Seal, L. J.; Franklin, S.; Richards, C.; Shishkareva, A.; Sinclaire, C.; Barrett, J. Predictive Markers for Mammoplasty and a Comparison of Side Effect Profiles in Transwomen Taking Various Hormonal Regimens. The Journal of Clinical Endocrinology & Metabolism. 2012, 97 (12): 4422–4428. ISSN 0021-972X. doi:10.1210/jc.2012-2030.
Boccardo, Francesco. Hormone therapy of prostate cancer: is there a role for antiandrogen monotherapy?. Critical Reviews in Oncology/Hematology. 2000, 35 (2): 121–132. ISSN 1040-8428. doi:10.1016/S1040-8428(00)00051-2.
Christians U, Schmitz V, Haschke M. Functional interactions between P-glycoprotein and CYP3A in drug metabolism. Expert Opin Drug Metab Toxicol. December 2005, 1 (4): 641–54. PMID 16863430. doi:10.1517/17425255.1.4.641.
Rabe T, Kowald A, Ortmann J, Rehberger-Schneider S. Inhibition of skin 5 alpha-reductase by oral contraceptive progestins in vitro. Gynecol. Endocrinol. 2000, 14 (4): 223–30. PMID 11075290. doi:10.3109/09513590009167685.
Tartagni M, Schonauer LM, De Salvia MA, Cicinelli E, De Pergola G, D'Addario V. Comparison of Diane 35 and Diane 35 plus finasteride in the treatment of hirsutism. Fertil. Steril. 2000, 73 (4): 718–23. PMID 10731531. doi:10.1016/s0015-0282(99)00633-0.
Sahin Y, Dilber S, Keleştimur F. Comparison of Diane 35 and Diane 35 plus finasteride in the treatment of hirsutism. Fertil. Steril. 2001, 75 (3): 496–500. PMID 11239530. doi:10.1016/s0015-0282(00)01764-7.
Gutiérrez M, Menéndez L, Ruiz-Gayo M, Hidalgo A, Baamonde A. Cyproterone acetate displaces opiate binding in mouse brain. Eur. J. Pharmacol. 1997, 328 (1): 99–102. PMID 9203575. doi:10.1016/s0014-2999(97)83034-8.
Neumann F, Kalmus J. Cyproterone acetate in the treatment of sexual disorders: pharmacological base and clinical experience. Exp. Clin. Endocrinol. 1991, 98 (2): 71–80. PMID 1838080. doi:10.1055/s-0029-1211103.
Herbert DC, Schuppler J, Poggel A, Günzel P, El Etreby MF. Effect of cyproterone acetate on prolactin secretion in the female Rhesus monkey. Cell Tissue Res. 1977, 183 (1): 51–60. PMID 411573. doi:10.1007/bf00219991.
Rost A, Schmidt-Gollwitzer M, Hantelmann W, Brosig W. Cyproterone acetate, testosterone, LH, FSH, and prolactin levels in plasma after intramuscular application of cyproterone acetate in patients with prostatic cancer. Prostate. 1981, 2 (3): 315–22. PMID 6458025. doi:10.1002/pros.2990020310.
Grunwald K, Rabe T, Schlereth G, Runnebaum B. [Serum hormones before and during therapy with cyproterone acetate and spironolactone in patients with androgenization]. Geburtshilfe Frauenheilkd. 1994, 54 (11): 634–45. PMID 8719011. doi:10.1055/s-2007-1022355(德语).
Girard J, Baumann JB, Bühler U, Zuppinger K, Haas HG, Staub JJ, Wyss HI. Cyproteroneacetate and ACTH adrenal function. J. Clin. Endocrinol. Metab. 1978, 47 (3): 581–6. PMID 233676. doi:10.1210/jcem-47-3-581.
Panesar NS, Herries DG, Stitch SR. Effects of cyproterone and cyproterone acetate on the adrenal gland in the rat: studies in vivo and in vitro. J. Endocrinol. 1979, 80 (2): 229–38. PMID 438696. doi:10.1677/joe.0.0800229.
El Etreby MF. Effect of cyproterone acetate, levonorgestrel and progesterone on adrenal glands and reproductive organs in the beagle bitch. Cell Tissue Res. 1979, 200 (2): 229–43. PMID 487397. doi:10.1007/bf00236416.
