Structural Genomics Consortium (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "Structural Genomics Consortium" in English language version.

refsWebsite

Global rank English rank

87nih.gov

4^th place

61doi.org

2^nd place

55worldcat.org

5^th place

22semanticscholar.org

11^th place

8^th place

7harvard.edu

18^th place

17^th place

5thesgc.org

low place

2biorxiv.org

5,061^st place

5,698^th place

1arxiv.org

69^th place

59^th place

1handle.net

102^nd place

76^th place

1ox.ac.uk

613^th place

456^th place

1vimiopen.org

low place

1nature.com

234^th place

397^th place

1unc.edu

1,538^th place

1,042^nd place

arxiv.org

Edwards, AM; et, al. (2011). "Too many roads not taken". Nature. 470 (2333): 163–165. arXiv:1102.0448. Bibcode:2011Natur.470..163E. doi:10.1038/470163a. PMID 21307913. S2CID 4429387.

biorxiv.org

Mann, Mandeep K.; Franzoni, Ivan; de Freitas, Renato Ferreira; Tempel, Wolfram; Houliston, Scott; Smith, Leanna; Vedadi, Masoud; Arrowsmith, Cheryl H.; Harding, Rachel J.; Schapira, Matthieu (27 November 2019). "Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain" (PDF). Journal of Medicinal Chemistry. 62 (22): 10144–10155. doi:10.1021/acs.jmedchem.9b00988. ISSN 1520-4804. PMID 31663737. S2CID 204975079.
Sorget, Nienke; et, al (2020). "Exploring the understudied human kinome for research and therapeutic opportunities" (PDF). www.biorxiv.org. doi:10.1101/2020.04.02.022277. S2CID 215404186.

