胍法辛 (Chinese Wikipedia)

Analysis of information sources in references of the Wikipedia article "胍法辛" in Chinese language version.

refsWebsite

Global rank Chinese rank

43nih.gov

4^th place

5^th place

34doi.org

2^nd place

23^rd place

17web.archive.org

1^st place

10semanticscholar.org

11^th place

332^nd place

2tga.gov.au

3,984^th place

1,603^rd place

2fda.gov

447^th place

581^st place

2clincalc.com

3,912^th place

5,917^th place

2archive.org

6^th place

4^th place

1drugs.com

399^th place

208^th place

1worldcat.org

5^th place

12^th place

1medscape.com

719^th place

889^th place

1harvard.edu

18^th place

57^th place

1medicines.org.uk

3,823^rd place

3,456^th place

1soton.ac.uk

6,219^th place

4,671^st place

1unc.edu

1,538^th place

1,766^th place

1ijest.org

low place

1urn.fi

8,035^th place

low place

1europa.eu

68^th place

209^th place

1racgp.org.au

low place

archive.org

Kornfield R, Watson S, Higashi AS, Conti RM, Dusetzina SB, Garfield CF, Dorsey ER, Huskamp HA, Alexander GC. Effects of FDA advisories on the pharmacologic treatment of ADHD, 2004-2008. Psychiatric Services. April 2013, 64 (4): 339–346. PMC 4023684 . PMID 23318985. doi:10.1176/appi.ps.201200147.
Jasper JR, Lesnick JD, Chang LK, Yamanishi SS, Chang TK, Hsu SA, et al. Ligand efficacy and potency at recombinant alpha2 adrenergic receptors: agonist-mediated [35S]GTPgammaS binding. Biochemical Pharmacology. April 1998, 55 (7): 1035–1043. PMID 9605427. doi:10.1016/s0006-2952(97)00631-x.

clincalc.com

The Top 300 of 2020. ClinCalc. [2022-10-07]. （原始内容存档于2021-01-12）.
Guanfacine - Drug Usage Statistics. ClinCalc. [2022-10-07]. （原始内容存档于2020-07-08）.

