References analysis of the Wikipedia article "Selective progesterone receptor modulator" in the English version

doi.org

Chwalisz K, Perez MC, Demanno D, Winkel C, Schubert G, Elger W (May 2005). "Selective progesterone receptor modulator development and use in the treatment of leiomyomata and endometriosis". Endocrine Reviews. 26 (3): 423–38. doi:10.1210/er.2005-0001. PMID 15857972.

Misrahi M, Loosfelt H, Atger M, Mériel C, Zerah V, Dessen P, Milgrom E (Jun 1988). "Organisation of the entire rabbit progesterone receptor mRNA and of the promoter and 5' flanking region of the gene". Nucleic Acids Research. 16 (12): 5459–72. doi:10.1093/nar/16.12.5459. PMC 336778. PMID 3387238.

Allen WM (Aug 1935). "The isolation of crystalline progestin". Science. 82 (2118): 89–93. Bibcode:1935Sci....82...89A. doi:10.1126/science.82.2118.89. PMID 17747122.

Karrer P, Schwarzenbach G (Jan 1934). "Nachtrag betreffend Acidität und Reduktions-Vermögen der Ascorbinsäure". Helvetica Chimica Acta. 17 (1): 58–59. doi:10.1002/hlca.19340170111. ISSN 1522-2675.

Sherman MR, Corvol PL, O'Malley BW (Nov 1970). "Progesterone-binding components of chick oviduct. I. Preliminary characterization of cytoplasmic components". The Journal of Biological Chemistry. 245 (22): 6085–96. doi:10.1016/S0021-9258(18)62667-5. PMID 5484467.

Groyer A, Le Bouc Y, Joab I, Radanyi C, Renoir JM, Robel P, Baulieu EE (Jun 1985). "Chick oviduct glucocorticosteroid receptor. Specific binding of the synthetic steroid RU 486 and immunological studies with antibodies to chick oviduct progesterone receptor". European Journal of Biochemistry. 149 (2): 445–51. doi:10.1111/j.1432-1033.1985.tb08945.x. PMID 3996417.

Gass EK, Leonhardt SA, Nordeen SK, Edwards DP (Apr 1998). "The antagonists RU486 and ZK98299 stimulate progesterone receptor binding to deoxyribonucleic acid in vitro and in vivo, but have distinct effects on receptor conformation". Endocrinology. 139 (4): 1905–19. doi:10.1210/endo.139.4.5944. PMID 9528977.

Lázár G, Lázár G, Husztik E, Duda E, Agarwal MK (Jun 1995). "The influence of antiglucocorticoids on stress and shock". Annals of the New York Academy of Sciences. 761 (1): 276–95. Bibcode:1995NYASA.761..276L. doi:10.1111/j.1749-6632.1995.tb31384.x. PMID 7625726. S2CID 40422188.

Spitz IM, Chwalisz K (Aug 2010). "Progesterone receptor modulators and progesterone antagonists in women's health". Steroids. 65 (10–11): 807–15. doi:10.1016/S0039-128X(00)00194-X. PMID 11108892. S2CID 27699000.

Chen W, Ohara N, Wang J, Xu Q, Liu J, Morikawa A, Sasaki H, Yoshida S, Demanno DA, Chwalisz K, Maruo T (Apr 2006). "A novel selective progesterone receptor modulator asoprisnil (J867) inhibits proliferation and induces apoptosis in cultured human uterine leiomyoma cells in the absence of comparable effects on myometrial cells". The Journal of Clinical Endocrinology and Metabolism. 91 (4): 1296–304. doi:10.1210/jc.2005-2379. PMID 16464945.

Chabbert-Buffet N, Meduri G, Bouchard P, Spitz IM (2005). "Selective progesterone receptor modulators and progesterone antagonists: mechanisms of action and clinical applications". Human Reproduction Update. 11 (3): 293–307. doi:10.1093/humupd/dmi002. PMID 15790602.

Elger W, Bartley J, Schneider B, Kaufmann G, Schubert G, Chwalisz K (2000-10-01). "Endocrine pharmacological characterization of progesterone antagonists and progesterone receptor modulators with respect to PR-agonistic and antagonistic activity". Steroids. 65 (10–11): 713–23. doi:10.1016/S0039-128X(00)00178-1. PMID 11108882. S2CID 46138800.

