3C様プロテアーゼ (Japanese Wikipedia)

Analysis of information sources in references of the Wikipedia article "3C様プロテアーゼ" in Japanese language version.

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clinicaltrials.gov

Pfizer (2021-06-23). A PHASE 1B, 2-PART, DOUBLE-BLIND, PLACEBO-CONTROLLED, SPONSOR-OPEN STUDY, TO EVALUATE THE SAFETY, TOLERABILITY AND PHARMACOKINETICS OF SINGLE ASCENDING (24-HOUR, PART 1) AND MULTIPLE ASCENDING (120-HOUR, PART 2) INTRAVENOUS INFUSIONS OF PF-07304814 IN HOSPITALIZED PARTICIPANTS WITH COVID-19.

doi.org

Goetz DH, Choe Y, Hansell E, Chen YT, McDowell M, Jonsson CB, Roush WR, McKerrow J, Craik CS (July 2007). “Substrate specificity profiling and identification of a new class of inhibitor for the major protease of the SARS coronavirus”. Biochemistry 46 (30): 8744–52. doi:10.1021/bi0621415. PMID 17605471.
Fan K, Wei P, Feng Q, Chen S, Huang C, Ma L, Lai B, Pei J, Liu Y, Chen J, Lai L (January 2004). “Biosynthesis, purification, and substrate specificity of severe acute respiratory syndrome coronavirus 3C-like proteinase”. The Journal of Biological Chemistry 279 (3): 1637–42. doi:10.1074/jbc.m310875200. PMC 7980035. PMID 14561748.
Akaji K, Konno H, Onozuka M, Makino A, Saito H, Nosaka K (November 2008). “Evaluation of peptide-aldehyde inhibitors using R188I mutant of SARS 3CL protease as a proteolysis-resistant mutant”. Bioorganic & Medicinal Chemistry 16 (21): 9400–8. doi:10.1016/j.bmc.2008.09.057. PMC 7126698. PMID 18845442.
Fehr AR, Perlman S (2015). “Coronaviruses: an overview of their replication and pathogenesis”. Coronaviruses. Methods in Molecular Biology. 1282. Springer. pp. 1–23. doi:10.1007/978-1-4939-2438-7_1. ISBN 978-1-4939-2438-7. PMC 4369385. PMID 25720466. "See section: Virion Structure."
Ryu, Young Bae; Park, Su-Jin; Kim, Young Min; Lee, Ju-Yeon; Seo, Woo Duck; Chang, Jong Sun; Park, Ki Hun; Rho, Mun-Chual et al. (2010-03-15). “SARS-CoV 3CLpro inhibitory effects of quinone-methide triterpenes from Tripterygium regelii” (英語). Bioorganic & Medicinal Chemistry Letters 20 (6): 1873–1876. doi:10.1016/j.bmcl.2010.01.152. ISSN 0960-894X. PMC 7127101. PMID 20167482.
Ocain TD, Rich DH (February 1992). “alpha-Keto amide inhibitors of aminopeptidases”. Journal of Medicinal Chemistry 35 (3): 451–6. doi:10.1021/jm00081a005. PMID 1738140.
Anand K, Ziebuhr J, Wadhwani P, Mesters JR, Hilgenfeld R (June 2003). “Coronavirus main proteinase (3CLpro) structure: basis for design of anti-SARS drugs”. Science 300 (5626): 1763–7. Bibcode: 2003Sci...300.1763A. doi:10.1126/science.1085658. PMID 12746549.
Pacifico S, Ferretti V, Albanese V, Fantinati A, Gallerani E, Nicoli F, Gavioli R, Zamberlan F, Preti D, Marastoni M (July 2019). “Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors”. ACS Medicinal Chemistry Letters 10 (7): 1086–1092. doi:10.1021/acsmedchemlett.9b00233. PMC 6627721. PMID 31312413.
Kusov Y, Tan J, Alvarez E, Enjuanes L, Hilgenfeld R (October 2015). “A G-quadruplex-binding macrodomain within the "SARS-unique domain" is essential for the activity of the SARS-coronavirus replication-transcription complex”. Virology 484: 313–22. doi:10.1016/j.virol.2015.06.016. PMC 4567502. PMID 26149721.
