Լիգանդ (կենսաքիմիա) (Armenian Wikipedia)

Analysis of information sources in references of the Wikipedia article "Լիգանդ (կենսաքիմիա)" in Armenian language version.

refsWebsite

Global rank Armenian rank

41nih.gov

4^th place

3^rd place

28doi.org

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4^th place

7harvard.edu

18^th place

38^th place

3semanticscholar.org

11^th place

428^th place

3jstor.org

26^th place

73^rd place

2web.archive.org

1^st place

1archive.org

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1arxiv.org

69^th place

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1sciencesnail.com

low place

1graphpad.com

low place

1physorg.com

6,156^th place

3,542^nd place

1ufl.edu

921^st place

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1books.google.com

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17^th place

1archives-ouvertes.fr

1,031^st place

3,920^th place

archive.org

Teif VB (October 2005). «Ligand-induced DNA condensation: choosing the model». Biophysical Journal. 89 (4): 2574–87. Bibcode:2005BpJ....89.2574T. doi:10.1529/biophysj.105.063909. PMC 1366757. PMID 16085765.

archives-ouvertes.fr

hal.archives-ouvertes.fr

Soulier JL, Russo O, Giner M, Rivail L, Berthouze M, Ongeri S, Maigret B, Fischmeister R, Lezoualc'h F, Sicsic S, Berque-Bestel I (October 2005). «Design and synthesis of specific probes for human 5-HT4 receptor dimerization studies» (PDF). Journal of Medicinal Chemistry. 48 (20): 6220–8. doi:10.1021/jm050234z. PMID 16190749.

arxiv.org

Teif VB, Rippe K (October 2010). «Statistical-mechanical lattice models for protein-DNA binding in chromatin». Journal of Physics: Condensed Matter. 22 (41): 414105. arXiv:1004.5514. Bibcode:2010JPCM...22O4105T. doi:10.1088/0953-8984/22/41/414105. PMID 21386588. S2CID 103345.

books.google.com

Kenakin TP (November 2006). A pharmacology primer: theory, applications, and methods. Academic Press. էջ 79. ISBN 978-0-12-370599-0.

