TIK-301 (English Wikipedia)

Analysis of information sources in references of the Wikipedia article "TIK-301" in English language version.

refsWebsite

Global rank English rank

18nih.gov

4^th place

15doi.org

2^nd place

4web.archive.org

1^st place

4semanticscholar.org

11^th place

8^th place

1chemdrug.com

low place

1prnewswire.com

406^th place

258^th place

1globenewswire.com

2,614^th place

1,549^th place

1biospace.com

low place

7,595^th place

1uca.edu.ar

low place

1fiercebiotech.com

low place

8,828^th place

1handle.net

102^nd place

76^th place

1espacenet.com

800^th place

676^th place

biospace.com

"Phase 2 Discovery, Inc. Receives Orphan Drug Designation From FDA For Synthetic Melatonin Analog PD-6735". BioSpace. 19 October 2005. Archived from the original on 4 March 2016.

chemdrug.com

"PD-6735, LY-156735,118702-11-7,C14-H17-Cl-N2-O2,N-[2(R)-(6-C--药物合成数据库". Archived from the original on 2009-09-27.

doi.org

Rivara S, Mor M, Bedini A, Spadoni G, Tarzia G (2008). "Melatonin receptor agonists: SAR and applications to the treatment of sleep-wake disorders". Current Topics in Medicinal Chemistry. 8 (11): 954–968. doi:10.2174/156802608784936719. PMID 18673165.
Kostiuk NV, Belyakova MB, Leshchenko DV, Zhigulina VV, Miniaev MV (2014). "Synthetic melatoninergic ligands: achievements and prospects". ISRN Biochemistry. 2014: 843478. doi:10.1155/2014/843478. PMC 4393004. PMID 25937968.
Zlotos DP (2012). "Recent progress in the development of agonists and antagonists for melatonin receptors". Current Medicinal Chemistry. 19 (21): 3532–3549. doi:10.2174/092986712801323153. PMID 22680635.
Carocci A, Catalano A, Sinicropi MS (2014). "Melatonergic drugs in development". Clinical Pharmacology. 6: 127–137. doi:10.2147/CPAA.S36600. PMC 4172069. PMID 25258560.
Zlotos DP, Jockers R, Cecon E, Rivara S, Witt-Enderby PA (April 2014). "MT1 and MT2 melatonin receptors: ligands, models, oligomers, and therapeutic potential". Journal of Medicinal Chemistry. 57 (8): 3161–3185. doi:10.1021/jm401343c. PMID 24228714.
Hardeland R, Poeggeler B (September 2012). "Melatonin and synthetic melatonergic agonists: actions and metabolism in the central nervous system". Central Nervous System Agents in Medicinal Chemistry. 12 (3): 189–216. doi:10.2174/187152412802430129. PMID 22640220.
Chan KH, Hu Y, Ho MK, Wong YH (2013). "Characterization of substituted phenylpropylamides as highly selective agonists at the melatonin MT2 receptor". Current Medicinal Chemistry. 20 (2): 289–300. doi:10.2174/0929867311320020009. PMID 23131177.
Mulchahey JJ, Goldwater DR, Zemlan FP (August 2004). "A single blind, placebo controlled, across groups dose escalation study of the safety, tolerability, pharmacokinetics and pharmacodynamics of the melatonin analog beta-methyl-6-chloromelatonin". Life Sciences. 75 (15): 1843–1856. doi:10.1016/j.lfs.2004.03.023. PMID 15302228.
Nickelsen T, Samel A, Vejvoda M, Wenzel J, Smith B, Gerzer R (September 2002). "Chronobiotic effects of the melatonin agonist LY 156735 following a simulated 9h time shift: results of a placebo-controlled trial". Chronobiology International. 19 (5): 915–936. doi:10.1081/cbi-120014108. PMID 12405554. S2CID 10363563.
Cardinali DP, Srinivasan V, Brzezinski A, Brown GM (May 2012). "Melatonin and its analogs in insomnia and depression" (PDF). Journal of Pineal Research. 52 (4): 365–375. doi:10.1111/j.1600-079x.2011.00962.x. PMID 21951153. S2CID 139480.
Zemlan FP, Mulchahey JJ, Scharf MB, Mayleben DW, Rosenberg R, Lankford A (March 2005). "The efficacy and safety of the melatonin agonist beta-methyl-6-chloromelatonin in primary insomnia: a randomized, placebo-controlled, crossover clinical trial". The Journal of Clinical Psychiatry. 66 (3): 384–390. doi:10.4088/jcp.v66n0316. PMID 15766306.
Turek FW, Gillette MU (November 2004). "Melatonin, sleep, and circadian rhythms: rationale for development of specific melatonin agonists". Sleep Medicine. 5 (6): 523–532. doi:10.1016/j.sleep.2004.07.009. PMID 15511698.
Doghramji K (August 2007). "Melatonin and its receptors: a new class of sleep-promoting agents". Journal of Clinical Sleep Medicine. 3 (5 Suppl): S17–S23. doi:10.5664/jcsm.26932. PMC 1978320. PMID 17824497.
Rivara S, Pala D, Bedini A, Spadoni G (April 2015). "Therapeutic uses of melatonin and melatonin derivatives: a patent review (2012 - 2014)". Expert Opinion on Therapeutic Patents. 25 (4): 425–441. doi:10.1517/13543776.2014.1001739. hdl:11576/2623397. PMID 25579320. S2CID 19644131.
Fee DB, Swartz KR, Scheff N, Roberts K, Gabbita P, Scheff S (June 2010). "Melatonin-analog, beta-methyl-6-chloromelatonin, supplementation in spinal cord injury". Brain Research. 1340: 81–85. doi:10.1016/j.brainres.2010.04.047. PMID 20420812. S2CID 27784753.