Zhang L, Lin D, Kusov Y, Nian Y, Ma Q, Wang J, von Brunn A, Leyssen P, Lanko K, Neyts J, de Wilde A, Snijder EJ, Liu H, Hilgenfeld R (February 2020). “α-Ketoamides as Broad-Spectrum Inhibitors of Coronavirus and Enterovirus Replication: Structure-Based Design, Synthesis, and Activity Assessment”. Journal of Medicinal Chemistry 63 (9): 4562–4578. doi:10.1021/acs.jmedchem.9b01828. PMC 7098070. PMID 32045235.
Zhang L, Lin D, Sun X, Curth U, Drosten C, Sauerhering L, Becker S, Rox K, Hilgenfeld R (March 2020). “Crystal structure of SARS-CoV-2 main protease provides a basis for design of improved α-ketoamide inhibitors”. Science 368 (6489): 409–412. Bibcode: 2020Sci...368..409Z. doi:10.1126/science.abb3405. PMC 7164518. PMID 32198291.
Morse JS, Lalonde T, Xu S, Liu WR (March 2020). “Learning from the Past: Possible Urgent Prevention and Treatment Options for Severe Acute Respiratory Infections Caused by 2019-nCoV”. ChemBioChem 21 (5): 730–738. doi:10.1002/cbic.202000047. PMC 7162020. PMID 32022370.
Liu C, Zhou Q, Li Y, Garner LV, Watkins SP, Carter LJ, Smoot J, Gregg AC, Daniels AD, Jervey S, Albaiu D (March 2020). “Research and Development on Therapeutic Agents and Vaccines for COVID-19 and Related Human Coronavirus Diseases”. ACS Central Science 6 (3): 315–331. doi:10.1021/acscentsci.0c00272. PMC 7094090. PMID 32226821.
Ramajayam R, Tan KP, Liang PH (October 2011). “Recent development of 3C and 3CL protease inhibitors for anti-coronavirus and anti-picornavirus drug discovery”. Biochemical Society Transactions 39 (5): 1371–5. doi:10.1042/BST0391371. PMID 21936817.
Dai, Wenhao; Zhang, Bing; Jiang, Xia-Ming; Su, Haixia; Li, Jian; Zhao, Yao; Xie, Xiong; Jin, Zhenming et al. (2020-06-19). “Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease” (英語). Science 368 (6497): 1331–1335. doi:10.1126/science.abb4489. ISSN 0036-8075. PMC 7179937. PMID 32321856.
Bhardwaj VK, Singh R, Sharma J, Rajendran V, Purohit R, Kumar S (May 2020). “Identification of bioactive molecules from tea plant as SARS-CoV-2 main protease inhibitors”. Journal of Biomolecular Structure and Dynamics: 1–10. doi:10.1080/07391102.2020.1766572. PMC 7256349. PMID 32397940.
Bhardwaj VK, Singh R, Das P, Purohit R (January 2021). “Evaluation of acridinedione analogs as potential SARS-CoV-2 main protease inhibitors and their comparison with repurposed anti-viral drugs”. Computers in Biology and Medicine 128 (1104117): 104117. doi:10.1016/j.compbiomed.2020.104117. PMC 7659809. PMID 33217661.
Kim Y, Lovell S, Tiew KC, Mandadapu SR, Alliston KR, Battaile KP, Groutas WC, Chang KO (November 2012). “Broad-spectrum antivirals against 3C or 3C-like proteases of picornaviruses, noroviruses, and coronaviruses”. Journal of Virology 86 (21): 11754–62. doi:10.1128/JVI.01348-12. PMC 3486288. PMID 22915796.
Ziebuhr J, Bayer S, Cowley JA, Gorbalenya AE (January 2003). “The 3C-like proteinase of an invertebrate nidovirus links coronavirus and potyvirus homologs”. Journal of Virology 77 (2): 1415–26. doi:10.1128/jvi.77.2.1415-1426.2003. PMC 140795. PMID 12502857.