doi.org

Teif VB (October 2005). «Ligand-induced DNA condensation: choosing the model». Biophysical Journal. 89 (4): 2574–87. Bibcode:2005BpJ....89.2574T. doi:10.1529/biophysj.105.063909. PMC 1366757. PMID 16085765.
Teif VB, Rippe K (October 2010). «Statistical-mechanical lattice models for protein-DNA binding in chromatin». Journal of Physics: Condensed Matter. 22 (41): 414105. arXiv:1004.5514. Bibcode:2010JPCM...22O4105T. doi:10.1088/0953-8984/22/41/414105. PMID 21386588. S2CID 103345.
Baron R, Setny P, McCammon JA (September 2010). «Water in cavity-ligand recognition». Journal of the American Chemical Society. 132 (34): 12091–7. doi:10.1021/ja1050082. PMC 2933114. PMID 20695475.
Baaske P, Wienken CJ, Reineck P, Duhr S, Braun D (March 2010). «Optical thermophoresis for quantifying the buffer dependence of aptamer binding». Angewandte Chemie. 49 (12): 2238–41. doi:10.1002/anie.200903998. PMID 20186894.
- «A hot road to new drugs». Phys.org. 2010 թ․ փետրվարի 24.
- Wienken CJ, Baaske P, Rothbauer U, Braun D, Duhr S (October 2010). «Protein-binding assays in biological liquids using microscale thermophoresis». Nature Communications. 1 (7): 100. Bibcode:2010NatCo...1..100W. doi:10.1038/ncomms1093. PMID 20981028.
- Cabanos, C; Wang, M; Han, X; Hansen, SB (2017 թ․ օգոստոսի 8). «A Soluble Fluorescent Binding Assay Reveals PIP₂ Antagonism of TREK-1 Channels». Cell Reports. 20 (6): 1287–1294. doi:10.1016/j.celrep.2017.07.034. PMC 5586213. PMID 28793254.
- Matera, Carlo; Pucci, Luca; Fiorentini, Chiara; Fucile, Sergio; Missale, Cristina; Grazioso, Giovanni; Clementi, Francesco; Zoli, Michele; De Amici, Marco (2015 թ․ օգոստոսի 28). «Bifunctional compounds targeting both D2 and non-α7 nACh receptors: Design, synthesis and pharmacological characterization». European Journal of Medicinal Chemistry. 101: 367–383. doi:10.1016/j.ejmech.2015.06.039. PMID 26164842.
- Matera, Carlo; Flammini, Lisa; Quadri, Marta; Vivo, Valentina; Ballabeni, Vigilio; Holzgrabe, Ulrike; Mohr, Klaus; De Amici, Marco; Barocelli, Elisabetta (2014 թ․ մարտի 21). «Bis(ammonio)alkane-type agonists of muscarinic acetylcholine receptors: Synthesis, in vitro functional characterization, and in vivo evaluation of their analgesic activity». European Journal of Medicinal Chemistry. 75: 222–232. doi:10.1016/j.ejmech.2014.01.032. PMID 24534538.
- Erez M, Takemori AE, Portoghese PS (July 1982). «Narcotic antagonistic potency of bivalent ligands which contain beta-naltrexamine. Evidence for bridging between proximal recognition sites». Journal of Medicinal Chemistry. 25 (7): 847–9. doi:10.1021/jm00349a016. PMID 7108900.
- Portoghese PS, Ronsisvalle G, Larson DL, Yim CB, Sayre LM, Takemori AE (1982). «Opioid agonist and antagonist bivalent ligands as receptor probes». Life Sciences. 31 (12–13): 1283–6. doi:10.1016/0024-3205(82)90362-9. PMID 6292615.
- Portoghese PS, Akgün E, Lunzer MM (January 2017). «Heteromer Induction: An Approach to Unique Pharmacology?». ACS Chemical Neuroscience. 8 (3): 426–428. doi:10.1021/acschemneuro.7b00002. PMID 28139906.
- Blum JJ, Conn PM (December 1982). «Gonadotropin-releasing hormone stimulation of luteinizing hormone release: A ligand-receptor-effector model». Proceedings of the National Academy of Sciences of the United States of America. 79 (23): 7307–11. Bibcode:1982PNAS...79.7307B. doi:10.1073/pnas.79.23.7307. JSTOR 13076. PMC 347328. PMID 6296828.
- Conn PM, Rogers DC, Stewart JM, Niedel J, Sheffield T (April 1982). «Conversion of a gonadotropin-releasing hormone antagonist to an agonist». Nature. 296 (5858): 653–5. Bibcode:1982Natur.296..653C. doi:10.1038/296653a0. PMID 6280058. S2CID 4303982.
- Nimczick M, Pemp D, Darras FH, Chen X, Heilmann J, Decker M (August 2014). «Synthesis and biological evaluation of bivalent cannabinoid receptor ligands based on hCB₂R selective benzimidazoles reveal unexpected intrinsic properties». Bioorganic & Medicinal Chemistry. 22 (15): 3938–46. doi:10.1016/j.bmc.2014.06.008. PMID 24984935.
- Soulier JL, Russo O, Giner M, Rivail L, Berthouze M, Ongeri S, Maigret B, Fischmeister R, Lezoualc'h F, Sicsic S, Berque-Bestel I (October 2005). «Design and synthesis of specific probes for human 5-HT4 receptor dimerization studies» (PDF). Journal of Medicinal Chemistry. 48 (20): 6220–8. doi:10.1021/jm050234z. PMID 16190749.
