Volpini R, Costanzi S, Lambertucci C, Taffi S, Vittori S, Klotz KN, Cristalli G (July 2002). „N(6)-alkyl-2-alkynyl derivatives of adenosine as potent and selective agonists at the human adenosine A(3) receptor and a starting point for searching A(2B) ligands”. Journal of Medicinal Chemistry45 (15): 3271–9. DOI:10.1021/jm0109762. PMID12109910.
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Carotti A, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Stefanachi A, Vidal B (January 2006). „Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor”. Journal of Medicinal Chemistry49 (1): 282–99. DOI:10.1021/jm0506221. PMID16392813.
Tabrizi MA, Baraldi PG, Preti D, Romagnoli R, Saponaro G, Baraldi S, Moorman AR, Zaid AN, Varani K, Borea PA (March 2008). „1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists”. Bioorganic & Medicinal Chemistry16 (5): 2419–30. DOI:10.1016/j.bmc.2007.11.058. PMID18077171.
Stefanachi A, Brea JM, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Vidal B, Carotti A (March 2008). „1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor”. Bioorganic & Medicinal Chemistry16 (6): 2852–69. DOI:10.1016/j.bmc.2008.01.002. PMID18226909.
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Kim MO, Kim MH, Lee SH, Suh HN, Lee YJ, Lee MY, Han HJ (June 2009). „5'-N-ethylcarboxamide induces IL-6 expression via MAPKs and NF-kappaB activation through Akt, Ca(2+)/PKC, cAMP signaling pathways in mouse embryonic stem cells”. Journal of Cellular Physiology219 (3): 752–9. DOI:10.1002/jcp.21721. PMID19194991.
Stefanachi A, Nicolotti O, Leonetti F, et al. (2008). „1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A(2B) adenosine receptor antagonists: Design, synthesis, structure-affinity and structure-selectivity relationships”. Bioorganic & medicinal chemistry16: 9780. DOI:10.1016/j.bmc.2008.09.067. PMID18938084.
Volpini R, Costanzi S, Lambertucci C, Taffi S, Vittori S, Klotz KN, Cristalli G (July 2002). „N(6)-alkyl-2-alkynyl derivatives of adenosine as potent and selective agonists at the human adenosine A(3) receptor and a starting point for searching A(2B) ligands”. Journal of Medicinal Chemistry45 (15): 3271–9. DOI:10.1021/jm0109762. PMID12109910.
Elzein E, Kalla R, Li X, Perry T, Parkhill E, Palle V, Varkhedkar V, Gimbel A, Zeng D, Lustig D, Leung K, Zablocki J (January 2006). „Novel 1,3-dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonists”. Bioorganic & Medicinal Chemistry Letters16 (2): 302–6. DOI:10.1016/j.bmcl.2005.10.002. PMID16275090.
Carotti A, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Stefanachi A, Vidal B (January 2006). „Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor”. Journal of Medicinal Chemistry49 (1): 282–99. DOI:10.1021/jm0506221. PMID16392813.
Tabrizi MA, Baraldi PG, Preti D, Romagnoli R, Saponaro G, Baraldi S, Moorman AR, Zaid AN, Varani K, Borea PA (March 2008). „1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists”. Bioorganic & Medicinal Chemistry16 (5): 2419–30. DOI:10.1016/j.bmc.2007.11.058. PMID18077171.
Stefanachi A, Brea JM, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Vidal B, Carotti A (March 2008). „1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor”. Bioorganic & Medicinal Chemistry16 (6): 2852–69. DOI:10.1016/j.bmc.2008.01.002. PMID18226909.
Kim MO, Kim MH, Lee SH, Suh HN, Lee YJ, Lee MY, Han HJ (June 2009). „5'-N-ethylcarboxamide induces IL-6 expression via MAPKs and NF-kappaB activation through Akt, Ca(2+)/PKC, cAMP signaling pathways in mouse embryonic stem cells”. Journal of Cellular Physiology219 (3): 752–9. DOI:10.1002/jcp.21721. PMID19194991.
Stefanachi A, Nicolotti O, Leonetti F, et al. (2008). „1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A(2B) adenosine receptor antagonists: Design, synthesis, structure-affinity and structure-selectivity relationships”. Bioorganic & medicinal chemistry16: 9780. DOI:10.1016/j.bmc.2008.09.067. PMID18938084.