. 18 (6): 839–49. doi:10.1517/13543780902953715. PMID19466874. S2CID21537130.
Taneja SS, Smith MR, Dalton JT, Raghow S, Barnette G, Steiner M, Veverka KA (Mar 2006). "Toremifene--a promising therapy for the prevention of prostate cancer and complications of androgen deprivation therapy". Expert Opinion on Investigational Drugs. 15 (3): 293–305. doi:10.1517/13543784.15.3.293. PMID16503765. S2CID29510508.
Archer DF (August 2020). "Ospemifene: less venous thrombosis than other selective estrogen receptor modulators in postmenopausal women with vulvo vaginal atrophy". Menopause. 27 (8): 846–847. doi:10.1097/GME.0000000000001600. PMID32576803. S2CID220045301.
Riggs BL, Hartmann LC (Feb 2003). "Selective estrogen-receptor modulators -- mechanisms of action and application to clinical practice". The New England Journal of Medicine. 348 (7): 618–29. doi:10.1056/NEJMra022219. PMID12584371.
Pickar JH, Komm BS (Sep 2015). "Selective estrogen receptor modulators and the combination therapy conjugated estrogens/bazedoxifene: A review of effects on the breast". Post Reproductive Health. 21 (3): 112–21. doi:10.1177/2053369115599090. PMID26289836. S2CID206825977.
Kremoser C, Albers M, Burris TP, Deuschle U, Koegl M (Oct 2007). "Panning for SNuRMs: using cofactor profiling for the rational discovery of selective nuclear receptor modulators". Drug Discovery Today. 12 (19–20): 860–9. doi:10.1016/j.drudis.2007.07.025. PMID17933688.
Rosano C, Stec-Martyna E, Lappano R, Maggiolini M (2011). "Structure-based approach for the discovery of novel selective estrogen receptor modulators". Current Medicinal Chemistry. 18 (8): 1188–94. doi:10.2174/092986711795029645. PMID21291367.
Xu X, Yang W, Li Y, Wang Y (Jan 2010). "Discovery of estrogen receptor modulators: a review of virtual screening and SAR efforts". Expert Opinion on Drug Discovery. 5 (1): 21–31. doi:10.1517/17460440903490395. PMID22823969. S2CID207492889.
Brzozowski AM, Pike AC, Dauter Z, Hubbard RE, Bonn T, Engström O, Öhman L, Greene GL, Gustafsson JÅ, Carlquist M (1997). "Molecular basis of agonism and antagonism in the oestrogen receptor". Nature. 389 (6652): 753–8. Bibcode:1997Natur.389..753B. doi:10.1038/39645. PMID9338790. S2CID4430999.
Musa MA, Khan MO, Cooperwood JS (2007). "Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs)". Current Medicinal Chemistry. 14 (11): 1249–61. doi:10.2174/092986707780598023. PMID17504144.
Lewis JS, Jordan VC (Dec 2005). "Selective estrogen receptor modulators (SERMs): mechanisms of anticarcinogenesis and drug resistance". Mutation Research. 591 (1–2): 247–63. doi:10.1016/j.mrfmmm.2005.02.028. PMID16083919.
Fang H, Tong W, Shi LM, Blair R, Perkins R, Branham W, Hass BS, Xie Q, Dial SL, Moland CL, Sheehan DM (Mar 2001). "Structure-activity relationships for a large diverse set of natural, synthetic, and environmental estrogens". Chemical Research in Toxicology. 14 (3): 280–94. CiteSeerX10.1.1.460.20. doi:10.1021/tx000208y. PMID11258977.
Clark JH, Markaverich BM (1981). "The agonistic-antagonistic properties of clomiphene: a review". Pharmacology & Therapeutics. 15 (3): 467–519. doi:10.1016/0163-7258(81)90055-3. PMID7048350.
Jensen EV, Jordan VC (Jun 2003). "The estrogen receptor: a model for molecular medicine". Clinical Cancer Research. 9 (6): 1980–9. PMID12796359.
Singh MN, Stringfellow HF, Paraskevaidis E, Martin-Hirsch PL, Martin FL (Apr 2007). "Tamoxifen: important considerations of a multi-functional compound with organ-specific properties". Cancer Treatment Reviews. 33 (2): 91–100. doi:10.1016/j.ctrv.2006.09.008. PMID17178195.]
de Médina P, Favre G, Poirot M (Nov 2004). "Multiple targeting by the antitumor drug tamoxifen: a structure-activity study". Current Medicinal Chemistry. Anti-Cancer Agents. 4 (6): 491–508. doi:10.2174/1568011043352696. PMID15579015.