- Russo O, Berthouze M, Giner M, Soulier JL, Rivail L, Sicsic S, Lezoualc'h F, Jockers R, Berque-Bestel I (September 2007). «Synthesis of specific bivalent probes that functionally interact with 5-HT(4) receptor dimers». Journal of Medicinal Chemistry. 50 (18): 4482–92. doi:10.1021/jm070552t. PMID 17676726.
- Busnelli M, Kleinau G, Muttenthaler M, Stoev S, Manning M, Bibic L, Howell LA, McCormick PJ, Di Lascio S, Braida D, Sala M, Rovati GE, Bellini T, Chini B (August 2016). «Design and Characterization of Superpotent Bivalent Ligands Targeting Oxytocin Receptor Dimers via a Channel-Like Structure». Journal of Medicinal Chemistry. 59 (15): 7152–66. doi:10.1021/acs.jmedchem.6b00564. PMID 27420737.
- Lensing CJ, Adank DN, Wilber SL, Freeman KT, Schnell SM, Speth RC, Zarth AT, Haskell-Luevano C (February 2017). «A Direct in Vivo Comparison of the Melanocortin Monovalent Agonist Ac-His-DPhe-Arg-Trp-NH2 versus the Bivalent Agonist Ac-His-DPhe-Arg-Trp-PEDG20-His-DPhe-Arg-Trp-NH2: A Bivalent Advantage». ACS Chemical Neuroscience. 8 (6): 1262–1278. doi:10.1021/acschemneuro.6b00399. PMC 5679024. PMID 28128928.
- Xu L, Josan JS, Vagner J, Caplan MR, Hruby VJ, Mash EA, Lynch RM, Morse DL, Gillies RJ (December 2012). «Heterobivalent ligands target cell-surface receptor combinations in vivo». Proceedings of the National Academy of Sciences of the United States of America. 109 (52): 21295–300. Bibcode:2012PNAS..10921295X. doi:10.1073/pnas.1211762109. JSTOR 42553664. PMC 3535626. PMID 23236171.
- Lensing CJ, Freeman KT, Schnell SM, Adank DN, Speth RC, Haskell-Luevano C (April 2016). «An in Vitro and in Vivo Investigation of Bivalent Ligands That Display Preferential Binding and Functional Activity for Different Melanocortin Receptor Homodimers». Journal of Medicinal Chemistry. 59 (7): 3112–28. doi:10.1021/acs.jmedchem.5b01894. PMC 5679017. PMID 26959173.
- Shonberg J, Scammells PJ, Capuano B (June 2011). «Design strategies for bivalent ligands targeting GPCRs». ChemMedChem. 6 (6): 963–74. doi:10.1002/cmdc.201100101. PMID 21520422. S2CID 10561038.
- Berque-Bestel I, Lezoualc'h F, Jockers R (December 2008). «Bivalent ligands as specific pharmacological tools for G protein-coupled receptor dimers». Current Drug Discovery Technologies. 5 (4): 312–8. doi:10.2174/157016308786733591. PMID 19075611.
- Akgün E, Javed MI, Lunzer MM, Powers MD, Sham YY, Watanabe Y, Portoghese PS (November 2015). «Inhibition of Inflammatory and Neuropathic Pain by Targeting a Mu Opioid Receptor/Chemokine Receptor5 Heteromer (MOR-CCR5)». Journal of Medicinal Chemistry. 58 (21): 8647–57. doi:10.1021/acs.jmedchem.5b01245. PMC 5055304. PMID 26451468.
- Smeester BA, Lunzer MM, Akgün E, Beitz AJ, Portoghese PS (November 2014). «Targeting putative mu opioid/metabotropic glutamate receptor-5 heteromers produces potent antinociception in a chronic murine bone cancer model». European Journal of Pharmacology. 743: 48–52. doi:10.1016/j.ejphar.2014.09.008. PMC 4259840. PMID 25239072.
- Daniels DJ, Lenard NR, Etienne CL, Law PY, Roerig SC, Portoghese PS (December 2005). «Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series». Proceedings of the National Academy of Sciences of the United States of America. 102 (52): 19208–13. Bibcode:2005PNAS..10219208D. doi:10.1073/pnas.0506627102. JSTOR 4152590. PMC 1323165. PMID 16365317.
- Abrusan G, Marsh JA (2019). «Ligand Binding Site Structure Shapes Folding, Assembly and Degradation of Homomeric Protein Complexes». Journal of Molecular Biology. 431 (19): 3871–3888. doi:10.1016/j.jmb.2019.07.014. PMC 6739599. PMID 31306664.
- Abrusan G, Marsh JA (2018). «Ligand Binding Site Structure Influences the Evolution of Protein Complex Function and Topology». Cell Reports. 22 (12): 3265–3276. doi:10.1016/j.celrep.2018.02.085. PMC 5873459. PMID 29562182.
- Abrusan G, Marsh JA (2019). «Ligand-Binding-Site Structure Shapes Allosteric Signal Transduction and the Evolution of Allostery in Protein Complexes». Molecular Biology and Evolution. 36 (8): 1711–1727. doi:10.1093/molbev/msz093. PMC 6657754. PMID 31004156.

