Holinka CF, Diczfalusy E, Coelingh Bennink HJ (maio de 2008). "Estetrol: a unique steroid in human pregnancy". The Journal of Steroid Biochemistry and Molecular Biology110 (1–2): 138–143. PMID18462934. doi:10.1016/j.jsbmb.2008.03.027.
Heikkilä J, Luukkainen T (xuño de 1971). "Urinary excretion of estriol and 15 alpha-hydroxyestriol in complicated pregnancies". American Journal of Obstetrics and Gynecology110 (4): 509–21. PMID5582006. doi:10.1016/0002-9378(71)90692-2.
Visser M, Foidart JM, Coelingh Bennink HJ (2008). "In vitro effects of estetrol on receptor binding, drug targets and human liver cell metabolism". Climacteric11 (Suppl 1): 64–68. PMID18464025. doi:10.1080/13697130802050340.
Gérard C, Blacher S, Communal L, Courtin A, Tskitishvili E, Mestdagt M, et al. (xaneiro de 2015). "Estetrol is a weak estrogen antagonizing estradiol-dependent mammary gland proliferation". The Journal of Endocrinology224 (1): 85–95. PMID25359896. doi:10.1530/JOE-14-0549.
Pluchino N, Santoro AN, Casarosa E, Giannini A, Genazzani A, Russo M, et al. (setembro de 2014). "Effect of estetrol administration on brain and serum allopregnanolone in intact and ovariectomized rats". The Journal of Steroid Biochemistry and Molecular Biology143: 285–290. PMID24787659. doi:10.1016/j.jsbmb.2014.04.011.
Coelingh Bennink HJ, Heegaard AM, Visser M, Holinka CF, Christiansen C (2008-01-01). "Oral bioavailability and bone-sparing effects of estetrol in an osteoporosis model". Climacteric11 (sup1): 2–14. PMID18464016. doi:10.1080/13697130701798692.
Benoit T, Valera MC, Fontaine C, Buscato M, Lenfant F, Raymond-Letron I, et al. (novembro de 2017). "Estetrol, a Fetal Selective Estrogen Receptor Modulator, Acts on the Vagina of Mice through Nuclear Estrogen Receptor α Activation". The American Journal of Pathology(en English)187 (11): 2499–2507. PMID28827141. doi:10.1016/j.ajpath.2017.07.013.
Klipping C, Duijkers I, Mawet M, Maillard C, Bastidas A, Jost M, Foidart JM (abril de 2021). "Endocrine and metabolic effects of an oral contraceptive containing estetrol and drospirenone". Contraception103 (4): 213–221. PMID33428907. doi:10.1016/j.contraception.2021.01.001.
Gérard C, Arnal JF, Jost M, Douxfils J, Lenfant F, Fontaine C, et al. (febreiro de 2022). "Profile of estetrol, a promising native estrogen for oral contraception and the relief of climacteric symptoms of menopause". Expert Review of Clinical Pharmacology15 (2): 121–137. PMID35306927. doi:10.1080/17512433.2022.2054413.
Schwers J, Eriksson G, Diczfalusy E (abril de 1965). "15a-hydroxylation: A new pathway of estrogen metabolism in the human fetus and newborn". Biochimica et Biophysica Acta100: 313–6. PMID14323645. doi:10.1016/0304-4165(65)90464-2.
Schwers J, Govaerts-Videtsky M, Wiqvist N, Diczfalusy E (decembro de 1965). "Metabolism of oestrone sulphate by the previable human foetus". Acta Endocrinologica50 (4): 597–610. PMID5897909. doi:10.1530/acta.0.0500597.
Mancuso S, Benagiano G, Dell'Acqua S, Shapiro M, Wiqvist N, Diczfalusy E (febreiro de 1968). "Studies on the metabolism of C-19 steroids in the human foeto-placental unit. 4. Aromatisation and hydroxylation products formed by previable foetuses perfused withandrostenedione and testosterone". Acta Endocrinologica57 (2): 208–27. PMID4229819. doi:10.1530/acta.0.0570208.