harvard.edu

ui.adsabs.harvard.edu

Anand K, Ziebuhr J, Wadhwani P, Mesters JR, Hilgenfeld R (June 2003). “Coronavirus main proteinase (3CLpro) structure: basis for design of anti-SARS drugs”. Science 300 (5626): 1763–7. Bibcode: 2003Sci...300.1763A. doi:10.1126/science.1085658. PMID 12746549.
Zhang L, Lin D, Sun X, Curth U, Drosten C, Sauerhering L, Becker S, Rox K, Hilgenfeld R (March 2020). “Crystal structure of SARS-CoV-2 main protease provides a basis for design of improved α-ketoamide inhibitors”. Science 368 (6489): 409–412. Bibcode: 2020Sci...368..409Z. doi:10.1126/science.abb3405. PMC 7164518. PMID 32198291.

nih.gov

pubmed.ncbi.nlm.nih.gov

Goetz DH, Choe Y, Hansell E, Chen YT, McDowell M, Jonsson CB, Roush WR, McKerrow J, Craik CS (July 2007). “Substrate specificity profiling and identification of a new class of inhibitor for the major protease of the SARS coronavirus”. Biochemistry 46 (30): 8744–52. doi:10.1021/bi0621415. PMID 17605471.
Fan K, Wei P, Feng Q, Chen S, Huang C, Ma L, Lai B, Pei J, Liu Y, Chen J, Lai L (January 2004). “Biosynthesis, purification, and substrate specificity of severe acute respiratory syndrome coronavirus 3C-like proteinase”. The Journal of Biological Chemistry 279 (3): 1637–42. doi:10.1074/jbc.m310875200. PMC 7980035. PMID 14561748.
Akaji K, Konno H, Onozuka M, Makino A, Saito H, Nosaka K (November 2008). “Evaluation of peptide-aldehyde inhibitors using R188I mutant of SARS 3CL protease as a proteolysis-resistant mutant”. Bioorganic & Medicinal Chemistry 16 (21): 9400–8. doi:10.1016/j.bmc.2008.09.057. PMC 7126698. PMID 18845442.
Fehr AR, Perlman S (2015). “Coronaviruses: an overview of their replication and pathogenesis”. Coronaviruses. Methods in Molecular Biology. 1282. Springer. pp. 1–23. doi:10.1007/978-1-4939-2438-7_1. ISBN 978-1-4939-2438-7. PMC 4369385. PMID 25720466. "See section: Virion Structure."
Ryu, Young Bae; Park, Su-Jin; Kim, Young Min; Lee, Ju-Yeon; Seo, Woo Duck; Chang, Jong Sun; Park, Ki Hun; Rho, Mun-Chual et al. (2010-03-15). “SARS-CoV 3CLpro inhibitory effects of quinone-methide triterpenes from Tripterygium regelii” (英語). Bioorganic & Medicinal Chemistry Letters 20 (6): 1873–1876. doi:10.1016/j.bmcl.2010.01.152. ISSN 0960-894X. PMC 7127101. PMID 20167482.
Ocain TD, Rich DH (February 1992). “alpha-Keto amide inhibitors of aminopeptidases”. Journal of Medicinal Chemistry 35 (3): 451–6. doi:10.1021/jm00081a005. PMID 1738140.
Anand K, Ziebuhr J, Wadhwani P, Mesters JR, Hilgenfeld R (June 2003). “Coronavirus main proteinase (3CLpro) structure: basis for design of anti-SARS drugs”. Science 300 (5626): 1763–7. Bibcode: 2003Sci...300.1763A. doi:10.1126/science.1085658. PMID 12746549.
Pacifico S, Ferretti V, Albanese V, Fantinati A, Gallerani E, Nicoli F, Gavioli R, Zamberlan F, Preti D, Marastoni M (July 2019). “Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors”. ACS Medicinal Chemistry Letters 10 (7): 1086–1092. doi:10.1021/acsmedchemlett.9b00233. PMC 6627721. PMID 31312413.
Kusov Y, Tan J, Alvarez E, Enjuanes L, Hilgenfeld R (October 2015). “A G-quadruplex-binding macrodomain within the "SARS-unique domain" is essential for the activity of the SARS-coronavirus replication-transcription complex”. Virology 484: 313–22. doi:10.1016/j.virol.2015.06.016. PMC 4567502. PMID 26149721.
