Cuccioloni, M; Mozzicafreddo, M; Bonfili, L; Cecarini, V; Eleuteri, A. M.; Angeletti, M (2009). “Natural occurring polyphenols as template for drug design. Focus on serine proteases”. 《Chemical Biology & Drug Design》 74 (1): 1–15. doi:10.1111/j.1747-0285.2009.00836.x. PMID19519739.
Chen, X; Kempf, D. J.; Li, L; Sham, H. L.; Vasavanonda, S; Wideburg, N. E.; Saldivar, A; Marsh, K. C.; McDonald, E; Norbeck, D. W. (2003). “Synthesis and SAR studies of potent HIV protease inhibitors containing novel dimethylphenoxyl acetates as P2 ligands”. 《Bioorganic & Medicinal Chemistry Letters》 13 (21): 3657–60. doi:10.1016/j.bmcl.2003.08.043. PMID14552751.
Brower, E. T.; Bacha, U. M.; Kawasaki, Y; Freire, E (2008). “Inhibition of HIV-2 protease by HIV-1 protease inhibitors in clinical use”. 《Chemical Biology & Drug Design》 71 (4): 298–305. doi:10.1111/j.1747-0285.2008.00647.x. PMID18312292. S2CID8461472.
Turk, Boris (2006). “Targeting proteases: successes, failures and future prospects”. 《Nature Reviews Drug Discovery》 5 (9): 785–99. doi:10.1038/nrd2092. PMID16955069. S2CID4156908.
Brower, E. T.; Bacha, U. M.; Kawasaki, Y; Freire, E (2008). “Inhibition of HIV-2 protease by HIV-1 protease inhibitors in clinical use”. 《Chemical Biology & Drug Design》 71 (4): 298–305. doi:10.1111/j.1747-0285.2008.00647.x. PMID18312292. S2CID8461472.
gsk.com
“Archived copy”. 2008년 12월 3일에 원본 문서에서 보존된 문서. 2008년 6월 11일에 확인함.GlaxoSmithKline discontinues clinical development of investigational protease inhibitor brecanavir (640385). Retrieved November 4th. 2009.
“Archived copy”. 2009년 8월 31일에 원본 문서에서 보존된 문서. 2009년 11월 5일에 확인함.GSK and Concert Pharmaceuticals form alliance to develop novel deuterium-modified drugs. Retrieved November 4th. 2009.
Cuccioloni, M; Mozzicafreddo, M; Bonfili, L; Cecarini, V; Eleuteri, A. M.; Angeletti, M (2009). “Natural occurring polyphenols as template for drug design. Focus on serine proteases”. 《Chemical Biology & Drug Design》 74 (1): 1–15. doi:10.1111/j.1747-0285.2009.00836.x. PMID19519739.
Chen, X; Kempf, D. J.; Li, L; Sham, H. L.; Vasavanonda, S; Wideburg, N. E.; Saldivar, A; Marsh, K. C.; McDonald, E; Norbeck, D. W. (2003). “Synthesis and SAR studies of potent HIV protease inhibitors containing novel dimethylphenoxyl acetates as P2 ligands”. 《Bioorganic & Medicinal Chemistry Letters》 13 (21): 3657–60. doi:10.1016/j.bmcl.2003.08.043. PMID14552751.
Brower, E. T.; Bacha, U. M.; Kawasaki, Y; Freire, E (2008). “Inhibition of HIV-2 protease by HIV-1 protease inhibitors in clinical use”. 《Chemical Biology & Drug Design》 71 (4): 298–305. doi:10.1111/j.1747-0285.2008.00647.x. PMID18312292. S2CID8461472.
Turk, Boris (2006). “Targeting proteases: successes, failures and future prospects”. 《Nature Reviews Drug Discovery》 5 (9): 785–99. doi:10.1038/nrd2092. PMID16955069. S2CID4156908.
Brower, E. T.; Bacha, U. M.; Kawasaki, Y; Freire, E (2008). “Inhibition of HIV-2 protease by HIV-1 protease inhibitors in clinical use”. 《Chemical Biology & Drug Design》 71 (4): 298–305. doi:10.1111/j.1747-0285.2008.00647.x. PMID18312292. S2CID8461472.
semanticscholar.org
api.semanticscholar.org
Brower, E. T.; Bacha, U. M.; Kawasaki, Y; Freire, E (2008). “Inhibition of HIV-2 protease by HIV-1 protease inhibitors in clinical use”. 《Chemical Biology & Drug Design》 71 (4): 298–305. doi:10.1111/j.1747-0285.2008.00647.x. PMID18312292. S2CID8461472.
Turk, Boris (2006). “Targeting proteases: successes, failures and future prospects”. 《Nature Reviews Drug Discovery》 5 (9): 785–99. doi:10.1038/nrd2092. PMID16955069. S2CID4156908.
Brower, E. T.; Bacha, U. M.; Kawasaki, Y; Freire, E (2008). “Inhibition of HIV-2 protease by HIV-1 protease inhibitors in clinical use”. 《Chemical Biology & Drug Design》 71 (4): 298–305. doi:10.1111/j.1747-0285.2008.00647.x. PMID18312292. S2CID8461472.
“Archived copy”. 2008년 12월 3일에 원본 문서에서 보존된 문서. 2008년 6월 11일에 확인함.GlaxoSmithKline discontinues clinical development of investigational protease inhibitor brecanavir (640385). Retrieved November 4th. 2009.
“Archived copy”. 2009년 8월 31일에 원본 문서에서 보존된 문서. 2009년 11월 5일에 확인함.GSK and Concert Pharmaceuticals form alliance to develop novel deuterium-modified drugs. Retrieved November 4th. 2009.