The synthesis and pharmacological properties of a series of 2-substituted aminomethyl-1,4-benzodioxanes. Journal of Medicinal Chemistry. March 1969, 12 (2): 326–9. PMID 5791620. doi:10.1021/jm00302a033.
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety. Pharmaceutica Acta Helvetiae. March 2000, 74 (2–3): 181–90. PMID 10812956. doi:10.1016/S0031-6865(99)00049-7.
Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist. European Journal of Medicinal Chemistry. December 2012, 58: 184–91. PMID 23124215. doi:10.1016/j.ejmech.2012.09.049.
6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist. Journal of Medicinal Chemistry. August 2013, 56 (16): 6402–12. PMID 23902232. doi:10.1021/jm400867d.
nih.gov
ncbi.nlm.nih.gov
The synthesis and pharmacological properties of a series of 2-substituted aminomethyl-1,4-benzodioxanes. Journal of Medicinal Chemistry. March 1969, 12 (2): 326–9. PMID 5791620. doi:10.1021/jm00302a033.
Characterization of alpha 1-adrenergic receptor subtypes in rat brain: a reevaluation of [3H]WB4104 and [3H]prazosin binding. Molecular Pharmacology. April 1986, 29 (4): 321–30. PMID 3010073.
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety. Pharmaceutica Acta Helvetiae. March 2000, 74 (2–3): 181–90. PMID 10812956. doi:10.1016/S0031-6865(99)00049-7.
Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist. European Journal of Medicinal Chemistry. December 2012, 58: 184–91. PMID 23124215. doi:10.1016/j.ejmech.2012.09.049.
6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist. Journal of Medicinal Chemistry. August 2013, 56 (16): 6402–12. PMID 23902232. doi:10.1021/jm400867d.