Palmer S, Campen CA, Allan GF, Rybczynski P, Haynes-Johnson D, Hutchins A, Kraft P, Kiddoe M, Lai M, Lombardi E, Pedersen P, Hodgen G, Combs DW (Dec 2000). "Nonsteroidal progesterone receptor ligands with unprecedented receptor selectivity". The Journal of Steroid Biochemistry and Molecular Biology. 75 (1): 33–42. doi:10.1016/S0960-0760(00)00134-5. PMID 11179906. S2CID 19167595.

DeManno D, Elger W, Garg R, Lee R, Schneider B, Hess-Stumpp H, Schubert G, Chwalisz K (Nov 2003). "Asoprisnil (J867): a selective progesterone receptor modulator for gynecological therapy". Steroids. 68 (10–13): 1019–32. doi:10.1016/j.steroids.2003.09.008. PMID 14667995. S2CID 23074350.

Donnez J, Vázquez F, Tomaszewski J, Nouri K, Bouchard P, Fauser BC, Barlow DH, Palacios S, Donnez O, Bestel E, Osterloh I, Loumaye E (Jun 2014). "Long-term treatment of uterine fibroids with ulipristal acetate". Fertility and Sterility. 101 (6): 1565–73.e1–18. doi:10.1016/j.fertnstert.2014.02.008. PMID 24630081.

Mangelsdorf DJ, Thummel C, Beato M, Herrlich P, Schütz G, Umesono K, Blumberg B, Kastner P, Mark M, Chambon P, Evans RM (Dec 1995). "The nuclear receptor superfamily: the second decade". Cell. 83 (6): 835–9. doi:10.1016/0092-8674(95)90199-X. PMC 6159888. PMID 8521507.

Conneely OM, Maxwell BL, Toft DO, Schrader WT, O'Malley BW (Dec 1987). "The A and B forms of the chicken progesterone receptor arise by alternate initiation of translation of a unique mRNA". Biochemical and Biophysical Research Communications. 149 (2): 493–501. doi:10.1016/0006-291X(87)90395-0. PMID 3426587.

Kastner P, Krust A, Turcotte B, Stropp U, Tora L, Gronemeyer H, Chambon P (May 1990). "Two distinct estrogen-regulated promoters generate transcripts encoding the two functionally different human progesterone receptor forms A and B". The EMBO Journal. 9 (5): 1603–14. doi:10.1002/j.1460-2075.1990.tb08280.x. PMC 551856. PMID 2328727.

Hirata S, Shoda T, Kato J, Hoshi K (Dec 2002). "Novel isoforms of the mRNA for human female sex steroid hormone receptors". The Journal of Steroid Biochemistry and Molecular Biology. 83 (1–5): 25–30. doi:10.1016/S0960-0760(02)00255-8. PMID 12650698. S2CID 23588169.

Hirata S, Shoda T, Kato J, Hoshi K (Apr 2003). "Isoform/variant mRNAs for sex steroid hormone receptors in humans". Trends in Endocrinology and Metabolism. 14 (3): 124–9. doi:10.1016/S1043-2760(03)00028-6. PMID 12670738. S2CID 46220794.

Brinton RD, Thompson RF, Foy MR, Baudry M, Wang J, Finch CE, Morgan TE, Pike CJ, Mack WJ, Stanczyk FZ, Nilsen J (May 2008). "Progesterone receptors: form and function in brain". Frontiers in Neuroendocrinology. 29 (2): 313–39. doi:10.1016/j.yfrne.2008.02.001. PMC 2398769. PMID 18374402.

Ellmann S, Sticht H, Thiel F, Beckmann MW, Strick R, Strissel PL (Aug 2009). "Estrogen and progesterone receptors: from molecular structures to clinical targets". Cellular and Molecular Life Sciences. 66 (15): 2405–26. doi:10.1007/s00018-009-0017-3. PMC 11115849. PMID 19333551. S2CID 19975774.

Winneker RC, Fensome A, Zhang P, Yudt MR, McComas CC, Unwalla RJ (Aug 2008). "A new generation of progesterone receptor modulators". Steroids. 73 (7): 689–701. doi:10.1016/j.steroids.2008.03.005. PMID 18472121. S2CID 25094160.