doi.org

Kornfield R, Watson S, Higashi AS, Conti RM, Dusetzina SB, Garfield CF, Dorsey ER, Huskamp HA, Alexander GC. Effects of FDA advisories on the pharmacologic treatment of ADHD, 2004-2008. Psychiatric Services. April 2013, 64 (4): 339–346. PMC 4023684 . PMID 23318985. doi:10.1176/appi.ps.201200147.
Zito JM, Derivan AT, Kratochvil CJ, Safer DJ, Fegert JM, Greenhill LL. Off-label psychopharmacologic prescribing for children: history supports close clinical monitoring. Child and Adolescent Psychiatry and Mental Health //www.ncbi.nlm.nih.gov/pmc/articles/PMC2566553 |PMC=缺少标题 (帮助). September 2008, 2 (1): 24. PMC 2566553 . PMID 18793403. doi:10.1186/1753-2000-2-24 .
Clemow, DB; Walker, DJ. The potential for misuse and abuse of medications in ADHD: a review.. Postgraduate Medicine. September 2014, 126 (5): 64–81. PMID 25295651. S2CID 207580823. doi:10.3810/pgm.2014.09.2801.
Radonjić NV, Bellato A, Khoury NM, Cortese S, Faraone SV. Nonstimulant Medications for Attention-Deficit/Hyperactivity Disorder (ADHD) in Adults: Systematic Review and Meta-analysis. CNS Drugs. May 2023, 37 (5): 381–397. PMID 37166701. S2CID 258616507. doi:10.1007/s40263-023-01005-8.
Yu S, Shen S, Tao M. Guanfacine for the Treatment of Attention-Deficit Hyperactivity Disorder: An Updated Systematic Review and Meta-Analysis. J Child Adolesc Psychopharmacol. March 2023, 33 (2): 40–50. PMID 36944092. S2CID 257664282. doi:10.1089/cap.2022.0038.
Catalá-López F, Hutton B, Núñez-Beltrán A, Page MJ, Ridao M, Macías Saint-Gerons D, Catalá MA, Tabarés-Seisdedos R, Moher D. The pharmacological and non-pharmacological treatment of attention deficit hyperactivity disorder in children and adolescents: A systematic review with network meta-analyses of randomised trials. PLOS ONE. 2017, 12 (7): e0180355. Bibcode:2017PLoSO..1280355C. PMC 5507500 . PMID 28700715. doi:10.1371/journal.pone.0180355 .
Pringsheim T, Hirsch L, Gardner D, Gorman DA. The pharmacological management of oppositional behaviour, conduct problems, and aggression in children and adolescents with attention-deficit hyperactivity disorder, oppositional defiant disorder, and conduct disorder: a systematic review and meta-analysis. Part 1: psychostimulants, alpha-2 agonists, and atomoxetine. Can J Psychiatry. February 2015, 60 (2): 42–51. PMC 4344946 . PMID 25886655. doi:10.1177/070674371506000202.
Padilha SC, Virtuoso S, Tonin FS, Borba HH, Pontarolo R. Efficacy and safety of drugs for attention deficit hyperactivity disorder in children and adolescents: a network meta-analysis. Eur Child Adolesc Psychiatry. October 2018, 27 (10): 1335–1345. PMID 29460165. S2CID 3402756. doi:10.1007/s00787-018-1125-0.
Morrow BA, George TP, Roth RH. Noradrenergic alpha-2 agonists have anxiolytic-like actions on stress-related behavior and mesoprefrontal dopamine biochemistry. Brain Research. November 2004, 1027 (1–2): 173–178. PMID 15494168. S2CID 7066842. doi:10.1016/j.brainres.2004.08.057.
Arnsten AF, Raskind MA, Taylor FB, Connor DF. The Effects of Stress Exposure on Prefrontal Cortex: Translating Basic Research into Successful Treatments for Post-Traumatic Stress Disorder. Neurobiology of Stress. January 2015, 1: 89–99. PMC 4244027 . PMID 25436222. doi:10.1016/j.ynstr.2014.10.002.
Kozaric-Kovacic D. Psychopharmacotherapy of posttraumatic stress disorder. Croatian Medical Journal. August 2008, 49 (4): 459–475. PMC 2525822 . PMID 18716993. doi:10.3325/cmj.2008.4.459.