Heikkilä J, Adlercreutz H (setembro de 1970). "A method for the determination of urinary 15α-hydroxyestriol and estriol: Preliminary results of 15α-hydroxyestriol determinations in pregnancy urine.". Journal of Steroid Biochemistry1 (3): 243–253. doi:10.1016/0022-4731(70)90020-8.
Heikkilä J (febreiro de 1971). "Excretion of 15α-hydroxyestriol and estriol in maternal urine during normal pregnancy.". Journal of Steroid Biochemistry2 (83–93): 83–93. doi:10.1016/0022-4731(71)90012-4.
Visser M, Holinka CF, Coelingh Bennink HJ (2008). "First human exposure to exogenous single-dose oral estetrol in early postmenopausal women". Climacteric. 11 Suppl 1: 31–40. PMID18464021. doi:10.1080/13697130802056511.
Hammond GL, Hogeveen KN, Visser M, Coelingh Bennink HJ (2008). "Estetrol does not bind sex hormone binding globulin or increase its production by human HepG2 cells". Climacteric. 11 Suppl 1: 41–46. PMID18464022. doi:10.1080/13697130701851814.
Stanczyk FZ, Archer DF, Bhavnani BR (xuño de 2013). "Ethinyl estradiol and 17β-estradiol in combined oral contraceptives: pharmacokinetics, pharmacodynamics and risk assessment". Contraception(en English)87 (6): 706–727. PMID23375353. doi:10.1016/j.contraception.2012.12.011.
Warmerdam EG, Visser M, Coelingh Bennink HJ, Groen M (2008). "A new route of synthesis of estetrol". Climacteric. 11 Suppl 1: 59–63. PMID18464024. doi:10.1080/13697130802054078.
Hagen AA, Barr M, Diczfalusy E (xuño de 1965). "METABOLISM OF 17β-OESTRADIOL-4-14C IN EARLY INFANCY". Acta Endocrinologica49 (2): 207–220. PMID14303250. doi:10.1530/acta.0.0490207.
Zucconi G, Lisboa BP, Simonitsch E, Roth L, Hagen AA, Diczfalusy E (novembro de 1967). "Isolation of 15-alpha-hydroxy-oestriol from pregnancy urine and from the urine of newborn infants". Acta Endocrinologica56 (3): 413–423. PMID6072461. doi:10.1530/acta.0.0560413.
Holinka CF, Diczfalusy E, Coelingh Bennink HJ (maio de 2008). "Estetrol: a unique steroid in human pregnancy". The Journal of Steroid Biochemistry and Molecular Biology110 (1–2): 138–143. PMID18462934. doi:10.1016/j.jsbmb.2008.03.027.
Heikkilä J, Luukkainen T (xuño de 1971). "Urinary excretion of estriol and 15 alpha-hydroxyestriol in complicated pregnancies". American Journal of Obstetrics and Gynecology110 (4): 509–21. PMID5582006. doi:10.1016/0002-9378(71)90692-2.
Visser M, Foidart JM, Coelingh Bennink HJ (2008). "In vitro effects of estetrol on receptor binding, drug targets and human liver cell metabolism". Climacteric11 (Suppl 1): 64–68. PMID18464025. doi:10.1080/13697130802050340.
Gérard C, Blacher S, Communal L, Courtin A, Tskitishvili E, Mestdagt M, et al. (xaneiro de 2015). "Estetrol is a weak estrogen antagonizing estradiol-dependent mammary gland proliferation". The Journal of Endocrinology224 (1): 85–95. PMID25359896. doi:10.1530/JOE-14-0549.
Pluchino N, Santoro AN, Casarosa E, Giannini A, Genazzani A, Russo M, et al. (setembro de 2014). "Effect of estetrol administration on brain and serum allopregnanolone in intact and ovariectomized rats". The Journal of Steroid Biochemistry and Molecular Biology143: 285–290. PMID24787659. doi:10.1016/j.jsbmb.2014.04.011.
