Huixian Wu, Daniel Wacker, Mauro Mileni, Vsevolod Katritch, GyeWon Han, Eyal Vardy, Wei Liu, Aaron A. Thompson, Xi-Ping Huang, F. Ivy Carroll, S. Wayne Mascarella, Richard B. Westkaemper, Philip D. Mosier, Bryan L. Roth, Vadim Cherezov & Raymond C. Stevens (2012). „Structure of the human k-opioid receptor in complex with JDTic”. Nature. DOI:10.1038/nature10939.
King N, Hittinger CT, Carroll SB (2003). „Evolution of key cell signaling and adhesion protein families predates animal origins”. Science301 (5631): 361–3. DOI:10.1126/science.1083853. PMID12869759.
Overington JP, Al-Lazikani B, Hopkins AL (December 2006). „How many drug targets are there?”. Nat Rev Drug Discov5 (12): 993–6. DOI:10.1038/nrd2199. PMID17139284.
Bjarnadottir TK, Gloriam DE, Hellstrand SH, Kristiansson H, Fredriksson R, Schioth HB (2006). „Comprehensive repertoire and phylogenetic analysis of the G protein-coupled receptors in human and mouse”. Genomics88 (3): 263–73. DOI:10.1016/j.ygeno.2006.04.001. PMID16753280.
Qiu JD, Huang JH, Liang RP, Lu XQ (July 2009). „Prediction of G-protein-coupled receptor classes based on the concept of Chou's pseudo amino acid composition: an approach from discrete wavelet transform”. Anal. Biochem.390 (1): 68–73. DOI:10.1016/j.ab.2009.04.009. PMID19364489.
Gu Q, Ding YS, Zhang TL (May 2010). „Prediction of G-Protein-Coupled Receptor Classes in Low Homology Using Chou's pseudo amino acid composition with Approximate Entropy and Hydrophobicity Patterns”. Protein Pept. Lett.17 (5): 559–67. DOI:10.2174/092986610791112693. PMID19594431.
Grigorieff N, Ceska TA, Downing KH, Baldwin JM, Henderson R (1996). „Electron-crystallographic refinement of the structure of bacteriorhodopsin”. J. Mol. Biol.259 (3): 393–421. DOI:10.1006/jmbi.1996.0328. PMID8676377.
Kimura Y, Vassylyev DG, Miyazawa A, Kidera A, Matsushima M, Mitsuoka K, Murata K, Hirai T, Fujiyoshi Y (1997). „Surface of bacteriorhodopsin revealed by high-resolution electron crystallography”. Nature389 (6647): 206–11. DOI:10.1038/38323. PMID9296502.
Pebay-Peyroula E, Rummel G, Rosenbusch JP, Landau EM (1997). „X-ray structure of bacteriorhodopsin at 2.5 angstroms from microcrystals grown in lipidic cubic phases”. Science277 (5332): 1676–81. DOI:10.1126/science.277.5332.1676. PMID9287223.
Palczewski K, Kumasaka T, Hori T, Behnke CA, Motoshima H, Fox BA, Trong IL, Teller DC, Okada T, Stenkamp RE, Yamamoto M, Miyano M (2000). „Crystal structure of rhodopsin: A G protein-coupled receptor.”. Science289 (5480): 739–45. DOI:10.1126/science.289.5480.739. PMID10926528.
Rasmussen SG, Choi HJ, Rosenbaum DM, Kobilka TS, Thian FS, Edwards PC, Burghammer M, Ratnala VR, Sanishvili R, Fischetti RF, Schertler GF, Weis WI, Kobilka BK (2007). „Crystal structure of the human β2-adrenergic G-protein-coupled receptor”. Nature450 (7168): 383–7. DOI:10.1038/nature06325. PMID17952055.
Millar RP, Newton CL (January 2010). „The year in G protein-coupled receptor research”. Mol. Endocrinol.24 (1): 261–74. DOI:10.1210/me.2009-0473. PMID20019124.
Duchene J, Schanstra JP, Pecher C, Pizard A, Susini C, Esteve JP, Bascands JL, Girolami JP (2002). „A novel protein-protein interaction between a G protein-coupled receptor and the phosphatase SHP-2 is involved in bradykinin-induced inhibition of cell proliferation”. J Biol Chem277 (43): 40375–83. DOI:10.1074/jbc.M202744200. PMID12177051.
Krueger KM, Daaka Y, Pitcher JA, Lefkowitz RJ (1997). „The role of sequestration in G protein-coupled receptor resensitization. Regulation of β2-adrenergic receptor dephosphorylation by vesicular acidification”. J. Biol. Chem.272 (1): 5–8. DOI:10.1074/jbc.272.1.5. PMID8995214.