Jerie P. Clinical experience with guanfacine in long-term treatment of hypertension. Part II: adverse reactions to guanfacine. British Journal of Clinical Pharmacology. 1980, 10 (Suppl 1): 157S–164S. PMC 1430125 . PMID 6994770. doi:10.1111/j.1365-2125.1980.tb04924.x.
Anand S, Tong H, Besag FM, Chan EW, Cortese S, Wong IC. Safety, Tolerability and Efficacy of Drugs for Treating Behavioural Insomnia in Children with Attention-Deficit/Hyperactivity Disorder: A Systematic Review with Methodological Quality Assessment. Paediatr Drugs. June 2017, 19 (3): 235–250 [2024-02-22]. PMID 28391425. S2CID 2220464. doi:10.1007/s40272-017-0224-6. （原始内容存档于2024-02-22）.
Rugino TA. Effect on Primary Sleep Disorders When Children With ADHD Are Administered Guanfacine Extended Release. J Atten Disord. January 2018, 22 (1): 14–24. PMID 25376194. S2CID 22675882. doi:10.1177/1087054714554932.
Solmi M, Fornaro M, Ostinelli EG, Zangani C, Croatto G, Monaco F, Krinitski D, Fusar-Poli P, Correll CU. Safety of 80 antidepressants, antipsychotics, anti-attention-deficit/hyperactivity medications and mood stabilizers in children and adolescents with psychiatric disorders: a large scale systematic meta-review of 78 adverse effects. World Psychiatry. June 2020, 19 (2): 214–232. PMC 7215080 . PMID 32394557. doi:10.1002/wps.20765.
Jasper JR, Lesnick JD, Chang LK, Yamanishi SS, Chang TK, Hsu SA, et al. Ligand efficacy and potency at recombinant alpha2 adrenergic receptors: agonist-mediated [35S]GTPgammaS binding. Biochemical Pharmacology. April 1998, 55 (7): 1035–1043. PMID 9605427. doi:10.1016/s0006-2952(97)00631-x.
Bender AM, Parr LC, Livingston WB, Lindsley CW, Merryman WD. 2B Determined: The Future of the Serotonin Receptor 2B in Drug Discovery. J Med Chem. August 2023, 66 (16): 11027–11039. PMID 37584406. S2CID 260924858. doi:10.1021/acs.jmedchem.3c01178. These results strongly indicate substantial risks for treatments involving 5-HT2B agonists, and it has been recommended that all serotonergic drugs be screened for this functional profile.43,59 [...] Additionally, there are cases of marketed drugs that were only later determined to have 5-HT2B activity. Of particular note is guanfacine, an FDA-approved medication for the treatment of attention deficit hyperactivity disorder (ADHD) that possesses potent 5-HT2B agonist activity in functional readouts to a similar degree as known valvulopathogens.66
Hutcheson JD, Setola V, Roth BL, Merryman WD. Serotonin receptors and heart valve disease--it was meant 2B. Pharmacol Ther. November 2011, 132 (2): 146–57. PMC 3179857 . PMID 21440001. doi:10.1016/j.pharmthera.2011.03.008.
Huang XP, Setola V, Yadav PN, Allen JA, Rogan SC, Hanson BJ, Revankar C, Robers M, Doucette C, Roth BL. Parallel functional activity profiling reveals valvulopathogens are potent 5-hydroxytryptamine(2B) receptor agonists: implications for drug safety assessment. Molecular Pharmacology. October 2009, 76 (4): 710–722. PMC 2769050 . PMID 19570945. doi:10.1124/mol.109.058057.
Unett DJ, Gatlin J, Anthony TL, Buzard DJ, Chang S, Chen C, Chen X, Dang HT, Frazer J, Le MK, Sadeque AJ, Xing C, Gaidarov I. Kinetics of 5-HT2B receptor signaling: profound agonist-dependent effects on signaling onset and duration. J Pharmacol Exp Ther. December 2013, 347 (3): 645–59. PMID 24049061. S2CID 8013309. doi:10.1124/jpet.113.207670.
van Zwieten PA, Timmermans PB. Centrally mediated hypotensive activity of B-HT 933 upon infusion via the cat's vertebral artery. Pharmacology. 1983, 21 (5): 327–332. PMC 1427667 . PMID 7433512. doi:10.1111/j.1365-2125.1983.tb00311.x.