graphpad.com

See Homologous competitive binding curves Արխիվացված 2007-12-19 Wayback Machine, A complete guide to nonlinear regression, curvefit.com.

harvard.edu

ui.adsabs.harvard.edu

Teif VB (October 2005). «Ligand-induced DNA condensation: choosing the model». Biophysical Journal. 89 (4): 2574–87. Bibcode:2005BpJ....89.2574T. doi:10.1529/biophysj.105.063909. PMC 1366757. PMID 16085765.
Teif VB, Rippe K (October 2010). «Statistical-mechanical lattice models for protein-DNA binding in chromatin». Journal of Physics: Condensed Matter. 22 (41): 414105. arXiv:1004.5514. Bibcode:2010JPCM...22O4105T. doi:10.1088/0953-8984/22/41/414105. PMID 21386588. S2CID 103345.
Wienken CJ, Baaske P, Rothbauer U, Braun D, Duhr S (October 2010). «Protein-binding assays in biological liquids using microscale thermophoresis». Nature Communications. 1 (7): 100. Bibcode:2010NatCo...1..100W. doi:10.1038/ncomms1093. PMID 20981028.
Blum JJ, Conn PM (December 1982). «Gonadotropin-releasing hormone stimulation of luteinizing hormone release: A ligand-receptor-effector model». Proceedings of the National Academy of Sciences of the United States of America. 79 (23): 7307–11. Bibcode:1982PNAS...79.7307B. doi:10.1073/pnas.79.23.7307. JSTOR 13076. PMC 347328. PMID 6296828.
Conn PM, Rogers DC, Stewart JM, Niedel J, Sheffield T (April 1982). «Conversion of a gonadotropin-releasing hormone antagonist to an agonist». Nature. 296 (5858): 653–5. Bibcode:1982Natur.296..653C. doi:10.1038/296653a0. PMID 6280058. S2CID 4303982.
Xu L, Josan JS, Vagner J, Caplan MR, Hruby VJ, Mash EA, Lynch RM, Morse DL, Gillies RJ (December 2012). «Heterobivalent ligands target cell-surface receptor combinations in vivo». Proceedings of the National Academy of Sciences of the United States of America. 109 (52): 21295–300. Bibcode:2012PNAS..10921295X. doi:10.1073/pnas.1211762109. JSTOR 42553664. PMC 3535626. PMID 23236171.
Daniels DJ, Lenard NR, Etienne CL, Law PY, Roerig SC, Portoghese PS (December 2005). «Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series». Proceedings of the National Academy of Sciences of the United States of America. 102 (52): 19208–13. Bibcode:2005PNAS..10219208D. doi:10.1073/pnas.0506627102. JSTOR 4152590. PMC 1323165. PMID 16365317.

jstor.org

Blum JJ, Conn PM (December 1982). «Gonadotropin-releasing hormone stimulation of luteinizing hormone release: A ligand-receptor-effector model». Proceedings of the National Academy of Sciences of the United States of America. 79 (23): 7307–11. Bibcode:1982PNAS...79.7307B. doi:10.1073/pnas.79.23.7307. JSTOR 13076. PMC 347328. PMID 6296828.
Xu L, Josan JS, Vagner J, Caplan MR, Hruby VJ, Mash EA, Lynch RM, Morse DL, Gillies RJ (December 2012). «Heterobivalent ligands target cell-surface receptor combinations in vivo». Proceedings of the National Academy of Sciences of the United States of America. 109 (52): 21295–300. Bibcode:2012PNAS..10921295X. doi:10.1073/pnas.1211762109. JSTOR 42553664. PMC 3535626. PMID 23236171.
Daniels DJ, Lenard NR, Etienne CL, Law PY, Roerig SC, Portoghese PS (December 2005). «Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series». Proceedings of the National Academy of Sciences of the United States of America. 102 (52): 19208–13. Bibcode:2005PNAS..10219208D. doi:10.1073/pnas.0506627102. JSTOR 4152590. PMC 1323165. PMID 16365317.