doi.org

Williamson, AR (2000). "Creating a structural genomics consortium". Nature Structural Biology. 7: 953. doi:10.1038/80726. PMID 11103997. S2CID 35185565.
Edwards, AM; et, al. (2011). "Too many roads not taken". Nature. 470 (2333): 163–165. arXiv:1102.0448. Bibcode:2011Natur.470..163E. doi:10.1038/470163a. PMID 21307913. S2CID 4429387.
Davis, Andrew M.; Engkvist, Ola; Fairclough, Rebecca J.; Feierberg, Isabella; Freeman, Adrian; Iyer, Preeti (2021-02-13). "Public-Private Partnerships: Compound and Data Sharing in Drug Discovery and Development". SLAS Discovery. 26 (5): 604–619. doi:10.1177/2472555220982268. ISSN 2472-5552. PMID 33586501. S2CID 231928371.
Edwards, Aled (September 2008). "Open-source science to enable drug discovery". Drug Discovery Today. 13 (17–18): 731–733. doi:10.1016/j.drudis.2008.04.011. ISSN 1359-6446. PMID 18790412.
Edwards, Aled M.; Bountra, Chas; Kerr, David J.; Willson, Timothy M. (July 2009). "Open access chemical and clinical probes to support drug discovery". Nature Chemical Biology. 5 (7): 436–440. doi:10.1038/nchembio0709-436. ISSN 1552-4469. PMID 19536100.
Masum, Hassan; Rao, Aarthi; Good, Benjamin M.; Todd, Matthew H.; Edwards, Aled M.; Chan, Leslie; Bunin, Barry A.; Su, Andrew I.; Thomas, Zakir; Bourne, Philip E. (2013). "Ten simple rules for cultivating open science and collaborative R&D". PLOS Computational Biology. 9 (9): e1003244. Bibcode:2013PLSCB...9E3244M. doi:10.1371/journal.pcbi.1003244. ISSN 1553-7358. PMC 3784487. PMID 24086123.
Morgan, Maxwell Robert; Roberts, Owen Gwilym; Edwards, Aled Morgan (2018). "Ideation and implementation of an open science drug discovery business model - M4K Pharma". Wellcome Open Research. 3: 154. doi:10.12688/wellcomeopenres.14947.1. ISSN 2398-502X. PMC 6346698. PMID 30705971.
Harding, Rachel J. (January 2019). "Open notebook science can maximize impact for rare disease projects". PLOS Biology. 17 (1): e3000120. doi:10.1371/journal.pbio.3000120. ISSN 1545-7885. PMC 6366684. PMID 30689629.
Schapira, Matthieu; Harding, Rachel J. (2019-04-02). "Open laboratory notebooks: good for science, good for society, good for scientists". F1000Research. 8: 87. doi:10.12688/f1000research.17710.2. ISSN 2046-1402. PMC 6694453. PMID 31448096.
Müller, Susanne; Ackloo, Suzanne; Arrowsmith, Cheryl H.; Bauser, Marcus; Baryza, Jeremy L.; Blagg, Julian; Böttcher, Jark; Bountra, Chas; Brown, Peter J.; Bunnage, Mark E.; Carter, Adrian J. (20 April 2018). "Donated chemical probes for open science". eLife. 7. doi:10.7554/eLife.34311. ISSN 2050-084X. PMC 5910019. PMID 29676732.
Drewry, David H.; Wells, Carrow I.; Zuercher, William J.; Willson, Timothy M. (June 2019). "A Perspective on Extreme Open Science: Companies Sharing Compounds without Restriction". SLAS Discovery. 24 (5): 505–514. doi:10.1177/2472555219838210. ISSN 2472-5560. PMC 6624833. PMID 31034310.
Wells, Carrow I.; Al-Ali, Hassan; Andrews, David M.; Asquith, Christopher R. M.; Axtman, Alison D.; Dikic, Ivan; Ebner, Daniel; Ettmayer, Peter; Fischer, Christian; Frederiksen, Mathias; Futrell, Robert E. (2021-01-08). "The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification". International Journal of Molecular Sciences. 22 (2): 566. doi:10.3390/ijms22020566. ISSN 1422-0067. PMC 7826789. PMID 33429995.
Laflamme, Carl; McKeever, Paul M.; Kumar, Rahul; Schwartz, Julie; Kolahdouzan, Mahshad; Chen, Carol X.; You, Zhipeng; Benaliouad, Faiza; Gileadi, Opher; McBride, Heidi M.; Durcan, Thomas M. (15 October 2019). "Implementation of an antibody characterization procedure and application to the major ALS/FTD disease gene C9ORF72". eLife. 8. doi:10.7554/eLife.48363. ISSN 2050-084X. PMC 6794092. PMID 31612854.
Ensan, Deeba; Smil, David; Zepeda-Velázquez, Carlos A.; Panagopoulos, Dimitrios; Wong, Jong Fu; Williams, Eleanor P.; Adamson, Roslin; Bullock, Alex N.; Kiyota, Taira; Aman, Ahmed; Roberts, Owen G. (2020-05-14). "Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma". Journal of Medicinal Chemistry. 63 (9): 4978–4996. doi:10.1021/acs.jmedchem.0c00395. ISSN 1520-4804. PMC 8213057. PMID 32369358.
Gold, E. Richard (June 2021). "The fall of the innovation empire and its possible rise through open science". Research Policy. 50 (5): 104226. doi:10.1016/j.respol.2021.104226. PMC 8024784. PMID 34083844.
Jones, Molly Morgan; Chataway, Joanna (2021-03-04). "The Structural Genomics Consortium: successful organisational technology experiment or new institutional infrastructure for health research?". Technology Analysis & Strategic Management. 33 (3): 296–306. doi:10.1080/09537325.2021.1882673. ISSN 0953-7325. S2CID 232245414.
Collins, Patrick M.; Douangamath, Alice; Talon, Romain; Dias, Alexandre; Brandao-Neto, Jose; Krojer, Tobias; von Delft, Frank (2018). "Achieving a Good Crystal System for Crystallographic X-Ray Fragment Screening". Modern Approaches in Drug Discovery. Methods in Enzymology. Vol. 610. pp. 251–264. doi:10.1016/bs.mie.2018.09.027. ISBN 9780128153833. ISSN 1557-7988. PMID 30390801. S2CID 53219679.
Arrowsmith, Cheryl H.; Bountra, Chas; Fish, Paul V.; Lee, Kevin; Schapira, Matthieu (2012-04-13). "Epigenetic protein families: a new frontier for drug discovery". Nature Reviews. Drug Discovery. 11 (5): 384–400. doi:10.1038/nrd3674. ISSN 1474-1784. PMID 22498752. S2CID 5478921.
Huston, Andrea; Arrowsmith, Cheryl H.; Knapp, Stefan; Schapira, Matthieu (August 2015). "Probing the epigenome". Nature Chemical Biology. 11 (8): 542–545. doi:10.1038/nchembio.1871. ISSN 1552-4469. PMID 26196765.
César-Razquin, Adrián; Snijder, Berend; Frappier-Brinton, Tristan; Isserlin, Ruth; Gyimesi, Gergely; Bai, Xiaoyun; Reithmeier, Reinhart A.; Hepworth, David; Hediger, Matthias A.; Edwards, Aled M.; Superti-Furga, Giulio (2015-07-30). "A Call for Systematic Research on Solute Carriers". Cell. 162 (3): 478–487. doi:10.1016/j.cell.2015.07.022. ISSN 1097-4172. PMID 26232220. S2CID 15427088.
Superti-Furga, Giulio; Lackner, Daniel; Wiedmer, Tabea; Ingles-Prieto, Alvaro; Barbosa, Barbara; Girardi, Enrico; Goldmann, Ulrich; Gürtl, Bettina; Klavins, Kristaps; Klimek, Christoph; Lindinger, Sabrina (July 2020). "The RESOLUTE consortium: unlocking SLC transporters for drug discovery". Nature Reviews. Drug Discovery. 19 (7): 429–430. doi:10.1038/d41573-020-00056-6. hdl:21.11116/0000-0006-0FF1-A. ISSN 1474-1784. PMID 32265506. S2CID 215406274.
Liu, Lihua; Damerell, David R.; Koukouflis, Leonidas; Tong, Yufeng; Marsden, Brian D.; Schapira, Matthieu (15 August 2019). "UbiHub: a data hub for the explorers of ubiquitination pathways". Bioinformatics. 35 (16): 2882–2884. doi:10.1093/bioinformatics/bty1067. ISSN 1367-4811. PMC 6691330. PMID 30601939.
Schapira, Matthieu; Calabrese, Matthew F.; Bullock, Alex N.; Crews, Craig M. (December 2019). "Targeted protein degradation: expanding the toolbox". Nature Reviews. Drug Discovery. 18 (12): 949–963. doi:10.1038/s41573-019-0047-y. ISSN 1474-1784. PMID 31666732. S2CID 204942300.
Harding, Rachel J.; Ferreira de Freitas, Renato; Collins, Patrick; Franzoni, Ivan; Ravichandran, Mani; Ouyang, Hui; Juarez-Ornelas, Kevin A.; Lautens, Mark; Schapira, Matthieu; von Delft, Frank; Santhakumar, Vjayaratnam (9 November 2017). "Small Molecule Antagonists of the Interaction between the Histone Deacetylase 6 Zinc-Finger Domain and Ubiquitin". Journal of Medicinal Chemistry. 60 (21): 9090–9096. doi:10.1021/acs.jmedchem.7b00933. ISSN 1520-4804. PMID 29019676.
Ferreira de Freitas, Renato; Harding, Rachel J.; Franzoni, Ivan; Ravichandran, Mani; Mann, Mandeep K.; Ouyang, Hui; Lautens, Mark; Santhakumar, Vijayaratnam; Arrowsmith, Cheryl H.; Schapira, Matthieu (24 May 2018). "Identification and Structure-Activity Relationship of HDAC6 Zinc-Finger Ubiquitin Binding Domain Inhibitors". Journal of Medicinal Chemistry. 61 (10): 4517–4527. doi:10.1021/acs.jmedchem.8b00258. ISSN 1520-4804. PMID 29741882.
Mann, Mandeep K.; Franzoni, Ivan; de Freitas, Renato Ferreira; Tempel, Wolfram; Houliston, Scott; Smith, Leanna; Vedadi, Masoud; Arrowsmith, Cheryl H.; Harding, Rachel J.; Schapira, Matthieu (27 November 2019). "Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain" (PDF). Journal of Medicinal Chemistry. 62 (22): 10144–10155. doi:10.1021/acs.jmedchem.9b00988. ISSN 1520-4804. PMID 31663737. S2CID 204975079.
Knapp, Stefan; Arruda, Paulo; Blagg, Julian; Burley, Stephen; Drewry, David H.; Edwards, Aled; Fabbro, Doriano; Gillespie, Paul; Gray, Nathanael S.; Kuster, Bernhard; Lackey, Karen E. (January 2013). "A public-private partnership to unlock the untargeted kinome". Nature Chemical Biology. 9 (1): 3–6. doi:10.1038/nchembio.1113. ISSN 1552-4469. PMID 23238671.
Drewry, David H.; Wells, Carrow I.; Andrews, David M.; Angell, Richard; Al-Ali, Hassan; Axtman, Alison D.; Capuzzi, Stephen J.; Elkins, Jonathan M.; Ettmayer, Peter; Frederiksen, Mathias; Gileadi, Opher (2017). "Progress towards a public chemogenomic set for protein kinases and a call for contributions". PLOS ONE. 12 (8): e0181585. Bibcode:2017PLoSO..1281585D. doi:10.1371/journal.pone.0181585. ISSN 1932-6203. PMC 5540273. PMID 28767711.
Wu, Qin; Heidenreich, David; Zhou, Stanley; Ackloo, Suzanne; Krämer, Andreas; Nakka, Kiran; Lima-Fernandes, Evelyne; Deblois, Genevieve; Duan, Shili; Vellanki, Ravi N.; Li, Fengling (23 April 2019). "A chemical toolbox for the study of bromodomains and epigenetic signaling". Nature Communications. 10 (1): 1915. Bibcode:2019NatCo..10.1915W. doi:10.1038/s41467-019-09672-2. ISSN 2041-1723. PMC 6478789. PMID 31015424.
