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A, Stefanachi; Nicolotti O; Leonetti F (2008). „1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A(2B) adenosine receptor antagonists: Design, synthesis, structure-affinity and structure-selectivity relationships”. Bioorganic & medicinal chemistry. 16: 9780. PMID18938084. doi:10.1016/j.bmc.2008.09.067.
Volpini R, Costanzi S, Lambertucci C, Taffi S, Vittori S, Klotz KN, Cristalli G (2002). „N(6)-alkyl-2-alkynyl derivatives of adenosine as potent and selective agonists at the human adenosine A(3) receptor and a starting point for searching A(2B) ligands”. Journal of Medicinal Chemistry. 45 (15): 3271—9. PMID12109910. doi:10.1021/jm0109762.
Elzein E, Kalla R, Li X, Perry T, Parkhill E, Palle V, Varkhedkar V, Gimbel A, Zeng D, Lustig D, Leung K, Zablocki J (2006). „Novel 1,3-dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonists”. Bioorganic & Medicinal Chemistry Letters. 16 (2): 302—6. PMID16275090. doi:10.1016/j.bmcl.2005.10.002.
Carotti A, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Stefanachi A, Vidal B (2006). „Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor”. Journal of Medicinal Chemistry. 49 (1): 282—99. PMID16392813. doi:10.1021/jm0506221.
Tabrizi MA, Baraldi PG, Preti D, Romagnoli R, Saponaro G, Baraldi S, Moorman AR, Zaid AN, Varani K, Borea PA (2008). „1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists”. Bioorganic & Medicinal Chemistry. 16 (5): 2419—30. PMID18077171. doi:10.1016/j.bmc.2007.11.058.
Stefanachi A, Brea JM, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Vidal B, Carotti A (2008). „1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor”. Bioorganic & Medicinal Chemistry. 16 (6): 2852—69. PMID18226909. doi:10.1016/j.bmc.2008.01.002.
Kim MO, Kim MH, Lee SH, Suh HN, Lee YJ, Lee MY, Han HJ (2009). „5'-N-ethylcarboxamide induces IL-6 expression via MAPKs and NF-kappaB activation through Akt, Ca(2+)/PKC, cAMP signaling pathways in mouse embryonic stem cells”. Journal of Cellular Physiology. 219 (3): 752—9. PMID19194991. doi:10.1002/jcp.21721.
A, Stefanachi; Nicolotti O; Leonetti F (2008). „1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A(2B) adenosine receptor antagonists: Design, synthesis, structure-affinity and structure-selectivity relationships”. Bioorganic & medicinal chemistry. 16: 9780. PMID18938084. doi:10.1016/j.bmc.2008.09.067.