Arnsten AF. The use of α-2A adrenergic agonists for the treatment of attention-deficit/hyperactivity disorder. Expert Review of Neurotherapeutics. October 2010, 10 (10): 1595–1605. PMC 3143019 . PMID 20925474. doi:10.1586/ern.10.133.
Wang M, Ramos BP, Paspalas CD, Shu Y, Simen A, Duque A, Vijayraghavan S, Brennan A, Dudley A, Nou E, Mazer JA, McCormick DA, Arnsten AF. Alpha2A-adrenoceptors strengthen working memory networks by inhibiting cAMP-HCN channel signaling in prefrontal cortex. Cell. April 2007, 129 (2): 397–410. PMID 17448997. S2CID 741677. doi:10.1016/j.cell.2007.03.015 .
Mladěnka P, Applová L, Patočka J, Costa VM, Remiao F, Pourová J, Mladěnka A, Karlíčková J, Jahodář L, Vopršalová M, Varner KJ, Štěrba M. Comprehensive review of cardiovascular toxicity of drugs and related agents. Med Res Rev. July 2018, 38 (4): 1332–1403. PMC 6033155 . PMID 29315692. doi:10.1002/med.21476. The list of valvulopathic drugs is short and can be seen in Table 7. According to a recent analysis, other drugs, in particular guanfacine, might possess some risk, but clinical data are yet not available.368–370
Kiechel JR. Pharmacokinetics and metabolism of guanfacine in man: a review. British Journal of Clinical Pharmacology. 1980, 10 (Suppl 1): 25S–32S. PMC 1430131 . PMID 6994775. doi:10.1111/j.1365-2125.1980.tb04901.x.
Kirch W, Köhler H, Braun W. Elimination of guanfacine in patients with normal and impaired renal function. British Journal of Clinical Pharmacology. 1980, 10 (Suppl 1): 33S–35S. PMC 1430110 . PMID 6994776. doi:10.1111/j.1365-2125.1980.tb04902.x.
Connor DF, Grasso DJ, Slivinsky MD, Pearson GS, Banga A. An open-label study of guanfacine extended release for traumatic stress related symptoms in children and adolescents. Journal of Child and Adolescent Psychopharmacology. May 2013, 23 (4): 244–251. PMC 3657282 . PMID 23683139. doi:10.1089/cap.2012.0119.
Belkin MR, Schwartz TL. Alpha-2 receptor agonists for the treatment of posttraumatic stress disorder. Drugs in Context. 2015, 4: 212286. PMC 4544272 . PMID 26322115. doi:10.7573/dic.212286.
Sofuoglu M, Sewell RA. Norepinephrine and stimulant addiction. Addiction Biology. April 2009, 14 (2): 119–129. PMC 2657197 . PMID 18811678. doi:10.1111/j.1369-1600.2008.00138.x.
McKee SA, Potenza MN, Kober H, Sofuoglu M, Arnsten AF, Picciotto MR, Weinberger AH, Ashare R, Sinha R. A translational investigation targeting stress-reactivity and prefrontal cognitive control with guanfacine for smoking cessation. Journal of Psychopharmacology. March 2015, 29 (3): 300–311. PMC 4376109 . PMID 25516371. doi:10.1177/0269881114562091.
Arnsten AF. Guanfacine's mechanism of action in treating prefrontal cortical disorders: Successful translation across species. Neurobiol Learn Mem. December 2020, 176: 107327. PMC 7567669 . PMID 33075480. doi:10.1016/j.nlm.2020.107327.
Fesharaki Zadeh A, Arnsten AF, Wang M. Scientific Rationale for the Treatment of Cognitive Deficits from Long COVID. Neurol Int. May 2023, 15 (2): 725–742. PMC 10303664 . PMID 37368329. doi:10.3390/neurolint15020045 .
Arnsten AF, Ishizawa Y, Xie Z. Scientific rationale for the use of α2A-adrenoceptor agonists in treating neuroinflammatory cognitive disorders. Mol Psychiatry. April 2023: 1–13. PMC 10080530 . PMID 37029295. doi:10.1038/s41380-023-02057-4.
Fesharaki-Zadeh, Arman; Lowe, Naomi; Arnsten, Amy F.T. Clinical experience with the α2A-adrenoceptor agonist, guanfacine, and N-acetylcysteine for the treatment of cognitive deficits in "Long-COVID19". Neuroimmunology Reports. 2023, 3: 100154. PMC 9691274 . doi:10.1016/j.nerep.2022.100154.