Scheer, Sebastian; Ackloo, Suzanne; Medina, Tiago S.; Schapira, Matthieu; Li, Fengling; Ward, Jennifer A.; Lewis, Andrew M.; Northrop, Jeffrey P.; Richardson, Paul L.; Kaniskan, H. Ümit; Shen, Yudao (3 January 2019). "A chemical biology toolbox to study protein methyltransferases and epigenetic signaling". Nature Communications. 10 (1): 19. Bibcode:2019NatCo..10...19S. doi:10.1038/s41467-018-07905-4. ISSN 2041-1723. PMC 6318333. PMID 30604761.
Frye, Stephen V. (March 2010). "The art of the chemical probe". Nature Chemical Biology. 6 (3): 159–161. doi:10.1038/nchembio.296. ISSN 1552-4469. PMID 20154659.
Arrowsmith, Cheryl H.; Audia, James E.; Austin, Christopher; Baell, Jonathan; Bennett, Jonathan; Blagg, Julian; Bountra, Chas; Brennan, Paul E.; Brown, Peter J.; Bunnage, Mark E.; Buser-Doepner, Carolyn (August 2015). "The promise and peril of chemical probes". Nature Chemical Biology. 11 (8): 536–541. doi:10.1038/nchembio.1867. ISSN 1552-4469. PMC 4706458. PMID 26196764.
Blagg, Julian; Workman, Paul (14 August 2017). "Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology". Cancer Cell. 32 (2): 268–270. doi:10.1016/j.ccell.2017.07.010. ISSN 1878-3686. PMC 5559281. PMID 28810148.
Antolin, Albert A.; Tym, Joseph E.; Komianou, Angeliki; Collins, Ian; Workman, Paul; Al-Lazikani, Bissan (15 February 2018). "Objective, Quantitative, Data-Driven Assessment of Chemical Probes". Cell Chemical Biology. 25 (2): 194–205.e5. doi:10.1016/j.chembiol.2017.11.004. ISSN 2451-9448. PMC 5814752. PMID 29249694.
Antolin, Albert A.; Workman, Paul; Al-Lazikani, Bissan (2019-11-28). "Public resources for chemical probes: the journey so far and the road ahead". Future Medicinal Chemistry. 13 (8): 731–747. doi:10.4155/fmc-2019-0231. ISSN 1756-8927. PMID 31778323.
Picaud, Sarah; Da Costa, David; Thanasopoulou, Angeliki; Filippakopoulos, Panagis; Fish, Paul V.; Philpott, Martin; Fedorov, Oleg; Brennan, Paul; Bunnage, Mark E.; Owen, Dafydd R.; Bradner, James E. (2013-06-01). "PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains". Cancer Research. 73 (11): 3336–3346. doi:10.1158/0008-5472.CAN-12-3292. ISSN 1538-7445. PMC 3673830. PMID 23576556.
Filippakopoulos, Panagis; Qi, Jun; Picaud, Sarah; Shen, Yao; Smith, William B.; Fedorov, Oleg; Morse, Elizabeth M.; Keates, Tracey; Hickman, Tyler T.; Felletar, Ildiko; Philpott, Martin (2010-12-23). "Selective inhibition of BET bromodomains". Nature. 468 (7327): 1067–1073. Bibcode:2010Natur.468.1067F. doi:10.1038/nature09504. ISSN 1476-4687. PMC 3010259. PMID 20871596.
Liu, Feng; Barsyte-Lovejoy, Dalia; Li, Fengling; Xiong, Yan; Korboukh, Victoria; Huang, Xi-Ping; Allali-Hassani, Abdellah; Janzen, William P.; Roth, Bryan L.; Frye, Stephen V.; Arrowsmith, Cheryl H. (2013-11-14). "Discovery of an in vivo chemical probe of the lysine methyltransferases G9a and GLP". Journal of Medicinal Chemistry. 56 (21): 8931–8942. doi:10.1021/jm401480r. ISSN 1520-4804. PMC 3880643. PMID 24102134.
Konze, Kyle D.; Ma, Anqi; Li, Fengling; Barsyte-Lovejoy, Dalia; Parton, Trevor; Macnevin, Christopher J.; Liu, Feng; Gao, Cen; Huang, Xi-Ping; Kuznetsova, Ekaterina; Rougie, Marie (2013). "An orally bioavailable chemical probe of the Lysine Methyltransferases EZH2 and EZH1". ACS Chemical Biology. 8 (6): 1324–1334. doi:10.1021/cb400133j. ISSN 1554-8937. PMC 3773059. PMID 23614352.
Bonday, Zahid Q.; Cortez, Guillermo S.; Grogan, Michael J.; Antonysamy, Stephen; Weichert, Ken; Bocchinfuso, Wayne P.; Li, Fengling; Kennedy, Steven; Li, Binghui; Mader, Mary M.; Arrowsmith, Cheryl H. (2018-04-23). "LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity". ACS Medicinal Chemistry Letters. 9 (7): 612–617. doi:10.1021/acsmedchemlett.8b00014. ISSN 1948-5875. PMC 6047023. PMID 30034588.
Duncan, Kenneth W.; Rioux, Nathalie; Boriack-Sjodin, P. Ann; Munchhof, Michael J.; Reiter, Lawrence A.; Majer, Christina R.; Jin, Lei; Johnston, L. Danielle; Chan-Penebre, Elayne; Kuplast, Kristy G.; Porter Scott, Margaret (2016-02-11). "Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666". ACS Medicinal Chemistry Letters. 7 (2): 162–166. doi:10.1021/acsmedchemlett.5b00380. ISSN 1948-5875. PMC 4753547. PMID 26985292.
Grebien, Florian; Vedadi, Masoud; Getlik, Matthäus; Giambruno, Roberto; Grover, Amit; Avellino, Roberto; Skucha, Anna; Vittori, Sarah; Kuznetsova, Ekaterina; Smil, David; Barsyte-Lovejoy, Dalia (August 2015). "Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia". Nature Chemical Biology. 11 (8): 571–578. doi:10.1038/nchembio.1859. ISSN 1552-4469. PMC 4511833. PMID 26167872.
Roskoski, Robert (June 2019). "Properties of FDA-approved small molecule protein kinase inhibitors". Pharmacological Research. 144: 19–50. doi:10.1016/j.phrs.2019.03.006. ISSN 1096-1186. PMID 30877063. S2CID 80625382.
Wilson, LJ; et, al. (2018). "New Perspectives, Opportunitiess, and Challenges in Exploring the Human Protein Kinome". Cancer Research. 78 (1): 15–29. doi:10.1158/0008-5472.CAN-17-2291. PMID 29254998.
Sorget, Nienke; et, al (2020). "Exploring the understudied human kinome for research and therapeutic opportunities" (PDF). www.biorxiv.org. doi:10.1101/2020.04.02.022277. S2CID 215404186.
Buljan, M; et, al. (2020). "Kinase Interaction Network Expands Functional and Disease Roles of Human Kinases". Molecular Cell. 79 (3): 504–520.e9. doi:10.1016/j.molcel.2020.07.001. PMC 7427327. PMID 32707033. S2CID 220746851.
Edwards, Aled M.; Arrowsmith, Cheryl H.; Bountra, Chas; Bunnage, Mark E.; Feldmann, Marc; Knight, Julian C.; Patel, Dhavalkumar D.; Prinos, Panagiotis; Taylor, Michael D.; Sundström, Michael; SGC Open Source Target-Discovery Partnership (March 2015). "Preclinical target validation using patient-derived cells". Nature Reviews. Drug Discovery. 14 (3): 149–150. doi:10.1038/nrd4565. ISSN 1474-1784. PMID 25722227. S2CID 2423838.
Hoag, Hannah (2009). "Richard Gold". Nature Biotechnology. 27 (5): 409. doi:10.1038/nbt0509-409. ISSN 1546-1696. PMID 19430435. S2CID 34394262.
Edwards, Aled; Morgan, Max; Al Chawaf, Arij; Andrusiak, Kerry; Charney, Rachel; Cynader, Zarya; ElDessouki, Ahmed; Lee, Yunjeong; Moeser, Andrew; Stern, Simon; Zuercher, William J. (31 May 2017). "A trust approach for sharing research reagents". Science Translational Medicine. 9 (392): eaai9055. doi:10.1126/scitranslmed.aai9055. ISSN 1946-6242. PMID 28566431. S2CID 4020927.
Vedadi, Masoud; Lew, Jocelyne; Artz, Jennifer; Amani, Mehrnaz; Zhao, Yong; Dong, Aiping; Wasney, Gregory A.; Gao, Mian; Hills, Tanya; Brokx, Stephen; Qiu, Wei (January 2007). "Genome-scale protein expression and structural biology of Plasmodium falciparum and related Apicomplexan organisms". Molecular and Biochemical Parasitology. 151 (1): 100–110. doi:10.1016/j.molbiopara.2006.10.011. ISSN 0166-6851. PMID 17125854.
Frye, Stephen V.; Arkin, Michelle R.; Arrowsmith, Cheryl H.; Conn, P. Jeffrey; Glicksman, Marcie A.; Hull-Ryde, Emily A.; Slusher, Barbara S. (November 2015). "Tackling reproducibility in academic preclinical drug discovery". Nature Reviews. Drug Discovery. 14 (11): 733–734. doi:10.1038/nrd4737. ISSN 1474-1784. PMID 26388229. S2CID 205478934.
Marcon, Edyta; Jain, Harshika; Bhattacharya, Anandi; Guo, Hongbo; Phanse, Sadhna; Pu, Shuye; Byram, Gregory; Collins, Ben C.; Dowdell, Evan; Fenner, Maria; Guo, Xinghua (August 2015). "Assessment of a method to characterize antibody selectivity and specificity for use in immunoprecipitation". Nature Methods. 12 (8): 725–731. doi:10.1038/nmeth.3472. ISSN 1548-7105. PMID 26121405. S2CID 205423964.
Gruetter, Markus (2012). "Open collaboration is key to new drugs". Nature. 491 (7422): 40. doi:10.1038/491040d. ISSN 0028-0836. PMID 23128216. S2CID 205074791.
Carter, Adrian J.; Kraemer, Oliver; Zwick, Matthias; Mueller-Fahrnow, Anke; Arrowsmith, Cheryl H.; Edwards, Aled M. (November 2019). "Target 2035: probing the human proteome". Drug Discovery Today. 24 (11): 2111–2115. doi:10.1016/j.drudis.2019.06.020. ISSN 1878-5832. PMID 31278990.
Schapira, Matthieu; Tyers, Mike; Torrent, Maricel; Arrowsmith, Cheryl H. (November 2017). "WD40 repeat domain proteins: a novel target class?". Nature Reviews. Drug Discovery. 16 (11): 773–786. doi:10.1038/nrd.2017.179. ISSN 1474-1784. PMC 5975957. PMID 29026209.
Song, Richard; Wang, Zhong-Duo; Schapira, Matthieu (6 October 2017). "Disease Association and Druggability of WD40 Repeat Proteins". Journal of Proteome Research. 16 (10): 3766–3773. doi:10.1021/acs.jproteome.7b00451. ISSN 1535-3907. PMID 28956604.
Wang, Jiayan; Yazdani, Setayesh; Han, Ana; Schapira, Matthieu (March 2020). "Structure-based view of the druggable genome". Drug Discovery Today. 25 (3): 561–567. doi:10.1016/j.drudis.2020.02.006. ISSN 1878-5832. PMID 32084498. S2CID 211246313.
Wacker, Daniel; Stevens, Raymond C.; Roth, Bryan L. (2017-07-27). "How Ligands Illuminate GPCR Molecular Pharmacology". Cell. 170 (3): 414–427. doi:10.1016/j.cell.2017.07.009. ISSN 1097-4172. PMC 5560499. PMID 28753422.
Roth, Bryan L.; Irwin, John J.; Shoichet, Brian K. (November 2017). "Discovery of new GPCR ligands to illuminate new biology". Nature Chemical Biology. 13 (11): 1143–1151. doi:10.1038/nchembio.2490. ISSN 1552-4469. PMC 5835362. PMID 29045379.
Roth, Bryan L. (August 2019). "How structure informs and transforms chemogenetics". Current Opinion in Structural Biology. 57: 9–16. doi:10.1016/j.sbi.2019.01.016. ISSN 1879-033X. PMID 30818201. S2CID 73479428.
Edwards, Aled (2016-03-17). "Reproducibility: Team up with industry". Nature. 531 (7594): 299–301. Bibcode:2016Natur.531..299E. doi:10.1038/531299a. ISSN 1476-4687. PMID 26983524. S2CID 4467772.