espacenet.com

worldwide.espacenet.com

WO 2014010603, Watanabe K, Kawabata Y, Watanabe K, Yuyama N, Burgard S, Bruce E, "Pharmaceutical composition for treatment or prevention of stress urinary incontinence or mixed urinary incontinence, and screening method for compounds contained in the pharmaceutical composition", published 16 January 2014, assigned to Astellas Pharma Inc.

fiercebiotech.com

"PRESS RELEASE: Tikvah Therapeutics Signs Agreement with Phase 2 Discovery". fiercebiotech.com. 29 August 2007. Archived from the original on 2018-11-01. Retrieved 7 April 2015.

globenewswire.com

"Tikvah Therapeutics Signs Agreement to Develop and Commercialize LY156735, a Second Generation Melatonin Agonist, for Circadian Rhythm and Sleep Disorders". Nasdaq Global Newswire (Press release). 2007-08-29.

handle.net

hdl.handle.net

Rivara S, Pala D, Bedini A, Spadoni G (April 2015). "Therapeutic uses of melatonin and melatonin derivatives: a patent review (2012 - 2014)". Expert Opinion on Therapeutic Patents. 25 (4): 425–441. doi:10.1517/13543776.2014.1001739. hdl:11576/2623397. PMID 25579320. S2CID 19644131.