Edwards DP, Altmann M, DeMarzo A, Zhang Y, Weigel NL, Beck CA (Jun 1995). "Progesterone receptor and the mechanism of action of progesterone antagonists". The Journal of Steroid Biochemistry and Molecular Biology. 53 (1–6): 449–58. doi:10.1016/0960-0760(95)00091-d. PMID 7626494. S2CID 41957428.

Lusher SJ, Raaijmakers HC, Vu-Pham D, Kazemier B, Bosch R, McGuire R, Azevedo R, Hamersma H, Dechering K, Oubrie A, van Duin M, de Vlieg J (Jun 2012). "X-ray structures of progesterone receptor ligand binding domain in its agonist state reveal differing mechanisms for mixed profiles of 11β-substituted steroids". The Journal of Biological Chemistry. 287 (24): 20333–43. doi:10.1074/jbc.M111.308403. PMC 3370215. PMID 22535964.

Jackson TA, Richer JK, Bain DL, Takimoto GS, Tung L, Horwitz KB (Jun 1997). "The partial agonist activity of antagonist-occupied steroid receptors is controlled by a novel hinge domain-binding coactivator L7/SPA and the corepressors N-CoR or SMRT". Molecular Endocrinology. 11 (6): 693–705. doi:10.1210/mend.11.6.0004. PMID 9171233. S2CID 21356045.

Smith CL, O'Malley BW (Feb 2004). "Coregulator function: a key to understanding tissue specificity of selective receptor modulators". Endocrine Reviews. 25 (1): 45–71. doi:10.1210/er.2003-0023. PMID 14769827.

Oñate SA, Estes PA, Welch WJ, Nordeen SK, Edwards DP (Dec 1991). "Evidence that heat shock protein-70 associated with progesterone receptors is not involved in receptor-DNA binding". Molecular Endocrinology. 5 (12): 1993–2004. doi:10.1210/mend-5-12-1993. PMID 1791844.

Smith DF, Stensgard BA, Welch WJ, Toft DO (Jan 1992). "Assembly of progesterone receptor with heat shock proteins and receptor activation are ATP mediated events". The Journal of Biological Chemistry. 267 (2): 1350–6. doi:10.1016/S0021-9258(18)48438-4. PMID 1730655.

DeMarzo AM, Beck CA, Onate SA, Edwards DP (Jan 1991). "Dimerization of mammalian progesterone receptors occurs in the absence of DNA and is related to the release of the 90-kDa heat shock protein". Proceedings of the National Academy of Sciences of the United States of America. 88 (1): 72–6. Bibcode:1991PNAS...88...72D. doi:10.1073/pnas.88.1.72. PMC 50750. PMID 1986383.

Guiochon-Mantel A, Loosfelt H, Lescop P, Sar S, Atger M, Perrot-Applanat M, Milgrom E (Jun 1989). "Mechanisms of nuclear localization of the progesterone receptor: evidence for interaction between monomers". Cell. 57 (7): 1147–54. doi:10.1016/0092-8674(89)90052-4. PMID 2736623.

O'Malley BW, Tsai MJ (Feb 1992). "Molecular pathways of steroid receptor action". Biology of Reproduction. 46 (2): 163–7. doi:10.1095/biolreprod46.2.163. PMID 1536890.

Bagchi MK, Tsai MJ, O'Malley BW, Tsai SY (Aug 1992). "Analysis of the mechanism of steroid hormone receptor-dependent gene activation in cell-free systems". Endocrine Reviews. 13 (3): 525–35. doi:10.1210/edrv-13-3-525. PMID 1425487.

McKenna NJ, O'Malley BW (Feb 2002). "Combinatorial control of gene expression by nuclear receptors and coregulators". Cell. 108 (4): 465–74. doi:10.1016/S0092-8674(02)00641-4. PMID 11909518.

Oñate SA, Tsai SY, Tsai MJ, O'Malley BW (Nov 1995). "Sequence and characterization of a coactivator for the steroid hormone receptor superfamily". Science. 270 (5240): 1354–7. Bibcode:1995Sci...270.1354O. doi:10.1126/science.270.5240.1354. PMID 7481822. S2CID 28749162.