nih.gov

pubmed.ncbi.nlm.nih.gov

Teif VB (October 2005). «Ligand-induced DNA condensation: choosing the model». Biophysical Journal. 89 (4): 2574–87. Bibcode:2005BpJ....89.2574T. doi:10.1529/biophysj.105.063909. PMC 1366757. PMID 16085765.
Teif VB, Rippe K (October 2010). «Statistical-mechanical lattice models for protein-DNA binding in chromatin». Journal of Physics: Condensed Matter. 22 (41): 414105. arXiv:1004.5514. Bibcode:2010JPCM...22O4105T. doi:10.1088/0953-8984/22/41/414105. PMID 21386588. S2CID 103345.
Baron R, Setny P, McCammon JA (September 2010). «Water in cavity-ligand recognition». Journal of the American Chemical Society. 132 (34): 12091–7. doi:10.1021/ja1050082. PMC 2933114. PMID 20695475.
Baaske P, Wienken CJ, Reineck P, Duhr S, Braun D (March 2010). «Optical thermophoresis for quantifying the buffer dependence of aptamer binding». Angewandte Chemie. 49 (12): 2238–41. doi:10.1002/anie.200903998. PMID 20186894.
- «A hot road to new drugs». Phys.org. 2010 թ․ փետրվարի 24.
- Wienken CJ, Baaske P, Rothbauer U, Braun D, Duhr S (October 2010). «Protein-binding assays in biological liquids using microscale thermophoresis». Nature Communications. 1 (7): 100. Bibcode:2010NatCo...1..100W. doi:10.1038/ncomms1093. PMID 20981028.
- Cabanos, C; Wang, M; Han, X; Hansen, SB (2017 թ․ օգոստոսի 8). «A Soluble Fluorescent Binding Assay Reveals PIP₂ Antagonism of TREK-1 Channels». Cell Reports. 20 (6): 1287–1294. doi:10.1016/j.celrep.2017.07.034. PMC 5586213. PMID 28793254.
- Matera, Carlo; Pucci, Luca; Fiorentini, Chiara; Fucile, Sergio; Missale, Cristina; Grazioso, Giovanni; Clementi, Francesco; Zoli, Michele; De Amici, Marco (2015 թ․ օգոստոսի 28). «Bifunctional compounds targeting both D2 and non-α7 nACh receptors: Design, synthesis and pharmacological characterization». European Journal of Medicinal Chemistry. 101: 367–383. doi:10.1016/j.ejmech.2015.06.039. PMID 26164842.
- Matera, Carlo; Flammini, Lisa; Quadri, Marta; Vivo, Valentina; Ballabeni, Vigilio; Holzgrabe, Ulrike; Mohr, Klaus; De Amici, Marco; Barocelli, Elisabetta (2014 թ․ մարտի 21). «Bis(ammonio)alkane-type agonists of muscarinic acetylcholine receptors: Synthesis, in vitro functional characterization, and in vivo evaluation of their analgesic activity». European Journal of Medicinal Chemistry. 75: 222–232. doi:10.1016/j.ejmech.2014.01.032. PMID 24534538.
- Erez M, Takemori AE, Portoghese PS (July 1982). «Narcotic antagonistic potency of bivalent ligands which contain beta-naltrexamine. Evidence for bridging between proximal recognition sites». Journal of Medicinal Chemistry. 25 (7): 847–9. doi:10.1021/jm00349a016. PMID 7108900.
- Portoghese PS, Ronsisvalle G, Larson DL, Yim CB, Sayre LM, Takemori AE (1982). «Opioid agonist and antagonist bivalent ligands as receptor probes». Life Sciences. 31 (12–13): 1283–6. doi:10.1016/0024-3205(82)90362-9. PMID 6292615.
- Portoghese PS, Akgün E, Lunzer MM (January 2017). «Heteromer Induction: An Approach to Unique Pharmacology?». ACS Chemical Neuroscience. 8 (3): 426–428. doi:10.1021/acschemneuro.7b00002. PMID 28139906.