handle.net

hdl.handle.net

Superti-Furga, Giulio; Lackner, Daniel; Wiedmer, Tabea; Ingles-Prieto, Alvaro; Barbosa, Barbara; Girardi, Enrico; Goldmann, Ulrich; Gürtl, Bettina; Klavins, Kristaps; Klimek, Christoph; Lindinger, Sabrina (July 2020). "The RESOLUTE consortium: unlocking SLC transporters for drug discovery". Nature Reviews. Drug Discovery. 19 (7): 429–430. doi:10.1038/d41573-020-00056-6. hdl:21.11116/0000-0006-0FF1-A. ISSN 1474-1784. PMID 32265506. S2CID 215406274.

harvard.edu

ui.adsabs.harvard.edu

Edwards, AM; et, al. (2011). "Too many roads not taken". Nature. 470 (2333): 163–165. arXiv:1102.0448. Bibcode:2011Natur.470..163E. doi:10.1038/470163a. PMID 21307913. S2CID 4429387.
Masum, Hassan; Rao, Aarthi; Good, Benjamin M.; Todd, Matthew H.; Edwards, Aled M.; Chan, Leslie; Bunin, Barry A.; Su, Andrew I.; Thomas, Zakir; Bourne, Philip E. (2013). "Ten simple rules for cultivating open science and collaborative R&D". PLOS Computational Biology. 9 (9): e1003244. Bibcode:2013PLSCB...9E3244M. doi:10.1371/journal.pcbi.1003244. ISSN 1553-7358. PMC 3784487. PMID 24086123.
Drewry, David H.; Wells, Carrow I.; Andrews, David M.; Angell, Richard; Al-Ali, Hassan; Axtman, Alison D.; Capuzzi, Stephen J.; Elkins, Jonathan M.; Ettmayer, Peter; Frederiksen, Mathias; Gileadi, Opher (2017). "Progress towards a public chemogenomic set for protein kinases and a call for contributions". PLOS ONE. 12 (8): e0181585. Bibcode:2017PLoSO..1281585D. doi:10.1371/journal.pone.0181585. ISSN 1932-6203. PMC 5540273. PMID 28767711.
Wu, Qin; Heidenreich, David; Zhou, Stanley; Ackloo, Suzanne; Krämer, Andreas; Nakka, Kiran; Lima-Fernandes, Evelyne; Deblois, Genevieve; Duan, Shili; Vellanki, Ravi N.; Li, Fengling (23 April 2019). "A chemical toolbox for the study of bromodomains and epigenetic signaling". Nature Communications. 10 (1): 1915. Bibcode:2019NatCo..10.1915W. doi:10.1038/s41467-019-09672-2. ISSN 2041-1723. PMC 6478789. PMID 31015424.
Scheer, Sebastian; Ackloo, Suzanne; Medina, Tiago S.; Schapira, Matthieu; Li, Fengling; Ward, Jennifer A.; Lewis, Andrew M.; Northrop, Jeffrey P.; Richardson, Paul L.; Kaniskan, H. Ümit; Shen, Yudao (3 January 2019). "A chemical biology toolbox to study protein methyltransferases and epigenetic signaling". Nature Communications. 10 (1): 19. Bibcode:2019NatCo..10...19S. doi:10.1038/s41467-018-07905-4. ISSN 2041-1723. PMC 6318333. PMID 30604761.
Filippakopoulos, Panagis; Qi, Jun; Picaud, Sarah; Shen, Yao; Smith, William B.; Fedorov, Oleg; Morse, Elizabeth M.; Keates, Tracey; Hickman, Tyler T.; Felletar, Ildiko; Philpott, Martin (2010-12-23). "Selective inhibition of BET bromodomains". Nature. 468 (7327): 1067–1073. Bibcode:2010Natur.468.1067F. doi:10.1038/nature09504. ISSN 1476-4687. PMC 3010259. PMID 20871596.
Edwards, Aled (2016-03-17). "Reproducibility: Team up with industry". Nature. 531 (7594): 299–301. Bibcode:2016Natur.531..299E. doi:10.1038/531299a. ISSN 1476-4687. PMID 26983524. S2CID 4467772.

nature.com

blogs.nature.com

Harding, Rachel (19 October 2016). "An Open Approach to Huntington's Disease Research". nature blogs.