Wagner BL, Norris JD, Knotts TA, Weigel NL, McDonnell DP (Mar 1998). "The nuclear corepressors NCoR and SMRT are key regulators of both ligand- and 8-bromo-cyclic AMP-dependent transcriptional activity of the human progesterone receptor". Molecular and Cellular Biology. 18 (3): 1369–78. doi:10.1128/mcb.18.3.1369. PMC 108850. PMID 9488452.

Liu Z, Auboeuf D, Wong J, Chen JD, Tsai SY, Tsai MJ, O'Malley BW (Jun 2002). "Coactivator/corepressor ratios modulate PR-mediated transcription by the selective receptor modulator RU486". Proceedings of the National Academy of Sciences of the United States of America. 99 (12): 7940–4. Bibcode:2002PNAS...99.7940L. doi:10.1073/pnas.122225699. PMC 122999. PMID 12048256.

Nickisch K, Elger W, Cessac J, Kesavaram N, Das B, Garfield R, Shi SQ, Amelkina O, Meister R (Feb 2013). "Synthesis and biological evaluation of partially fluorinated antiprogestins and mesoprogestins". Steroids. 78 (2): 255–67. doi:10.1016/j.steroids.2012.09.010. PMID 23178161. S2CID 17158416.

Nickisch K, Elger W, Santhamma B, Garfield R, Killeen Z, Amelkina O, Schneider B, Meister R (Dec 2014). "Synthesis and biological evaluation of 11' imidazolyl antiprogestins and mesoprogestins". Steroids. 92: 45–55. doi:10.1016/j.steroids.2014.08.017. PMID 25174783. S2CID 6311225.

Rao PN, Wang Z, Cessac JW, Rosenberg RS, Jenkins DJ, Diamandis EP (Oct 1998). "New 11 beta-aryl-substituted steroids exhibit both progestational and antiprogestational activity". Steroids. 63 (10): 523–30. doi:10.1016/S0039-128X(98)00060-9. PMID 9800283. S2CID 42703467.

Wagner BL, Pollio G, Leonhardt S, Wani MC, Lee DY, Imhof MO, Edwards DP, Cook CE, McDonnell DP (Aug 1996). "16 alpha-substituted analogs of the antiprogestin RU486 induce a unique conformation in the human progesterone receptor resulting in mixed agonist activity". Proceedings of the National Academy of Sciences of the United States of America. 93 (16): 8739–44. Bibcode:1996PNAS...93.8739W. doi:10.1073/pnas.93.16.8739. PMC 38743. PMID 8710941.

Kang FA, Guan J, Jain N, Allan G, Linton O, Tannenbaum P, Chen X, Xu J, Zhu P, Gunnet J, Demarest K, Lundeen S, Sui Z (May 2007). "Parallel synthesis and SAR study of novel oxa-steroids as potent and selective progesterone receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 17 (9): 2531–4. doi:10.1016/j.bmcl.2007.02.013. PMID 17317167.

Kang FA, Allan G, Guan J, Jain N, Linton O, Tannenbaum P, Xu J, Zhu P, Gunnet J, Chen X, Demarest K, Lundeen S, Sui Z (Feb 2007). "Synthesis and identification of novel oxa-steroids as progesterone receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 17 (4): 907–10. doi:10.1016/j.bmcl.2006.11.062. PMID 17169557.

Rewinkel J, Enthoven M, Golstein I, van der Rijst M, Scholten A, van Tilborg M, de Weys D, Wisse J, Hamersma H (Mar 2008). "11-(pyridinylphenyl)steroids--a new class of mixed-profile progesterone agonists/antagonists". Bioorganic & Medicinal Chemistry. 16 (6): 2753–63. doi:10.1016/j.bmc.2008.01.010. PMID 18243712.

Jain N, Allan G, Linton O, Tannenbaum P, Chen X, Xu J, Zhu P, Gunnet J, Demarest K, Lundeen S, Murray W, Sui Z (Jul 2009). "Synthesis and SAR study of novel pseudo-steroids as potent and selective progesterone receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 19 (14): 3977–80. doi:10.1016/j.bmcl.2009.01.095. PMID 19217285.