- Blum JJ, Conn PM (December 1982). «Gonadotropin-releasing hormone stimulation of luteinizing hormone release: A ligand-receptor-effector model». Proceedings of the National Academy of Sciences of the United States of America. 79 (23): 7307–11. Bibcode:1982PNAS...79.7307B. doi:10.1073/pnas.79.23.7307. JSTOR 13076. PMC 347328. PMID 6296828.
- Conn PM, Rogers DC, Stewart JM, Niedel J, Sheffield T (April 1982). «Conversion of a gonadotropin-releasing hormone antagonist to an agonist». Nature. 296 (5858): 653–5. Bibcode:1982Natur.296..653C. doi:10.1038/296653a0. PMID 6280058. S2CID 4303982.
- Nimczick M, Pemp D, Darras FH, Chen X, Heilmann J, Decker M (August 2014). «Synthesis and biological evaluation of bivalent cannabinoid receptor ligands based on hCB₂R selective benzimidazoles reveal unexpected intrinsic properties». Bioorganic & Medicinal Chemistry. 22 (15): 3938–46. doi:10.1016/j.bmc.2014.06.008. PMID 24984935.
- Soulier JL, Russo O, Giner M, Rivail L, Berthouze M, Ongeri S, Maigret B, Fischmeister R, Lezoualc'h F, Sicsic S, Berque-Bestel I (October 2005). «Design and synthesis of specific probes for human 5-HT4 receptor dimerization studies» (PDF). Journal of Medicinal Chemistry. 48 (20): 6220–8. doi:10.1021/jm050234z. PMID 16190749.
- Russo O, Berthouze M, Giner M, Soulier JL, Rivail L, Sicsic S, Lezoualc'h F, Jockers R, Berque-Bestel I (September 2007). «Synthesis of specific bivalent probes that functionally interact with 5-HT(4) receptor dimers». Journal of Medicinal Chemistry. 50 (18): 4482–92. doi:10.1021/jm070552t. PMID 17676726.
- Busnelli M, Kleinau G, Muttenthaler M, Stoev S, Manning M, Bibic L, Howell LA, McCormick PJ, Di Lascio S, Braida D, Sala M, Rovati GE, Bellini T, Chini B (August 2016). «Design and Characterization of Superpotent Bivalent Ligands Targeting Oxytocin Receptor Dimers via a Channel-Like Structure». Journal of Medicinal Chemistry. 59 (15): 7152–66. doi:10.1021/acs.jmedchem.6b00564. PMID 27420737.
- Lensing CJ, Adank DN, Wilber SL, Freeman KT, Schnell SM, Speth RC, Zarth AT, Haskell-Luevano C (February 2017). «A Direct in Vivo Comparison of the Melanocortin Monovalent Agonist Ac-His-DPhe-Arg-Trp-NH2 versus the Bivalent Agonist Ac-His-DPhe-Arg-Trp-PEDG20-His-DPhe-Arg-Trp-NH2: A Bivalent Advantage». ACS Chemical Neuroscience. 8 (6): 1262–1278. doi:10.1021/acschemneuro.6b00399. PMC 5679024. PMID 28128928.
- Xu L, Josan JS, Vagner J, Caplan MR, Hruby VJ, Mash EA, Lynch RM, Morse DL, Gillies RJ (December 2012). «Heterobivalent ligands target cell-surface receptor combinations in vivo». Proceedings of the National Academy of Sciences of the United States of America. 109 (52): 21295–300. Bibcode:2012PNAS..10921295X. doi:10.1073/pnas.1211762109. JSTOR 42553664. PMC 3535626. PMID 23236171.
- Lensing CJ, Freeman KT, Schnell SM, Adank DN, Speth RC, Haskell-Luevano C (April 2016). «An in Vitro and in Vivo Investigation of Bivalent Ligands That Display Preferential Binding and Functional Activity for Different Melanocortin Receptor Homodimers». Journal of Medicinal Chemistry. 59 (7): 3112–28. doi:10.1021/acs.jmedchem.5b01894. PMC 5679017. PMID 26959173.
- Shonberg J, Scammells PJ, Capuano B (June 2011). «Design strategies for bivalent ligands targeting GPCRs». ChemMedChem. 6 (6): 963–74. doi:10.1002/cmdc.201100101. PMID 21520422. S2CID 10561038.