Zhang L, Lin D, Kusov Y, Nian Y, Ma Q, Wang J, von Brunn A, Leyssen P, Lanko K, Neyts J, de Wilde A, Snijder EJ, Liu H, Hilgenfeld R (February 2020). “α-Ketoamides as Broad-Spectrum Inhibitors of Coronavirus and Enterovirus Replication: Structure-Based Design, Synthesis, and Activity Assessment”. Journal of Medicinal Chemistry 63 (9): 4562–4578. doi:10.1021/acs.jmedchem.9b01828. PMC 7098070. PMID 32045235.
Zhang L, Lin D, Sun X, Curth U, Drosten C, Sauerhering L, Becker S, Rox K, Hilgenfeld R (March 2020). “Crystal structure of SARS-CoV-2 main protease provides a basis for design of improved α-ketoamide inhibitors”. Science 368 (6489): 409–412. Bibcode: 2020Sci...368..409Z. doi:10.1126/science.abb3405. PMC 7164518. PMID 32198291.
Morse JS, Lalonde T, Xu S, Liu WR (March 2020). “Learning from the Past: Possible Urgent Prevention and Treatment Options for Severe Acute Respiratory Infections Caused by 2019-nCoV”. ChemBioChem 21 (5): 730–738. doi:10.1002/cbic.202000047. PMC 7162020. PMID 32022370.
Liu C, Zhou Q, Li Y, Garner LV, Watkins SP, Carter LJ, Smoot J, Gregg AC, Daniels AD, Jervey S, Albaiu D (March 2020). “Research and Development on Therapeutic Agents and Vaccines for COVID-19 and Related Human Coronavirus Diseases”. ACS Central Science 6 (3): 315–331. doi:10.1021/acscentsci.0c00272. PMC 7094090. PMID 32226821.
Ramajayam R, Tan KP, Liang PH (October 2011). “Recent development of 3C and 3CL protease inhibitors for anti-coronavirus and anti-picornavirus drug discovery”. Biochemical Society Transactions 39 (5): 1371–5. doi:10.1042/BST0391371. PMID 21936817.
Dai, Wenhao; Zhang, Bing; Jiang, Xia-Ming; Su, Haixia; Li, Jian; Zhao, Yao; Xie, Xiong; Jin, Zhenming et al. (2020-06-19). “Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease” (英語). Science 368 (6497): 1331–1335. doi:10.1126/science.abb4489. ISSN 0036-8075. PMC 7179937. PMID 32321856.
Bhardwaj VK, Singh R, Sharma J, Rajendran V, Purohit R, Kumar S (May 2020). “Identification of bioactive molecules from tea plant as SARS-CoV-2 main protease inhibitors”. Journal of Biomolecular Structure and Dynamics: 1–10. doi:10.1080/07391102.2020.1766572. PMC 7256349. PMID 32397940.
Bhardwaj VK, Singh R, Das P, Purohit R (January 2021). “Evaluation of acridinedione analogs as potential SARS-CoV-2 main protease inhibitors and their comparison with repurposed anti-viral drugs”. Computers in Biology and Medicine 128 (1104117): 104117. doi:10.1016/j.compbiomed.2020.104117. PMC 7659809. PMID 33217661.
Kim Y, Lovell S, Tiew KC, Mandadapu SR, Alliston KR, Battaile KP, Groutas WC, Chang KO (November 2012). “Broad-spectrum antivirals against 3C or 3C-like proteases of picornaviruses, noroviruses, and coronaviruses”. Journal of Virology 86 (21): 11754–62. doi:10.1128/JVI.01348-12. PMC 3486288. PMID 22915796.
Ziebuhr J, Bayer S, Cowley JA, Gorbalenya AE (January 2003). “The 3C-like proteinase of an invertebrate nidovirus links coronavirus and potyvirus homologs”. Journal of Virology 77 (2): 1415–26. doi:10.1128/jvi.77.2.1415-1426.2003. PMC 140795. PMID 12502857.