Hague WM, Munro DS, Sawers RS, Duncan SL, Honour JW. Long-term effects of cyproterone acetate on the pituitary adrenal axis in adult women. Br J Obstet Gynaecol. 1982, 89 (12): 981–4. PMID 6216913. doi:10.1111/j.1471-0528.1982.tb04650.x.
Mercier L, Miller PA, Simons SS. Antiglucocorticoid steroids have increased agonist activity in those hepatoma cell lines that are more sensitive to glucocorticoids. J. Steroid Biochem. 1986, 25 (1): 11–20. PMID 2875214. doi:10.1016/0022-4731(86)90275-x.
Poulin R, Baker D, Poirier D, Labrie F. Multiple actions of synthetic 'progestins' on the growth of ZR-75-1 human breast cancer cells: an in vitro model for the simultaneous assay of androgen, progestin, estrogen, and glucocorticoid agonistic and antagonistic activities of steroids. Breast Cancer Research and Treatment. 1991, 17 (3): 197–210. PMID 1645605. doi:10.1007/BF01806369.
Pham-Huu-Trung MT, de Smitter N, Bogyo A, Girard F. Effects of cyproterone acetate on adrenal steroidogenesis in vitro. Horm. Res. 1984, 20 (2): 108–15. PMID 6237971. doi:10.1159/000179982.
Lambert A, Mitchell RM, Robertson WR. On the site of action of the anti-adrenal steroidogenic effect of cyproterone acetate. Biochem. Pharmacol. 1985, 34 (12): 2091–5. PMID 2988566. doi:10.1016/0006-2952(85)90400-9.
Heinze F, Teller WM, Fehm HL, Joos A. The effect of cyproterone acetate on adrenal cortical function in children with precocious puberty. Eur. J. Pediatr. 1978, 128 (2): 81–8. PMID 208851. doi:10.1007/bf00496993.
Frith RG, Phillipou G. 15-Hydroxycyproterone acetate and cyproterone acetate levels in plasma and urine. J. Chromatogr. 1985, 338 (1): 179–86. PMID 3160716. doi:10.1016/0378-4347(85)80082-7.
Broulik PD, Starka L. Corticosteroid-like effect of cyproterone and cyproterone acetate in mice. Experientia. 1975, 31 (11): 1364–5. PMID 1204803. doi:10.1007/bf01945829.
van Wayjen RG, van den Ende A. Effect of cyproterone acetate on pituitary-adrenocortical function in man. Acta Endocrinol. 1981, 96 (1): 112–22. PMID 6257015. doi:10.1530/acta.0.0960112.
Schürmeyer T, Graff J, Senge T, Nieschlag E. Effect of oestrogen or cyproterone acetate treatment on adrenocortical function in prostate carcinoma patients. Acta Endocrinol. 1986, 111 (3): 360–7. PMID 2421511. doi:10.1530/acta.0.1110360.
van Wayjen RG, van den Ende A. Experience in the long-term treatment of patients with hirsutism and/or acne with cyproterone acetate-containing preparations: efficacy, metabolic and endocrine effects. Exp. Clin. Endocrinol. Diabetes. 1995, 103 (4): 241–51. PMID 7584530. doi:10.1055/s-0029-1211357.
Holdaway IM, Croxson MS, Evans MC, France J, Sheehan A, Wilson T, Ibbertson HK. Effect of cyproterone acetate on glucocorticoid secretion in patients treated for hirsutism. Acta Endocrinol. 1983, 104 (2): 222–6. PMID 6227191. doi:10.1530/acta.0.1040222.
Christians U, Schmitz V, Haschke M. Functional interactions between P-glycoprotein and CYP3A in drug metabolism. Expert Opin Drug Metab Toxicol. December 2005, 1 (4): 641–54. PMID 16863430. doi:10.1517/17425255.1.4.641.
Rabe T, Kowald A, Ortmann J, Rehberger-Schneider S. Inhibition of skin 5 alpha-reductase by oral contraceptive progestins in vitro. Gynecol. Endocrinol. 2000, 14 (4): 223–30. PMID 11075290. doi:10.3109/09513590009167685.
Stárka L, Sulcová J, Broulík P. Effect of cyproterone acetate on the action and metabolism of testosterone in the mouse kidney. Endokrinologie. 1976, 68 (2): 155–63. PMID 1009901.
