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Balani SK, Miwa GT, Gan LS, Wu JT, Lee FW. Strategy of utilizing in vitro and in vivo ADME tools for lead optimization and drug candidate selection. Current Topics in Medicinal Chemistry. 2005, 5 (11): 1033–1038. PMID 16181128. doi:10.2174/156802605774297038.
Singh SS. Preclinical pharmacokinetics: an approach towards safer and efficacious drugs. Current Drug Metabolism. February 2006, 7 (2): 165–182. PMID 16472106. doi:10.2174/138920006775541552.