nih.gov

pubmed.ncbi.nlm.nih.gov

Rivara S, Mor M, Bedini A, Spadoni G, Tarzia G (2008). "Melatonin receptor agonists: SAR and applications to the treatment of sleep-wake disorders". Current Topics in Medicinal Chemistry. 8 (11): 954–968. doi:10.2174/156802608784936719. PMID 18673165.
Kostiuk NV, Belyakova MB, Leshchenko DV, Zhigulina VV, Miniaev MV (2014). "Synthetic melatoninergic ligands: achievements and prospects". ISRN Biochemistry. 2014: 843478. doi:10.1155/2014/843478. PMC 4393004. PMID 25937968.
Zlotos DP (2012). "Recent progress in the development of agonists and antagonists for melatonin receptors". Current Medicinal Chemistry. 19 (21): 3532–3549. doi:10.2174/092986712801323153. PMID 22680635.
Carocci A, Catalano A, Sinicropi MS (2014). "Melatonergic drugs in development". Clinical Pharmacology. 6: 127–137. doi:10.2147/CPAA.S36600. PMC 4172069. PMID 25258560.
Zlotos DP, Jockers R, Cecon E, Rivara S, Witt-Enderby PA (April 2014). "MT1 and MT2 melatonin receptors: ligands, models, oligomers, and therapeutic potential". Journal of Medicinal Chemistry. 57 (8): 3161–3185. doi:10.1021/jm401343c. PMID 24228714.
Hardeland R, Poeggeler B (September 2012). "Melatonin and synthetic melatonergic agonists: actions and metabolism in the central nervous system". Central Nervous System Agents in Medicinal Chemistry. 12 (3): 189–216. doi:10.2174/187152412802430129. PMID 22640220.
Chan KH, Hu Y, Ho MK, Wong YH (2013). "Characterization of substituted phenylpropylamides as highly selective agonists at the melatonin MT2 receptor". Current Medicinal Chemistry. 20 (2): 289–300. doi:10.2174/0929867311320020009. PMID 23131177.
Mulchahey JJ, Goldwater DR, Zemlan FP (August 2004). "A single blind, placebo controlled, across groups dose escalation study of the safety, tolerability, pharmacokinetics and pharmacodynamics of the melatonin analog beta-methyl-6-chloromelatonin". Life Sciences. 75 (15): 1843–1856. doi:10.1016/j.lfs.2004.03.023. PMID 15302228.
Nickelsen T, Samel A, Vejvoda M, Wenzel J, Smith B, Gerzer R (September 2002). "Chronobiotic effects of the melatonin agonist LY 156735 following a simulated 9h time shift: results of a placebo-controlled trial". Chronobiology International. 19 (5): 915–936. doi:10.1081/cbi-120014108. PMID 12405554. S2CID 10363563.
Cardinali DP, Srinivasan V, Brzezinski A, Brown GM (May 2012). "Melatonin and its analogs in insomnia and depression" (PDF). Journal of Pineal Research. 52 (4): 365–375. doi:10.1111/j.1600-079x.2011.00962.x. PMID 21951153. S2CID 139480.
Zemlan FP, Mulchahey JJ, Scharf MB, Mayleben DW, Rosenberg R, Lankford A (March 2005). "The efficacy and safety of the melatonin agonist beta-methyl-6-chloromelatonin in primary insomnia: a randomized, placebo-controlled, crossover clinical trial". The Journal of Clinical Psychiatry. 66 (3): 384–390. doi:10.4088/jcp.v66n0316. PMID 15766306.
Turek FW, Gillette MU (November 2004). "Melatonin, sleep, and circadian rhythms: rationale for development of specific melatonin agonists". Sleep Medicine. 5 (6): 523–532. doi:10.1016/j.sleep.2004.07.009. PMID 15511698.
Doghramji K (August 2007). "Melatonin and its receptors: a new class of sleep-promoting agents". Journal of Clinical Sleep Medicine. 3 (5 Suppl): S17–S23. doi:10.5664/jcsm.26932. PMC 1978320. PMID 17824497.
Rivara S, Pala D, Bedini A, Spadoni G (April 2015). "Therapeutic uses of melatonin and melatonin derivatives: a patent review (2012 - 2014)". Expert Opinion on Therapeutic Patents. 25 (4): 425–441. doi:10.1517/13543776.2014.1001739. hdl:11576/2623397. PMID 25579320. S2CID 19644131.
Fee DB, Swartz KR, Scheff N, Roberts K, Gabbita P, Scheff S (June 2010). "Melatonin-analog, beta-methyl-6-chloromelatonin, supplementation in spinal cord injury". Brain Research. 1340: 81–85. doi:10.1016/j.brainres.2010.04.047. PMID 20420812. S2CID 27784753.