nih.gov

pubmed.ncbi.nlm.nih.gov

Williamson, AR (2000). "Creating a structural genomics consortium". Nature Structural Biology. 7: 953. doi:10.1038/80726. PMID 11103997. S2CID 35185565.
Edwards, AM; et, al. (2011). "Too many roads not taken". Nature. 470 (2333): 163–165. arXiv:1102.0448. Bibcode:2011Natur.470..163E. doi:10.1038/470163a. PMID 21307913. S2CID 4429387.
Davis, Andrew M.; Engkvist, Ola; Fairclough, Rebecca J.; Feierberg, Isabella; Freeman, Adrian; Iyer, Preeti (2021-02-13). "Public-Private Partnerships: Compound and Data Sharing in Drug Discovery and Development". SLAS Discovery. 26 (5): 604–619. doi:10.1177/2472555220982268. ISSN 2472-5552. PMID 33586501. S2CID 231928371.
Edwards, Aled (September 2008). "Open-source science to enable drug discovery". Drug Discovery Today. 13 (17–18): 731–733. doi:10.1016/j.drudis.2008.04.011. ISSN 1359-6446. PMID 18790412.
Edwards, Aled M.; Bountra, Chas; Kerr, David J.; Willson, Timothy M. (July 2009). "Open access chemical and clinical probes to support drug discovery". Nature Chemical Biology. 5 (7): 436–440. doi:10.1038/nchembio0709-436. ISSN 1552-4469. PMID 19536100.
Masum, Hassan; Rao, Aarthi; Good, Benjamin M.; Todd, Matthew H.; Edwards, Aled M.; Chan, Leslie; Bunin, Barry A.; Su, Andrew I.; Thomas, Zakir; Bourne, Philip E. (2013). "Ten simple rules for cultivating open science and collaborative R&D". PLOS Computational Biology. 9 (9): e1003244. Bibcode:2013PLSCB...9E3244M. doi:10.1371/journal.pcbi.1003244. ISSN 1553-7358. PMC 3784487. PMID 24086123.
Morgan, Maxwell Robert; Roberts, Owen Gwilym; Edwards, Aled Morgan (2018). "Ideation and implementation of an open science drug discovery business model - M4K Pharma". Wellcome Open Research. 3: 154. doi:10.12688/wellcomeopenres.14947.1. ISSN 2398-502X. PMC 6346698. PMID 30705971.
Harding, Rachel J. (January 2019). "Open notebook science can maximize impact for rare disease projects". PLOS Biology. 17 (1): e3000120. doi:10.1371/journal.pbio.3000120. ISSN 1545-7885. PMC 6366684. PMID 30689629.
Schapira, Matthieu; Harding, Rachel J. (2019-04-02). "Open laboratory notebooks: good for science, good for society, good for scientists". F1000Research. 8: 87. doi:10.12688/f1000research.17710.2. ISSN 2046-1402. PMC 6694453. PMID 31448096.
Müller, Susanne; Ackloo, Suzanne; Arrowsmith, Cheryl H.; Bauser, Marcus; Baryza, Jeremy L.; Blagg, Julian; Böttcher, Jark; Bountra, Chas; Brown, Peter J.; Bunnage, Mark E.; Carter, Adrian J. (20 April 2018). "Donated chemical probes for open science". eLife. 7. doi:10.7554/eLife.34311. ISSN 2050-084X. PMC 5910019. PMID 29676732.
Drewry, David H.; Wells, Carrow I.; Zuercher, William J.; Willson, Timothy M. (June 2019). "A Perspective on Extreme Open Science: Companies Sharing Compounds without Restriction". SLAS Discovery. 24 (5): 505–514. doi:10.1177/2472555219838210. ISSN 2472-5560. PMC 6624833. PMID 31034310.
Wells, Carrow I.; Al-Ali, Hassan; Andrews, David M.; Asquith, Christopher R. M.; Axtman, Alison D.; Dikic, Ivan; Ebner, Daniel; Ettmayer, Peter; Fischer, Christian; Frederiksen, Mathias; Futrell, Robert E. (2021-01-08). "The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification". International Journal of Molecular Sciences. 22 (2): 566. doi:10.3390/ijms22020566. ISSN 1422-0067. PMC 7826789. PMID 33429995.
Laflamme, Carl; McKeever, Paul M.; Kumar, Rahul; Schwartz, Julie; Kolahdouzan, Mahshad; Chen, Carol X.; You, Zhipeng; Benaliouad, Faiza; Gileadi, Opher; McBride, Heidi M.; Durcan, Thomas M. (15 October 2019). "Implementation of an antibody characterization procedure and application to the major ALS/FTD disease gene C9ORF72". eLife. 8. doi:10.7554/eLife.48363. ISSN 2050-084X. PMC 6794092. PMID 31612854.
Ensan, Deeba; Smil, David; Zepeda-Velázquez, Carlos A.; Panagopoulos, Dimitrios; Wong, Jong Fu; Williams, Eleanor P.; Adamson, Roslin; Bullock, Alex N.; Kiyota, Taira; Aman, Ahmed; Roberts, Owen G. (2020-05-14). "Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma". Journal of Medicinal Chemistry. 63 (9): 4978–4996. doi:10.1021/acs.jmedchem.0c00395. ISSN 1520-4804. PMC 8213057. PMID 32369358.
Gold, E. Richard (June 2021). "The fall of the innovation empire and its possible rise through open science". Research Policy. 50 (5): 104226. doi:10.1016/j.respol.2021.104226. PMC 8024784. PMID 34083844.
Collins, Patrick M.; Douangamath, Alice; Talon, Romain; Dias, Alexandre; Brandao-Neto, Jose; Krojer, Tobias; von Delft, Frank (2018). "Achieving a Good Crystal System for Crystallographic X-Ray Fragment Screening". Modern Approaches in Drug Discovery. Methods in Enzymology. Vol. 610. pp. 251–264. doi:10.1016/bs.mie.2018.09.027. ISBN 9780128153833. ISSN 1557-7988. PMID 30390801. S2CID 53219679.
Arrowsmith, Cheryl H.; Bountra, Chas; Fish, Paul V.; Lee, Kevin; Schapira, Matthieu (2012-04-13). "Epigenetic protein families: a new frontier for drug discovery". Nature Reviews. Drug Discovery. 11 (5): 384–400. doi:10.1038/nrd3674. ISSN 1474-1784. PMID 22498752. S2CID 5478921.
Huston, Andrea; Arrowsmith, Cheryl H.; Knapp, Stefan; Schapira, Matthieu (August 2015). "Probing the epigenome". Nature Chemical Biology. 11 (8): 542–545. doi:10.1038/nchembio.1871. ISSN 1552-4469. PMID 26196765.
César-Razquin, Adrián; Snijder, Berend; Frappier-Brinton, Tristan; Isserlin, Ruth; Gyimesi, Gergely; Bai, Xiaoyun; Reithmeier, Reinhart A.; Hepworth, David; Hediger, Matthias A.; Edwards, Aled M.; Superti-Furga, Giulio (2015-07-30). "A Call for Systematic Research on Solute Carriers". Cell. 162 (3): 478–487. doi:10.1016/j.cell.2015.07.022. ISSN 1097-4172. PMID 26232220. S2CID 15427088.
Superti-Furga, Giulio; Lackner, Daniel; Wiedmer, Tabea; Ingles-Prieto, Alvaro; Barbosa, Barbara; Girardi, Enrico; Goldmann, Ulrich; Gürtl, Bettina; Klavins, Kristaps; Klimek, Christoph; Lindinger, Sabrina (July 2020). "The RESOLUTE consortium: unlocking SLC transporters for drug discovery". Nature Reviews. Drug Discovery. 19 (7): 429–430. doi:10.1038/d41573-020-00056-6. hdl:21.11116/0000-0006-0FF1-A. ISSN 1474-1784. PMID 32265506. S2CID 215406274.
Liu, Lihua; Damerell, David R.; Koukouflis, Leonidas; Tong, Yufeng; Marsden, Brian D.; Schapira, Matthieu (15 August 2019). "UbiHub: a data hub for the explorers of ubiquitination pathways". Bioinformatics. 35 (16): 2882–2884. doi:10.1093/bioinformatics/bty1067. ISSN 1367-4811. PMC 6691330. PMID 30601939.
Schapira, Matthieu; Calabrese, Matthew F.; Bullock, Alex N.; Crews, Craig M. (December 2019). "Targeted protein degradation: expanding the toolbox". Nature Reviews. Drug Discovery. 18 (12): 949–963. doi:10.1038/s41573-019-0047-y. ISSN 1474-1784. PMID 31666732. S2CID 204942300.
Harding, Rachel J.; Ferreira de Freitas, Renato; Collins, Patrick; Franzoni, Ivan; Ravichandran, Mani; Ouyang, Hui; Juarez-Ornelas, Kevin A.; Lautens, Mark; Schapira, Matthieu; von Delft, Frank; Santhakumar, Vjayaratnam (9 November 2017). "Small Molecule Antagonists of the Interaction between the Histone Deacetylase 6 Zinc-Finger Domain and Ubiquitin". Journal of Medicinal Chemistry. 60 (21): 9090–9096. doi:10.1021/acs.jmedchem.7b00933. ISSN 1520-4804. PMID 29019676.
Ferreira de Freitas, Renato; Harding, Rachel J.; Franzoni, Ivan; Ravichandran, Mani; Mann, Mandeep K.; Ouyang, Hui; Lautens, Mark; Santhakumar, Vijayaratnam; Arrowsmith, Cheryl H.; Schapira, Matthieu (24 May 2018). "Identification and Structure-Activity Relationship of HDAC6 Zinc-Finger Ubiquitin Binding Domain Inhibitors". Journal of Medicinal Chemistry. 61 (10): 4517–4527. doi:10.1021/acs.jmedchem.8b00258. ISSN 1520-4804. PMID 29741882.
Mann, Mandeep K.; Franzoni, Ivan; de Freitas, Renato Ferreira; Tempel, Wolfram; Houliston, Scott; Smith, Leanna; Vedadi, Masoud; Arrowsmith, Cheryl H.; Harding, Rachel J.; Schapira, Matthieu (27 November 2019). "Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain" (PDF). Journal of Medicinal Chemistry. 62 (22): 10144–10155. doi:10.1021/acs.jmedchem.9b00988. ISSN 1520-4804. PMID 31663737. S2CID 204975079.
Knapp, Stefan; Arruda, Paulo; Blagg, Julian; Burley, Stephen; Drewry, David H.; Edwards, Aled; Fabbro, Doriano; Gillespie, Paul; Gray, Nathanael S.; Kuster, Bernhard; Lackey, Karen E. (January 2013). "A public-private partnership to unlock the untargeted kinome". Nature Chemical Biology. 9 (1): 3–6. doi:10.1038/nchembio.1113. ISSN 1552-4469. PMID 23238671.
Drewry, David H.; Wells, Carrow I.; Andrews, David M.; Angell, Richard; Al-Ali, Hassan; Axtman, Alison D.; Capuzzi, Stephen J.; Elkins, Jonathan M.; Ettmayer, Peter; Frederiksen, Mathias; Gileadi, Opher (2017). "Progress towards a public chemogenomic set for protein kinases and a call for contributions". PLOS ONE. 12 (8): e0181585. Bibcode:2017PLoSO..1281585D. doi:10.1371/journal.pone.0181585. ISSN 1932-6203. PMC 5540273. PMID 28767711.
Wu, Qin; Heidenreich, David; Zhou, Stanley; Ackloo, Suzanne; Krämer, Andreas; Nakka, Kiran; Lima-Fernandes, Evelyne; Deblois, Genevieve; Duan, Shili; Vellanki, Ravi N.; Li, Fengling (23 April 2019). "A chemical toolbox for the study of bromodomains and epigenetic signaling". Nature Communications. 10 (1): 1915. Bibcode:2019NatCo..10.1915W. doi:10.1038/s41467-019-09672-2. ISSN 2041-1723. PMC 6478789. PMID 31015424.
Scheer, Sebastian; Ackloo, Suzanne; Medina, Tiago S.; Schapira, Matthieu; Li, Fengling; Ward, Jennifer A.; Lewis, Andrew M.; Northrop, Jeffrey P.; Richardson, Paul L.; Kaniskan, H. Ümit; Shen, Yudao (3 January 2019). "A chemical biology toolbox to study protein methyltransferases and epigenetic signaling". Nature Communications. 10 (1): 19. Bibcode:2019NatCo..10...19S. doi:10.1038/s41467-018-07905-4. ISSN 2041-1723. PMC 6318333. PMID 30604761.
Frye, Stephen V. (March 2010). "The art of the chemical probe". Nature Chemical Biology. 6 (3): 159–161. doi:10.1038/nchembio.296. ISSN 1552-4469. PMID 20154659.
Arrowsmith, Cheryl H.; Audia, James E.; Austin, Christopher; Baell, Jonathan; Bennett, Jonathan; Blagg, Julian; Bountra, Chas; Brennan, Paul E.; Brown, Peter J.; Bunnage, Mark E.; Buser-Doepner, Carolyn (August 2015). "The promise and peril of chemical probes". Nature Chemical Biology. 11 (8): 536–541. doi:10.1038/nchembio.1867. ISSN 1552-4469. PMC 4706458. PMID 26196764.
Blagg, Julian; Workman, Paul (14 August 2017). "Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology". Cancer Cell. 32 (2): 268–270. doi:10.1016/j.ccell.2017.07.010. ISSN 1878-3686. PMC 5559281. PMID 28810148.
Antolin, Albert A.; Tym, Joseph E.; Komianou, Angeliki; Collins, Ian; Workman, Paul; Al-Lazikani, Bissan (15 February 2018). "Objective, Quantitative, Data-Driven Assessment of Chemical Probes". Cell Chemical Biology. 25 (2): 194–205.e5. doi:10.1016/j.chembiol.2017.11.004. ISSN 2451-9448. PMC 5814752. PMID 29249694.
Antolin, Albert A.; Workman, Paul; Al-Lazikani, Bissan (2019-11-28). "Public resources for chemical probes: the journey so far and the road ahead". Future Medicinal Chemistry. 13 (8): 731–747. doi:10.4155/fmc-2019-0231. ISSN 1756-8927. PMID 31778323.
Picaud, Sarah; Da Costa, David; Thanasopoulou, Angeliki; Filippakopoulos, Panagis; Fish, Paul V.; Philpott, Martin; Fedorov, Oleg; Brennan, Paul; Bunnage, Mark E.; Owen, Dafydd R.; Bradner, James E. (2013-06-01). "PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains". Cancer Research. 73 (11): 3336–3346. doi:10.1158/0008-5472.CAN-12-3292. ISSN 1538-7445. PMC 3673830. PMID 23576556.
Filippakopoulos, Panagis; Qi, Jun; Picaud, Sarah; Shen, Yao; Smith, William B.; Fedorov, Oleg; Morse, Elizabeth M.; Keates, Tracey; Hickman, Tyler T.; Felletar, Ildiko; Philpott, Martin (2010-12-23). "Selective inhibition of BET bromodomains". Nature. 468 (7327): 1067–1073. Bibcode:2010Natur.468.1067F. doi:10.1038/nature09504. ISSN 1476-4687. PMC 3010259. PMID 20871596.
Liu, Feng; Barsyte-Lovejoy, Dalia; Li, Fengling; Xiong, Yan; Korboukh, Victoria; Huang, Xi-Ping; Allali-Hassani, Abdellah; Janzen, William P.; Roth, Bryan L.; Frye, Stephen V.; Arrowsmith, Cheryl H. (2013-11-14). "Discovery of an in vivo chemical probe of the lysine methyltransferases G9a and GLP". Journal of Medicinal Chemistry. 56 (21): 8931–8942. doi:10.1021/jm401480r. ISSN 1520-4804. PMC 3880643. PMID 24102134.
Konze, Kyle D.; Ma, Anqi; Li, Fengling; Barsyte-Lovejoy, Dalia; Parton, Trevor; Macnevin, Christopher J.; Liu, Feng; Gao, Cen; Huang, Xi-Ping; Kuznetsova, Ekaterina; Rougie, Marie (2013). "An orally bioavailable chemical probe of the Lysine Methyltransferases EZH2 and EZH1". ACS Chemical Biology. 8 (6): 1324–1334. doi:10.1021/cb400133j. ISSN 1554-8937. PMC 3773059. PMID 23614352.
Bonday, Zahid Q.; Cortez, Guillermo S.; Grogan, Michael J.; Antonysamy, Stephen; Weichert, Ken; Bocchinfuso, Wayne P.; Li, Fengling; Kennedy, Steven; Li, Binghui; Mader, Mary M.; Arrowsmith, Cheryl H. (2018-04-23). "LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity". ACS Medicinal Chemistry Letters. 9 (7): 612–617. doi:10.1021/acsmedchemlett.8b00014. ISSN 1948-5875. PMC 6047023. PMID 30034588.
Duncan, Kenneth W.; Rioux, Nathalie; Boriack-Sjodin, P. Ann; Munchhof, Michael J.; Reiter, Lawrence A.; Majer, Christina R.; Jin, Lei; Johnston, L. Danielle; Chan-Penebre, Elayne; Kuplast, Kristy G.; Porter Scott, Margaret (2016-02-11). "Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666". ACS Medicinal Chemistry Letters. 7 (2): 162–166. doi:10.1021/acsmedchemlett.5b00380. ISSN 1948-5875. PMC 4753547. PMID 26985292.
Grebien, Florian; Vedadi, Masoud; Getlik, Matthäus; Giambruno, Roberto; Grover, Amit; Avellino, Roberto; Skucha, Anna; Vittori, Sarah; Kuznetsova, Ekaterina; Smil, David; Barsyte-Lovejoy, Dalia (August 2015). "Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia". Nature Chemical Biology. 11 (8): 571–578. doi:10.1038/nchembio.1859. ISSN 1552-4469. PMC 4511833. PMID 26167872.
Roskoski, Robert (June 2019). "Properties of FDA-approved small molecule protein kinase inhibitors". Pharmacological Research. 144: 19–50. doi:10.1016/j.phrs.2019.03.006. ISSN 1096-1186. PMID 30877063. S2CID 80625382.
Wilson, LJ; et, al. (2018). "New Perspectives, Opportunitiess, and Challenges in Exploring the Human Protein Kinome". Cancer Research. 78 (1): 15–29. doi:10.1158/0008-5472.CAN-17-2291. PMID 29254998.
Buljan, M; et, al. (2020). "Kinase Interaction Network Expands Functional and Disease Roles of Human Kinases". Molecular Cell. 79 (3): 504–520.e9. doi:10.1016/j.molcel.2020.07.001. PMC 7427327. PMID 32707033. S2CID 220746851.
Edwards, Aled M.; Arrowsmith, Cheryl H.; Bountra, Chas; Bunnage, Mark E.; Feldmann, Marc; Knight, Julian C.; Patel, Dhavalkumar D.; Prinos, Panagiotis; Taylor, Michael D.; Sundström, Michael; SGC Open Source Target-Discovery Partnership (March 2015). "Preclinical target validation using patient-derived cells". Nature Reviews. Drug Discovery. 14 (3): 149–150. doi:10.1038/nrd4565. ISSN 1474-1784. PMID 25722227. S2CID 2423838.
Hoag, Hannah (2009). "Richard Gold". Nature Biotechnology. 27 (5): 409. doi:10.1038/nbt0509-409. ISSN 1546-1696. PMID 19430435. S2CID 34394262.
Edwards, Aled; Morgan, Max; Al Chawaf, Arij; Andrusiak, Kerry; Charney, Rachel; Cynader, Zarya; ElDessouki, Ahmed; Lee, Yunjeong; Moeser, Andrew; Stern, Simon; Zuercher, William J. (31 May 2017). "A trust approach for sharing research reagents". Science Translational Medicine. 9 (392): eaai9055. doi:10.1126/scitranslmed.aai9055. ISSN 1946-6242. PMID 28566431. S2CID 4020927.
Vedadi, Masoud; Lew, Jocelyne; Artz, Jennifer; Amani, Mehrnaz; Zhao, Yong; Dong, Aiping; Wasney, Gregory A.; Gao, Mian; Hills, Tanya; Brokx, Stephen; Qiu, Wei (January 2007). "Genome-scale protein expression and structural biology of Plasmodium falciparum and related Apicomplexan organisms". Molecular and Biochemical Parasitology. 151 (1): 100–110. doi:10.1016/j.molbiopara.2006.10.011. ISSN 0166-6851. PMID 17125854.
Frye, Stephen V.; Arkin, Michelle R.; Arrowsmith, Cheryl H.; Conn, P. Jeffrey; Glicksman, Marcie A.; Hull-Ryde, Emily A.; Slusher, Barbara S. (November 2015). "Tackling reproducibility in academic preclinical drug discovery". Nature Reviews. Drug Discovery. 14 (11): 733–734. doi:10.1038/nrd4737. ISSN 1474-1784. PMID 26388229. S2CID 205478934.
Marcon, Edyta; Jain, Harshika; Bhattacharya, Anandi; Guo, Hongbo; Phanse, Sadhna; Pu, Shuye; Byram, Gregory; Collins, Ben C.; Dowdell, Evan; Fenner, Maria; Guo, Xinghua (August 2015). "Assessment of a method to characterize antibody selectivity and specificity for use in immunoprecipitation". Nature Methods. 12 (8): 725–731. doi:10.1038/nmeth.3472. ISSN 1548-7105. PMID 26121405. S2CID 205423964.
Gruetter, Markus (2012). "Open collaboration is key to new drugs". Nature. 491 (7422): 40. doi:10.1038/491040d. ISSN 0028-0836. PMID 23128216. S2CID 205074791.
Carter, Adrian J.; Kraemer, Oliver; Zwick, Matthias; Mueller-Fahrnow, Anke; Arrowsmith, Cheryl H.; Edwards, Aled M. (November 2019). "Target 2035: probing the human proteome". Drug Discovery Today. 24 (11): 2111–2115. doi:10.1016/j.drudis.2019.06.020. ISSN 1878-5832. PMID 31278990.
Schapira, Matthieu; Tyers, Mike; Torrent, Maricel; Arrowsmith, Cheryl H. (November 2017). "WD40 repeat domain proteins: a novel target class?". Nature Reviews. Drug Discovery. 16 (11): 773–786. doi:10.1038/nrd.2017.179. ISSN 1474-1784. PMC 5975957. PMID 29026209.
Song, Richard; Wang, Zhong-Duo; Schapira, Matthieu (6 October 2017). "Disease Association and Druggability of WD40 Repeat Proteins". Journal of Proteome Research. 16 (10): 3766–3773. doi:10.1021/acs.jproteome.7b00451. ISSN 1535-3907. PMID 28956604.
Wang, Jiayan; Yazdani, Setayesh; Han, Ana; Schapira, Matthieu (March 2020). "Structure-based view of the druggable genome". Drug Discovery Today. 25 (3): 561–567. doi:10.1016/j.drudis.2020.02.006. ISSN 1878-5832. PMID 32084498. S2CID 211246313.
Wacker, Daniel; Stevens, Raymond C.; Roth, Bryan L. (2017-07-27). "How Ligands Illuminate GPCR Molecular Pharmacology". Cell. 170 (3): 414–427. doi:10.1016/j.cell.2017.07.009. ISSN 1097-4172. PMC 5560499. PMID 28753422.
Roth, Bryan L.; Irwin, John J.; Shoichet, Brian K. (November 2017). "Discovery of new GPCR ligands to illuminate new biology". Nature Chemical Biology. 13 (11): 1143–1151. doi:10.1038/nchembio.2490. ISSN 1552-4469. PMC 5835362. PMID 29045379.
Roth, Bryan L. (August 2019). "How structure informs and transforms chemogenetics". Current Opinion in Structural Biology. 57: 9–16. doi:10.1016/j.sbi.2019.01.016. ISSN 1879-033X. PMID 30818201. S2CID 73479428.
Edwards, Aled (2016-03-17). "Reproducibility: Team up with industry". Nature. 531 (7594): 299–301. Bibcode:2016Natur.531..299E. doi:10.1038/531299a. ISSN 1476-4687. PMID 26983524. S2CID 4467772.