Tartagni M, Schonauer LM, De Salvia MA, Cicinelli E, De Pergola G, D'Addario V. Comparison of Diane 35 and Diane 35 plus finasteride in the treatment of hirsutism. Fertil. Steril. 2000, 73 (4): 718–23. PMID 10731531. doi:10.1016/s0015-0282(99)00633-0.
Sahin Y, Dilber S, Keleştimur F. Comparison of Diane 35 and Diane 35 plus finasteride in the treatment of hirsutism. Fertil. Steril. 2001, 75 (3): 496–500. PMID 11239530. doi:10.1016/s0015-0282(00)01764-7.
Gutiérrez M, Menéndez L, Ruiz-Gayo M, Hidalgo A, Baamonde A. Cyproterone acetate displaces opiate binding in mouse brain. Eur. J. Pharmacol. 1997, 328 (1): 99–102. PMID 9203575. doi:10.1016/s0014-2999(97)83034-8.
Neumann F, Kalmus J. Cyproterone acetate in the treatment of sexual disorders: pharmacological base and clinical experience. Exp. Clin. Endocrinol. 1991, 98 (2): 71–80. PMID 1838080. doi:10.1055/s-0029-1211103.
Schröder FH. Antiandrogens as monotherapy for prostate cancer. Eur. Urol. 1998,. 34 Suppl 3: 12–7. PMID 9854190.
Herbert DC, Schuppler J, Poggel A, Günzel P, El Etreby MF. Effect of cyproterone acetate on prolactin secretion in the female Rhesus monkey. Cell Tissue Res. 1977, 183 (1): 51–60. PMID 411573. doi:10.1007/bf00219991.
Donald RA, Espiner EA, Cowles RJ, Fazackerley JE. The effect of cyproterone acetate on the plasma gonadotrophin response to gonadotrophin releasing hormone. Acta Endocrinologica. April 1976, 81 (4): 680–4. PMID 769466.
Rost A, Schmidt-Gollwitzer M, Hantelmann W, Brosig W. Cyproterone acetate, testosterone, LH, FSH, and prolactin levels in plasma after intramuscular application of cyproterone acetate in patients with prostatic cancer. Prostate. 1981, 2 (3): 315–22. PMID 6458025. doi:10.1002/pros.2990020310.
Grunwald K, Rabe T, Schlereth G, Runnebaum B. [Serum hormones before and during therapy with cyproterone acetate and spironolactone in patients with androgenization]. Geburtshilfe Frauenheilkd. 1994, 54 (11): 634–45. PMID 8719011. doi:10.1055/s-2007-1022355(德语).
Schürenkämper P, Lisse K. Effects of cyproterone on the steroid biosynthesis in the human ovary in vitro. Endokrinologie. 1982, 80 (3): 281–6. PMID 7166160.
Girard J, Baumann JB, Bühler U, Zuppinger K, Haas HG, Staub JJ, Wyss HI. Cyproteroneacetate and ACTH adrenal function. J. Clin. Endocrinol. Metab. 1978, 47 (3): 581–6. PMID 233676. doi:10.1210/jcem-47-3-581.
Panesar NS, Herries DG, Stitch SR. Effects of cyproterone and cyproterone acetate on the adrenal gland in the rat: studies in vivo and in vitro. J. Endocrinol. 1979, 80 (2): 229–38. PMID 438696. doi:10.1677/joe.0.0800229.
El Etreby MF. Effect of cyproterone acetate, levonorgestrel and progesterone on adrenal glands and reproductive organs in the beagle bitch. Cell Tissue Res. 1979, 200 (2): 229–43. PMID 487397. doi:10.1007/bf00236416.
Hague WM, Munro DS, Sawers RS, Duncan SL, Honour JW. Long-term effects of cyproterone acetate on the pituitary adrenal axis in adult women. Br J Obstet Gynaecol. 1982, 89 (12): 981–4. PMID 6216913. doi:10.1111/j.1471-0528.1982.tb04650.x.
Mercier L, Miller PA, Simons SS. Antiglucocorticoid steroids have increased agonist activity in those hepatoma cell lines that are more sensitive to glucocorticoids. J. Steroid Biochem. 1986, 25 (1): 11–20. PMID 2875214. doi:10.1016/0022-4731(86)90275-x.