ncbi.nlm.nih.gov

Fan K, Wei P, Feng Q, Chen S, Huang C, Ma L, Lai B, Pei J, Liu Y, Chen J, Lai L (January 2004). “Biosynthesis, purification, and substrate specificity of severe acute respiratory syndrome coronavirus 3C-like proteinase”. The Journal of Biological Chemistry 279 (3): 1637–42. doi:10.1074/jbc.m310875200. PMC 7980035. PMID 14561748.
Akaji K, Konno H, Onozuka M, Makino A, Saito H, Nosaka K (November 2008). “Evaluation of peptide-aldehyde inhibitors using R188I mutant of SARS 3CL protease as a proteolysis-resistant mutant”. Bioorganic & Medicinal Chemistry 16 (21): 9400–8. doi:10.1016/j.bmc.2008.09.057. PMC 7126698. PMID 18845442.
Fehr AR, Perlman S (2015). “Coronaviruses: an overview of their replication and pathogenesis”. Coronaviruses. Methods in Molecular Biology. 1282. Springer. pp. 1–23. doi:10.1007/978-1-4939-2438-7_1. ISBN 978-1-4939-2438-7. PMC 4369385. PMID 25720466. "See section: Virion Structure."
Ryu, Young Bae; Park, Su-Jin; Kim, Young Min; Lee, Ju-Yeon; Seo, Woo Duck; Chang, Jong Sun; Park, Ki Hun; Rho, Mun-Chual et al. (2010-03-15). “SARS-CoV 3CLpro inhibitory effects of quinone-methide triterpenes from Tripterygium regelii” (英語). Bioorganic & Medicinal Chemistry Letters 20 (6): 1873–1876. doi:10.1016/j.bmcl.2010.01.152. ISSN 0960-894X. PMC 7127101. PMID 20167482.
Pacifico S, Ferretti V, Albanese V, Fantinati A, Gallerani E, Nicoli F, Gavioli R, Zamberlan F, Preti D, Marastoni M (July 2019). “Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors”. ACS Medicinal Chemistry Letters 10 (7): 1086–1092. doi:10.1021/acsmedchemlett.9b00233. PMC 6627721. PMID 31312413.
Kusov Y, Tan J, Alvarez E, Enjuanes L, Hilgenfeld R (October 2015). “A G-quadruplex-binding macrodomain within the "SARS-unique domain" is essential for the activity of the SARS-coronavirus replication-transcription complex”. Virology 484: 313–22. doi:10.1016/j.virol.2015.06.016. PMC 4567502. PMID 26149721.
Zhang L, Lin D, Kusov Y, Nian Y, Ma Q, Wang J, von Brunn A, Leyssen P, Lanko K, Neyts J, de Wilde A, Snijder EJ, Liu H, Hilgenfeld R (February 2020). “α-Ketoamides as Broad-Spectrum Inhibitors of Coronavirus and Enterovirus Replication: Structure-Based Design, Synthesis, and Activity Assessment”. Journal of Medicinal Chemistry 63 (9): 4562–4578. doi:10.1021/acs.jmedchem.9b01828. PMC 7098070. PMID 32045235.
Zhang L, Lin D, Sun X, Curth U, Drosten C, Sauerhering L, Becker S, Rox K, Hilgenfeld R (March 2020). “Crystal structure of SARS-CoV-2 main protease provides a basis for design of improved α-ketoamide inhibitors”. Science 368 (6489): 409–412. Bibcode: 2020Sci...368..409Z. doi:10.1126/science.abb3405. PMC 7164518. PMID 32198291.