drugs.com

Guanfacine Monograph for Professionals. Drugs.com. American Society of Health-System Pharmacists. [2019-03-18]. （原始内容存档于2018-01-15）（英语）.

europa.eu

ema.europa.eu

European Medicines Agency: Intuniv. Europa (web portal). October 2015 [2016-02-03]. （原始内容存档于2018-08-16）.

fda.gov

accessdata.fda.gov

Patient Information. INTUNIV (in-TOO-niv) (guanfacine). Extended-Release Tablets (PDF). FDA.gov. [2022-10-12]. （原始内容存档 (PDF)于2022-10-13）.
Drugs@FDA: FDA-Approved Drugs. [2024-02-22]. （原始内容存档于2017-06-29）.

harvard.edu

ui.adsabs.harvard.edu

Catalá-López F, Hutton B, Núñez-Beltrán A, Page MJ, Ridao M, Macías Saint-Gerons D, Catalá MA, Tabarés-Seisdedos R, Moher D. The pharmacological and non-pharmacological treatment of attention deficit hyperactivity disorder in children and adolescents: A systematic review with network meta-analyses of randomised trials. PLOS ONE. 2017, 12 (7): e0180355. Bibcode:2017PLoSO..1280355C. PMC 5507500 . PMID 28700715. doi:10.1371/journal.pone.0180355 .

ijest.org

Tardner, Paul. A Comprehensive Literature Review on Guanfacine as a Potential Treatment for Attention-Deficit/Hyperactivity Disorder (ADHD). International Journal of Environmental Science and Technology. May 2023 [2024-02-22]. （原始内容存档于2023-09-21）.