Poulin R, Baker D, Poirier D, Labrie F. Multiple actions of synthetic 'progestins' on the growth of ZR-75-1 human breast cancer cells: an in vitro model for the simultaneous assay of androgen, progestin, estrogen, and glucocorticoid agonistic and antagonistic activities of steroids. Breast Cancer Research and Treatment. 1991, 17 (3): 197–210. PMID 1645605. doi:10.1007/BF01806369.
Pham-Huu-Trung MT, de Smitter N, Bogyo A, Girard F. Effects of cyproterone acetate on adrenal steroidogenesis in vitro. Horm. Res. 1984, 20 (2): 108–15. PMID 6237971. doi:10.1159/000179982.
Lambert A, Mitchell RM, Robertson WR. On the site of action of the anti-adrenal steroidogenic effect of cyproterone acetate. Biochem. Pharmacol. 1985, 34 (12): 2091–5. PMID 2988566. doi:10.1016/0006-2952(85)90400-9.
Heinze F, Teller WM, Fehm HL, Joos A. The effect of cyproterone acetate on adrenal cortical function in children with precocious puberty. Eur. J. Pediatr. 1978, 128 (2): 81–8. PMID 208851. doi:10.1007/bf00496993.
Frith RG, Phillipou G. 15-Hydroxycyproterone acetate and cyproterone acetate levels in plasma and urine. J. Chromatogr. 1985, 338 (1): 179–86. PMID 3160716. doi:10.1016/0378-4347(85)80082-7.
Bhargava AS, Kapp JF, Poggel HA, Heinick J, Nieuweboer B, Günzel P. Effect of cyproterone acetate and its metabolites on the adrenal function in man, rhesus monkey and rat. Arzneimittelforschung. 1981, 31 (6): 1005–9. PMID 6266428.
Broulik PD, Starka L. Corticosteroid-like effect of cyproterone and cyproterone acetate in mice. Experientia. 1975, 31 (11): 1364–5. PMID 1204803. doi:10.1007/bf01945829.
van Wayjen RG, van den Ende A. Effect of cyproterone acetate on pituitary-adrenocortical function in man. Acta Endocrinol. 1981, 96 (1): 112–22. PMID 6257015. doi:10.1530/acta.0.0960112.
Schürmeyer T, Graff J, Senge T, Nieschlag E. Effect of oestrogen or cyproterone acetate treatment on adrenocortical function in prostate carcinoma patients. Acta Endocrinol. 1986, 111 (3): 360–7. PMID 2421511. doi:10.1530/acta.0.1110360.
van Wayjen RG, van den Ende A. Experience in the long-term treatment of patients with hirsutism and/or acne with cyproterone acetate-containing preparations: efficacy, metabolic and endocrine effects. Exp. Clin. Endocrinol. Diabetes. 1995, 103 (4): 241–51. PMID 7584530. doi:10.1055/s-0029-1211357.
Holdaway IM, Croxson MS, Evans MC, France J, Sheehan A, Wilson T, Ibbertson HK. Effect of cyproterone acetate on glucocorticoid secretion in patients treated for hirsutism. Acta Endocrinol. 1983, 104 (2): 222–6. PMID 6227191. doi:10.1530/acta.0.1040222.
Tamm J, Voigt KD, Schönrock M, Ludwig E. The effect of orally administered cyproterone on the serum production in human subjects. Acta Endocrinol (Copenh). Jan 1970, 63 (1): 50–8. PMID 5467021.
Seal, L. J.; Franklin, S.; Richards, C.; Shishkareva, A.; Sinclaire, C.; Barrett, J. Predictive Markers for Mammoplasty and a Comparison of Side Effect Profiles in Transwomen Taking Various Hormonal Regimens. The Journal of Clinical Endocrinology & Metabolism. 2012, 97 (12): 4422–4428. ISSN 0021-972X. doi:10.1210/jc.2012-2030.
Boccardo, Francesco. Hormone therapy of prostate cancer: is there a role for antiandrogen monotherapy?. Critical Reviews in Oncology/Hematology. 2000, 35 (2): 121–132. ISSN 1040-8428. doi:10.1016/S1040-8428(00)00051-2.