ncbi.nlm.nih.gov

Kostiuk NV, Belyakova MB, Leshchenko DV, Zhigulina VV, Miniaev MV (2014). "Synthetic melatoninergic ligands: achievements and prospects". ISRN Biochemistry. 2014: 843478. doi:10.1155/2014/843478. PMC 4393004. PMID 25937968.
Carocci A, Catalano A, Sinicropi MS (2014). "Melatonergic drugs in development". Clinical Pharmacology. 6: 127–137. doi:10.2147/CPAA.S36600. PMC 4172069. PMID 25258560.
Doghramji K (August 2007). "Melatonin and its receptors: a new class of sleep-promoting agents". Journal of Clinical Sleep Medicine. 3 (5 Suppl): S17–S23. doi:10.5664/jcsm.26932. PMC 1978320. PMID 17824497.

prnewswire.com

"Phase 2 Discovery, Inc. Acquires Drug in Clinical Development to Treat Sleep Disorders". Phase 2 Discovery, Inc. Acquires Drug in Clinical Development to Treat Sleep Disorders. Archived from the original on 2016-10-30. Retrieved 15 March 2015.

semanticscholar.org

api.semanticscholar.org

Nickelsen T, Samel A, Vejvoda M, Wenzel J, Smith B, Gerzer R (September 2002). "Chronobiotic effects of the melatonin agonist LY 156735 following a simulated 9h time shift: results of a placebo-controlled trial". Chronobiology International. 19 (5): 915–936. doi:10.1081/cbi-120014108. PMID 12405554. S2CID 10363563.
Cardinali DP, Srinivasan V, Brzezinski A, Brown GM (May 2012). "Melatonin and its analogs in insomnia and depression" (PDF). Journal of Pineal Research. 52 (4): 365–375. doi:10.1111/j.1600-079x.2011.00962.x. PMID 21951153. S2CID 139480.
Rivara S, Pala D, Bedini A, Spadoni G (April 2015). "Therapeutic uses of melatonin and melatonin derivatives: a patent review (2012 - 2014)". Expert Opinion on Therapeutic Patents. 25 (4): 425–441. doi:10.1517/13543776.2014.1001739. hdl:11576/2623397. PMID 25579320. S2CID 19644131.
Fee DB, Swartz KR, Scheff N, Roberts K, Gabbita P, Scheff S (June 2010). "Melatonin-analog, beta-methyl-6-chloromelatonin, supplementation in spinal cord injury". Brain Research. 1340: 81–85. doi:10.1016/j.brainres.2010.04.047. PMID 20420812. S2CID 27784753.

uca.edu.ar

repositorio.uca.edu.ar

Cardinali DP, Srinivasan V, Brzezinski A, Brown GM (May 2012). "Melatonin and its analogs in insomnia and depression" (PDF). Journal of Pineal Research. 52 (4): 365–375. doi:10.1111/j.1600-079x.2011.00962.x. PMID 21951153. S2CID 139480.

web.archive.org

"PD-6735, LY-156735,118702-11-7,C14-H17-Cl-N2-O2,N-[2(R)-(6-C--药物合成数据库". Archived from the original on 2009-09-27.
"Phase 2 Discovery, Inc. Acquires Drug in Clinical Development to Treat Sleep Disorders". Phase 2 Discovery, Inc. Acquires Drug in Clinical Development to Treat Sleep Disorders. Archived from the original on 2016-10-30. Retrieved 15 March 2015.
"Phase 2 Discovery, Inc. Receives Orphan Drug Designation From FDA For Synthetic Melatonin Analog PD-6735". BioSpace. 19 October 2005. Archived from the original on 4 March 2016.
"PRESS RELEASE: Tikvah Therapeutics Signs Agreement with Phase 2 Discovery". fiercebiotech.com. 29 August 2007. Archived from the original on 2018-11-01. Retrieved 7 April 2015.