Morse JS, Lalonde T, Xu S, Liu WR (March 2020). “Learning from the Past: Possible Urgent Prevention and Treatment Options for Severe Acute Respiratory Infections Caused by 2019-nCoV”. ChemBioChem 21 (5): 730–738. doi:10.1002/cbic.202000047. PMC 7162020. PMID 32022370.
Liu C, Zhou Q, Li Y, Garner LV, Watkins SP, Carter LJ, Smoot J, Gregg AC, Daniels AD, Jervey S, Albaiu D (March 2020). “Research and Development on Therapeutic Agents and Vaccines for COVID-19 and Related Human Coronavirus Diseases”. ACS Central Science 6 (3): 315–331. doi:10.1021/acscentsci.0c00272. PMC 7094090. PMID 32226821.
Dai, Wenhao; Zhang, Bing; Jiang, Xia-Ming; Su, Haixia; Li, Jian; Zhao, Yao; Xie, Xiong; Jin, Zhenming et al. (2020-06-19). “Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease” (英語). Science 368 (6497): 1331–1335. doi:10.1126/science.abb4489. ISSN 0036-8075. PMC 7179937. PMID 32321856.
Bhardwaj VK, Singh R, Sharma J, Rajendran V, Purohit R, Kumar S (May 2020). “Identification of bioactive molecules from tea plant as SARS-CoV-2 main protease inhibitors”. Journal of Biomolecular Structure and Dynamics: 1–10. doi:10.1080/07391102.2020.1766572. PMC 7256349. PMID 32397940.
Bhardwaj VK, Singh R, Das P, Purohit R (January 2021). “Evaluation of acridinedione analogs as potential SARS-CoV-2 main protease inhibitors and their comparison with repurposed anti-viral drugs”. Computers in Biology and Medicine 128 (1104117): 104117. doi:10.1016/j.compbiomed.2020.104117. PMC 7659809. PMID 33217661.
Kim Y, Lovell S, Tiew KC, Mandadapu SR, Alliston KR, Battaile KP, Groutas WC, Chang KO (November 2012). “Broad-spectrum antivirals against 3C or 3C-like proteases of picornaviruses, noroviruses, and coronaviruses”. Journal of Virology 86 (21): 11754–62. doi:10.1128/JVI.01348-12. PMC 3486288. PMID 22915796.
Ziebuhr J, Bayer S, Cowley JA, Gorbalenya AE (January 2003). “The 3C-like proteinase of an invertebrate nidovirus links coronavirus and potyvirus homologs”. Journal of Virology 77 (2): 1415–26. doi:10.1128/jvi.77.2.1415-1426.2003. PMC 140795. PMID 12502857.

worldcat.org

search.worldcat.org

Ryu, Young Bae; Park, Su-Jin; Kim, Young Min; Lee, Ju-Yeon; Seo, Woo Duck; Chang, Jong Sun; Park, Ki Hun; Rho, Mun-Chual et al. (2010-03-15). “SARS-CoV 3CLpro inhibitory effects of quinone-methide triterpenes from Tripterygium regelii” (英語). Bioorganic & Medicinal Chemistry Letters 20 (6): 1873–1876. doi:10.1016/j.bmcl.2010.01.152. ISSN 0960-894X. PMC 7127101. PMID 20167482.
Dai, Wenhao; Zhang, Bing; Jiang, Xia-Ming; Su, Haixia; Li, Jian; Zhao, Yao; Xie, Xiong; Jin, Zhenming et al. (2020-06-19). “Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease” (英語). Science 368 (6497): 1331–1335. doi:10.1126/science.abb4489. ISSN 0036-8075. PMC 7179937. PMID 32321856.