Laporte SA, Oakley RH, Holt JA, Barak LS, Caron MG (2000). „The interaction of β-arrestin with the AP-2 adaptor is required for the clustering of β2-adrenergic receptor into clathrin-coated pits”. J. Biol. Chem.275 (30): 23120–6. DOI:10.1074/jbc.M002581200. PMID10770944.
Margeta-Mitrovic M, Jan YN, Jan LY (2000). „A trafficking checkpoint controls GABA(B) receptor heterodimerization”. Neuron27 (1): 97–106. DOI:10.1016/S0896-6273(00)00012-X. PMID10939334.
White JH, Wise A, Main MJ, Green A, Fraser NJ, Disney GH, Barnes AA, Emson P, Foord SM, Marshall FH (1998). „Heterodimerization is required for the formation of a functional GABA(B) receptor”. Nature396 (6712): 679–82. DOI:10.1038/25354. PMID9872316.
Krishnan A, Alme´n MS, Fredriksson R, Schiöth HB (2012). „The Origin of GPCRs: Identification of Mammalian like Rhodopsin, Adhesion, Glutamate and Frizzled GPCRs in Fungi”. PLoS ONE: e29817. DOI:10.1371/journal.pone.0029817. PMID22238661.
Nordström KJ, Sällman Almén M, Edstam MM, Fredriksson R, Schiöth HB (2011). „Independent HHsearch, Needleman–Wunsch-Based, and Motif Analyses Reveal the Overall Hierarchy for Most of the G Protein-Coupled Receptor Families”. Mol Biol Evol: 2471–80. DOI:10.1093/molbev/msr061. PMID21402729.
Bakthavatsalam D, Brazill D, Gomer RH, Eichinger L, Rivero F, Noegel AA (2007). „A G protein-coupled receptor with a lipid kinase domain is involved in cell-density sensing”. Curr Biol17 (10): 892–7. DOI:10.1016/j.cub.2007.04.029. PMID17481898.
Huixian Wu, Daniel Wacker, Mauro Mileni, Vsevolod Katritch, GyeWon Han, Eyal Vardy, Wei Liu, Aaron A. Thompson, Xi-Ping Huang, F. Ivy Carroll, S. Wayne Mascarella, Richard B. Westkaemper, Philip D. Mosier, Bryan L. Roth, Vadim Cherezov & Raymond C. Stevens (2012). „Structure of the human k-opioid receptor in complex with JDTic”. Nature. DOI:10.1038/nature10939.
King N, Hittinger CT, Carroll SB (2003). „Evolution of key cell signaling and adhesion protein families predates animal origins”. Science301 (5631): 361–3. DOI:10.1126/science.1083853. PMID12869759.
Overington JP, Al-Lazikani B, Hopkins AL (December 2006). „How many drug targets are there?”. Nat Rev Drug Discov5 (12): 993–6. DOI:10.1038/nrd2199. PMID17139284.
Bjarnadottir TK, Gloriam DE, Hellstrand SH, Kristiansson H, Fredriksson R, Schioth HB (2006). „Comprehensive repertoire and phylogenetic analysis of the G protein-coupled receptors in human and mouse”. Genomics88 (3): 263–73. DOI:10.1016/j.ygeno.2006.04.001. PMID16753280.
Qiu JD, Huang JH, Liang RP, Lu XQ (July 2009). „Prediction of G-protein-coupled receptor classes based on the concept of Chou's pseudo amino acid composition: an approach from discrete wavelet transform”. Anal. Biochem.390 (1): 68–73. DOI:10.1016/j.ab.2009.04.009. PMID19364489.
Gu Q, Ding YS, Zhang TL (May 2010). „Prediction of G-Protein-Coupled Receptor Classes in Low Homology Using Chou's pseudo amino acid composition with Approximate Entropy and Hydrophobicity Patterns”. Protein Pept. Lett.17 (5): 559–67. DOI:10.2174/092986610791112693. PMID19594431.
Grigorieff N, Ceska TA, Downing KH, Baldwin JM, Henderson R (1996). „Electron-crystallographic refinement of the structure of bacteriorhodopsin”. J. Mol. Biol.259 (3): 393–421. DOI:10.1006/jmbi.1996.0328. PMID8676377.
Kimura Y, Vassylyev DG, Miyazawa A, Kidera A, Matsushima M, Mitsuoka K, Murata K, Hirai T, Fujiyoshi Y (1997). „Surface of bacteriorhodopsin revealed by high-resolution electron crystallography”. Nature389 (6647): 206–11. DOI:10.1038/38323. PMID9296502.