ncbi.nlm.nih.gov

Masum, Hassan; Rao, Aarthi; Good, Benjamin M.; Todd, Matthew H.; Edwards, Aled M.; Chan, Leslie; Bunin, Barry A.; Su, Andrew I.; Thomas, Zakir; Bourne, Philip E. (2013). "Ten simple rules for cultivating open science and collaborative R&D". PLOS Computational Biology. 9 (9): e1003244. Bibcode:2013PLSCB...9E3244M. doi:10.1371/journal.pcbi.1003244. ISSN 1553-7358. PMC 3784487. PMID 24086123.
Morgan, Maxwell Robert; Roberts, Owen Gwilym; Edwards, Aled Morgan (2018). "Ideation and implementation of an open science drug discovery business model - M4K Pharma". Wellcome Open Research. 3: 154. doi:10.12688/wellcomeopenres.14947.1. ISSN 2398-502X. PMC 6346698. PMID 30705971.
Harding, Rachel J. (January 2019). "Open notebook science can maximize impact for rare disease projects". PLOS Biology. 17 (1): e3000120. doi:10.1371/journal.pbio.3000120. ISSN 1545-7885. PMC 6366684. PMID 30689629.
Schapira, Matthieu; Harding, Rachel J. (2019-04-02). "Open laboratory notebooks: good for science, good for society, good for scientists". F1000Research. 8: 87. doi:10.12688/f1000research.17710.2. ISSN 2046-1402. PMC 6694453. PMID 31448096.
Müller, Susanne; Ackloo, Suzanne; Arrowsmith, Cheryl H.; Bauser, Marcus; Baryza, Jeremy L.; Blagg, Julian; Böttcher, Jark; Bountra, Chas; Brown, Peter J.; Bunnage, Mark E.; Carter, Adrian J. (20 April 2018). "Donated chemical probes for open science". eLife. 7. doi:10.7554/eLife.34311. ISSN 2050-084X. PMC 5910019. PMID 29676732.
Drewry, David H.; Wells, Carrow I.; Zuercher, William J.; Willson, Timothy M. (June 2019). "A Perspective on Extreme Open Science: Companies Sharing Compounds without Restriction". SLAS Discovery. 24 (5): 505–514. doi:10.1177/2472555219838210. ISSN 2472-5560. PMC 6624833. PMID 31034310.
Wells, Carrow I.; Al-Ali, Hassan; Andrews, David M.; Asquith, Christopher R. M.; Axtman, Alison D.; Dikic, Ivan; Ebner, Daniel; Ettmayer, Peter; Fischer, Christian; Frederiksen, Mathias; Futrell, Robert E. (2021-01-08). "The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification". International Journal of Molecular Sciences. 22 (2): 566. doi:10.3390/ijms22020566. ISSN 1422-0067. PMC 7826789. PMID 33429995.
Laflamme, Carl; McKeever, Paul M.; Kumar, Rahul; Schwartz, Julie; Kolahdouzan, Mahshad; Chen, Carol X.; You, Zhipeng; Benaliouad, Faiza; Gileadi, Opher; McBride, Heidi M.; Durcan, Thomas M. (15 October 2019). "Implementation of an antibody characterization procedure and application to the major ALS/FTD disease gene C9ORF72". eLife. 8. doi:10.7554/eLife.48363. ISSN 2050-084X. PMC 6794092. PMID 31612854.
Ensan, Deeba; Smil, David; Zepeda-Velázquez, Carlos A.; Panagopoulos, Dimitrios; Wong, Jong Fu; Williams, Eleanor P.; Adamson, Roslin; Bullock, Alex N.; Kiyota, Taira; Aman, Ahmed; Roberts, Owen G. (2020-05-14). "Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma". Journal of Medicinal Chemistry. 63 (9): 4978–4996. doi:10.1021/acs.jmedchem.0c00395. ISSN 1520-4804. PMC 8213057. PMID 32369358.
Gold, E. Richard (June 2021). "The fall of the innovation empire and its possible rise through open science". Research Policy. 50 (5): 104226. doi:10.1016/j.respol.2021.104226. PMC 8024784. PMID 34083844.
Liu, Lihua; Damerell, David R.; Koukouflis, Leonidas; Tong, Yufeng; Marsden, Brian D.; Schapira, Matthieu (15 August 2019). "UbiHub: a data hub for the explorers of ubiquitination pathways". Bioinformatics. 35 (16): 2882–2884. doi:10.1093/bioinformatics/bty1067. ISSN 1367-4811. PMC 6691330. PMID 30601939.
Drewry, David H.; Wells, Carrow I.; Andrews, David M.; Angell, Richard; Al-Ali, Hassan; Axtman, Alison D.; Capuzzi, Stephen J.; Elkins, Jonathan M.; Ettmayer, Peter; Frederiksen, Mathias; Gileadi, Opher (2017). "Progress towards a public chemogenomic set for protein kinases and a call for contributions". PLOS ONE. 12 (8): e0181585. Bibcode:2017PLoSO..1281585D. doi:10.1371/journal.pone.0181585. ISSN 1932-6203. PMC 5540273. PMID 28767711.
Wu, Qin; Heidenreich, David; Zhou, Stanley; Ackloo, Suzanne; Krämer, Andreas; Nakka, Kiran; Lima-Fernandes, Evelyne; Deblois, Genevieve; Duan, Shili; Vellanki, Ravi N.; Li, Fengling (23 April 2019). "A chemical toolbox for the study of bromodomains and epigenetic signaling". Nature Communications. 10 (1): 1915. Bibcode:2019NatCo..10.1915W. doi:10.1038/s41467-019-09672-2. ISSN 2041-1723. PMC 6478789. PMID 31015424.
Scheer, Sebastian; Ackloo, Suzanne; Medina, Tiago S.; Schapira, Matthieu; Li, Fengling; Ward, Jennifer A.; Lewis, Andrew M.; Northrop, Jeffrey P.; Richardson, Paul L.; Kaniskan, H. Ümit; Shen, Yudao (3 January 2019). "A chemical biology toolbox to study protein methyltransferases and epigenetic signaling". Nature Communications. 10 (1): 19. Bibcode:2019NatCo..10...19S. doi:10.1038/s41467-018-07905-4. ISSN 2041-1723. PMC 6318333. PMID 30604761.
Arrowsmith, Cheryl H.; Audia, James E.; Austin, Christopher; Baell, Jonathan; Bennett, Jonathan; Blagg, Julian; Bountra, Chas; Brennan, Paul E.; Brown, Peter J.; Bunnage, Mark E.; Buser-Doepner, Carolyn (August 2015). "The promise and peril of chemical probes". Nature Chemical Biology. 11 (8): 536–541. doi:10.1038/nchembio.1867. ISSN 1552-4469. PMC 4706458. PMID 26196764.
Blagg, Julian; Workman, Paul (14 August 2017). "Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology". Cancer Cell. 32 (2): 268–270. doi:10.1016/j.ccell.2017.07.010. ISSN 1878-3686. PMC 5559281. PMID 28810148.
Antolin, Albert A.; Tym, Joseph E.; Komianou, Angeliki; Collins, Ian; Workman, Paul; Al-Lazikani, Bissan (15 February 2018). "Objective, Quantitative, Data-Driven Assessment of Chemical Probes". Cell Chemical Biology. 25 (2): 194–205.e5. doi:10.1016/j.chembiol.2017.11.004. ISSN 2451-9448. PMC 5814752. PMID 29249694.
Picaud, Sarah; Da Costa, David; Thanasopoulou, Angeliki; Filippakopoulos, Panagis; Fish, Paul V.; Philpott, Martin; Fedorov, Oleg; Brennan, Paul; Bunnage, Mark E.; Owen, Dafydd R.; Bradner, James E. (2013-06-01). "PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains". Cancer Research. 73 (11): 3336–3346. doi:10.1158/0008-5472.CAN-12-3292. ISSN 1538-7445. PMC 3673830. PMID 23576556.
Filippakopoulos, Panagis; Qi, Jun; Picaud, Sarah; Shen, Yao; Smith, William B.; Fedorov, Oleg; Morse, Elizabeth M.; Keates, Tracey; Hickman, Tyler T.; Felletar, Ildiko; Philpott, Martin (2010-12-23). "Selective inhibition of BET bromodomains". Nature. 468 (7327): 1067–1073. Bibcode:2010Natur.468.1067F. doi:10.1038/nature09504. ISSN 1476-4687. PMC 3010259. PMID 20871596.
Liu, Feng; Barsyte-Lovejoy, Dalia; Li, Fengling; Xiong, Yan; Korboukh, Victoria; Huang, Xi-Ping; Allali-Hassani, Abdellah; Janzen, William P.; Roth, Bryan L.; Frye, Stephen V.; Arrowsmith, Cheryl H. (2013-11-14). "Discovery of an in vivo chemical probe of the lysine methyltransferases G9a and GLP". Journal of Medicinal Chemistry. 56 (21): 8931–8942. doi:10.1021/jm401480r. ISSN 1520-4804. PMC 3880643. PMID 24102134.
Konze, Kyle D.; Ma, Anqi; Li, Fengling; Barsyte-Lovejoy, Dalia; Parton, Trevor; Macnevin, Christopher J.; Liu, Feng; Gao, Cen; Huang, Xi-Ping; Kuznetsova, Ekaterina; Rougie, Marie (2013). "An orally bioavailable chemical probe of the Lysine Methyltransferases EZH2 and EZH1". ACS Chemical Biology. 8 (6): 1324–1334. doi:10.1021/cb400133j. ISSN 1554-8937. PMC 3773059. PMID 23614352.
Bonday, Zahid Q.; Cortez, Guillermo S.; Grogan, Michael J.; Antonysamy, Stephen; Weichert, Ken; Bocchinfuso, Wayne P.; Li, Fengling; Kennedy, Steven; Li, Binghui; Mader, Mary M.; Arrowsmith, Cheryl H. (2018-04-23). "LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity". ACS Medicinal Chemistry Letters. 9 (7): 612–617. doi:10.1021/acsmedchemlett.8b00014. ISSN 1948-5875. PMC 6047023. PMID 30034588.
Duncan, Kenneth W.; Rioux, Nathalie; Boriack-Sjodin, P. Ann; Munchhof, Michael J.; Reiter, Lawrence A.; Majer, Christina R.; Jin, Lei; Johnston, L. Danielle; Chan-Penebre, Elayne; Kuplast, Kristy G.; Porter Scott, Margaret (2016-02-11). "Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666". ACS Medicinal Chemistry Letters. 7 (2): 162–166. doi:10.1021/acsmedchemlett.5b00380. ISSN 1948-5875. PMC 4753547. PMID 26985292.
Grebien, Florian; Vedadi, Masoud; Getlik, Matthäus; Giambruno, Roberto; Grover, Amit; Avellino, Roberto; Skucha, Anna; Vittori, Sarah; Kuznetsova, Ekaterina; Smil, David; Barsyte-Lovejoy, Dalia (August 2015). "Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia". Nature Chemical Biology. 11 (8): 571–578. doi:10.1038/nchembio.1859. ISSN 1552-4469. PMC 4511833. PMID 26167872.
Buljan, M; et, al. (2020). "Kinase Interaction Network Expands Functional and Disease Roles of Human Kinases". Molecular Cell. 79 (3): 504–520.e9. doi:10.1016/j.molcel.2020.07.001. PMC 7427327. PMID 32707033. S2CID 220746851.
Schapira, Matthieu; Tyers, Mike; Torrent, Maricel; Arrowsmith, Cheryl H. (November 2017). "WD40 repeat domain proteins: a novel target class?". Nature Reviews. Drug Discovery. 16 (11): 773–786. doi:10.1038/nrd.2017.179. ISSN 1474-1784. PMC 5975957. PMID 29026209.
Wacker, Daniel; Stevens, Raymond C.; Roth, Bryan L. (2017-07-27). "How Ligands Illuminate GPCR Molecular Pharmacology". Cell. 170 (3): 414–427. doi:10.1016/j.cell.2017.07.009. ISSN 1097-4172. PMC 5560499. PMID 28753422.
Roth, Bryan L.; Irwin, John J.; Shoichet, Brian K. (November 2017). "Discovery of new GPCR ligands to illuminate new biology". Nature Chemical Biology. 13 (11): 1143–1151. doi:10.1038/nchembio.2490. ISSN 1552-4469. PMC 5835362. PMID 29045379.

