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Burris HA, Hurwitz HI, Dees EC, et al. (agosto de 2005). «Phase I safety, pharmacokinetics, and clinical activity study of lapatinib (GW572016), a reversible dual inhibitor of epidermal growth factor receptor tyrosine kinases, in heavily pretreated patients with metastatic carcinomas». J. Clin. Oncol.23 (23): 5305-13. PMID15955900. doi:10.1200/JCO.2005.16.584.
«Data Sheet: TYKERB». Medsafe. New Zealand Medicines and Medical Devices Safety Authority. 12 de marzo de 2008. Archivado desde el original el 14 de octubre de 2008. Retrieved December 2, 2008.
Wood ER, Truesdale AT, McDonald OB, Yuan D, Hassell A, Dickerson SH, Ellis B, Pennisi C, Horne E, Lackey K, Alligood KJ, Rusnak DW, Gilmer TM, Shewchuk L. A unique structure for epidermal growth factor receptor bound to GW572016 (Lapatinib): relationships among protein conformation, inhibitor off-rate, and receptor activity in tumor cells. Cancer Res. 2004 Sep 15;64(18):6652-9. PMID 15374980
Geyer CE, Forster J, Lindquist D, et al. (diciembre de 2006). «Lapatinib plus capecitabine for HER2-positive advanced breast cancer». N. Engl. J. Med.355 (26): 2733-43. PMID17192538. doi:10.1056/NEJMoa064320.
Burris HA, Hurwitz HI, Dees EC, et al. (agosto de 2005). «Phase I safety, pharmacokinetics, and clinical activity study of lapatinib (GW572016), a reversible dual inhibitor of epidermal growth factor receptor tyrosine kinases, in heavily pretreated patients with metastatic carcinomas». J. Clin. Oncol.23 (23): 5305-13. PMID15955900. doi:10.1200/JCO.2005.16.584.
«Data Sheet: TYKERB». Medsafe. New Zealand Medicines and Medical Devices Safety Authority. 12 de marzo de 2008. Archivado desde el original el 14 de octubre de 2008. Retrieved December 2, 2008.