Coelingh Bennink HJ, Heegaard AM, Visser M, Holinka CF, Christiansen C (2008-01-01). "Oral bioavailability and bone-sparing effects of estetrol in an osteoporosis model". Climacteric11 (sup1): 2–14. PMID18464016. doi:10.1080/13697130701798692.
Benoit T, Valera MC, Fontaine C, Buscato M, Lenfant F, Raymond-Letron I, et al. (novembro de 2017). "Estetrol, a Fetal Selective Estrogen Receptor Modulator, Acts on the Vagina of Mice through Nuclear Estrogen Receptor α Activation". The American Journal of Pathology(en English)187 (11): 2499–2507. PMID28827141. doi:10.1016/j.ajpath.2017.07.013.
Klipping C, Duijkers I, Mawet M, Maillard C, Bastidas A, Jost M, Foidart JM (abril de 2021). "Endocrine and metabolic effects of an oral contraceptive containing estetrol and drospirenone". Contraception103 (4): 213–221. PMID33428907. doi:10.1016/j.contraception.2021.01.001.
Gérard C, Arnal JF, Jost M, Douxfils J, Lenfant F, Fontaine C, et al. (febreiro de 2022). "Profile of estetrol, a promising native estrogen for oral contraception and the relief of climacteric symptoms of menopause". Expert Review of Clinical Pharmacology15 (2): 121–137. PMID35306927. doi:10.1080/17512433.2022.2054413.
Schwers J, Eriksson G, Diczfalusy E (abril de 1965). "15a-hydroxylation: A new pathway of estrogen metabolism in the human fetus and newborn". Biochimica et Biophysica Acta100: 313–6. PMID14323645. doi:10.1016/0304-4165(65)90464-2.
Schwers J, Govaerts-Videtsky M, Wiqvist N, Diczfalusy E (decembro de 1965). "Metabolism of oestrone sulphate by the previable human foetus". Acta Endocrinologica50 (4): 597–610. PMID5897909. doi:10.1530/acta.0.0500597.
Mancuso S, Benagiano G, Dell'Acqua S, Shapiro M, Wiqvist N, Diczfalusy E (febreiro de 1968). "Studies on the metabolism of C-19 steroids in the human foeto-placental unit. 4. Aromatisation and hydroxylation products formed by previable foetuses perfused withandrostenedione and testosterone". Acta Endocrinologica57 (2): 208–27. PMID4229819. doi:10.1530/acta.0.0570208.
Visser M, Holinka CF, Coelingh Bennink HJ (2008). "First human exposure to exogenous single-dose oral estetrol in early postmenopausal women". Climacteric. 11 Suppl 1: 31–40. PMID18464021. doi:10.1080/13697130802056511.
Hammond GL, Hogeveen KN, Visser M, Coelingh Bennink HJ (2008). "Estetrol does not bind sex hormone binding globulin or increase its production by human HepG2 cells". Climacteric. 11 Suppl 1: 41–46. PMID18464022. doi:10.1080/13697130701851814.
Stanczyk FZ, Archer DF, Bhavnani BR (xuño de 2013). "Ethinyl estradiol and 17β-estradiol in combined oral contraceptives: pharmacokinetics, pharmacodynamics and risk assessment". Contraception(en English)87 (6): 706–727. PMID23375353. doi:10.1016/j.contraception.2012.12.011.
Warmerdam EG, Visser M, Coelingh Bennink HJ, Groen M (2008). "A new route of synthesis of estetrol". Climacteric. 11 Suppl 1: 59–63. PMID18464024. doi:10.1080/13697130802054078.
Hagen AA, Barr M, Diczfalusy E (xuño de 1965). "METABOLISM OF 17β-OESTRADIOL-4-14C IN EARLY INFANCY". Acta Endocrinologica49 (2): 207–220. PMID14303250. doi:10.1530/acta.0.0490207.
Zucconi G, Lisboa BP, Simonitsch E, Roth L, Hagen AA, Diczfalusy E (novembro de 1967). "Isolation of 15-alpha-hydroxy-oestriol from pregnancy urine and from the urine of newborn infants". Acta Endocrinologica56 (3): 413–423. PMID6072461. doi:10.1530/acta.0.0560413.