ox.ac.uk

ora.ox.ac.uk

Schapira, Matthieu; Calabrese, Matthew F.; Bullock, Alex N.; Crews, Craig M. (December 2019). "Targeted protein degradation: expanding the toolbox". Nature Reviews. Drug Discovery. 18 (12): 949–963. doi:10.1038/s41573-019-0047-y. ISSN 1474-1784. PMID 31666732. S2CID 204942300.

semanticscholar.org

api.semanticscholar.org

Williamson, AR (2000). "Creating a structural genomics consortium". Nature Structural Biology. 7: 953. doi:10.1038/80726. PMID 11103997. S2CID 35185565.
Edwards, AM; et, al. (2011). "Too many roads not taken". Nature. 470 (2333): 163–165. arXiv:1102.0448. Bibcode:2011Natur.470..163E. doi:10.1038/470163a. PMID 21307913. S2CID 4429387.
Davis, Andrew M.; Engkvist, Ola; Fairclough, Rebecca J.; Feierberg, Isabella; Freeman, Adrian; Iyer, Preeti (2021-02-13). "Public-Private Partnerships: Compound and Data Sharing in Drug Discovery and Development". SLAS Discovery. 26 (5): 604–619. doi:10.1177/2472555220982268. ISSN 2472-5552. PMID 33586501. S2CID 231928371.
Jones, Molly Morgan; Chataway, Joanna (2021-03-04). "The Structural Genomics Consortium: successful organisational technology experiment or new institutional infrastructure for health research?". Technology Analysis & Strategic Management. 33 (3): 296–306. doi:10.1080/09537325.2021.1882673. ISSN 0953-7325. S2CID 232245414.
Collins, Patrick M.; Douangamath, Alice; Talon, Romain; Dias, Alexandre; Brandao-Neto, Jose; Krojer, Tobias; von Delft, Frank (2018). "Achieving a Good Crystal System for Crystallographic X-Ray Fragment Screening". Modern Approaches in Drug Discovery. Methods in Enzymology. Vol. 610. pp. 251–264. doi:10.1016/bs.mie.2018.09.027. ISBN 9780128153833. ISSN 1557-7988. PMID 30390801. S2CID 53219679.
Arrowsmith, Cheryl H.; Bountra, Chas; Fish, Paul V.; Lee, Kevin; Schapira, Matthieu (2012-04-13). "Epigenetic protein families: a new frontier for drug discovery". Nature Reviews. Drug Discovery. 11 (5): 384–400. doi:10.1038/nrd3674. ISSN 1474-1784. PMID 22498752. S2CID 5478921.
César-Razquin, Adrián; Snijder, Berend; Frappier-Brinton, Tristan; Isserlin, Ruth; Gyimesi, Gergely; Bai, Xiaoyun; Reithmeier, Reinhart A.; Hepworth, David; Hediger, Matthias A.; Edwards, Aled M.; Superti-Furga, Giulio (2015-07-30). "A Call for Systematic Research on Solute Carriers". Cell. 162 (3): 478–487. doi:10.1016/j.cell.2015.07.022. ISSN 1097-4172. PMID 26232220. S2CID 15427088.
Superti-Furga, Giulio; Lackner, Daniel; Wiedmer, Tabea; Ingles-Prieto, Alvaro; Barbosa, Barbara; Girardi, Enrico; Goldmann, Ulrich; Gürtl, Bettina; Klavins, Kristaps; Klimek, Christoph; Lindinger, Sabrina (July 2020). "The RESOLUTE consortium: unlocking SLC transporters for drug discovery". Nature Reviews. Drug Discovery. 19 (7): 429–430. doi:10.1038/d41573-020-00056-6. hdl:21.11116/0000-0006-0FF1-A. ISSN 1474-1784. PMID 32265506. S2CID 215406274.
Schapira, Matthieu; Calabrese, Matthew F.; Bullock, Alex N.; Crews, Craig M. (December 2019). "Targeted protein degradation: expanding the toolbox". Nature Reviews. Drug Discovery. 18 (12): 949–963. doi:10.1038/s41573-019-0047-y. ISSN 1474-1784. PMID 31666732. S2CID 204942300.
Mann, Mandeep K.; Franzoni, Ivan; de Freitas, Renato Ferreira; Tempel, Wolfram; Houliston, Scott; Smith, Leanna; Vedadi, Masoud; Arrowsmith, Cheryl H.; Harding, Rachel J.; Schapira, Matthieu (27 November 2019). "Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain" (PDF). Journal of Medicinal Chemistry. 62 (22): 10144–10155. doi:10.1021/acs.jmedchem.9b00988. ISSN 1520-4804. PMID 31663737. S2CID 204975079.
Roskoski, Robert (June 2019). "Properties of FDA-approved small molecule protein kinase inhibitors". Pharmacological Research. 144: 19–50. doi:10.1016/j.phrs.2019.03.006. ISSN 1096-1186. PMID 30877063. S2CID 80625382.
Sorget, Nienke; et, al (2020). "Exploring the understudied human kinome for research and therapeutic opportunities" (PDF). www.biorxiv.org. doi:10.1101/2020.04.02.022277. S2CID 215404186.
Buljan, M; et, al. (2020). "Kinase Interaction Network Expands Functional and Disease Roles of Human Kinases". Molecular Cell. 79 (3): 504–520.e9. doi:10.1016/j.molcel.2020.07.001. PMC 7427327. PMID 32707033. S2CID 220746851.
Edwards, Aled M.; Arrowsmith, Cheryl H.; Bountra, Chas; Bunnage, Mark E.; Feldmann, Marc; Knight, Julian C.; Patel, Dhavalkumar D.; Prinos, Panagiotis; Taylor, Michael D.; Sundström, Michael; SGC Open Source Target-Discovery Partnership (March 2015). "Preclinical target validation using patient-derived cells". Nature Reviews. Drug Discovery. 14 (3): 149–150. doi:10.1038/nrd4565. ISSN 1474-1784. PMID 25722227. S2CID 2423838.
Hoag, Hannah (2009). "Richard Gold". Nature Biotechnology. 27 (5): 409. doi:10.1038/nbt0509-409. ISSN 1546-1696. PMID 19430435. S2CID 34394262.
Edwards, Aled; Morgan, Max; Al Chawaf, Arij; Andrusiak, Kerry; Charney, Rachel; Cynader, Zarya; ElDessouki, Ahmed; Lee, Yunjeong; Moeser, Andrew; Stern, Simon; Zuercher, William J. (31 May 2017). "A trust approach for sharing research reagents". Science Translational Medicine. 9 (392): eaai9055. doi:10.1126/scitranslmed.aai9055. ISSN 1946-6242. PMID 28566431. S2CID 4020927.
Frye, Stephen V.; Arkin, Michelle R.; Arrowsmith, Cheryl H.; Conn, P. Jeffrey; Glicksman, Marcie A.; Hull-Ryde, Emily A.; Slusher, Barbara S. (November 2015). "Tackling reproducibility in academic preclinical drug discovery". Nature Reviews. Drug Discovery. 14 (11): 733–734. doi:10.1038/nrd4737. ISSN 1474-1784. PMID 26388229. S2CID 205478934.
Marcon, Edyta; Jain, Harshika; Bhattacharya, Anandi; Guo, Hongbo; Phanse, Sadhna; Pu, Shuye; Byram, Gregory; Collins, Ben C.; Dowdell, Evan; Fenner, Maria; Guo, Xinghua (August 2015). "Assessment of a method to characterize antibody selectivity and specificity for use in immunoprecipitation". Nature Methods. 12 (8): 725–731. doi:10.1038/nmeth.3472. ISSN 1548-7105. PMID 26121405. S2CID 205423964.
Gruetter, Markus (2012). "Open collaboration is key to new drugs". Nature. 491 (7422): 40. doi:10.1038/491040d. ISSN 0028-0836. PMID 23128216. S2CID 205074791.
Wang, Jiayan; Yazdani, Setayesh; Han, Ana; Schapira, Matthieu (March 2020). "Structure-based view of the druggable genome". Drug Discovery Today. 25 (3): 561–567. doi:10.1016/j.drudis.2020.02.006. ISSN 1878-5832. PMID 32084498. S2CID 211246313.
Roth, Bryan L. (August 2019). "How structure informs and transforms chemogenetics". Current Opinion in Structural Biology. 57: 9–16. doi:10.1016/j.sbi.2019.01.016. ISSN 1879-033X. PMID 30818201. S2CID 73479428.
Edwards, Aled (2016-03-17). "Reproducibility: Team up with industry". Nature. 531 (7594): 299–301. Bibcode:2016Natur.531..299E. doi:10.1038/531299a. ISSN 1476-4687. PMID 26983524. S2CID 4467772.