- Berque-Bestel I, Lezoualc'h F, Jockers R (December 2008). «Bivalent ligands as specific pharmacological tools for G protein-coupled receptor dimers». Current Drug Discovery Technologies. 5 (4): 312–8. doi:10.2174/157016308786733591. PMID 19075611.
- Akgün E, Javed MI, Lunzer MM, Powers MD, Sham YY, Watanabe Y, Portoghese PS (November 2015). «Inhibition of Inflammatory and Neuropathic Pain by Targeting a Mu Opioid Receptor/Chemokine Receptor5 Heteromer (MOR-CCR5)». Journal of Medicinal Chemistry. 58 (21): 8647–57. doi:10.1021/acs.jmedchem.5b01245. PMC 5055304. PMID 26451468.
- Smeester BA, Lunzer MM, Akgün E, Beitz AJ, Portoghese PS (November 2014). «Targeting putative mu opioid/metabotropic glutamate receptor-5 heteromers produces potent antinociception in a chronic murine bone cancer model». European Journal of Pharmacology. 743: 48–52. doi:10.1016/j.ejphar.2014.09.008. PMC 4259840. PMID 25239072.
- Daniels DJ, Lenard NR, Etienne CL, Law PY, Roerig SC, Portoghese PS (December 2005). «Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series». Proceedings of the National Academy of Sciences of the United States of America. 102 (52): 19208–13. Bibcode:2005PNAS..10219208D. doi:10.1073/pnas.0506627102. JSTOR 4152590. PMC 1323165. PMID 16365317.
- Abrusan G, Marsh JA (2019). «Ligand Binding Site Structure Shapes Folding, Assembly and Degradation of Homomeric Protein Complexes». Journal of Molecular Biology. 431 (19): 3871–3888. doi:10.1016/j.jmb.2019.07.014. PMC 6739599. PMID 31306664.
- Abrusan G, Marsh JA (2018). «Ligand Binding Site Structure Influences the Evolution of Protein Complex Function and Topology». Cell Reports. 22 (12): 3265–3276. doi:10.1016/j.celrep.2018.02.085. PMC 5873459. PMID 29562182.
- Abrusan G, Marsh JA (2019). «Ligand-Binding-Site Structure Shapes Allosteric Signal Transduction and the Evolution of Allostery in Protein Complexes». Molecular Biology and Evolution. 36 (8): 1711–1727. doi:10.1093/molbev/msz093. PMC 6657754. PMID 31004156.
ncbi.nlm.nih.gov
- Teif VB (October 2005). «Ligand-induced DNA condensation: choosing the model». Biophysical Journal. 89 (4): 2574–87. Bibcode:2005BpJ....89.2574T. doi:10.1529/biophysj.105.063909. PMC 1366757. PMID 16085765.
- Baron R, Setny P, McCammon JA (September 2010). «Water in cavity-ligand recognition». Journal of the American Chemical Society. 132 (34): 12091–7. doi:10.1021/ja1050082. PMC 2933114. PMID 20695475.
- Cabanos, C; Wang, M; Han, X; Hansen, SB (2017 թ․ օգոստոսի 8). «A Soluble Fluorescent Binding Assay Reveals PIP₂ Antagonism of TREK-1 Channels». Cell Reports. 20 (6): 1287–1294. doi:10.1016/j.celrep.2017.07.034. PMC 5586213. PMID 28793254.
- Blum JJ, Conn PM (December 1982). «Gonadotropin-releasing hormone stimulation of luteinizing hormone release: A ligand-receptor-effector model». Proceedings of the National Academy of Sciences of the United States of America. 79 (23): 7307–11. Bibcode:1982PNAS...79.7307B. doi:10.1073/pnas.79.23.7307. JSTOR 13076. PMC 347328. PMID 6296828.
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Vu-Quoc, L., Configuration integral (statistical mechanics), 2008. this wiki site is down; see this article in the web archive on 2012 April 28.