medicines.org.uk

Intuniv 1 mg, 2 mg, 3 mg, 4 mg prolonged-release tablets - Summary of Product Characteristics. UK Electronic Medicines Compendium. June 2017 [2017-07-07]. （原始内容存档于2018-01-15）.

medscape.com

reference.medscape.com

guanfacine (Rx) - Intuniv, Tenex. Medscape Reference. WebMD. [2013-11-09]. （原始内容存档于2019-05-18）.

nih.gov

ncbi.nlm.nih.gov

Kornfield R, Watson S, Higashi AS, Conti RM, Dusetzina SB, Garfield CF, Dorsey ER, Huskamp HA, Alexander GC. Effects of FDA advisories on the pharmacologic treatment of ADHD, 2004-2008. Psychiatric Services. April 2013, 64 (4): 339–346. PMC 4023684 . PMID 23318985. doi:10.1176/appi.ps.201200147.
Zito JM, Derivan AT, Kratochvil CJ, Safer DJ, Fegert JM, Greenhill LL. Off-label psychopharmacologic prescribing for children: history supports close clinical monitoring. Child and Adolescent Psychiatry and Mental Health //www.ncbi.nlm.nih.gov/pmc/articles/PMC2566553 |PMC=缺少标题 (帮助). September 2008, 2 (1): 24. PMC 2566553 . PMID 18793403. doi:10.1186/1753-2000-2-24 .
Clemow, DB; Walker, DJ. The potential for misuse and abuse of medications in ADHD: a review.. Postgraduate Medicine. September 2014, 126 (5): 64–81. PMID 25295651. S2CID 207580823. doi:10.3810/pgm.2014.09.2801.
Arnsten AF, Jin LE. Guanfacine for the treatment of cognitive disorders: a century of discoveries at Yale. The Yale Journal of Biology and Medicine. March 2012, 85 (1): 45–58. PMC 3313539 . PMID 22461743.
Radonjić NV, Bellato A, Khoury NM, Cortese S, Faraone SV. Nonstimulant Medications for Attention-Deficit/Hyperactivity Disorder (ADHD) in Adults: Systematic Review and Meta-analysis. CNS Drugs. May 2023, 37 (5): 381–397. PMID 37166701. S2CID 258616507. doi:10.1007/s40263-023-01005-8.
Yu S, Shen S, Tao M. Guanfacine for the Treatment of Attention-Deficit Hyperactivity Disorder: An Updated Systematic Review and Meta-Analysis. J Child Adolesc Psychopharmacol. March 2023, 33 (2): 40–50. PMID 36944092. S2CID 257664282. doi:10.1089/cap.2022.0038.
Catalá-López F, Hutton B, Núñez-Beltrán A, Page MJ, Ridao M, Macías Saint-Gerons D, Catalá MA, Tabarés-Seisdedos R, Moher D. The pharmacological and non-pharmacological treatment of attention deficit hyperactivity disorder in children and adolescents: A systematic review with network meta-analyses of randomised trials. PLOS ONE. 2017, 12 (7): e0180355. Bibcode:2017PLoSO..1280355C. PMC 5507500 . PMID 28700715. doi:10.1371/journal.pone.0180355 .
Pringsheim T, Hirsch L, Gardner D, Gorman DA. The pharmacological management of oppositional behaviour, conduct problems, and aggression in children and adolescents with attention-deficit hyperactivity disorder, oppositional defiant disorder, and conduct disorder: a systematic review and meta-analysis. Part 1: psychostimulants, alpha-2 agonists, and atomoxetine. Can J Psychiatry. February 2015, 60 (2): 42–51. PMC 4344946 . PMID 25886655. doi:10.1177/070674371506000202.
Padilha SC, Virtuoso S, Tonin FS, Borba HH, Pontarolo R. Efficacy and safety of drugs for attention deficit hyperactivity disorder in children and adolescents: a network meta-analysis. Eur Child Adolesc Psychiatry. October 2018, 27 (10): 1335–1345. PMID 29460165. S2CID 3402756. doi:10.1007/s00787-018-1125-0.
Morrow BA, George TP, Roth RH. Noradrenergic alpha-2 agonists have anxiolytic-like actions on stress-related behavior and mesoprefrontal dopamine biochemistry. Brain Research. November 2004, 1027 (1–2): 173–178. PMID 15494168. S2CID 7066842. doi:10.1016/j.brainres.2004.08.057.
Arnsten AF, Raskind MA, Taylor FB, Connor DF. The Effects of Stress Exposure on Prefrontal Cortex: Translating Basic Research into Successful Treatments for Post-Traumatic Stress Disorder. Neurobiology of Stress. January 2015, 1: 89–99. PMC 4244027 . PMID 25436222. doi:10.1016/j.ynstr.2014.10.002.
Kozaric-Kovacic D. Psychopharmacotherapy of posttraumatic stress disorder. Croatian Medical Journal. August 2008, 49 (4): 459–475. PMC 2525822 . PMID 18716993. doi:10.3325/cmj.2008.4.459.
Kaminer D, Seedat S, Stein DJ. Post-traumatic stress disorder in children. World Psychiatry. June 2005, 4 (2): 121–125. PMC 1414752 . PMID 16633528.
Jerie P. Clinical experience with guanfacine in long-term treatment of hypertension. Part II: adverse reactions to guanfacine. British Journal of Clinical Pharmacology. 1980, 10 (Suppl 1): 157S–164S. PMC 1430125 . PMID 6994770. doi:10.1111/j.1365-2125.1980.tb04924.x.
Anand S, Tong H, Besag FM, Chan EW, Cortese S, Wong IC. Safety, Tolerability and Efficacy of Drugs for Treating Behavioural Insomnia in Children with Attention-Deficit/Hyperactivity Disorder: A Systematic Review with Methodological Quality Assessment. Paediatr Drugs. June 2017, 19 (3): 235–250 [2024-02-22]. PMID 28391425. S2CID 2220464. doi:10.1007/s40272-017-0224-6. （原始内容存档于2024-02-22）.
Rugino TA. Effect on Primary Sleep Disorders When Children With ADHD Are Administered Guanfacine Extended Release. J Atten Disord. January 2018, 22 (1): 14–24. PMID 25376194. S2CID 22675882. doi:10.1177/1087054714554932.