thesgc.org

"Structure Gallery". SGC. Retrieved 2020-09-09.
"Target Enabling Packages (TEPs)". SGC. 2016-06-13. Retrieved 2020-09-09.
"Chemical Probes". SGC. 2019-04-08. Retrieved 2020-09-09.

chromohub.thesgc.org

"ChromoHub". chromohub.thesgc.org. Retrieved 2020-09-09.

ubihub.thesgc.org

"UbiHub". ubihub.thesgc.org. Retrieved 2020-09-09.

unc.edu

cdr.lib.unc.edu

Roth, Bryan L. (August 2019). "How structure informs and transforms chemogenetics". Current Opinion in Structural Biology. 57: 9–16. doi:10.1016/j.sbi.2019.01.016. ISSN 1879-033X. PMID 30818201. S2CID 73479428.

vimiopen.org

"Viral Interruption Medicines Initiative (VIMI)". Viral Interruption Medicines Initiative (VIMI). Retrieved 2021-03-21.

worldcat.org

Davis, Andrew M.; Engkvist, Ola; Fairclough, Rebecca J.; Feierberg, Isabella; Freeman, Adrian; Iyer, Preeti (2021-02-13). "Public-Private Partnerships: Compound and Data Sharing in Drug Discovery and Development". SLAS Discovery. 26 (5): 604–619. doi:10.1177/2472555220982268. ISSN 2472-5552. PMID 33586501. S2CID 231928371.
Edwards, Aled (September 2008). "Open-source science to enable drug discovery". Drug Discovery Today. 13 (17–18): 731–733. doi:10.1016/j.drudis.2008.04.011. ISSN 1359-6446. PMID 18790412.
Edwards, Aled M.; Bountra, Chas; Kerr, David J.; Willson, Timothy M. (July 2009). "Open access chemical and clinical probes to support drug discovery". Nature Chemical Biology. 5 (7): 436–440. doi:10.1038/nchembio0709-436. ISSN 1552-4469. PMID 19536100.
Masum, Hassan; Rao, Aarthi; Good, Benjamin M.; Todd, Matthew H.; Edwards, Aled M.; Chan, Leslie; Bunin, Barry A.; Su, Andrew I.; Thomas, Zakir; Bourne, Philip E. (2013). "Ten simple rules for cultivating open science and collaborative R&D". PLOS Computational Biology. 9 (9): e1003244. Bibcode:2013PLSCB...9E3244M. doi:10.1371/journal.pcbi.1003244. ISSN 1553-7358. PMC 3784487. PMID 24086123.
Morgan, Maxwell Robert; Roberts, Owen Gwilym; Edwards, Aled Morgan (2018). "Ideation and implementation of an open science drug discovery business model - M4K Pharma". Wellcome Open Research. 3: 154. doi:10.12688/wellcomeopenres.14947.1. ISSN 2398-502X. PMC 6346698. PMID 30705971.
Harding, Rachel J. (January 2019). "Open notebook science can maximize impact for rare disease projects". PLOS Biology. 17 (1): e3000120. doi:10.1371/journal.pbio.3000120. ISSN 1545-7885. PMC 6366684. PMID 30689629.
Schapira, Matthieu; Harding, Rachel J. (2019-04-02). "Open laboratory notebooks: good for science, good for society, good for scientists". F1000Research. 8: 87. doi:10.12688/f1000research.17710.2. ISSN 2046-1402. PMC 6694453. PMID 31448096.
Müller, Susanne; Ackloo, Suzanne; Arrowsmith, Cheryl H.; Bauser, Marcus; Baryza, Jeremy L.; Blagg, Julian; Böttcher, Jark; Bountra, Chas; Brown, Peter J.; Bunnage, Mark E.; Carter, Adrian J. (20 April 2018). "Donated chemical probes for open science". eLife. 7. doi:10.7554/eLife.34311. ISSN 2050-084X. PMC 5910019. PMID 29676732.
Drewry, David H.; Wells, Carrow I.; Zuercher, William J.; Willson, Timothy M. (June 2019). "A Perspective on Extreme Open Science: Companies Sharing Compounds without Restriction". SLAS Discovery. 24 (5): 505–514. doi:10.1177/2472555219838210. ISSN 2472-5560. PMC 6624833. PMID 31034310.
Wells, Carrow I.; Al-Ali, Hassan; Andrews, David M.; Asquith, Christopher R. M.; Axtman, Alison D.; Dikic, Ivan; Ebner, Daniel; Ettmayer, Peter; Fischer, Christian; Frederiksen, Mathias; Futrell, Robert E. (2021-01-08). "The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification". International Journal of Molecular Sciences. 22 (2): 566. doi:10.3390/ijms22020566. ISSN 1422-0067. PMC 7826789. PMID 33429995.
Laflamme, Carl; McKeever, Paul M.; Kumar, Rahul; Schwartz, Julie; Kolahdouzan, Mahshad; Chen, Carol X.; You, Zhipeng; Benaliouad, Faiza; Gileadi, Opher; McBride, Heidi M.; Durcan, Thomas M. (15 October 2019). "Implementation of an antibody characterization procedure and application to the major ALS/FTD disease gene C9ORF72". eLife. 8. doi:10.7554/eLife.48363. ISSN 2050-084X. PMC 6794092. PMID 31612854.
Ensan, Deeba; Smil, David; Zepeda-Velázquez, Carlos A.; Panagopoulos, Dimitrios; Wong, Jong Fu; Williams, Eleanor P.; Adamson, Roslin; Bullock, Alex N.; Kiyota, Taira; Aman, Ahmed; Roberts, Owen G. (2020-05-14). "Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma". Journal of Medicinal Chemistry. 63 (9): 4978–4996. doi:10.1021/acs.jmedchem.0c00395. ISSN 1520-4804. PMC 8213057. PMID 32369358.
Jones, Molly Morgan; Chataway, Joanna (2021-03-04). "The Structural Genomics Consortium: successful organisational technology experiment or new institutional infrastructure for health research?". Technology Analysis & Strategic Management. 33 (3): 296–306. doi:10.1080/09537325.2021.1882673. ISSN 0953-7325. S2CID 232245414.
Collins, Patrick M.; Douangamath, Alice; Talon, Romain; Dias, Alexandre; Brandao-Neto, Jose; Krojer, Tobias; von Delft, Frank (2018). "Achieving a Good Crystal System for Crystallographic X-Ray Fragment Screening". Modern Approaches in Drug Discovery. Methods in Enzymology. Vol. 610. pp. 251–264. doi:10.1016/bs.mie.2018.09.027. ISBN 9780128153833. ISSN 1557-7988. PMID 30390801. S2CID 53219679.
Arrowsmith, Cheryl H.; Bountra, Chas; Fish, Paul V.; Lee, Kevin; Schapira, Matthieu (2012-04-13). "Epigenetic protein families: a new frontier for drug discovery". Nature Reviews. Drug Discovery. 11 (5): 384–400. doi:10.1038/nrd3674. ISSN 1474-1784. PMID 22498752. S2CID 5478921.
Huston, Andrea; Arrowsmith, Cheryl H.; Knapp, Stefan; Schapira, Matthieu (August 2015). "Probing the epigenome". Nature Chemical Biology. 11 (8): 542–545. doi:10.1038/nchembio.1871. ISSN 1552-4469. PMID 26196765.
César-Razquin, Adrián; Snijder, Berend; Frappier-Brinton, Tristan; Isserlin, Ruth; Gyimesi, Gergely; Bai, Xiaoyun; Reithmeier, Reinhart A.; Hepworth, David; Hediger, Matthias A.; Edwards, Aled M.; Superti-Furga, Giulio (2015-07-30). "A Call for Systematic Research on Solute Carriers". Cell. 162 (3): 478–487. doi:10.1016/j.cell.2015.07.022. ISSN 1097-4172. PMID 26232220. S2CID 15427088.
Superti-Furga, Giulio; Lackner, Daniel; Wiedmer, Tabea; Ingles-Prieto, Alvaro; Barbosa, Barbara; Girardi, Enrico; Goldmann, Ulrich; Gürtl, Bettina; Klavins, Kristaps; Klimek, Christoph; Lindinger, Sabrina (July 2020). "The RESOLUTE consortium: unlocking SLC transporters for drug discovery". Nature Reviews. Drug Discovery. 19 (7): 429–430. doi:10.1038/d41573-020-00056-6. hdl:21.11116/0000-0006-0FF1-A. ISSN 1474-1784. PMID 32265506. S2CID 215406274.
Liu, Lihua; Damerell, David R.; Koukouflis, Leonidas; Tong, Yufeng; Marsden, Brian D.; Schapira, Matthieu (15 August 2019). "UbiHub: a data hub for the explorers of ubiquitination pathways". Bioinformatics. 35 (16): 2882–2884. doi:10.1093/bioinformatics/bty1067. ISSN 1367-4811. PMC 6691330. PMID 30601939.
Schapira, Matthieu; Calabrese, Matthew F.; Bullock, Alex N.; Crews, Craig M. (December 2019). "Targeted protein degradation: expanding the toolbox". Nature Reviews. Drug Discovery. 18 (12): 949–963. doi:10.1038/s41573-019-0047-y. ISSN 1474-1784. PMID 31666732. S2CID 204942300.
Harding, Rachel J.; Ferreira de Freitas, Renato; Collins, Patrick; Franzoni, Ivan; Ravichandran, Mani; Ouyang, Hui; Juarez-Ornelas, Kevin A.; Lautens, Mark; Schapira, Matthieu; von Delft, Frank; Santhakumar, Vjayaratnam (9 November 2017). "Small Molecule Antagonists of the Interaction between the Histone Deacetylase 6 Zinc-Finger Domain and Ubiquitin". Journal of Medicinal Chemistry. 60 (21): 9090–9096. doi:10.1021/acs.jmedchem.7b00933. ISSN 1520-4804. PMID 29019676.
Ferreira de Freitas, Renato; Harding, Rachel J.; Franzoni, Ivan; Ravichandran, Mani; Mann, Mandeep K.; Ouyang, Hui; Lautens, Mark; Santhakumar, Vijayaratnam; Arrowsmith, Cheryl H.; Schapira, Matthieu (24 May 2018). "Identification and Structure-Activity Relationship of HDAC6 Zinc-Finger Ubiquitin Binding Domain Inhibitors". Journal of Medicinal Chemistry. 61 (10): 4517–4527. doi:10.1021/acs.jmedchem.8b00258. ISSN 1520-4804. PMID 29741882.
Mann, Mandeep K.; Franzoni, Ivan; de Freitas, Renato Ferreira; Tempel, Wolfram; Houliston, Scott; Smith, Leanna; Vedadi, Masoud; Arrowsmith, Cheryl H.; Harding, Rachel J.; Schapira, Matthieu (27 November 2019). "Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain" (PDF). Journal of Medicinal Chemistry. 62 (22): 10144–10155. doi:10.1021/acs.jmedchem.9b00988. ISSN 1520-4804. PMID 31663737. S2CID 204975079.
Knapp, Stefan; Arruda, Paulo; Blagg, Julian; Burley, Stephen; Drewry, David H.; Edwards, Aled; Fabbro, Doriano; Gillespie, Paul; Gray, Nathanael S.; Kuster, Bernhard; Lackey, Karen E. (January 2013). "A public-private partnership to unlock the untargeted kinome". Nature Chemical Biology. 9 (1): 3–6. doi:10.1038/nchembio.1113. ISSN 1552-4469. PMID 23238671.
Drewry, David H.; Wells, Carrow I.; Andrews, David M.; Angell, Richard; Al-Ali, Hassan; Axtman, Alison D.; Capuzzi, Stephen J.; Elkins, Jonathan M.; Ettmayer, Peter; Frederiksen, Mathias; Gileadi, Opher (2017). "Progress towards a public chemogenomic set for protein kinases and a call for contributions". PLOS ONE. 12 (8): e0181585. Bibcode:2017PLoSO..1281585D. doi:10.1371/journal.pone.0181585. ISSN 1932-6203. PMC 5540273. PMID 28767711.
Wu, Qin; Heidenreich, David; Zhou, Stanley; Ackloo, Suzanne; Krämer, Andreas; Nakka, Kiran; Lima-Fernandes, Evelyne; Deblois, Genevieve; Duan, Shili; Vellanki, Ravi N.; Li, Fengling (23 April 2019). "A chemical toolbox for the study of bromodomains and epigenetic signaling". Nature Communications. 10 (1): 1915. Bibcode:2019NatCo..10.1915W. doi:10.1038/s41467-019-09672-2. ISSN 2041-1723. PMC 6478789. PMID 31015424.
Scheer, Sebastian; Ackloo, Suzanne; Medina, Tiago S.; Schapira, Matthieu; Li, Fengling; Ward, Jennifer A.; Lewis, Andrew M.; Northrop, Jeffrey P.; Richardson, Paul L.; Kaniskan, H. Ümit; Shen, Yudao (3 January 2019). "A chemical biology toolbox to study protein methyltransferases and epigenetic signaling". Nature Communications. 10 (1): 19. Bibcode:2019NatCo..10...19S. doi:10.1038/s41467-018-07905-4. ISSN 2041-1723. PMC 6318333. PMID 30604761.
Frye, Stephen V. (March 2010). "The art of the chemical probe". Nature Chemical Biology. 6 (3): 159–161. doi:10.1038/nchembio.296. ISSN 1552-4469. PMID 20154659.
Arrowsmith, Cheryl H.; Audia, James E.; Austin, Christopher; Baell, Jonathan; Bennett, Jonathan; Blagg, Julian; Bountra, Chas; Brennan, Paul E.; Brown, Peter J.; Bunnage, Mark E.; Buser-Doepner, Carolyn (August 2015). "The promise and peril of chemical probes". Nature Chemical Biology. 11 (8): 536–541. doi:10.1038/nchembio.1867. ISSN 1552-4469. PMC 4706458. PMID 26196764.
Blagg, Julian; Workman, Paul (14 August 2017). "Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology". Cancer Cell. 32 (2): 268–270. doi:10.1016/j.ccell.2017.07.010. ISSN 1878-3686. PMC 5559281. PMID 28810148.
Antolin, Albert A.; Tym, Joseph E.; Komianou, Angeliki; Collins, Ian; Workman, Paul; Al-Lazikani, Bissan (15 February 2018). "Objective, Quantitative, Data-Driven Assessment of Chemical Probes". Cell Chemical Biology. 25 (2): 194–205.e5. doi:10.1016/j.chembiol.2017.11.004. ISSN 2451-9448. PMC 5814752. PMID 29249694.
Antolin, Albert A.; Workman, Paul; Al-Lazikani, Bissan (2019-11-28). "Public resources for chemical probes: the journey so far and the road ahead". Future Medicinal Chemistry. 13 (8): 731–747. doi:10.4155/fmc-2019-0231. ISSN 1756-8927. PMID 31778323.
Picaud, Sarah; Da Costa, David; Thanasopoulou, Angeliki; Filippakopoulos, Panagis; Fish, Paul V.; Philpott, Martin; Fedorov, Oleg; Brennan, Paul; Bunnage, Mark E.; Owen, Dafydd R.; Bradner, James E. (2013-06-01). "PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains". Cancer Research. 73 (11): 3336–3346. doi:10.1158/0008-5472.CAN-12-3292. ISSN 1538-7445. PMC 3673830. PMID 23576556.
Filippakopoulos, Panagis; Qi, Jun; Picaud, Sarah; Shen, Yao; Smith, William B.; Fedorov, Oleg; Morse, Elizabeth M.; Keates, Tracey; Hickman, Tyler T.; Felletar, Ildiko; Philpott, Martin (2010-12-23). "Selective inhibition of BET bromodomains". Nature. 468 (7327): 1067–1073. Bibcode:2010Natur.468.1067F. doi:10.1038/nature09504. ISSN 1476-4687. PMC 3010259. PMID 20871596.
Liu, Feng; Barsyte-Lovejoy, Dalia; Li, Fengling; Xiong, Yan; Korboukh, Victoria; Huang, Xi-Ping; Allali-Hassani, Abdellah; Janzen, William P.; Roth, Bryan L.; Frye, Stephen V.; Arrowsmith, Cheryl H. (2013-11-14). "Discovery of an in vivo chemical probe of the lysine methyltransferases G9a and GLP". Journal of Medicinal Chemistry. 56 (21): 8931–8942. doi:10.1021/jm401480r. ISSN 1520-4804. PMC 3880643. PMID 24102134.
Konze, Kyle D.; Ma, Anqi; Li, Fengling; Barsyte-Lovejoy, Dalia; Parton, Trevor; Macnevin, Christopher J.; Liu, Feng; Gao, Cen; Huang, Xi-Ping; Kuznetsova, Ekaterina; Rougie, Marie (2013). "An orally bioavailable chemical probe of the Lysine Methyltransferases EZH2 and EZH1". ACS Chemical Biology. 8 (6): 1324–1334. doi:10.1021/cb400133j. ISSN 1554-8937. PMC 3773059. PMID 23614352.
Bonday, Zahid Q.; Cortez, Guillermo S.; Grogan, Michael J.; Antonysamy, Stephen; Weichert, Ken; Bocchinfuso, Wayne P.; Li, Fengling; Kennedy, Steven; Li, Binghui; Mader, Mary M.; Arrowsmith, Cheryl H. (2018-04-23). "LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity". ACS Medicinal Chemistry Letters. 9 (7): 612–617. doi:10.1021/acsmedchemlett.8b00014. ISSN 1948-5875. PMC 6047023. PMID 30034588.
Duncan, Kenneth W.; Rioux, Nathalie; Boriack-Sjodin, P. Ann; Munchhof, Michael J.; Reiter, Lawrence A.; Majer, Christina R.; Jin, Lei; Johnston, L. Danielle; Chan-Penebre, Elayne; Kuplast, Kristy G.; Porter Scott, Margaret (2016-02-11). "Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666". ACS Medicinal Chemistry Letters. 7 (2): 162–166. doi:10.1021/acsmedchemlett.5b00380. ISSN 1948-5875. PMC 4753547. PMID 26985292.
Grebien, Florian; Vedadi, Masoud; Getlik, Matthäus; Giambruno, Roberto; Grover, Amit; Avellino, Roberto; Skucha, Anna; Vittori, Sarah; Kuznetsova, Ekaterina; Smil, David; Barsyte-Lovejoy, Dalia (August 2015). "Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia". Nature Chemical Biology. 11 (8): 571–578. doi:10.1038/nchembio.1859. ISSN 1552-4469. PMC 4511833. PMID 26167872.
Roskoski, Robert (June 2019). "Properties of FDA-approved small molecule protein kinase inhibitors". Pharmacological Research. 144: 19–50. doi:10.1016/j.phrs.2019.03.006. ISSN 1096-1186. PMID 30877063. S2CID 80625382.
Edwards, Aled M.; Arrowsmith, Cheryl H.; Bountra, Chas; Bunnage, Mark E.; Feldmann, Marc; Knight, Julian C.; Patel, Dhavalkumar D.; Prinos, Panagiotis; Taylor, Michael D.; Sundström, Michael; SGC Open Source Target-Discovery Partnership (March 2015). "Preclinical target validation using patient-derived cells". Nature Reviews. Drug Discovery. 14 (3): 149–150. doi:10.1038/nrd4565. ISSN 1474-1784. PMID 25722227. S2CID 2423838.
Hoag, Hannah (2009). "Richard Gold". Nature Biotechnology. 27 (5): 409. doi:10.1038/nbt0509-409. ISSN 1546-1696. PMID 19430435. S2CID 34394262.
Edwards, Aled; Morgan, Max; Al Chawaf, Arij; Andrusiak, Kerry; Charney, Rachel; Cynader, Zarya; ElDessouki, Ahmed; Lee, Yunjeong; Moeser, Andrew; Stern, Simon; Zuercher, William J. (31 May 2017). "A trust approach for sharing research reagents". Science Translational Medicine. 9 (392): eaai9055. doi:10.1126/scitranslmed.aai9055. ISSN 1946-6242. PMID 28566431. S2CID 4020927.
Vedadi, Masoud; Lew, Jocelyne; Artz, Jennifer; Amani, Mehrnaz; Zhao, Yong; Dong, Aiping; Wasney, Gregory A.; Gao, Mian; Hills, Tanya; Brokx, Stephen; Qiu, Wei (January 2007). "Genome-scale protein expression and structural biology of Plasmodium falciparum and related Apicomplexan organisms". Molecular and Biochemical Parasitology. 151 (1): 100–110. doi:10.1016/j.molbiopara.2006.10.011. ISSN 0166-6851. PMID 17125854.
Frye, Stephen V.; Arkin, Michelle R.; Arrowsmith, Cheryl H.; Conn, P. Jeffrey; Glicksman, Marcie A.; Hull-Ryde, Emily A.; Slusher, Barbara S. (November 2015). "Tackling reproducibility in academic preclinical drug discovery". Nature Reviews. Drug Discovery. 14 (11): 733–734. doi:10.1038/nrd4737. ISSN 1474-1784. PMID 26388229. S2CID 205478934.
Marcon, Edyta; Jain, Harshika; Bhattacharya, Anandi; Guo, Hongbo; Phanse, Sadhna; Pu, Shuye; Byram, Gregory; Collins, Ben C.; Dowdell, Evan; Fenner, Maria; Guo, Xinghua (August 2015). "Assessment of a method to characterize antibody selectivity and specificity for use in immunoprecipitation". Nature Methods. 12 (8): 725–731. doi:10.1038/nmeth.3472. ISSN 1548-7105. PMID 26121405. S2CID 205423964.
Gruetter, Markus (2012). "Open collaboration is key to new drugs". Nature. 491 (7422): 40. doi:10.1038/491040d. ISSN 0028-0836. PMID 23128216. S2CID 205074791.
Carter, Adrian J.; Kraemer, Oliver; Zwick, Matthias; Mueller-Fahrnow, Anke; Arrowsmith, Cheryl H.; Edwards, Aled M. (November 2019). "Target 2035: probing the human proteome". Drug Discovery Today. 24 (11): 2111–2115. doi:10.1016/j.drudis.2019.06.020. ISSN 1878-5832. PMID 31278990.
Schapira, Matthieu; Tyers, Mike; Torrent, Maricel; Arrowsmith, Cheryl H. (November 2017). "WD40 repeat domain proteins: a novel target class?". Nature Reviews. Drug Discovery. 16 (11): 773–786. doi:10.1038/nrd.2017.179. ISSN 1474-1784. PMC 5975957. PMID 29026209.
Song, Richard; Wang, Zhong-Duo; Schapira, Matthieu (6 October 2017). "Disease Association and Druggability of WD40 Repeat Proteins". Journal of Proteome Research. 16 (10): 3766–3773. doi:10.1021/acs.jproteome.7b00451. ISSN 1535-3907. PMID 28956604.
Wang, Jiayan; Yazdani, Setayesh; Han, Ana; Schapira, Matthieu (March 2020). "Structure-based view of the druggable genome". Drug Discovery Today. 25 (3): 561–567. doi:10.1016/j.drudis.2020.02.006. ISSN 1878-5832. PMID 32084498. S2CID 211246313.
Wacker, Daniel; Stevens, Raymond C.; Roth, Bryan L. (2017-07-27). "How Ligands Illuminate GPCR Molecular Pharmacology". Cell. 170 (3): 414–427. doi:10.1016/j.cell.2017.07.009. ISSN 1097-4172. PMC 5560499. PMID 28753422.
Roth, Bryan L.; Irwin, John J.; Shoichet, Brian K. (November 2017). "Discovery of new GPCR ligands to illuminate new biology". Nature Chemical Biology. 13 (11): 1143–1151. doi:10.1038/nchembio.2490. ISSN 1552-4469. PMC 5835362. PMID 29045379.
Roth, Bryan L. (August 2019). "How structure informs and transforms chemogenetics". Current Opinion in Structural Biology. 57: 9–16. doi:10.1016/j.sbi.2019.01.016. ISSN 1879-033X. PMID 30818201. S2CID 73479428.
Edwards, Aled (2016-03-17). "Reproducibility: Team up with industry". Nature. 531 (7594): 299–301. Bibcode:2016Natur.531..299E. doi:10.1038/531299a. ISSN 1476-4687. PMID 26983524. S2CID 4467772.