Kang FA, Chen X, Jain N, Allan G, Tannenbaum P, Lundeen S, Sui Z (Jul 2008). "Insight from molecular modeling into different conformation and SAR of natural steroids and unnatural 7-oxa-steroids". Bioorganic & Medicinal Chemistry Letters. 18 (13): 3687–90. doi:10.1016/j.bmcl.2008.05.070. PMID 18539027.

Benagiano G, Bastianelli C, Farris M, Brosens I (Jul 2014). "Selective progesterone receptor modulators: an update". Expert Opinion on Pharmacotherapy. 15 (10): 1403–15. doi:10.1517/14656566.2014.914494. PMID 24787486. S2CID 31746942.

Brache V, Cochon L, Jesam C, Maldonado R, Salvatierra AM, Levy DP, Gainer E, Croxatto HB (Sep 2010). "Immediate pre-ovulatory administration of 30 mg ulipristal acetate significantly delays follicular rupture". Human Reproduction. 25 (9): 2256–63. doi:10.1093/humrep/deq157. PMID 20634186.

Aiken AR, Trussell J (2014). "Recent advances in contraception". F1000Prime Reports. 6: 113. doi:10.12703/p6-113. PMC 4251416. PMID 25580267.

Spitz IM (Nov 2003). "Progesterone antagonists and progesterone receptor modulators: an overview". Steroids. 68 (10–13): 981–93. doi:10.1016/j.steroids.2003.08.007. PMID 14667991. S2CID 23054270.

Lindsay SF, Luciano DE, Luciano AA (Sep 2015). "Emerging therapy for endometriosis". Expert Opinion on Emerging Drugs. 20 (3): 449–61. doi:10.1517/14728214.2015.1051966. PMID 26050551. S2CID 19276904.

Eckstein N, Haas B, Hass MD, Pfeifer V (Aug 2014). "Systemic therapy of Cushing's syndrome". Orphanet Journal of Rare Diseases. 9 (1): 122. doi:10.1186/s13023-014-0122-8. PMC 4237936. PMID 25091295.

Taylor DK, Holthouser K, Segars JH, Leppert PC (2015). "Recent scientific advances in leiomyoma (uterine fibroids) research facilitates better understanding and management". F1000Research. 4 (F1000 Faculty Rev): 183. doi:10.12688/f1000research.6189.1. PMC 4513689. PMID 26236472.

Pabla B, Bissonnette M, Konda VJ (Oct 2015). "Colon cancer and the epidermal growth factor receptor: Current treatment paradigms, the importance of diet, and the role of chemoprevention". World Journal of Clinical Oncology. 6 (5): 133–41. doi:10.5306/wjco.v6.i5.133. PMC 4600187. PMID 26468449.

Spitz IM (Aug 2009). "Clinical utility of progesterone receptor modulators and their effect on the endometrium". Current Opinion in Obstetrics and Gynecology. 21 (4): 318–24. doi:10.1097/GCO.0b013e32832e07e8. PMID 19602929. S2CID 2121292.

Bouchard P, Chabbert-Buffet N, Fauser BC (Nov 2011). "Selective progesterone receptor modulators in reproductive medicine: pharmacology, clinical efficacy and safety". Fertility and Sterility. 96 (5): 1175–89. doi:10.1016/j.fertnstert.2011.08.021. PMID 21944187.

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Allen WM (Aug 1935). "The isolation of crystalline progestin". Science. 82 (2118): 89–93. Bibcode:1935Sci....82...89A. doi:10.1126/science.82.2118.89. PMID 17747122.

O'Malley BW, Tsai MJ (Feb 1992). "Molecular pathways of steroid receptor action". Biology of Reproduction. 46 (2): 163–7. doi:10.1095/biolreprod46.2.163. PMID 1536890.

McKenna NJ, O'Malley BW (Feb 2002). "Combinatorial control of gene expression by nuclear receptors and coregulators". Cell. 108 (4): 465–74. doi:10.1016/S0092-8674(02)00641-4. PMID 11909518.

Aiken AR, Trussell J (2014). "Recent advances in contraception". F1000Prime Reports. 6: 113. doi:10.12703/p6-113. PMC 4251416. PMID 25580267.

Ohara N (2008). "Action of progesterone receptor modulators on uterine leiomyomas". Clinical and Experimental Obstetrics & Gynecology. 35 (3): 165–6. PMID 18754282.

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Selective progesterone receptor modulator (English Wikipedia)

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