Pebay-Peyroula E, Rummel G, Rosenbusch JP, Landau EM (1997). „X-ray structure of bacteriorhodopsin at 2.5 angstroms from microcrystals grown in lipidic cubic phases”. Science277 (5332): 1676–81. DOI:10.1126/science.277.5332.1676. PMID9287223.
Palczewski K, Kumasaka T, Hori T, Behnke CA, Motoshima H, Fox BA, Trong IL, Teller DC, Okada T, Stenkamp RE, Yamamoto M, Miyano M (2000). „Crystal structure of rhodopsin: A G protein-coupled receptor.”. Science289 (5480): 739–45. DOI:10.1126/science.289.5480.739. PMID10926528.
Rasmussen SG, Choi HJ, Rosenbaum DM, Kobilka TS, Thian FS, Edwards PC, Burghammer M, Ratnala VR, Sanishvili R, Fischetti RF, Schertler GF, Weis WI, Kobilka BK (2007). „Crystal structure of the human β2-adrenergic G-protein-coupled receptor”. Nature450 (7168): 383–7. DOI:10.1038/nature06325. PMID17952055.
Luttrell LM, Lefkowitz RJ (February 2002). „The role of beta-arrestins in the termination and transduction of G-protein-coupled receptor signals”. J. Cell. Sci.115 (Pt 3): 455–65. PMID11861753.
Millar RP, Newton CL (January 2010). „The year in G protein-coupled receptor research”. Mol. Endocrinol.24 (1): 261–74. DOI:10.1210/me.2009-0473. PMID20019124.
Duchene J, Schanstra JP, Pecher C, Pizard A, Susini C, Esteve JP, Bascands JL, Girolami JP (2002). „A novel protein-protein interaction between a G protein-coupled receptor and the phosphatase SHP-2 is involved in bradykinin-induced inhibition of cell proliferation”. J Biol Chem277 (43): 40375–83. DOI:10.1074/jbc.M202744200. PMID12177051.
Krueger KM, Daaka Y, Pitcher JA, Lefkowitz RJ (1997). „The role of sequestration in G protein-coupled receptor resensitization. Regulation of β2-adrenergic receptor dephosphorylation by vesicular acidification”. J. Biol. Chem.272 (1): 5–8. DOI:10.1074/jbc.272.1.5. PMID8995214.
Laporte SA, Oakley RH, Holt JA, Barak LS, Caron MG (2000). „The interaction of β-arrestin with the AP-2 adaptor is required for the clustering of β2-adrenergic receptor into clathrin-coated pits”. J. Biol. Chem.275 (30): 23120–6. DOI:10.1074/jbc.M002581200. PMID10770944.
Margeta-Mitrovic M, Jan YN, Jan LY (2000). „A trafficking checkpoint controls GABA(B) receptor heterodimerization”. Neuron27 (1): 97–106. DOI:10.1016/S0896-6273(00)00012-X. PMID10939334.
White JH, Wise A, Main MJ, Green A, Fraser NJ, Disney GH, Barnes AA, Emson P, Foord SM, Marshall FH (1998). „Heterodimerization is required for the formation of a functional GABA(B) receptor”. Nature396 (6712): 679–82. DOI:10.1038/25354. PMID9872316.
Dean, M. K.; Higgs, C.; Smith, R. E.; Bywater, R. P.; Snell, C. R.; Scott, P. D.; Upton, G. J.; Howe, T. J.; Reynolds, C. A. (2001). „Dimerization of G-protein-coupled receptors”. J. Med. Chem.44: 4595.
Krishnan A, Alme´n MS, Fredriksson R, Schiöth HB (2012). „The Origin of GPCRs: Identification of Mammalian like Rhodopsin, Adhesion, Glutamate and Frizzled GPCRs in Fungi”. PLoS ONE: e29817. DOI:10.1371/journal.pone.0029817. PMID22238661.
Nordström KJ, Sällman Almén M, Edstam MM, Fredriksson R, Schiöth HB (2011). „Independent HHsearch, Needleman–Wunsch-Based, and Motif Analyses Reveal the Overall Hierarchy for Most of the G Protein-Coupled Receptor Families”. Mol Biol Evol: 2471–80. DOI:10.1093/molbev/msr061. PMID21402729.
Bakthavatsalam D, Brazill D, Gomer RH, Eichinger L, Rivero F, Noegel AA (2007). „A G protein-coupled receptor with a lipid kinase domain is involved in cell-density sensing”. Curr Biol17 (10): 892–7. DOI:10.1016/j.cub.2007.04.029. PMID17481898.