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(en) Asher Mullard, « First targeted protein degrader hits the clinic », Nature Reviews Drug Discovery, vol. 18, no 4, , p. 237–239 (DOI10.1038/d41573-019-00043-6, lire en ligne, consulté le )
Ian Churcher, « Protac-Induced Protein Degradation in Drug Discovery: Breaking the Rules or Just Making New Ones? », Journal of Medicinal Chemistry, vol. 61, no 2, , p. 444–452 (ISSN0022-2623, DOI10.1021/acs.jmedchem.7b01272, lire en ligne, consulté le )
doi.org
Ian Churcher, « Protac-Induced Protein Degradation in Drug Discovery: Breaking the Rules or Just Making New Ones? », Journal of Medicinal Chemistry, vol. 61, no 2, , p. 444–452 (ISSN0022-2623, DOI10.1021/acs.jmedchem.7b01272, lire en ligne, consulté le )
David B. Beck, Achim Werner, Daniel L. Kastner et Ivona Aksentijevich, « Disorders of ubiquitylation: unchained inflammation », Nature Reviews Rheumatology, vol. 18, no 8, , p. 435–447 (ISSN1759-4790 et 1759-4804, DOI10.1038/s41584-022-00778-4, lire en ligne, consulté le )
Ian Churcher, « Protac-Induced Protein Degradation in Drug Discovery: Breaking the Rules or Just Making New Ones? », Journal of Medicinal Chemistry, vol. 61, no 2, , p. 444–452 (ISSN0022-2623, DOI10.1021/acs.jmedchem.7b01272, lire en ligne, consulté le )
(en) Asher Mullard, « First targeted protein degrader hits the clinic », Nature Reviews Drug Discovery, vol. 18, no 4, , p. 237–239 (DOI10.1038/d41573-019-00043-6, lire en ligne, consulté le )