Solmi M, Fornaro M, Ostinelli EG, Zangani C, Croatto G, Monaco F, Krinitski D, Fusar-Poli P, Correll CU. Safety of 80 antidepressants, antipsychotics, anti-attention-deficit/hyperactivity medications and mood stabilizers in children and adolescents with psychiatric disorders: a large scale systematic meta-review of 78 adverse effects. World Psychiatry. June 2020, 19 (2): 214–232. PMC 7215080 . PMID 32394557. doi:10.1002/wps.20765.
Jasper JR, Lesnick JD, Chang LK, Yamanishi SS, Chang TK, Hsu SA, et al. Ligand efficacy and potency at recombinant alpha2 adrenergic receptors: agonist-mediated [35S]GTPgammaS binding. Biochemical Pharmacology. April 1998, 55 (7): 1035–1043. PMID 9605427. doi:10.1016/s0006-2952(97)00631-x.
Uhlén S, Porter AC, Neubig RR. The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors. The Journal of Pharmacology and Experimental Therapeutics. December 1994, 271 (3): 1558–1565. PMID 7996470.
Bender AM, Parr LC, Livingston WB, Lindsley CW, Merryman WD. 2B Determined: The Future of the Serotonin Receptor 2B in Drug Discovery. J Med Chem. August 2023, 66 (16): 11027–11039. PMID 37584406. S2CID 260924858. doi:10.1021/acs.jmedchem.3c01178. These results strongly indicate substantial risks for treatments involving 5-HT2B agonists, and it has been recommended that all serotonergic drugs be screened for this functional profile.43,59 [...] Additionally, there are cases of marketed drugs that were only later determined to have 5-HT2B activity. Of particular note is guanfacine, an FDA-approved medication for the treatment of attention deficit hyperactivity disorder (ADHD) that possesses potent 5-HT2B agonist activity in functional readouts to a similar degree as known valvulopathogens.66
Hutcheson JD, Setola V, Roth BL, Merryman WD. Serotonin receptors and heart valve disease--it was meant 2B. Pharmacol Ther. November 2011, 132 (2): 146–57. PMC 3179857 . PMID 21440001. doi:10.1016/j.pharmthera.2011.03.008.
Huang XP, Setola V, Yadav PN, Allen JA, Rogan SC, Hanson BJ, Revankar C, Robers M, Doucette C, Roth BL. Parallel functional activity profiling reveals valvulopathogens are potent 5-hydroxytryptamine(2B) receptor agonists: implications for drug safety assessment. Molecular Pharmacology. October 2009, 76 (4): 710–722. PMC 2769050 . PMID 19570945. doi:10.1124/mol.109.058057.
Unett DJ, Gatlin J, Anthony TL, Buzard DJ, Chang S, Chen C, Chen X, Dang HT, Frazer J, Le MK, Sadeque AJ, Xing C, Gaidarov I. Kinetics of 5-HT2B receptor signaling: profound agonist-dependent effects on signaling onset and duration. J Pharmacol Exp Ther. December 2013, 347 (3): 645–59. PMID 24049061. S2CID 8013309. doi:10.1124/jpet.113.207670.
van Zwieten PA, Timmermans PB. Centrally mediated hypotensive activity of B-HT 933 upon infusion via the cat's vertebral artery. Pharmacology. 1983, 21 (5): 327–332. PMC 1427667 . PMID 7433512. doi:10.1111/j.1365-2125.1983.tb00311.x.
Arnsten AF. The use of α-2A adrenergic agonists for the treatment of attention-deficit/hyperactivity disorder. Expert Review of Neurotherapeutics. October 2010, 10 (10): 1595–1605. PMC 3143019 . PMID 20925474. doi:10.1586/ern.10.133.
Wang M, Ramos BP, Paspalas CD, Shu Y, Simen A, Duque A, Vijayraghavan S, Brennan A, Dudley A, Nou E, Mazer JA, McCormick DA, Arnsten AF. Alpha2A-adrenoceptors strengthen working memory networks by inhibiting cAMP-HCN channel signaling in prefrontal cortex. Cell. April 2007, 129 (2): 397–410. PMID 17448997. S2CID 741677. doi:10.1016/j.cell.2007.03.015 .
Mladěnka P, Applová L, Patočka J, Costa VM, Remiao F, Pourová J, Mladěnka A, Karlíčková J, Jahodář L, Vopršalová M, Varner KJ, Štěrba M. Comprehensive review of cardiovascular toxicity of drugs and related agents. Med Res Rev. July 2018, 38 (4): 1332–1403. PMC 6033155 . PMID 29315692. doi:10.1002/med.21476. The list of valvulopathic drugs is short and can be seen in Table 7. According to a recent analysis, other drugs, in particular guanfacine, might possess some risk, but clinical data are yet not available.368–370
Kiechel JR. Pharmacokinetics and metabolism of guanfacine in man: a review. British Journal of Clinical Pharmacology. 1980, 10 (Suppl 1): 25S–32S. PMC 1430131 . PMID 6994775. doi:10.1111/j.1365-2125.1980.tb04901.x.
Kirch W, Köhler H, Braun W. Elimination of guanfacine in patients with normal and impaired renal function. British Journal of Clinical Pharmacology. 1980, 10 (Suppl 1): 33S–35S. PMC 1430110 . PMID 6994776. doi:10.1111/j.1365-2125.1980.tb04902.x.
Scholtysik G. Proceedings: Inhibition of effects of accelerator nerve stimulation in cats and rabbits by BS 100-141 and guanabenz. Naunyn Schmiedebergs Arch Pharmacol. 1974, 282 (Suppl): suppl 282:R86. PMID 4276642.
Bream JB, Lauener H, Picard CW, Scholtysik G, White TG. Substituted phenylacetylguanidines: a new class of antihypertensive agents. Arzneimittelforschung. October 1975, 25 (10): 1477–82. PMID 1243024.
Saameli K, Scholtysik G, Waite R. Pharmacology of BS 100-141, a centrally acting antihypertensive drug. Clin Exp Pharmacol Physiol. 1975,. Suppl 2: 207–12. PMID 241524.
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Boland RJ, Verduin ML, Sadock BJ. Ruiz P , 编. Kaplan & Sadock's Concise Textbook of Clinical Psychiatry 5th. Philadelphia. 2023: 1811–1812 [2023-01-12]. ISBN 978-1-9751-6748-6. OCLC 1264172789. （原始内容存档于2023-02-08）.