Gauthier S, Mailhot J, Labrie F (May 1996). "New Highly Stereoselective Synthesis of (Z)-4-Hydroxytamoxifen and (Z)-4-Hydroxytoremifene via McMurry Reaction". The Journal of Organic Chemistry. 61 (11): 3890–3893. doi:10.1021/jo952279l. PMID11667248.
Jordan VC (Mar 2003). "Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents". Journal of Medicinal Chemistry. 46 (7): 1081–111. doi:10.1021/jm020450x. PMID12646017.
Kung AW, Chu EY, Xu L (Jun 2009). "Bazedoxifene: a new selective estrogen receptor modulator for the treatment of postmenopausal osteoporosis". Expert Opinion on Pharmacotherapy. 10 (8): 1377–85. doi:10.1517/14656560902980228. PMID19445558. S2CID20781017.
Gennari L, Merlotti D, Valleggi F, Nuti R (Jun 2009). "Ospemifene use in postmenopausal women". Expert Opinion on Investigational Drugs. 18 (6): 839–49. doi:10.1517/13543780902953715. PMID19466874. S2CID21537130.
Taneja SS, Smith MR, Dalton JT, Raghow S, Barnette G, Steiner M, Veverka KA (Mar 2006). "Toremifene--a promising therapy for the prevention of prostate cancer and complications of androgen deprivation therapy". Expert Opinion on Investigational Drugs. 15 (3): 293–305. doi:10.1517/13543784.15.3.293. PMID16503765. S2CID29510508.
Fang H, Tong W, Shi LM, Blair R, Perkins R, Branham W, Hass BS, Xie Q, Dial SL, Moland CL, Sheehan DM (Mar 2001). "Structure-activity relationships for a large diverse set of natural, synthetic, and environmental estrogens". Chemical Research in Toxicology. 14 (3): 280–94. CiteSeerX10.1.1.460.20. doi:10.1021/tx000208y. PMID11258977.
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Archer DF (August 2020). "Ospemifene: less venous thrombosis than other selective estrogen receptor modulators in postmenopausal women with vulvo vaginal atrophy". Menopause. 27 (8): 846–847. doi:10.1097/GME.0000000000001600. PMID32576803. S2CID220045301.
Pickar JH, Komm BS (Sep 2015). "Selective estrogen receptor modulators and the combination therapy conjugated estrogens/bazedoxifene: A review of effects on the breast". Post Reproductive Health. 21 (3): 112–21. doi:10.1177/2053369115599090. PMID26289836. S2CID206825977.
Xu X, Yang W, Li Y, Wang Y (Jan 2010). "Discovery of estrogen receptor modulators: a review of virtual screening and SAR efforts". Expert Opinion on Drug Discovery. 5 (1): 21–31. doi:10.1517/17460440903490395. PMID22823969. S2CID207492889.
Brzozowski AM, Pike AC, Dauter Z, Hubbard RE, Bonn T, Engström O, Öhman L, Greene GL, Gustafsson JÅ, Carlquist M (1997). "Molecular basis of agonism and antagonism in the oestrogen receptor". Nature. 389 (6652): 753–8. Bibcode:1997Natur.389..753B. doi:10.1038/39645. PMID9338790. S2CID4430999.
Kung AW, Chu EY, Xu L (Jun 2009). "Bazedoxifene: a new selective estrogen receptor modulator for the treatment of postmenopausal osteoporosis". Expert Opinion on Pharmacotherapy. 10 (8): 1377–85. doi:10.1517/14656560902980228. PMID19445558. S2CID20781017.
Gennari L, Merlotti D, Valleggi F, Nuti R (Jun 2009). "Ospemifene use in postmenopausal women". Expert Opinion on Investigational Drugs. 18 (6): 839–49. doi:10.1517/13543780902953715. PMID19466874. S2CID21537130.
Taneja SS, Smith MR, Dalton JT, Raghow S, Barnette G, Steiner M, Veverka KA (Mar 2006). "Toremifene--a promising therapy for the prevention of prostate cancer and complications of androgen deprivation therapy". Expert Opinion on Investigational Drugs. 15 (3): 293–305. doi:10.1517/13543784.15.3.293. PMID16503765. S2CID29510508.